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NameHistamine H1 receptor
Kindprotein
OrganismHuman
Polypeptides
NameUniProt ID
Histamine H1 receptorP35367 Details

Drugs

DrugBank IDNameDrug groupPharmacological action?ActionsDetails
DB00283ClemastineapprovedyesantagonistDetails
DB00341CetirizineapprovedyesantagonistDetails
DB00342TerfenadinewithdrawnyesantagonistDetails
DB00354BuclizineapprovedyesantagonistDetails
DB00366DoxylamineapprovedyesantagonistDetails
DB00405DexbrompheniramineapprovedyesantagonistDetails
DB00427TriprolidineapprovedyesantagonistDetails
DB00455LoratadineapprovedyesantagonistDetails
DB00557HydroxyzineapprovedyesantagonistDetails
DB00568CinnarizineapprovedyesantagonistDetails
DB00637Astemizoleapproved, withdrawnyesantagonistDetails
DB00667Histamine PhosphateapprovedyesagonistDetails
DB00719AzatadineapprovedyesantagonistDetails
DB00734Risperidoneapproved, investigationalunknownantagonistDetails
DB00737MeclizineapprovedyesantagonistDetails
DB00748CarbinoxamineapprovedyesantagonistDetails
DB00768OlopatadineapprovedyesantagonistDetails
DB00792TripelennamineapprovedyesantagonistDetails
DB00835BrompheniramineapprovedyesantagonistDetails
DB00902MethdilazineapprovedyesantagonistDetails
DB00934MaprotilineapprovednoantagonistDetails
DB00950FexofenadineapprovedyesantagonistDetails
DB00967Desloratadineapproved, investigationalyesantagonistDetails
DB00972AzelastineapprovedyesantagonistDetails
DB00985DimenhydrinateapprovedyesantagonistDetails
DB01071MequitazineapprovedyesantagonistDetails
DB01075DiphenhydramineapprovedyesantagonistDetails
DB01084EmedastineapprovedyesantagonistDetails
DB01114ChlorphenamineapprovedyesantagonistDetails
DB01146DiphenylpyralineapprovedyesantagonistDetails
DB01176CyclizineapprovedyesantagonistDetails
DB01237BromodiphenhydramineapprovedyesantagonistDetails
DB01246AlimemazineapprovedyesantagonistDetails
DB00246ZiprasidoneapprovednoantagonistDetails
DB00334Olanzapineapproved, investigationalunknownantagonistDetails
DB00363ClozapineapprovednoantagonistDetails
DB00420PromazineunknownantagonistDetails
DB00656Trazodoneapproved, investigationalunknownantagonistDetails
DB00767BenzquinamidewithdrawnyesantagonistDetails
DB00777PropiomazineapprovedyesantagonistDetails
DB00920KetotifenapprovedyesantagonistDetails
DB01069PromethazineapprovedyesantagonistDetails
DB01106LevocabastineapprovedyesantagonistDetails
DB01142DoxepinapprovedyesantagonistDetails
DB01151DesipramineapprovednoantagonistDetails
DB01173OrphenadrineapprovedyesantagonistDetails
DB01403MethotrimeprazineapprovedunknownantagonistDetails
DB01619PhenindamineapprovedyesantagonistDetails
DB01620PheniramineapprovedyesantagonistDetails
DB04837Clofedanolapproved, withdrawnyesantagonistDetails
DB04841FlunarizineapprovedunknownantagonistDetails
DB01615AceprometazineapprovedyesantagonistDetails
DB01239Chlorprothixeneapproved, withdrawnunknownantagonistDetails
DB00370MirtazapineapprovednoantagonistDetails
DB01224QuetiapineapprovedunknownantagonistDetails
DB00434CyproheptadineapprovedyesantagonistDetails
DB04890BepotastineapprovedyesantagonistDetails
DB00751Epinastineapproved, investigationalyesantagonistDetails
DB06148MianserinapprovedunknownantagonistDetails
DB04905TesmilifeneinvestigationalunknownantagonistDetails
DB05079HY10275investigationalunknownDetails
DB05345SO-101investigationalunknownDetails
DB05080OBE101investigationalunknownDetails
DB05492Epicept NP-1investigationalunknownDetails
DB06216AsenapineapprovedunknownantagonistDetails
DB06229ocaperidoneinvestigationalunknownDetails
DB00245BenzatropineapprovedunknownantagonistDetails
DB01267PaliperidoneapprovedunknownagonistDetails
DB01238Aripiprazoleapproved, investigationalnoantagonistDetails
DB00321AmitriptylineapprovednoantagonistDetails
DB00458ImipramineapprovednoantagonistDetails
DB00540NortriptylineapprovednoantagonistDetails
DB01175Escitalopramapproved, investigationalunknownantagonistDetails
DB00726TrimipramineapprovedunknownantagonistDetails
DB00797TolazolineapprovedunknownagonistDetails
DB06766AlcaftadineapprovedunknownantagonistDetails
DB08799AntazolineapprovedyesantagonistDetails
DB08800ChloropyramineapprovedyesantagonistDetails
DB08801DimetindeneapprovedyesantagonistDetails
DB08802IsothipendylapprovedyesantagonistDetails
DB06698BetahistineapprovedyesagonistDetails
DB06691MepyramineapprovedyesantagonistDetails
DB00477ChlorpromazineapprovedyesantagonistDetails
DB04946IloperidoneapprovedunknownantagonistDetails
DB00215CitalopramapprovedunknownbinderDetails
DB01624Zuclopenthixolexperimental, investigationalunknownantagonistDetails
DB08920Zuclopenthixol decanoateexperimental, investigationalunknownantagonistDetails
DB08919Zuclopenthixol acetateexperimental, investigationalunknownantagonistDetails
DB08936ChlorcyclizineapprovedyesantagonistDetails