Anti-Bacterial Agents

Name
Anti-Bacterial Agents
Accession Number
DBCAT000104
Description

Substances produced by microorganisms that can inhibit or suppress the growth of other microorganisms.

ATC Classification
Drugs
DrugDrug Description
Gramicidin DA bactericidal antibiotic used in the treatment of dermatological and ophthalmic infections.
ErythromycinA macrolide antibiotic used to treat and prevent a variety of bacterial infections.
CycloserineA broad-spectrum antibiotic used in the treatment of tuberculosis and certain urinary tract infections (UTI).
CapreomycinAn aminoglycoside antibiotic used as an adjunct drug in tuberculosis.
FramycetinAn aminoglycoside antibiotic used in various formulations and combinations with other agents to treat hemorrhoids, eye and ear infections, and to reduce nasal carriage of staphylococcus.
OxytetracyclineA tetracycline antibiotic used to treat a wide variety of susceptible bacterial infections.
RifabutinAn antibiotic used to treat mycobacterium avium complex disease in patients with HIV.
BacitracinA cyclic polypeptide antibiotic used to prevent wound infections, treat pneumonia and empyema in infants, and to treat skin and eye infections.
BenzylpenicillinA penicillin used for the treatment of infections caused by gram-positive cocci, in particular streptococcal infections. This form of penicillin is typically used in intravenous or long-acting injectable formulations due to poor oral absorption.
StreptomycinAn aminoglycoside antibiotic indicated to treat multi-drug resistant mycobacterium tuberculosis and various non-tuberculosis infections.
CandicidinUsed in the topical treatment of vulvovaginal candidiasis.
RifapentineAn antibiotic agent used in the treatment of pulmonary tuberculosis.
ParomomycinAn aminoglycoside antibiotic used in the treatment of acute and chronic intestinal amebiasis, and as an adjunct for the management of hepatic coma.
Fusidic acidA topical antibacterial agent used to prevent and treat mild to moderate skin infections caused by susceptible bacteria.
DihydrostreptomycinDihydrostreptomycin is an aminoglycoside antibiotic. In humans, the use of dihydrostreptomycin has been associated with ototoxicity. The FDA withdrew its approval for the use of all drug products containing dihydrostreptomycin...
MicronomicinMicronomicin is an aminoglycoside antibiotic which is marketed in Japan, and sold under the brand names Sagamicin and Luxomicina.
TyrothricinA topical antibiotic with broad spectrum activity against Gram positive bacteria and some fungal infections.
CarfecillinNot Annotated
MepartricinA medication indicated in the treatment of benign prostatic hyperplasia, vaginal candidiasis, or trichomoniasis.
NeomycinAn aminoglycoside antibiotic agent used orally and topically to treat a wide variety of infections in the body.
AzithromycinA macrolide antibiotic used to treat a variety of bacterial infections.
MoxifloxacinA fluoroquinolone antibiotic used to treat various bacterial infections.
MupirocinAn antibacterial ointment used to treat impetigo and secondary skin infections caused by Staphylococcus aureus and Streptococcus pyogenes.
ChloramphenicolA broad spectrum antibiotic that is effective against a variety of susceptible and serious bacterial infections but is not frequently used because of its high risk of bone marrow toxicity.
CiprofloxacinA second generation fluoroquinolone used to treat various susceptible bacterial infections.
TobramycinAn aminoglycoside antibiotic used to treat cystic fibrosis-associated bacterial, lower respiratory tract, urinary tract, eye, skin, bone, and skin structure infections.
TetracyclineAn antibiotic used to treat a wide variety of susceptible infections.
GentamicinAn aminoglycoside used to treat a wide variety of aerobic infections in the body.
MinocyclineA tetracycline analog used to treat a wide variety of infections in the body.
GatifloxacinA fourth generation fluoroquinolone used to treat a wide variety of infections in the body.
NorfloxacinA broad-spectrum fluoroquinolone antibiotic with variable activity against gram-positive and gram-negative bacteria. Typically reserved for the treatment of UTIs due to accumulation in the urine.
OfloxacinAn antibacterial agent used for the treatment of bacterial infections in many parts of the body, including the respiratory tract, kidney, skin, soft tissue, and urinary tract.
ClindamycinA lincosamide antibiotic used to treat serious infections caused by susceptible anaerobic, streptococcal, staphylococcal, and pneumococcal bacteria.
KanamycinAn aminoglycoside antibiotic agent used in the treatment of various infections caused by susceptible bacteria.
Amphotericin BAn antifungal used to treat fungal infections in neutropenic patients, cryptococcal meningitis in HIV infection, fungal infections, and leishmaniasis.
NatamycinA macrolide antifungal used to treat fungal infections of the eye.
DaptomycinA cyclic lipopeptide antibiotic used to treat complicated skin and skin structure infections by susceptible Gram-positive bacteria and bacteremia due to Staphylococcus aureus.
CefotiamA cephalosporin antibiotic used to treat a variety of bacterial infections.
Aminosalicylic acidAn aminosalicylate drug used to induce remission in ulcerative colitis.
DapsoneA sulfone drug used to treat acne vulgaris, Hansen's disease, and dermatitis herpetiformis.
SulfanilamideA sulfonamide anti-infective used to treat vulvovaginal candidiasis caused by Candida albicans.
CefmenoximeUsed to treat female gynecologic and obstetric infections caused by susceptible aerobic (including the gonococcus) and anaerobic bacteria.
CefmetazoleA cephalosporin antibiotic used to treat a variety of bacterial infections.
FlucloxacillinA narrow spectrum penicillin antibiotic that exerts specific activity against Gram positive organisms in skin and soft tissue infections, except those caused by methicillin resistant staphylococcus aureus (MRSA).
ErtapenemA carbapenem antibiotic used for the treatment of moderate to severe infections caused by susceptible bacteria.
PiperacillinA penicillin antibiotic combined with tazobactam to treat piperacillin-resistant, piperacillin/tazobactam­ susceptible, β-lactamase generating strains of several bacteria.
EthambutolAn antituberculosis agent used in the prophylaxis and treatment of tuberculosis (TB).
PyrazinamideAn antituberculosis agent used as a component of tuberculosis (TB) treatment.
AztreonamA beta-lactam antibiotic used to treat select aztreonam sensitive gram negative bacteria.
GrepafloxacinA fluoroquinolone antibiotic used to treat various gram positive and gram negative bacterial infections.
AmpicillinA penicillin derivative used for the treatment of a variety of infections caused by gram-positive and gram-negative bacteria as well as some anaerobes.
PhenoxymethylpenicillinA penicillin antibiotic used to prevent and treat mild to moderately severe infections in the respiratory tract, skin, and soft tissues.
CefpiramideFor treatment of severe infections caused by susceptible bacteria such as P. aeruginosa.
CeftazidimeAn injected broad-spectrum third-generation cephalosporin beta-lactam antibiotic used to treat or prevent a variety of bacterial infections, including pneumonia, gynecological infections, bone and joint infections, and septicemia, among others.
LoracarbefUsed to treat upper respiratory tract bacterial infections, chronic bronchitis, pneumonia, sinusitis, pharyntitis and tonsillitis, skin absceses, urinary tract infections and pyelonephritis caused by E. coli, S. pyogenes, S. aureus,...
CefalotinA broad-spectrum cephalosporin antibiotic used for the treatment of serious bacterial infections in various locations, such as the urinary tract, skin, bone, and lower respiratory tract.
EnoxacinFor the treatment of adults (≥18 years of age) with the following infections caused by susceptible strains of the designated microorganisms: (1) uncomplicated urethral or cervical gonorrhea due to Neisseria...
AmikacinAn aminoglycoside used to treat infections caused by more resistant strains of Gram negative bacteria and some Gram positive bacteria.
DicloxacillinA penicillin used to treat penicillinase-producing bacterial infections that are susceptible to the drug.
PefloxacinAn antibiotic used to treat a variety of bacterial infections.
CefotaximeA third generation cephalosporin used to treat susceptible Gram negative and Gram positive bacterial infections.
VancomycinA glycopeptide antibiotic used to treat severe but susceptible bacterial infections such as MRSA (methicillin-resistant Staphylococcus aureus) infections.
CefdinirA third generation cephalosporin used to treat susceptible Gram negative and Gram positive bacterial infections.
CephalexinA first generation cephalosporin used to treat certain susceptible bacterial infections.
CarbenicillinFor the treatment of acute and chronic infections of the upper and lower urinary tract and in asymptomatic bacteriuria due to susceptible strains of bacteria.
LinezolidAn oxazolidinone antibiotic used to treat infections by susceptible strains of aerobic Gram-positive bacteria.
NafcillinA penicillin derivative antibiotic used to treat susceptible staphylococcal infections.
EthionamideA second line antitubercular agent used to treat tuberculosis when other treatments have failed.
CefiximeA third generation cephalosporin used to treat susceptible Gram-negative and Gram-positive bacterial infections.
CephaloglycinFor treatment of severe infections caused by susceptible bacteria.
OxacillinA penicillin antibiotic used to treat a number of susceptible bacterial infections.
MeropenemA carbapenem antibiotic used to treat a wide variety of infections in the body.
Clavulanic acidA beta lactamase inhibitor used to enhance the effectiveness of beta lactam antibiotics.
RoxithromycinAn antibiotic used to treat a variety of susceptible bacterial infections.
Nalidixic acidA quinolone antibiotic used to treat urinary tract infections.
ColistinA polymyxin antibiotic used to treat bacterial infections caused by susceptible Gram negative bacteria.
FosfomycinA broad spectrum antibiotic used to treat uncomplicated urinary tract infections.
CefaclorA second generation cephalosporin used to treat a wide variety of infections in the body.
ClofazimineA riminophenazine antimycobacterial used to treat leprosy.
SirolimusAn mTOR inhibitor immunosuppressant used to prevent organ transplant rejections, treat lymphangioleiomyomatosis, and treat adults with perivascular epithelioid cell tumors.
SpectinomycinAn aminocyclitol antibiotic used to treat susceptible strains of Neisseria gonorrhoeae.
CeforanideFor the treatment of infections caused by susceptible organisms.
MezlocillinUsed to treat serious gram–negative infections of the lungs, urinary tract, and skin.
DirithromycinAn antibiotic used to treat a variety of respiratory, skin, and other infections.
NetilmicinAn aminoglycoside used to treat a wide variety of infections in the body.
TelithromycinAn ketolide used to treat community acquired pneumonia of mild to moderate severity.
LomefloxacinA fluoroquinolone used to prevent and treat a wide variety of infections in the body.
CyclacillinFor the treatment of bacterial infections caused by susceptible organisms.
RifampicinAn antibiotic used to treat several types of mycobacterial infections including Mycobacterium avium complex, leprosy, and in combination with other antibacterials to treat latent or active tuberculosis.
NovobiocinFor the treatment of infections due to staphylococci and other susceptible organisms
AmoxicillinA penicillin derivative used for the treatment of infections caused by gram-positive bacteria, in particular streptococcal bacteria causing upper respiratory tract infections.
AzlocillinFor the treatment of infections caused by Pseudomonas aeruginosa, Escherichia coli, and Haemophilus influenzae.
CefditorenA broad-spectrum third-generation cephalosporin antibiotic typically used to treat bacterial infections of the skin and respiratory tract.
CefuroximeA cephalosporin indicated for the treatment of a variety of infections including acute bacterial otitis media, several upper respiratory tract infections, skin infections, urinary tract infections, gonorrhea, early Lyme disease, and impetigo.
LevofloxacinA fluoroquinolone antibiotic used to treat infections caused by susceptible bacteria of the upper respiratory tract, skin and skin structures, urinary tract, and prostate, as well as for post-exposure treatment of inhaled anthrax and the plague.
CefapirinA first generation cephalosporin indicated in the treatment of susceptible bacterial infections.
CefadroxilA cephalosporin antibiotic used in the treatment of various bacterial infections, such as urinary tract infections, skin and skin structure infections, and tonsillitis.
CloxacillinAn antibiotic agent used for the treatment of beta-hemolytic streptococcal and pneumococcal infections as well as staphylococcal infections.
CefprozilA cephalosporin antibiotic used in the treatment of various bacterial infections, such as pharyngitis, tonsillitis, otitis media, and uncomplicated skin infections.
GemifloxacinA quinolone antibacterial agent used for the treatment of acute bacterial exacerbation of chronic bronchitis and mild to moderate community-acquired pneumonia caused by susceptible bacteria.
AmdinocillinUsed in the treatment of urinary tract infections caused by some strains of E. coli and klebsiella and enterobacter species. Used mainly against Gram negative organisms.
SparfloxacinA fluoroquinolone antibiotic used to treat bacterial respiratory infections and sinusitis.
ClarithromycinA macrolide antibiotic used for the treatment of a wide variety of bacterial infections such as acute otitis, pharyngitis, tonsillitis, respiratory tract infections, uncomplicated skin infections, and helicobacter pylori infection.
CeftriaxoneA broad-spectrum cephalosporin antibiotic used for the treatment of bacterial infections in various locations, such as in the respiratory tract, skin, soft tissue, and urinary tract.
ChloroxineAn antibacterial agent used for the treatment of dandruff and mild to moderately severe seborrheic dermatitis of the scalp.
JosamycinA macrolide antibiotic used for the treatment of various susceptible bacterial infections.
CefamandoleA beta-lactam antibiotic used in the treatment of various infections caused by susceptible strains of bacteria, such as lower respiratory infections, urinary tract infections, skin infections, and bone and joint infections.
CefazolinA broad-spectrum cephalosporin antibiotic mainly used for the treatment of skin bacterial infections and other moderate to severe bacterial infections in the lung, bone, joint, stomach, blood, heart valve, and urinary tract.
CefonicidFor the treatment of bacterial infections caused by susceptible microorganisms.
CefoperazoneA broad-spectrum cephalosporin antibiotic used for the treatment of bacterial infections in various locations, including the respiratory tract, abdomen, skin, and female genital tracts.
CefotetanAn antibiotic medication used for the prophylaxis and treatment of various bacterial infections, including urinary tract infections, bone and joint infection, and lower respiratory tract infections.
CefoxitinA semi-synthetic, broad-spectrum antibiotic for parenteral administration used for the treatment of serious bacterial infections, such as urinary tract infection, blood infection, bone and joint infection, and lower respiratory tract infection.
CeftizoximeA third-generation cephalosporin antibiotic used in the treatment of various bacterial infections, including lower respiratory tract infection, urinary tract infection, and gonorrhea.
CefradineA first-generation cephalosporin antibiotic used in the treatment of bacterial infections of the respiratory and urinary tracts and of the skin and soft tissues.
QuinupristinAn antibiotic agent used in the treatment of serious vancomycin-resistant Enterococcus faecium bacteremia as well as complicated skin and skin structure infections.
TemafloxacinFor the treatment of lower respiratory tract infections, genital and urinary infections like prostatitis, and skin infections.
CefepimeA fourth-generation cephalosporin antibiotic used in the treatment of infections caused by susceptible bacteria, such as pneumonia, urinary tract infections, and skin infections.
CefacetrileA broad-spectrum first-generation cephalosporin used for the treatment of susceptible bacterial infections.
CeftibutenA third-generation cephalosporin antibiotic commonly used in the treatment of acute bacterial exacerbations of chronic bronchitis (ABECB), acute bacterial otitis media, pharyngitis, and tonsillitis.
CefpodoximeA third-generation cephalosporin antibiotic used in the treatment of various bacterial infections, including gonorrhea, community acquired pneumonia, and sinusitis.
ImipenemA carbapenem antibiotic normally administered with cilastatin to treat a variety of infections.
BacampicillinAn ampicillin prodrug used to treat various susceptible bacterial infections in the body, such as respiratory infections and skin and subcutaneous tissue infections.
MeticillinUsed to treat infections caused by susceptible Gram-positive bacteria, particularly beta-lactamase-producing organisms such as Staphylococcus aureus that would otherwise be resistant to most penicillins.
PivampicillinAn ampicillin prodrug used to treat a variety of infections.
PivmecillinamA prodrug of the beta lactam antibiotic mecillinam, indicated for the treatment of uncomplicated urinary tract infections (UTIs).
TicarcillinA beta lactam antibiotic used to treat a variety of infections in the body.
LincomycinAn antibiotic indicated only for the treatment of serious infections and is typically reserved for use in cases of penicillin allergy or where penicillin is inappropriate.
Virginiamycin M1For the treatment of bacterial infections.
DalfopristinAn antibiotic used with quinupristin to treat severe or life-threatening infections of vancomycin-resistant Enterococcus faecium (VREF), and skin infections caused by methicillin susceptible staphylococcus aureus or streptococcus pyogenes.
MaltotetraoseNot Available
GE-2270ANot Available
UbenimexAn adjuvant therapy used for acute and chronic myelonous leukemia, lung cancer and nasopharyngeal cancer. It is also used to treat hypercholesterolaemia.
RibostamycinA broad spectrum aminoglycoside antibiotic on the list of WHO critical antimicrobials for human medicine.
AurodoxAurodox is an antibiotic obtained from a streptomyces variant considered as possibly effective against streptococcus pyogenes infections. It may promote growth in poultry.
LatamoxefLatamoxef is an oxacephem antibiotic usually grouped with the cephalosporins. It is used to treat bacterial infections. Latamoxef is primarily indicated in conditions like Bone and joint infection, GI infections,...
ApramycinAn aminoglycoside antibiotic for veterinary use that is used to treat infections in animals.
OritavancinAn antibacterial agent used to treat acute bacterial skin and skin structure infections caused by susceptible Gram-positive bacteria.
CeftobiproleA cephalosporin antibiotic used to treat both community and hospital-acquired pneumonia caused by susceptible bacteria.
RifalazilInvestigated for use/treatment in atherosclerosis, bacterial infection, and peripheral vascular disease.
RamoplaninFor the treatment of bacterial infections.
SpiramycinA macrolide antimicrobial agent used in the treatment of various bacterial infections.
TeicoplaninA glycopeptide antibiotic with a similar mechanism of action and spectrum of activity to vancomycin used to treat various infections caused by gram-positive bacteria.
GarenoxacinInvestigated for use/treatment in bacterial infection.
DalbavancinAn antibacterial used to treat acute bacterial skin and skin structure infections (ABSSSI) caused by susceptible strains of Gram-positive bacteria.
TelavancinAn antibacterial agent used in the treatment of complicated skin and skin structure infections and types of hospital-acquired bacterial pneumonia.
CethromycinA ketolide antibiotic with broad-spectrum activity against Gram-positive, Gram-negative, and atypical bacteria that may be useful for treating several conditions including community-acquired pneumonia, inhalation anthrax, plague, and tularemia.
SqualamineInvestigated for use/treatment in ovarian cancer, lung cancer, and macular degeneration.
ViomycinViomycin is an essential component in the drug cocktail currently used to fight infections of Mycobacterium tuberculosis.
Brefeldin AA metabolite from Penicillium brefeldianum that exhibits a wide range of antibiotic activity.
AnisomycinAnisomycin (sometimes known as flagecidin), is an antibiotic retrieved from the bacteria Streptomyces griseolus. This drug acts to inhibit bacterial protein and DNA synthesis.
Chloramphenicol succinateA broad-spectrum antibiotic agent used for the treatment of acute and severe infections caused by susceptible bacterial strains.
ThiamphenicolA semisynthetic derivative of chloramphenicol with a broad spectrum of antibacterial activity.
BedaquilineA diarylquinoline antimycobacterial used in combination with other antibacterials to treat pulmonary multidrug resistant tuberculosis (MDR-TB).
EnviomycinCyclic basic peptide related to viomycin. It is isolated from an induced mutant of Streptomyces griseoverticillatus var. tuberacticus and acts as an antitubercular agent with less ototoxicity than tuberactinomycin.
CefaloridineCephaloridine or cefaloridine is a first generation semisynthetic cephalosporin. It is derived from cephalosporin C and is a zwitterion at physiological pH.
Tedizolid phosphateAn oxazolidinone class antibiotic that inhibits bacterial protein synthesis and is proven to be effective in the treatment of certain Gram-positive bacterial infections.
CefminoxCefminox (INN) is a second generation cephalosporin antibiotic. It is approved for use in Japan.
ChlortetracyclineThe first tetracycline antibiotic most commonly used for veterinary purposes.
KitasamycinKitasamycin is a macrolide antibiotic derived from Streptomyces kitasatoensis.
CarindacillinA penicillin antibiotic used to treat a variety of infections, but is no longer marketed in the USA.
Procaine benzylpenicillinA local anesthetic and antibiotic combination for intramuscular injection to treat a variety of bacterial infections while reducing pain from a deep intramuscular injection.
AvilamycinNot Annotated
BambermycinsBambermycins are antibiotic complexes which are retrieved from the organism, Streptomyces bambergiensis. They are used as an additive in food ingested by chickens and swine. The bambermycin complex of antibiotics...
EfrotomycinNot Annotated
FlorfenicolFlorfenicol is a fluorinated synthetic analog of thiamphenicol.
GamithromycinGamithromycin is an antibiotic used in cattle.
MarbofloxacinMarbofloxacin is a carboxylic acid, part of the third generation of antibiotic fluoroquinolones. It is used in veterinary medicine. A formulation of marbofloxacin combined with clotrimazole and dexamethasone is available...
OleandomycinOleandomycin is a macrolide antibiotic, though it is less effective than erythromycin. It is synthesized from strains of Streptomyces antibioticus.
RoxarsoneRoxarsone is an organoarsenic molecule added to poultry feed. The addition of this compound to poultry feed improves weight gain and feed efficiency as well as prevent the growth of...
ThiostreptonThiostrepton is a natural cyclic oligopeptide antibiotic, derived from several strains of streptomycetes including Streptomyces azureus and Streptomyces laurentii. Thiostrepton is a natural product of the ribosomally synthesized and post-translationally...
TiamulinTiamulin is a pleuromutilin antibiotic drug that is used in veterinary medicine particularly for pigs and poultry.
TilmicosinTilmicosin is a macrolide antibiotic. It is used in veterinary medicine for the treatment of bovine respiratory disease and ovine respiratory disease associated with Mannheimia haemolytica.
TylosinTylosin is a bacteriostatic macrolide antibiotic and feed additive used in veterinary medicine. It has a broad spectrum of activity against Gram-positive organisms and a limited range of Gram-negative organisms....
VirginiamycinVirginiamycin is a streptogramin antibiotic similar to pristinamycin and quinupristin/dalfopristin. It is a combination of pristinamycin IIA and virginiamycin S1. Virginiamycin is used in the fuel ethanol industry to prevent...
CeftiofurCeftiofur is a third generation cephalosporin antibiotic, first described in 1987, and now used in veterinary medicine. It is marketed by pharmaceutical company Zoetis as Excenel, and is the active...
Hygromycin BHygromycin B is an aminoglycoside antibiotic produced by the bacterium Streptomyces hygroscopicus which kills bacteria, fungi and higher eukaryotic cells by inhibiting protein synthesis.
MaduramicinMaduramicin is an antiprotozoal agent used in veterinary medicine as prophylaxis against coccidiosis. It is a naturally occurring compound which was first isolated from the actinomycete, Actinomadura rubra.
SalinomycinNot Annotated
Isatoic anhydrideNot Available
EpetraboroleEpetraborole has been used in trials studying the treatment of Infections, Bacterial, Infections, Intestinal, Infections, Urinary Tract, and Community-acquired Infection.
PazufloxacinPazufloxacin is under investigation in clinical trial NCT02592096 (Pazufloxacin Mesilate Ear Drops Clinical Trial Protocol).
PrulifloxacinA broad-spectrum fluoroquinolone antibiotic used to treat a variety of susceptible bacterial infections.
LanopepdenLanopepden has been used in trials studying the treatment of Pneumonia, Infections, Bacterial, Skin Diseases, Infectious, and Skin Infections, Bacterial.
SultamicillinA mutual prodrug of ampicillin and sulbactam useful in the treatment of infections caused by beta-lactamase-producing bacteria.
NadifloxacinA topical fluoroquinolone used in the treatment of acne and topical bacterial skin infections.
SisomicinSisomicin has been used in trials studying the treatment of Pyoderma.
ProtionamideAn antitubercular thioamide-derivative used in the treatment of multi-drug resistant (MDR) tuberculosis and leprosy.
AmithiozoneAmithiozone has been used in trials studying the treatment of Mycobacterium Avium-intracellulare Infection.
TunicamycinTunicamycin is a mixture of homologous nucleoside antibiotics that inhibits the UDP-HexNAc: polyprenol-P HexNAc-1-P family of enzymes. One member of this family is the enzyme GlcNAc phosphotransferase (GPT), which catalyzes...
TroleandomycinFor the treatment of bacterial infection.
SitafloxacinA fluoroquinolone antibiotic indicated in the treatment of susceptible bacterial infections.
CefatrizineNot Annotated
DibekacinDibekacin is an aminoglycoside antibiotic marketed in Japan .
MiocamycinMiocamycin is a macrolide type antimicrobial . This drug may be marketed in Japan for clinical use as it is listed in the Japanese pharmacopeia . It has shown to...
EpicillinNot Annotated
MidecamycinA macrolide antibiotic used to treat a variety of infections caused by susceptible bacteria.
CefodizimeA broad-spectrum, third-generation cephalosporin used to treat serious infections caused by susceptible bacteria.
CefsulodinNot Annotated
CefetametNot Annotated
IsepamicinNot Annotated
Oxolinic acidNot Annotated
PropicillinNot Annotated
BekanamycinAn aminoglycoside antibiotic indicated in the treatment of eye infections.
CefpiromeAn antibiotic indicated in the treatment of a wide variety of infections in the body.
SulbenicillinNot Annotated
PristinamycinNot Annotated
DecamethoxineNot Annotated
SulfamethoxypyridazineA sulphonamide antibiotic indicated in the treatment of gonorrhea, inflammation, urinary tract ulcers, and bronchitis.
CefazedoneNot Annotated
TalampicillinNot Annotated
CeftezoleNot Annotated
Pipemidic acidA quinolone antibiotic indicated in the treatment of susceptible urinary tract infections.
MetampicillinMetampicillin is a penicillin antibiotic prepared by the reaction of ampicillin with formaldehyde. It is hydrolysed in aqueous solution to form ampicillin. Hydrolysis is rapid under acid conditions like the...
ClinafloxacinClinafloxacin is a fluoroquinolone antibacterial currently under research. It has been proven to present good antibiotic properties. However, its approval and release have been halted due to the presence of...
RifaximinA rifamycin-based non-systemic antibiotic used for the treatment of gastrointestinal bacterial infections, such as traveler's diarrhea and irritable bowel syndrome, and reduction of overt hepatic encephalopathy recurrence in adults.
FidaxomicinA macrolide antibiotic used to treat diarrhea associated with Clostridium difficile infection.
FusafungineFusafungine is an antibiotic from Fusarium lateririum, and is used for the treatment of respiratory infections.
AzidamfenicolNot Annotated
SulfacetamideA sulfonamide used to treat inflammatory ocular conditions and acne vulgaris.
MetronidazoleA nitroimidazole used to treat trichomoniasis, amebiasis, inflammatory lesions of rosacea, and bacterial infections, as well as prevent postoperative infections.
RetapamulinA topical antibiotic agent used for the treatment of impetigo caused by methicillin-susceptible Staphylococcus aureus or Streptococcus pyogenes.
BesifloxacinA fluoroquinolone antibiotic agent used for the treatment of bacterial conjunctivitis.
FinafloxacinFinafloxacin is indicated for the treatment of acute otitis externa (AOE) with or without an otowick, caused by susceptible strains of Pseudomonas aeruginosa and Staphylococcus aureus in patients age 1...
OzenoxacinA quinolone antibiotic used to treat impetigo caused by susceptible bacteria.
SolithromycinInvestigated for the treatment of community-acquired pneumonia (CAP).
FlurithromycinNot Annotated
RokitamycinNot Annotated
EverolimusA mammalian target of rapamycin (mTOR) kinase inhibitor used to treat various types of malignancies.
Epothilone DInvestigated for use/treatment in colorectal cancer, lung cancer, breast cancer, solid tumors, and prostate cancer.
PatupiloneInvestigated for use/treatment in ovarian cancer, lung cancer, brain cancer, breast cancer, and gastric cancer.
6-Deoxyerythronolide BNot Available
IxabepiloneA microtubule inhibitor administered in combination with capecitabine or alone in the treatment of metastatic or locally advanced breast cancer that has shown inadequate response to taxanes and anthracyclines.
KOS-1584Investigated for use/treatment in solid tumors.
RidaforolimusInvestigated for use/treatment in solid tumors, sarcoma, cancer/tumors (unspecified), endometrial cancer, prostate cancer, and bone metastases.
TemsirolimusA antineoplastic agent used in the treatment of renal cell carcinoma (RCC) that works by inhibiting mTOR.
AVE9633Investigated for use/treatment in leukemia (myeloid).
Coltuximab ravtansineInvestigated for use/treatment in lymphoma (non-hodgkin's).
MitemcinalInvestigated for use/treatment in gastroparesis and irritable bowel syndrome (IBS).
CarbomycinCarbomycin, also called magnamycin, is crystalline macrolide antibiotic. This antibacterial is obtained from Streptomyces halstedii and it presents a large inhibitory effect against Gram-positive bacteria and some Mycoplasma strains. The...
DoramectinDoramectin is a veterinary drug approved by the Food and Drug Administration for the treatment of parasites such as gastrointestinal roundworms, lungworms, eyeworms, grubs, sucking lice and mange mites in...
EprinomectinNot Annotated
SelamectinSelamectin is a topical parasiticide and antihelminthic used on dogs and cats to treat and prevent infections of heartworms, fleas, ear mites, sarcoptic mange, and certain types of ticks in...
TildipirosinTildipirosin is a veterinary antibiotic.
TylvalosinNot Annotated
Bryostatin 1Bryostatin 1 has been investigated for the treatment of HIV Infection and Alzheimer's Disease.
Lorvotuzumab mertansineLorvotuzumab mertansine has been used in trials studying the treatment of SCLC, Leukemia, Ovarian Cancer, Multiple Myeloma, and Merkel Cell Carcinoma, among others.
EpofolateEpofolate has been used in trials studying the treatment of Advanced Solid Tumors. Epofolate (BMS-753493) is a folate conjugate of the epothilone analog BMS-748285 that was designed to selectively target...
SagopiloneSagopilone has been used in trials studying the treatment of Melanoma, Neoplasms, CNS Disease, Breast Cancer, and Breast Neoplasms, among others. It is a so-called fully synthetic epothilone and is...
CefroxadineWas used for the treatment of bacterial infections.
CefbuperazoneNot Annotated
Ceftaroline fosamilAn antibacterial agent used to treat various bacterial infections, such as acute bacterial skin and skin structure infections and community-acquired bacterial pneumonia.
CefcapeneNot Annotated
CefozopranNot Annotated
Benzylpenicilloyl polylysineA penicillin derivative used to determine penicillin allergies.
AzidocillinFor treatment of infection (Respiratory, GI, UTI and meningitis) due to E. coli, P. mirabilis, enterococci, Shigella, S. typhosa and other Salmonella, nonpenicillinase-producing N. gononhoeae, H. influenzae, staphylococci, streptococci including...
PenamecillinNot Annotated
AspoxicillinNot Annotated
BiapenemA carbapenem antibiotic indicated in the treatment of bacterial infections.
DoripenemAn antibiotic of the penem class used to treat complicated intra-abdominal and urinary tract infections.
Technetium Tc-99m ciprofloxacinInvestigated for use/treatment in infectious and parasitic disease (unspecified).
OrbifloxacinOrbifloxacin is a fluoroquinolone antibiotic. It is marketed by Schering-Plough Animal Health and approved for certain infections in dogs.
SarafloxacinSarafloxacin is a quinolone antibiotic drug, which was discontinued by its manufacturer, Abbott Laboratories, before receiving approval for use in the US or Canada.
DifloxacinDifloxacin is a synthetic fluoroquinolone used in veterinary. As an antibacterial, it presents a broad bactericidal spectrum and its effects are dependent on its concentration. However, it presents a reduced...
TrovafloxacinAn antibiotic used to treat gonorrhea and chlamydia.
RosoxacinFor the treatment of bacterial infection of respiratory tract, urinary tract, GI, CNS and immuno compromised patients.
CinoxacinFor the treatment of initial and recurrent urinary tract infections in adults caused by the following susceptible microorganisms: Escherichia coli, Proteus mirabilis, Proteus vulgaris, Klebsiella species (including K. pneumoniae), and...
FleroxacinFleroxacin is a broad-spectrum antimicrobial fluoroquinolone.
NemonoxacinInvestigated for use/treatment in bacterial infection and pneumonia.
FlumequineFlumequine is a synthetic chemotherapeutic antibiotic of the fluoroquinolone drug class used to treat bacterial infections.
RufloxacinA fluoroquinolone antibiotic indicated in the treatment of susceptible respiratory infections and uncomplicated cystitis.
SulfamethoxazoleAn oral sulfonamide antibiotic, given in combination with trimethoprim, used to treat a variety of infections of the urinary tract, respiratory system, and gastrointestinal tract.
SulfisoxazoleA sulfonamide antibiotic used with other antibiotics to prevent and treat a variety of bacterial infections.
SulfadiazineA sulfonamide antibiotic used in a variety of infections, such as urinary tract infections, trachoma, and chancroid.
Silver sulfadiazineA topical sulfonamide antibiotic that acts on the bacterial cell wall and cell membrane; approved for the treatment of burns.
FlomoxefFlomoxef has been used in trials studying the treatment of Urinary Tract Infection.
IsoniazidAn antibiotic used to treat mycobacterial infections; most commonly use in combination with other antimycobacterial agents for the treatment of active or latent tuberculosis.
GeneticinGeneticin (also known as G418) is an aminoglycoside antibiotic similar in structure to gentamicin B1, produced by Micromonospora rhodorangea. Geneticin blocks polypeptide synthesis by inhibiting the elongation step in both...
Gentamicin C1aNot Available
NeamineNot Available
ArbekacinArbekacin is used for the short term treatment of multi-resistant bacterial infections, such as methicillin-resistant Staphylococcus aureus (MRSA).
PuromycinPuromycin is an antibiotic that prevents bacterial protein translation. It is utilized as a selective agent in laboratory cell cultures. Puromycin is toxic to both prokaryotic and eukaryotic cells, resulting...
PlazomicinAn aminoglycoside antibiotic used to treat complicated urinary tract infections.
SulfamerazineAn antibacterial agent used in the treatment of various bacterial infections, such as bronchitis, prostatitis, and urinary tract infections.
LasalocidLasalocid is an agent that presents antibacterial and coccidiostat activities. It is produced by strains of Streptomyces lasaliensis.
NarasinNarasin is an agent with coccidiostatic and antibacterial properties.
SulfameterLong acting sulfonamide used in leprosy, urinary, and respiratory tract infections.
TemocillinTemocillin has been investigated in Infection, Liver Dysfunction, and Urinary Tract Infection.
NigericinA polyether antibiotic which affects ion transport and ATPase activity in mitochondria. It is produced by Streptomyces hygroscopicus. (From Merck Index, 11th ed)
ValinomycinA cyclododecadepsipeptide ionophore antibiotic produced by Streptomyces fulvissimus and related to the enniatins. It is composed of 3 moles each of L-valine, D-alpha-hydroxyisovaleric acid, D-valine, and L-lactic acid linked alternately...
MafenideAn antimicrobial topical agent indicated for use as an adjunctive treatment to control bacterial infection when used under moist dressings over meshed autografts on excised burn wounds.
DoxycyclineA tetracycline antibiotic used to treat a wide variety of bacterial infections.
LymecyclineA tetracycline antibiotic used for the treatment of acne vulgaris and other susceptible infections.
TigecyclineA glycylcycline antibiotic used to treat a number of susceptible bacterial infections.
DemeclocyclineA tetracycline antibiotic used to treat a wide variety of susceptible bacterial infections.
MetacyclineFor the treatment of acute bacterial exacerbations of chronic bronchitis
RolitetracyclineA broad-spectrum tetracycline antibiotic used in cases needing high concentrations or when oral administration is impractical.
PenimepicyclinePenimepicycline is a tetracycline-class antibiotic. It is mentioned on List A produced by the Government of Canada, which is a list of antimicrobial active pharmaceutical ingredients . In the classification...
TedizolidAn oxazolidinone class antibiotic that inhibits bacterial protein synthesis and is proven to be effective in the treatment of certain Gram-positive bacterial infections.
RifamycinAn antibacterial used to treat traveler's diarrhea.
CeftolozaneA cephalosporin antibiotic used to treat complicated intra-abdominal infections in combination with metronidazole, complicated urinary tract infections, and hospital-acquired pneumonia.
Acetyl sulfisoxazoleAcute, recurrent or chronic urinary tract infections (primarily pyelonephritis, pyelitis and cystitis) due to susceptible organisms (usually Escherichia coli, Klebsiella-Enterobacter, staphylococcus, Proteus mirabilis and, less frequently, Proteus vulgaris) in the...
DelafloxacinA fluoroquinolone antibiotic used to treat skin and skin structure infections.
PirlimycinPirlimycin hydrochloride is an antibiotic belonging to the lincosamide class. Often marketed as Pirsue, this drug is used to treat mastitis in cattle.
ClomocyclineFor the treatment and management of Brucellosis, mycoplasma infection, acne vulgaris, chlamydial infection;Chronic bronchitis
SarecyclineA tetracycline antibiotic used to treat inflammatory lesions of non-nodular moderate to severe acne vulgaris.
OmadacyclineA tetracycline antibiotic used to treat community acquired bacterial pneumonia.
RadezolidRadezolid has been used in trials studying the treatment of Abscess, Bacterial Skin Diseases, Streptococcal Infections, Infectious Skin Diseases, and Staphylococcal Skin Infections, among others.
MeclocyclineA tetracycline antibiotic indicated in the treatment of susceptible skin infections, bacterial vaginitis, vulvovaginitis, and cervicitis.
Cefamandole nafateA second generation cephalosporin indicated in the prevention of infections during surgery.
Ceftobiprole medocarilA cephalosporin indicated in the treatment of pneumonia.
Polymyxin BA polymyxin antibiotic used to treat a wide variety of infections in the body.
EravacyclineA tetracycline antibiotic used to treat complicated intra-abdominal infections.
25-desacetylrifapentine25-desacetylrifapentine is under investigation in clinical trial NCT00023387 (TBTC Study 25PK: Intensive Pharmacokinetic Study of Three Doses of Rifapentine and 25-Desacetyl Rifapentine).
PheneticillinPheneticillin (or phenethicillin) is a penicillin antibiotic which is approved for use internationally.
HetacillinHetacillin is a beta-lactam antibiotic prodrug used to treat bacterial infections. In the body it gets converted to ampicillin.
ClometocillinNot Annotated
Mycophenolate mofetilAn inosine monophosphate dehydrogenase inhibitor used to prevent the rejection of kidney, heart, or liver transplants.
NitrofurantoinAn antibiotic used to treat urinary tract infections.
TinidazoleA nitroimidazole used to treat trichomoniasis, giardiasis, amebiasis, and bacterial vaginosis.
Mycophenolic acidAn immunosuppressant used to prevent organ transplant rejections.
FosmidomycinNot Available
Acetic acidAn antimicrobial agent used to treat susceptible infections of the external auditory canal.
StreptolydiginStreptolydigin is an antibiotic isolated from culture filtrates of Streptomyces lydicus. It is active against gram-postive bacteria except micrococci.
MethenamineA urinary tract antiseptic and antibacterial drug used for the prophylaxis and treatment of frequently recurring urinary tract infections requiring a long-term therapy.
EnrofloxacinEnrofloxacin is an antibiotic agent from the fluoroquinolone family produced by the Bayer Corporation. Enrofloxacin is approved by the FDA for its veterinary use. Due to the identification of fluoroquinolone-resistant...
Tulathromycin ATulathromycin is a macrolide antibiotic used to treat bovine respiratory disease in cattle and swine respiratory disease in pigs. It is marketed by Pfizer Inc. under the tradename Draxxin.
DelpazolidDelpazolid (LCB01-0371) is under investigation in clinical trial NCT01554995 (A Clinical Study, Randomized, Double-blind, Placebo-controlled, Single Dose Study).
Malacidin AMalacidin A is being investigated for its antibiotic action and has potential for use as an antibacterial agent in the future .
Malacidin BMalacidin B is being investigated for its antibiotic action and has potential for use as an antibacterial agent in the future .
MurepavadinMurepavadin is under investigation in clinical trial NCT02110459 (Pharmacokinetics and Safety of POL7080 in Patients With Renal Impairment).
UmirolimusNot Annotated
CefiderocolA cephalosporin antibiotic used in complicated urinary tract infections.
AmphomycinNot Annotated
PradofloxacinPradofloxacin is a 3rd generation fluoroquinolone antibiotic developed by Bayer HealthCare AG, Animal Health GmBH. It was approved by the European Commission in April 2011 for bacterial infections in dogs...
Ala-geninthiocinAla-geninthiocin is a novel thiopeptide antibacterial compound derived from marine Streptomyces species. It has exhibited potent in vitro activity against gram-positive bacteria including Staphylococcus aureus, Bacillus subtilis, Mycobacterium smegmatis, and...
Sulbactam pivoxilA prodrug of a beta-lactamase inhibitor used to improve the efficacy of beta lactam antibiotics
PexigananPexiganan is under investigation in clinical trial NCT01594762 (Pexiganan Versus Placebo Control for the Treatment of Mild Infections of Diabetic Foot Ulcers).
Tetracycline phosphate complexNot Annotated
EvernimicinInvestigated for use/treatment in bacterial infection.
DurlobactamDurlobactam is co-packaged with sulbactam as a single combination product, and is indicated for the treatment of hospital-acquired bacterial pneumonia and ventilator-associated bacterial pneumonia caused by susceptible isolates of Acinetobacter...
DequaliniumA quaternary ammonium cation antimicrobial agent used to treat common infections of the mouth and throat, as well as vaginal candidiasis.
SulfamethizoleA sulfonamide antibiotic used to treat a wide variety of susceptible bacterial infections.
LefamulinA pleuromutilin antibacterial used to treat community-acquired bacterial pneumonia (CABP).
EchinomycinEchinomycin is a cytotoxic polypeptide quinoxaline antibiotic isolated from Streptomyces echinatus that binds to DNA and inhibits RNA synthesis.
NafithromycinNafithromycin is under investigation in clinical trial NCT02903836 (Phase II Study of Oral Nafithromycin in CABP).
MacozinoneMacozinone is under investigation in clinical trial NCT03036163 (Phase 1 Study of PBTZ169).
LevonadifloxacinLevonadifloxacin is under investigation in clinical trial NCT03405064 (Comparative Study of Levonadifloxacin (IV and Oral) With Linezolid (IV and Oral) in Acute Bacterial Skin and Skin Structure Infections (ABSSSI)).
Josamycin propionateNot Annotated
Indatuximab ravtansineIndatuximab ravtansine is under investigation in clinical trial NCT01001442 (Safety and Dose Determining Multi-dose Study of BT062 in Patients With Relapsed or Refractory Multiple Myeloma).
CarrimycinNot Available
Nanoparticle EpirubicinNanoparticle Epirubicin is under investigation in clinical trial NCT03168061 (Dose-escalation and Expansion Trial of NC-6300 in Patients With Advanced Solid Tumors or Soft Tissue Sarcoma). It is a novel epirubicin...
Tebipenem pivoxilNot Annotated
TosufloxacinNot Annotated
ChelerythrineA benzophenanthridine alkaloid evaluated as a kinase-inhibitor.
BerubicinNot Annotated
Cantuzumab mertansineNot Annotated
NC-6300NC-6300, also known as K-912, is a novel epirubicin drug-conjugated polymeric micelle.
CRS-3123CRS3123 has been used in trials studying the treatment of Clostridial Infection and Clostridium Difficile Colitis.
LFF-571LFF571 has been used in trials studying the treatment of Moderate Clostridium Difficile Infection.
AfabicinAfabicin is under investigation in clinical trial NCT03723551 (Study to Assess Safety, Tolerability and Efficacy of Afabicin in The Treatment of Participants With Bone or Joint Infection Due to Staphylococcus).
RidinilazoleRidinilazole is under investigation in clinical trial NCT02092935 (A Study of SMT19969 Compared With Vancomycin for the Treatment of Clostridium Difficile-Associated Diarrhoea (CDAD)).
AconiazideNot Annotated
Gentamicin C2Not Annotated
EnmetazobactamA beta-lactamase inhibitor used to treat complicated urinary tract infections in combination with cefepime.
Drugs & Drug Targets
DrugTargetType
Gramicidin DP-glycoprotein 1transporter
Erythromycin23S ribosomal RNAtarget
ErythromycinCytochrome P450 3A4enzyme
ErythromycinCytochrome P450 3A7enzyme
ErythromycinP-glycoprotein 1transporter
ErythromycinSolute carrier organic anion transporter family member 1B1transporter
ErythromycinMotilin receptortarget
ErythromycinPotassium voltage-gated channel subfamily H member 2target
ErythromycinCytochrome P450 3A5enzyme
ErythromycinSolute carrier organic anion transporter family member 1B3transporter
ErythromycinBile salt export pumptransporter
ErythromycinCanalicular multispecific organic anion transporter 1transporter
ErythromycinSolute carrier organic anion transporter family member 1A2transporter
CycloserineD-alanine--D-alanine ligase Atarget
CycloserineAlanine racemasetarget
CycloserineAromatic-L-amino-acid decarboxylaseenzyme
CycloserineProton-coupled amino acid transporter 2transporter
Capreomycin16S/23S rRNA (cytidine-2'-O)-methyltransferase TlyAtarget
Framycetin30S ribosomal protein S12target
Framycetin16S ribosomal RNAtarget
FramycetinC-X-C chemokine receptor type 4target
Oxytetracycline30S ribosomal protein S4target
Oxytetracycline30S ribosomal protein S9target
Oxytetracycline16S ribosomal RNAtarget
OxytetracyclineSolute carrier family 22 member 6transporter
OxytetracyclineSolute carrier family 22 member 8transporter
OxytetracyclineSolute carrier family 22 member 11transporter
OxytetracyclineSolute carrier family 22 member 7transporter
OxytetracyclineSerum albumincarrier
RifabutinDNA-directed RNA polymerase subunit alphatarget
RifabutinHeat shock protein HSP 90-alphatarget
RifabutinEndoplasmintarget
RifabutinCytochrome P450 3A4enzyme
RifabutinDNA-directed RNA polymerase subunit betatarget
RifabutinDNA-directed RNA polymerase subunit beta'target
RifabutinCytochrome P450 2C19enzyme
RifabutinCytochrome P450 2B6enzyme
RifabutinCytochrome P450 2C8enzyme
RifabutinCytochrome P450 2C9enzyme
RifabutinP-glycoprotein 1transporter
BacitracinAlpha-2-macroglobulintarget
BacitracinInsulin-degrading enzymetarget
BacitracinC55-isoprenyl pyrophosphatetarget
BacitracinBacitracin transport ATP-binding protein BcrAtransporter
BacitracinBacitracin transport permease protein BCRBtransporter
BacitracinBacitracin transport permease protein BcrCtransporter
BenzylpenicillinSolute carrier family 22 member 5transporter
BenzylpenicillinSolute carrier family 15 member 1transporter
BenzylpenicillinSolute carrier family 15 member 2transporter
BenzylpenicillinSolute carrier family 22 member 6transporter
BenzylpenicillinSolute carrier family 22 member 8transporter
BenzylpenicillinSolute carrier family 22 member 4transporter
BenzylpenicillinSolute carrier family 22 member 11transporter
BenzylpenicillinSolute carrier organic anion transporter family member 2B1transporter
BenzylpenicillinSolute carrier organic anion transporter family member 4A1transporter
BenzylpenicillinSolute carrier organic anion transporter family member 3A1transporter
BenzylpenicillinSolute carrier organic anion transporter family member 1B1transporter
BenzylpenicillinPenicillin-binding protein 3target
BenzylpenicillinSolute carrier family 22 member 8target
BenzylpenicillinSolute carrier family 15 member 1target
BenzylpenicillinSolute carrier family 15 member 2target
BenzylpenicillinBeta-lactamase TEMenzyme
BenzylpenicillinSerum albumincarrier
Streptomycin30S ribosomal protein S12target
Streptomycin16S ribosomal RNAtarget
StreptomycinProtein-arginine deiminase type-4target
Streptomycin23S ribosomal RNAtarget
StreptomycinBacterial outer membranetarget
StreptomycinCytoplasmic membranetarget
CandicidinErgosteroltarget
CandicidinCytochrome P450 3A4enzyme
RifapentineDNA-directed RNA polymerase subunit beta'target
RifapentineCytochrome P450 2C8enzyme
RifapentineCytochrome P450 2C9enzyme
RifapentineCytochrome P450 3A4enzyme
RifapentineCytochrome P450 2C19enzyme
RifapentineCytochrome P450 2B6enzyme
RifapentineCytochrome P450 3A Subfamilyenzyme
Paromomycin16S ribosomal RNAtarget
Paromomycin30S ribosomal protein S10target
Paromomycin40S ribosomal protein SAtarget
Paromomycin60S ribosomal protein L10-liketarget
Fusidic acidChloramphenicol acetyltransferase 3target
Fusidic acidChloramphenicol acetyltransferasetarget
Fusidic acidBile salt export pumptransporter
Fusidic acidCanalicular multispecific organic anion transporter 1transporter
Fusidic acidElongation factor Gtarget
Fusidic acidCytochrome P450 2D6enzyme
Fusidic acidCytochrome P450 3A4enzyme
Fusidic acidUDP-glucuronosyltransferase 1-1enzyme
Fusidic acidATP-binding cassette sub-family G member 2transporter
Fusidic acidSolute carrier organic anion transporter family member 1B1transporter
TyrothricinAcetylcholinesterasetarget
TyrothricinBeta-galactosidasetarget
TyrothricinPhospholipid membranetarget
Neomycin30S ribosomal protein S12target
Neomycin16S ribosomal RNAtarget
NeomycinExtracellular calcium-sensing receptortarget
Azithromycin23S ribosomal RNAtarget
AzithromycinP-glycoprotein 1transporter
AzithromycinCytochrome P450 3A4enzyme
AzithromycinProtein-arginine deiminase type-4target
AzithromycinCanalicular multispecific organic anion transporter 1transporter
MoxifloxacinDNA gyrase subunit Atarget
MoxifloxacinDNA topoisomerase 4 subunit Atarget
MoxifloxacinDNA topoisomerase 2-alphatarget
MoxifloxacinCytochrome P450 1A2enzyme
MoxifloxacinSerum paraoxonase/arylesterase 1target
MupirocinIsoleucine--tRNA ligasetarget
ChloramphenicolComplement decay-accelerating factortarget
ChloramphenicolDr hemagglutinin structural subunittarget
ChloramphenicolCytochrome P450 2C19enzyme
ChloramphenicolCytochrome P450 3A4enzyme
ChloramphenicolCytochrome P450 3A5enzyme
ChloramphenicolCytochrome P450 3A7enzyme
ChloramphenicolSolute carrier family 22 member 6transporter
Chloramphenicol50S ribosomal protein L16target
ChloramphenicolChloramphenicol acetyltransferase 3enzyme
ChloramphenicolChloramphenicol acetyltransferaseenzyme
ChloramphenicolChloramphenicol 3-O phosphotransferaseenzyme
CiprofloxacinDNA gyrase subunit Atarget
CiprofloxacinDNA topoisomerase 4 subunit Atarget
CiprofloxacinDNA topoisomerase 2-alphatarget
CiprofloxacinCytochrome P450 1A2enzyme
CiprofloxacinCytochrome P450 3A4enzyme
CiprofloxacinCytochrome P450 3A5enzyme
CiprofloxacinCytochrome P450 3A7enzyme
CiprofloxacinP-glycoprotein 1transporter
CiprofloxacinPotassium voltage-gated channel subfamily H member 2target
CiprofloxacinDNA gyrase subunit Atarget
CiprofloxacinDNA topoisomerase 4 subunit Atarget
CiprofloxacinDNA topoisomerase 4 subunit Btarget
CiprofloxacinDNA gyrase subunit Atarget
CiprofloxacinMultidrug resistance protein MdtKtarget
CiprofloxacinGyrase Atarget
CiprofloxacinDNA gyrase subunit Atarget
CiprofloxacinMultidrug and toxin extrusion protein 1transporter
CiprofloxacinMultidrug and toxin extrusion protein 2transporter
CiprofloxacinSerum albumincarrier
Tobramycin16S ribosomal RNAtarget
TobramycinBacterial outer membranetarget
TobramycinCytoplasmic membranetarget
Tobramycin23S ribosomal RNAtarget
Tetracycline16S ribosomal RNAtarget
TetracyclineMajor prion proteintarget
TetracyclineSerum albumincarrier
TetracyclineCytochrome P450 3A4enzyme
TetracyclineSolute carrier family 22 member 6transporter
TetracyclineSolute carrier family 22 member 8transporter
TetracyclineSolute carrier family 22 member 11transporter
TetracyclineSolute carrier family 22 member 7transporter
Tetracycline30S ribosomal protein S3target
Tetracycline30S ribosomal protein S8target
Tetracycline30S ribosomal protein S19target
Tetracycline30S ribosomal protein S14target
Tetracycline30S ribosomal protein S7target
TetracyclineMultidrug translocase MdfAtarget
TetracyclineProtein-arginine deiminase type-4target
TetracyclineSolute carrier organic anion transporter family member 2B1transporter
Gentamicin30S ribosomal protein S12target
Gentamicin16S ribosomal RNAtarget
GentamicinNH(3)-dependent NAD(+) synthetasetarget
GentamicinDihydrofolate reductasetarget
Gentamicin23S ribosomal RNAtarget
GentamicinBacterial outer membranetarget
GentamicinCytoplasmic membranetarget
GentamicinLow-density lipoprotein receptor-related protein 2transporter
GentamicinSolute carrier family 22 member 2transporter
GentamicinCanalicular multispecific organic anion transporter 1transporter
Minocycline30S ribosomal protein S4target
Minocycline30S ribosomal protein S9target
Minocycline16S ribosomal RNAtarget
MinocyclineInterleukin-1 betatarget
MinocyclineArachidonate 5-lipoxygenasetarget
MinocyclineMatrix metalloproteinase-9target
MinocyclineVascular endothelial growth factor Atarget
MinocyclineCaspase-1target
MinocyclineCaspase-3target
MinocyclineCytochrome ctarget
MinocyclineSolute carrier family 22 member 6transporter
MinocyclineSolute carrier family 22 member 7transporter
MinocyclineOuter membrane protein Ftransporter
MinocyclineOuter membrane porin Ctransporter
MinocyclineMitogen-activated Protein Kinasestarget
MinocyclineNitric oxide synthase, inducibletarget
GatifloxacinSerum albumincarrier
GatifloxacinDNA gyrase subunit Atarget
GatifloxacinDNA gyrase subunit Btarget
GatifloxacinDNA topoisomerase 4 subunit Atarget
GatifloxacinDNA topoisomerase 4 subunit Btarget
GatifloxacinCytochrome P450 1A2enzyme
NorfloxacinDNA gyrase subunit Atarget
NorfloxacinDNA topoisomerase 4 subunit Atarget
NorfloxacinDNA topoisomerase 2-alphatarget
NorfloxacinCytochrome P450 1A2enzyme
NorfloxacinCytochrome P450 3A4enzyme
NorfloxacinSolute carrier family 22 member 5transporter
NorfloxacinSolute carrier family 22 member 6transporter
NorfloxacinCytochrome P450 1A1enzyme
NorfloxacinCytochrome P450 3A7enzyme
NorfloxacinDNA gyrase subunit Atarget
NorfloxacinDNA topoisomerase 2target
NorfloxacinDNA topoisomerase 4 subunit Atarget
OfloxacinDNA gyrase subunit Atarget
OfloxacinDNA topoisomerase 4 subunit Atarget
OfloxacinDNA topoisomerase 2-alphatarget
OfloxacinCytochrome P450 1A2enzyme
OfloxacinSolute carrier family 22 member 5transporter
OfloxacinMultidrug resistance-associated protein 1transporter
OfloxacinSolute carrier family 22 member 6transporter
OfloxacinCanalicular multispecific organic anion transporter 1transporter
OfloxacinSolute carrier family 22 member 4transporter
OfloxacinBile salt export pumptransporter
ClindamycinCytochrome P450 3A4enzyme
ClindamycinCytochrome P450 3A5enzyme
ClindamycinAlpha-1-acid glycoprotein 1carrier
ClindamycinP-glycoprotein 1transporter
Clindamycin50S ribosomal protein L1target
Kanamycin30S ribosomal protein S12target
Kanamycin16S ribosomal RNAtarget
KanamycinAminoglycoside 2'-N-acetyltransferaseenzyme
KanamycinKanamycin nucleotidyltransferaseenzyme
KanamycinAminoglycoside 3'-phosphotransferaseenzyme
Amphotericin BErgosteroltarget
NatamycinErgosteroltarget
DaptomycinCytoplasmic membranetarget
DaptomycinSerum albumincarrier
DaptomycinAlpha-1-acid glycoprotein 1carrier
DaptomycinAlpha-1-antitrypsincarrier
DaptomycinLow-density lipoprotein receptorcarrier
DaptomycinSex hormone-binding globulincarrier
DaptomycinHemopexincarrier
DaptomycinP-glycoprotein 1transporter
CefotiamPenicillin-binding protein 1Atarget
CefotiamSolute carrier family 22 member 6transporter
CefotiamSolute carrier family 22 member 8transporter
Aminosalicylic acidGroup IIE secretory phospholipase A2target
Aminosalicylic acidProstaglandin G/H synthase 2target
Aminosalicylic acidArachidonate 5-lipoxygenasetarget
Aminosalicylic acidInhibitor of nuclear factor kappa-B kinase subunit alphatarget
Aminosalicylic acidMyeloperoxidaseenzyme
DapsoneInactive dihydropteroate synthase 2target
DapsoneDihydropteroate synthase 1target
DapsoneCytochrome P450 2C9enzyme
DapsoneCytochrome P450 2E1enzyme
DapsoneCytochrome P450 3A4enzyme
DapsoneDimethylaniline monooxygenase [N-oxide-forming] 3enzyme
DapsoneProstaglandin G/H synthase 1enzyme
DapsoneProstaglandin G/H synthase 2enzyme
DapsoneCytochrome P450 2C8enzyme
DapsoneCytochrome P450 2C19enzyme
DapsoneArylamine N-acetyltransferase 2enzyme
DapsoneCytochrome P450 3A5enzyme
DapsoneCytochrome P450 3A7enzyme
DapsoneMyeloperoxidaseenzyme
DapsoneCytochrome P450 2C18enzyme
SulfanilamideDihydropteroate synthasetarget
CefmenoximePenicillin-binding protein 1Atarget
CefmenoximePeptidoglycan synthase FtsItarget
CefmetazolePenicillin binding protein 2atarget
CefmetazoleSerum albumincarrier
CefmetazoleSolute carrier family 15 member 1transporter
CefmetazoleSolute carrier family 15 member 2transporter
CefmetazolePenicillin-binding protein 1Atarget
CefmetazolePenicillin-binding protein 1Btarget
CefmetazolePeptidoglycan synthase FtsItarget
CefmetazoleD-alanyl-D-alanine carboxypeptidase DacAtarget
CefmetazoleD-alanyl-D-alanine carboxypeptidase DacCtarget
FlucloxacillinPenicillin-binding protein 1Atarget
FlucloxacillinCytochrome P450 3A4enzyme
FlucloxacillinBile salt export pumptransporter
ErtapenemPenicillin-binding protein 2target
ErtapenemPeptidoglycan synthase FtsItarget
ErtapenemPenicillin-binding protein 1Atarget
ErtapenemD-alanyl-D-alanine carboxypeptidase DacCtarget
ErtapenemD-alanyl-D-alanine carboxypeptidase DacBtarget
ErtapenemPenicillin-binding protein 1Btarget
ErtapenemPeptidoglycan synthase FtsItarget
ErtapenemPenicillin-binding protein 2target
ErtapenemSerum albumincarrier
ErtapenemDipeptidase 1enzyme
PiperacillinSolute carrier family 22 member 6transporter
PiperacillinPenicillin-binding protein 3target
PiperacillinPenicillin-binding protein 2Btarget
PiperacillinPenicillin-binding protein 2atarget
PiperacillinPenicillin-binding protein 1btarget
PiperacillinSolute carrier family 22 member 8transporter
EthambutolProbable arabinosyltransferase Btarget
EthambutolProbable arabinosyltransferase Atarget
EthambutolProbable arabinosyltransferase Ctarget
EthambutolCytochrome P450 1A2enzyme
EthambutolCytochrome P450 2E1enzyme
EthambutolCytochrome P450 2C19enzyme
EthambutolCytochrome P450 2D6enzyme
EthambutolCytochrome P450 2A6enzyme
EthambutolCytochrome P450 2C9enzyme
EthambutolCytochrome P450 3A4enzyme
PyrazinamideXanthine dehydrogenase/oxidaseenzyme
PyrazinamideFatty acid synthetasetarget
PyrazinamideAldehyde oxidaseenzyme
AztreonamPenicillin-binding protein 3target
AztreonamBeta-lactamasetarget
AztreonamBeta-lactamase Toho-1target
GrepafloxacinDNA gyrase subunit Atarget
GrepafloxacinDNA topoisomerase 4 subunit Atarget
GrepafloxacinCytochrome P450 3A4enzyme
GrepafloxacinCytochrome P450 1A2enzyme
GrepafloxacinSolute carrier family 22 member 2transporter
GrepafloxacinSolute carrier family 22 member 5transporter
GrepafloxacinCanalicular multispecific organic anion transporter 1transporter
GrepafloxacinP-glycoprotein 1transporter
GrepafloxacinMultidrug resistance-associated protein 1transporter
GrepafloxacinSolute carrier family 22 member 6transporter
AmpicillinSerum albumincarrier
AmpicillinSolute carrier family 22 member 5transporter
AmpicillinSolute carrier family 15 member 1transporter
AmpicillinSolute carrier family 15 member 2transporter
AmpicillinPenicillin-binding protein 2atarget
AmpicillinPenicillin-binding protein 1btarget
AmpicillinPenicillin-binding protein 3target
AmpicillinPenicillin-binding protein 1Atarget
AmpicillinPenicillin-binding protein 2Btarget
AmpicillinMonocarboxylate transporter 1transporter
AmpicillinSolute carrier family 15 member 1target
AmpicillinSolute carrier family 15 member 2target
AmpicillinAngiopoietin-1 receptortarget
PhenoxymethylpenicillinPenicillin-binding protein 1Atarget
PhenoxymethylpenicillinMecA PBP2' (penicillin binding protein 2')target
PhenoxymethylpenicillinD-alanyl-D-alanine carboxypeptidase DacBtarget
PhenoxymethylpenicillinPenicillin acylasetarget
PhenoxymethylpenicillinSolute carrier family 15 member 1target
CefpiramidePenicillin binding protein 2atarget
CefpiramideSerum albumincarrier
CefpiramidePeptidoglycan synthase FtsItarget
CefpiramidePenicillin-binding protein 1Btarget
CefpiramidePenicillin-binding protein 1Atarget
CefpiramidePenicillin-binding protein 1Btarget
CefpiramideD-alanyl-D-alanine carboxypeptidase DacCtarget
CefpiramidePenicillin-binding protein 1Atarget
CeftazidimeSolute carrier family 22 member 6transporter
CeftazidimePeptidoglycan synthase FtsItarget
CeftazidimePenicillin-binding protein 1Atarget
CeftazidimePenicillin-binding protein 1Btarget
CeftazidimePenicillin-binding protein 2target
CeftazidimeSerum albumincarrier
CeftazidimeBeta-lactamase Toho-1target
LoracarbefPenicillin-binding protein 1Atarget
LoracarbefSolute carrier family 15 member 1transporter
LoracarbefSolute carrier family 15 member 2transporter
LoracarbefPenicillin-binding protein 3target
CefalotinPenicillin-binding protein 1Atarget
CefalotinD-alanyl-D-alanine carboxypeptidasetarget
CefalotinBeta-lactamasetarget
CefalotinSolute carrier family 22 member 5transporter
CefalotinSolute carrier family 15 member 1transporter
CefalotinSolute carrier family 15 member 2transporter
CefalotinSolute carrier family 22 member 6transporter
CefalotinSolute carrier family 22 member 8transporter
CefalotinSolute carrier family 22 member 11transporter
CefalotinSolute carrier family 22 member 7transporter
CefalotinPenicillin-binding protein 1Atarget
CefalotinPenicillin-binding protein 1btarget
CefalotinPenicillin-binding protein 3target
CefalotinPenicillin-binding protein 2atarget
CefalotinPenicillin-binding protein 2Btarget
CefalotinSerum albumincarrier
EnoxacinDNA gyrase subunit Atarget
EnoxacinDNA topoisomerase 4 subunit Atarget
EnoxacinDNA topoisomerase 2-alphatarget
EnoxacinCytochrome P450 1A2enzyme
Amikacin30S ribosomal protein S12target
DicloxacillinSolute carrier family 15 member 1transporter
DicloxacillinSolute carrier family 15 member 2transporter
DicloxacillinPenicillin-binding protein 3target
DicloxacillinPenicillin-binding protein 1btarget
DicloxacillinPenicillin-binding protein 2atarget
DicloxacillinPenicillin-binding protein 3target
DicloxacillinPenicillin-binding protein 1Atarget
DicloxacillinPenicillin-binding protein 2Btarget
DicloxacillinCytochrome P450 3A4enzyme
DicloxacillinSerum albumincarrier
PefloxacinDNA gyrase subunit Atarget
PefloxacinDNA topoisomerase 4 subunit Atarget
PefloxacinDNA topoisomerase 2-alphatarget
PefloxacinCytochrome P450 1A2enzyme
PefloxacinDNA topoisomerase 1target
CefotaximePenicillin-binding protein 3target
CefotaximeSolute carrier family 15 member 1transporter
CefotaximeSolute carrier family 15 member 2transporter
CefotaximeSolute carrier family 22 member 6transporter
CefotaximeSolute carrier family 22 member 8transporter
CefotaximeSolute carrier family 22 member 11transporter
CefotaximeSolute carrier family 22 member 7transporter
CefotaximePenicillin-binding protein 1btarget
CefotaximePenicillin-binding protein 2atarget
CefotaximePenicillin-binding protein 1Atarget
CefotaximePenicillin-binding protein 2Btarget
CefotaximeSolute carrier family 22 member 6target
CefotaximeSolute carrier family 22 member 8target
CefotaximeSolute carrier family 22 member 11target
CefotaximeSolute carrier family 22 member 7target
CefotaximeSolute carrier family 15 member 1target
CefotaximeSerum albumintarget
CefotaximeBeta-lactamasetarget
CefotaximeSolute carrier family 15 member 2target
VancomycinD-Ala-D-Ala moiety of NAM/NAG peptide subunits of peptidoglycantarget
VancomycinSerum albumincarrier
Vancomycinalpha1-acid glycoproteincarrier
VancomycinHistamine H1 receptorcarrier
CefdinirMyeloperoxidasetarget
CefdinirPenicillin-binding protein 2target
CefdinirPBP3target
CefdinirSolute carrier family 22 member 5transporter
CefdinirSolute carrier family 15 member 1transporter
CefdinirSolute carrier family 15 member 2transporter
CefdinirSolute carrier family 22 member 6transporter
CefdinirSolute carrier family 22 member 8transporter
CefdinirPeptidoglycan transpeptidasetarget
CephalexinSerum albumincarrier
CephalexinSolute carrier family 22 member 5transporter
CephalexinSolute carrier family 15 member 1transporter
CephalexinSolute carrier family 15 member 2transporter
CephalexinSolute carrier family 22 member 6transporter
CephalexinSolute carrier family 22 member 8transporter
CephalexinMultidrug and toxin extrusion protein 1transporter
CephalexinPenicillin-binding protein 3target
CephalexinPenicillin-binding protein 2atarget
CephalexinPenicillin-binding protein 1btarget
CephalexinPenicillin-binding protein 1Atarget
CephalexinPenicillin-binding protein 2Btarget
CarbenicillinSolute carrier family 22 member 6transporter
CarbenicillinPenicillin-binding proteintarget
CarbenicillinCytosolic phospholipase A2enzyme
CarbenicillinBeta-lactamase Toho-1target
Linezolid23S ribosomal RNAtarget
LinezolidAmine oxidase [flavin-containing] Aenzyme
LinezolidAmine oxidase [flavin-containing] Benzyme
LinezolidSerum albumincarrier
LinezolidSolute carrier family 22 member 6transporter
LinezolidSolute carrier family 22 member 8transporter
NafcillinCytochrome P450 1A2enzyme
NafcillinCytochrome P450 3A4enzyme
NafcillinSolute carrier family 22 member 6transporter
NafcillinPenicillin-binding protein 1btarget
NafcillinPenicillin-binding protein 2Btarget
NafcillinPenicillin-binding protein 2atarget
NafcillinPenicillin-binding protein 3target
NafcillinPenicillin-binding protein 1Atarget
NafcillinSerum albumincarrier
EthionamideCatalase-peroxidasetarget
EthionamideEnoyl-[acyl-carrier-protein] reductase [NADH]target
CefiximePenicillin-binding protein 2target
CefiximeSolute carrier family 22 member 5transporter
CefiximeSolute carrier family 15 member 1transporter
CefiximeSolute carrier family 15 member 2transporter
CephaloglycinSolute carrier family 22 member 5transporter
CephaloglycinPenicillin-binding protein 1Btarget
OxacillinPenicillin-binding protein 1Atarget
OxacillinSolute carrier family 15 member 1transporter
OxacillinSolute carrier family 15 member 2transporter
OxacillinPenicillin-binding protein 3target
OxacillinPenicillin-binding protein 2atarget
OxacillinPenicillin-binding protein 1Atarget
OxacillinPenicillin-binding protein 2Btarget
OxacillinPenicillin-binding protein 1btarget
OxacillinSolute carrier family 15 member 1target
OxacillinPenicillin-binding protein 2target
OxacillinSolute carrier family 15 member 2target
OxacillinBeta-lactamase Toho-1target
MeropenemD-alanyl-D-alanine carboxypeptidase DacBtarget
MeropenemBeta-lactamase OXA-10enzyme
MeropenemDipeptidase 1enzyme
Clavulanic acidBacterial beta-lactamase enzymestarget
Clavulanic acidSodium/glucose cotransporter 1transporter
Roxithromycin50S ribosomal protein L10target
RoxithromycinP-glycoprotein 1target
RoxithromycinCytochrome P450 3A4enzyme
RoxithromycinCytochrome P450 2B6enzyme
Nalidixic acidDNAtarget
Nalidixic acidSolute carrier family 22 member 6transporter
Nalidixic acidTryptophan 2,3-dioxygenaseenzyme
Nalidixic acidCytochrome P450 1A2enzyme
ColistinBacterial outer membranetarget
FosfomycinUDP-N-acetylglucosamine 1-carboxyvinyltransferasetarget
CefaclorPenicillin-binding protein 1Atarget
CefaclorSolute carrier family 15 member 1transporter
CefaclorSolute carrier family 15 member 2transporter
CefaclorPenicillin-binding protein 3target
CefaclorMyeloperoxidaseenzyme
CefaclorSolute carrier family 22 member 8transporter
CefaclorBile salt export pumptransporter
ClofazimineCytochrome P450 3A4enzyme
ClofaziminePeroxisome proliferator-activated receptor gammatarget
ClofazimineCytochrome P450 2C8enzyme
ClofazimineCytochrome P450 2D6enzyme
ClofazimineCytochrome P450 3A5enzyme
ClofaziminePotassium voltage-gated channel subfamily A member 3target
ClofazimineSerum albumincarrier
ClofazimineP-glycoprotein 1transporter
ClofazimineATP-binding cassette sub-family G member 2transporter
ClofazimineMultidrug resistance-associated protein 1transporter
SirolimusCytochrome P450 3A4enzyme
SirolimusSerine/threonine-protein kinase mTORtarget
SirolimusCytochrome P450 3A5enzyme
SirolimusCytochrome P450 3A7enzyme
SirolimusP-glycoprotein 1transporter
SirolimusSolute carrier organic anion transporter family member 1B1transporter
SirolimusMultidrug and toxin extrusion protein 1transporter
SirolimusSerum albumincarrier
SirolimusAlpha-1-acid glycoprotein 1carrier
SirolimusApolipoproteinscarrier
Spectinomycin30S ribosomal protein S12target
CeforanidePenicillin-binding protein 2target
MezlocillinPenicillin-binding protein 1Atarget
MezlocillinPenicillin-binding protein 2target
MezlocillinPenicillin-binding protein 3target
Dirithromycin23S ribosomal RNAtarget
DirithromycinCytochrome P450 3A4enzyme
Netilmicin30S ribosomal protein S12target
Netilmicin16S ribosomal RNAtarget
Telithromycin23S ribosomal RNAtarget
TelithromycinCytochrome P450 3A4enzyme
TelithromycinSolute carrier organic anion transporter family member 1B1transporter
TelithromycinSolute carrier organic anion transporter family member 1B3transporter
LomefloxacinDNA gyrase subunit Atarget
LomefloxacinDNA topoisomerase 4 subunit Atarget
LomefloxacinDNA topoisomerase 2-alphatarget
LomefloxacinCytochrome P450 1A2enzyme
LomefloxacinSolute carrier family 22 member 5transporter
LomefloxacinCanalicular multispecific organic anion transporter 1transporter
CyclacillinSolute carrier family 22 member 5transporter
CyclacillinSolute carrier family 15 member 1transporter
CyclacillinSolute carrier family 15 member 2transporter
CyclacillinPenicillin-binding protein 1Atarget
CyclacillinPenicillin-binding protein 3target
CyclacillinPenicillin binding protein 2atarget
CyclacillinPenicillin-binding proteintarget
RifampicinDNA-directed RNA polymerase subunit betatarget
RifampicinNuclear receptor subfamily 1 group I member 2target
RifampicinCytochrome P450 3A4enzyme
RifampicinCytochrome P450 1A2enzyme
RifampicinCytochrome P450 2C8enzyme
RifampicinUDP-glucuronosyltransferase 1-1enzyme
RifampicinCytochrome P450 2C9enzyme
RifampicinCytochrome P450 2B6enzyme
RifampicinCytochrome P450 2C19enzyme
RifampicinCanalicular multispecific organic anion transporter 2transporter
RifampicinMultidrug resistance-associated protein 5transporter
RifampicinP-glycoprotein 1transporter
RifampicinCanalicular multispecific organic anion transporter 1transporter
RifampicinSolute carrier organic anion transporter family member 2B1transporter
RifampicinBile salt export pumptransporter
RifampicinMultidrug resistance-associated protein 1transporter
RifampicinSolute carrier organic anion transporter family member 1A2transporter
RifampicinSolute carrier organic anion transporter family member 1B3transporter
RifampicinSolute carrier family 22 member 7transporter
RifampicinSolute carrier organic anion transporter family member 1B1transporter
RifampicinCytochrome P450 2A6enzyme
RifampicinCytochrome P450 2E1enzyme
RifampicinCytochrome P450 3A43enzyme
RifampicinCytochrome P450 3A7enzyme
RifampicinSolute carrier family 22 member 6transporter
RifampicinSolute carrier family 22 member 8transporter
RifampicinUDP-glucuronosyltransferase 1-9enzyme
RifampicinCytochrome P450 3A5enzyme
RifampicinSerum albumincarrier
Rifampicinalpha1-acid glycoproteincarrier
NovobiocinDNA gyrase subunit Btarget
NovobiocinSolute carrier family 22 member 6transporter
NovobiocinSolute carrier family 22 member 8transporter
NovobiocinSolute carrier family 22 member 11transporter
NovobiocinATP-binding cassette sub-family G member 2transporter
NovobiocinDNA topoisomerase 1target
NovobiocinSolute carrier organic anion transporter family member 1B1transporter
NovobiocinSolute carrier organic anion transporter family member 1B3transporter
NovobiocinSolute carrier organic anion transporter family member 2B1transporter
AmoxicillinSolute carrier family 15 member 1transporter
AmoxicillinSolute carrier family 15 member 2transporter
AmoxicillinSolute carrier family 22 member 6transporter
AmoxicillinCytochrome P450 2C8enzyme
AmoxicillinSerum albumincarrier
AmoxicillinBeta-lactamase 2enzyme
AmoxicillinPenicillin binding proteintarget
AzlocillinPenicillin-binding protein 1Atarget
CefditorenPenicillin-binding protein 1Atarget
CefditorenPenicillin-binding protein 2Btarget
CefuroximePenicillin-binding protein 1Atarget
CefuroximeSolute carrier family 15 member 1transporter
CefuroximeSolute carrier family 15 member 2transporter
LevofloxacinDNA gyrase subunit Atarget
LevofloxacinDNA topoisomerase 4 subunit Atarget
LevofloxacinSolute carrier family 22 member 2transporter
LevofloxacinP-glycoprotein 1transporter
LevofloxacinSolute carrier family 22 member 4transporter
LevofloxacinMultidrug and toxin extrusion protein 1transporter
LevofloxacinMultidrug and toxin extrusion protein 2transporter
LevofloxacinCytochrome P450 2C9enzyme
LevofloxacinSerum albumincarrier
LevofloxacinSolute carrier organic anion transporter family member 4C1transporter
LevofloxacinSolute carrier family 22 member 1transporter
LevofloxacinSolute carrier organic anion transporter family member 1A2transporter
CefapirinPenicillin-binding protein 1Atarget
CefadroxilSolute carrier family 22 member 5transporter
CefadroxilSolute carrier family 15 member 1transporter
CefadroxilSolute carrier family 15 member 2transporter
CefadroxilSolute carrier family 22 member 6transporter
CefadroxilSolute carrier family 22 member 8transporter
CefadroxilPenicillin-binding protein 3target
CefadroxilPenicillin-binding protein 1Atarget
CefadroxilPenicillin-binding protein 1btarget
CefadroxilPenicillin-binding protein 2Btarget
CloxacillinSerum albumincarrier
CloxacillinSolute carrier family 15 member 1transporter
CloxacillinSolute carrier family 15 member 2transporter
CloxacillinD-alanyl-D-alanine carboxypeptidase DacAtarget
CloxacillinSolute carrier family 22 member 8transporter
CloxacillinPenicillin-binding protein 2Xtarget
CloxacillinPenicillin-binding protein 1Atarget
CefprozilPenicillin-binding protein 1Atarget
CefprozilPenicillin-binding protein 2xtarget
CefprozilPenicillin-binding protein 2Btarget
GemifloxacinDNA gyrase subunit Atarget
GemifloxacinDNA topoisomerase 4 subunit Atarget
GemifloxacinCytochrome P450 1A2enzyme
AmdinocillinPenicillin-binding protein 2target
AmdinocillinPenicillin-binding protein 2atarget
AmdinocillinPenicillin-binding protein 3target
AmdinocillinPenicillin-binding protein 1Atarget
AmdinocillinPenicillin-binding protein 2Btarget
AmdinocillinPenicillin-binding protein 1btarget
SparfloxacinDNA gyrase subunit Atarget
SparfloxacinDNA topoisomerase 4 subunit Atarget
SparfloxacinDNA topoisomerase 2-alphatarget
SparfloxacinSolute carrier family 22 member 5transporter
SparfloxacinCanalicular multispecific organic anion transporter 1transporter
SparfloxacinP-glycoprotein 1transporter
SparfloxacinCytochrome P450 1A2enzyme
Clarithromycin50S ribosomal protein L10target
ClarithromycinCytochrome P450 3A4enzyme
ClarithromycinCytochrome P450 3A5enzyme
ClarithromycinP-glycoprotein 1transporter
ClarithromycinSolute carrier family 22 member 7transporter
ClarithromycinPotassium voltage-gated channel subfamily H member 2target
ClarithromycinSolute carrier organic anion transporter family member 1B1target
ClarithromycinSolute carrier organic anion transporter family member 1B3target
ClarithromycinBile salt export pumptransporter
ClarithromycinSolute carrier organic anion transporter family member 1B1transporter
ClarithromycinSolute carrier organic anion transporter family member 1B3transporter
CeftriaxoneSerum albumincarrier
CeftriaxoneSolute carrier family 15 member 1transporter
CeftriaxoneSolute carrier family 15 member 2transporter
CeftriaxoneSolute carrier family 22 member 6transporter
CeftriaxoneSolute carrier family 22 member 8transporter
CeftriaxoneSolute carrier family 22 member 11transporter
CeftriaxonePenicillin-binding protein 2Btarget
CeftriaxoneGlutamine synthetaseenzyme
CeftriaxoneSolute carrier family 22 member 11target
CeftriaxoneSolute carrier family 22 member 6target
CeftriaxoneSolute carrier family 22 member 8target
CeftriaxoneSolute carrier family 15 member 1target
CeftriaxoneP-glycoprotein 1transporter
Josamycin50S ribosomal protein L4target
CefamandoleSolute carrier family 22 member 6transporter
CefamandoleSolute carrier family 22 member 8transporter
CefamandoleSolute carrier family 22 member 11transporter
CefamandoleSolute carrier family 22 member 7transporter
CefamandolePenicillin-binding protein 2target
CefazolinSerum paraoxonase/arylesterase 1target
CefazolinSerum albumincarrier
CefazolinSolute carrier family 22 member 6transporter
CefazolinSolute carrier family 22 member 8transporter
CefazolinSolute carrier family 22 member 11transporter
CefazolinPenicillin-binding protein 1Atarget
CefazolinPenicillin-binding protein 1Btarget
CefazolinPenicillin-binding protein 2target
CefazolinPenicillin-binding protein 1Ctarget
CefazolinPeptidoglycan synthase FtsItarget
CefazolinMultidrug resistance-associated protein 4transporter
CefazolinThiopurine S-methyltransferaseenzyme
CefazolinInterleukin-15target
CefazolinInterleukin-2target
CefonicidSerum albumincarrier
CefonicidPenicillin-binding protein 1Atarget
CefonicidPeptidoglycan synthase FtsItarget
CefonicidPenicillin-binding protein 1Btarget
CefonicidD-alanyl-D-alanine carboxypeptidase DacBtarget
CefonicidPenicillin-binding protein 2target
CefoperazoneSerum albumincarrier
CefoperazoneSolute carrier family 22 member 6transporter
CefoperazoneSolute carrier family 22 member 8transporter
CefoperazoneSolute carrier family 22 member 11transporter
CefoperazoneSolute carrier family 22 member 7transporter
CefoperazonePeptidoglycan synthase FtsItarget
CefoperazonePenicillin-binding protein 1Btarget
CefoperazonePenicillin-binding protein 2target
CefoperazonePenicillin-binding protein 1Atarget
CefoperazoneD-alanyl-D-alanine carboxypeptidase DacCtarget
CefoperazoneD-alanyl-D-alanine carboxypeptidase DacAtarget
CefoperazoneD-alanyl-D-alanine carboxypeptidase DacBtarget
CefoperazonePenicillin-binding protein 1Atarget
CefoperazonePenicillin-binding protein 1Btarget
CefotetanSerum albumincarrier
CefotetanPenicillin-binding protein 3target
CefoxitinPenicillin-binding protein 1Atarget
CefoxitinPenicillin-binding protein 1Btarget
CefoxitinPeptidoglycan synthase FtsItarget
CefoxitinD-alanyl-D-alanine carboxypeptidase DacAtarget
CefoxitinD-alanyl-D-alanine carboxypeptidase DacBtarget
CefoxitinD-alanyl-D-alanine carboxypeptidase DacCtarget
CefoxitinD-alanyl-D-alanine endopeptidasetarget
CefoxitinBeta-lactamaseenzyme
CefoxitinPenicillin-binding protein 3target
CefoxitinPenicillin-binding protein 1btarget
CefoxitinPenicillin-binding protein 2atarget
CefoxitinPenicillin-binding protein 1Atarget
CefoxitinPenicillin-binding protein 2Btarget
CeftizoximeSolute carrier family 15 member 1transporter
CeftizoximePenicillin-binding protein 1Atarget
CeftizoximePenicillin-binding protein 1Btarget
CeftizoximeSolute carrier family 22 member 6transporter
CeftizoximeSolute carrier family 22 member 8transporter
CeftizoximePeptidoglycan transpeptidasetarget
CeftizoximeD-alanyl-D-alanine carboxypeptidase DacCtarget
CefradineSolute carrier family 22 member 5transporter
CefradineSolute carrier family 15 member 1transporter
CefradineSolute carrier family 15 member 2transporter
CefradineSolute carrier family 22 member 6transporter
CefradinePenicillin-binding protein 1Atarget
CefradineCytochrome P450 3A4enzyme
CefradineMultidrug and toxin extrusion protein 1transporter
Quinupristin23S ribosomal RNAtarget
Quinupristin50S ribosomal protein L10target
Quinupristin50S ribosomal protein L22target
QuinupristinCytochrome P450 3A4enzyme
TemafloxacinDNA gyrase subunit Atarget
TemafloxacinDNA topoisomerase 4 subunit Atarget
TemafloxacinCytochrome P450 1A2enzyme
CefepimeSolute carrier family 22 member 5transporter
CefepimeSolute carrier family 15 member 1transporter
CefepimeSolute carrier family 15 member 2transporter
CefepimePenicillin-binding protein 2target
CefepimePeptidoglycan synthase FtsItarget
CefepimePenicillin-binding protein 3target
CefepimePenicillin-binding protein 2target
CefepimePenicillin-binding protein 1Atarget
CefepimePenicillin-binding protein 1Btarget
CefepimePenicillin-binding protein 1Btarget
CefacetrilePenicillin-binding protein 1Atarget
CefacetrilePenicillin-binding protein 1Btarget
CefacetrileSolute carrier family 22 member 6transporter
CefacetrileSolute carrier family 22 member 8transporter
CeftibutenSolute carrier family 15 member 1transporter
CeftibutenSolute carrier family 15 member 2transporter
CeftibutenPeptidoglycan synthase FtsItarget
CeftibutenPenicillin-binding protein 1Atarget
CeftibutenPenicillin-binding protein 1Btarget
CeftibutenPenicillin-binding protein 2target
CeftibutenSolute carrier family 22 member 6transporter
CeftibutenSolute carrier family 22 member 8transporter
CefpodoximePeptidoglycan synthase FtsItarget
ImipenemPenicillin-binding protein 1Atarget
ImipenemPenicillin-binding protein 1Btarget
ImipenemPenicillin-binding protein 2target
ImipenemPenicillin-binding protein 3target
ImipenemDipeptidase 1enzyme
ImipenemPenicillin-binding protein 4target
ImipenemBeta-lactamase SHV-1enzyme
ImipenemBeta-lactamase TEMenzyme
ImipenemBeta-lactamase CTX-Menzyme
ImipenemBeta-lactamase (KPC-2)enzyme
ImipenemBeta-lactamasetarget
BacampicillinPenicillin-binding proteintarget
MeticillinMecA PBP2' (penicillin binding protein 2')target
MeticillinPenicillin-binding protein 2atarget
MeticillinPenicillin-binding protein 1btarget
MeticillinPenicillin-binding protein 2Btarget
MeticillinPenicillin-binding protein 3target
MeticillinPenicillin-binding protein 1Atarget
PivampicillinPenicillin-binding protein 1Atarget
PivmecillinamPenicillin-binding protein 1Atarget
TicarcillinPenicillin binding protein 2atarget
Lincomycin23S ribosomal RNAtarget
LincomycinAlpha-1-acid glycoprotein 1carrier
Virginiamycin M1Streptogramin A acetyltransferasetarget
DalfopristinStreptogramin A acetyltransferasetarget
DalfopristinCytochrome P450 3A4enzyme
MaltotetraoseGlucan 1,4-alpha-maltotetraohydrolasetarget
MaltotetraoseNeopullulanase 2target
GE-2270AElongation factor Tutarget
UbenimexBacterial leucyl aminopeptidasetarget
UbenimexLeukotriene A-4 hydrolasetarget
UbenimexSolute carrier family 15 member 1transporter
UbenimexSolute carrier family 15 member 2transporter
UbenimexDipeptidase 1enzyme
RibostamycinProtein disulfide-isomerasetarget
Ribostamycin30S ribosomal protein S12target
RibostamycinAminoglycoside N(6')-acetyltransferase type 1target
RibostamycinAminoglycoside 2'-N-acetyltransferasetarget
RibostamycinAminoglycoside 2'-N-acetyltransferaseenzyme
AurodoxElongation factor Tu-Btarget
LatamoxefPenicillin-binding protein 3target
LatamoxefPenicillin-binding protein 1Atarget
LatamoxefPenicillin-binding protein 1Btarget
LatamoxefD-alanyl-D-alanine carboxypeptidase DacBtarget
Apramycin16S ribosomal RNAtarget
OritavancinCytochrome P450 3A4enzyme
OritavancinCytochrome P450 2D6enzyme
OritavancinCytochrome P450 2C9enzyme
OritavancinCytochrome P450 2C19enzyme
OritavancinSerum albumincarrier
OritavancinPeptidoglycan precursorstarget
OritavancinBacterial cell wall peptide bridging segmentstarget
OritavancinPentaglycyl bridging segmenttarget
CeftobiproleMecAtarget
CeftobiprolePenicillin-binding protein 2xtarget
CeftobiprolePeptidoglycan synthase FtsItarget
RifalazilDNA-directed RNA polymerase subunit betatarget
RifalazilCytochrome P450 3A4enzyme
Spiramycin50S ribosomal protein L3target
TeicoplaninD-Ala-D-Ala moiety of NAM/NAG peptide subunits of peptidoglycantarget
GarenoxacinCytochrome P450 1A2enzyme
DalbavancinD-Ala-D-Ala moiety of NAM/NAG peptide subunits of peptidoglycantarget
Cethromycin23S ribosomal RNAtarget
CethromycinCytochrome P450 3A5enzyme
CethromycinCytochrome P450 3A4enzyme
CethromycinP-glycoprotein 1transporter
Viomycin16S/23S rRNA (cytidine-2'-O)-methyltransferase TlyAtarget
Brefeldin ACytohesin-2target
Brefeldin AADP-ribosylation factor 1target
Brefeldin ACytochrome P450 3A4enzyme
Anisomycin60S ribosomal protein L10-liketarget
Anisomycin60S ribosomal protein L13atarget
Anisomycin60S ribosomal protein L23target
Anisomycin60S ribosomal protein L15target
Anisomycin60S ribosomal protein L19target
Anisomycin60S ribosomal protein L23atarget
AnisomycinProbable ribosome biogenesis protein RLP24target
Anisomycin60S ribosomal protein L26-like 1target
Anisomycin60S ribosomal protein L8target
Anisomycin60S ribosomal protein L37target
Anisomycin60S ribosomal protein L3target
Anisomycin60S ribosomal protein L11target
AnisomycinNHP2-like protein 1target
Chloramphenicol succinateDr hemagglutinin structural subunittarget
Chloramphenicol succinateSerum albumincarrier
Chloramphenicol succinateP-glycoprotein 1transporter
Chloramphenicol succinateChloramphenicol acetyltransferase 3enzyme
ThiamphenicolDr hemagglutinin structural subunittarget
BedaquilineCytochrome P450 3A4enzyme
BedaquilineATP synthase subunit ctarget
BedaquilineSerum albumincarrier
BedaquilineAlpha-1-acid glycoprotein 1carrier
CefaloridineSolute carrier family 22 member 6transporter
CefaloridineSolute carrier family 22 member 8transporter
Tedizolid phosphate23S ribosomal RNAtarget
Tedizolid phosphateAmine oxidase [flavin-containing] Aenzyme
Tedizolid phosphateAmine oxidase [flavin-containing] Benzyme
Chlortetracycline16S ribosomal RNAtarget
ChlortetracyclineSerum albumincarrier
Chlortetracycline30S ribosomal protein S3target
Chlortetracycline30S ribosomal protein S8target
Chlortetracycline30S ribosomal protein S19target
Chlortetracycline30S ribosomal protein S14target
Chlortetracycline30S ribosomal protein S7target
ChlortetracyclineADP-ribosylation factor 1target
ChlortetracyclineCatalasetarget
ChlortetracyclineEphrin type-B receptor 1target
ChlortetracyclinePancreatic triacylglycerol lipasetarget
ChlortetracyclineProtein-arginine deiminase type-4target
KitasamycinCytochrome P450 3A4enzyme
CarindacillinPenicillin-binding proteintarget
OleandomycinCytochrome P450 3A4enzyme
SalinomycinP-glycoprotein 1transporter
PazufloxacinCytochrome P450 1A2enzyme
PrulifloxacinCytochrome P450 1A2enzyme
TroleandomycinCytochrome P450 3A5enzyme
TroleandomycinCytochrome P450 3A43enzyme
Troleandomycin50S ribosomal protein L4target
Troleandomycin50S ribosomal protein L32target
TroleandomycinP-glycoprotein 1transporter
TroleandomycinCytochrome P450 2C8enzyme
TroleandomycinCytochrome P450 3A4enzyme
TroleandomycinNuclear receptor subfamily 1 group I member 2target
TroleandomycinCytochrome P450 3A7enzyme
SitafloxacinCytochrome P450 1A2enzyme
MiocamycinCytochrome P450 3A4enzyme
MidecamycinCytochrome P450 3A4enzyme
Pipemidic acidCytochrome P450 1A2enzyme
ClinafloxacinCytochrome P450 1A2enzyme
ClinafloxacinCytochrome P450 2C19enzyme
ClinafloxacinCytochrome P450 2D6enzyme
ClinafloxacinCytochrome P450 2C9enzyme
RifaximinDNA-directed RNA polymerase subunit betatarget
RifaximinNuclear receptor subfamily 1 group I member 2target
RifaximinCytochrome P450 3A4enzyme
RifaximinCytochrome P450 2C19enzyme
RifaximinCytochrome P450 2C8enzyme
FidaxomicinP-glycoprotein 1transporter
FidaxomicinRNA polymerase sigma factortarget
FidaxomicinCytochrome P450 3A4enzyme
SulfacetamideDihydropteroate synthasetarget
SulfacetamideDihydropteroate synthase type-1target
SulfacetamideFolic acid synthesis protein FOL1target
MetronidazoleOxygen-insensitive NADPH nitroreductasetarget
MetronidazoleCytochrome P450 2C9enzyme
MetronidazoleCytochrome P450 3A4enzyme
MetronidazoleCytochrome P450 2C8enzyme
MetronidazoleUDP-glucuronosyltransferase 1-1enzyme
MetronidazoleAnaerobic bacterial DNAtarget
MetronidazoleProtozoal DNAtarget
MetronidazoleP-glycoprotein 1transporter
MetronidazoleCytochrome P450 2A6enzyme
MetronidazoleCytochrome P450 3A5enzyme
MetronidazoleCytochrome P450 3A7enzyme
Retapamulin50S ribosomal protein L3target
RetapamulinCytochrome P450 3A4enzyme
BesifloxacinDNA topoisomerase 4 subunit Atarget
BesifloxacinDNA topoisomerase 4 subunit Atarget
BesifloxacinDNA gyrase subunit Atarget
BesifloxacinDNA gyrase subunit Atarget
BesifloxacinCytochrome P450 1A2enzyme
FinafloxacinDNA gyrase subunit Atarget
FinafloxacinDNA topoisomerase 4 subunit Atarget
FinafloxacinDNA topoisomerase 2-alphatarget
OzenoxacinDNA gyrase subunit Atarget
OzenoxacinDNA topoisomerase 4 subunit Atarget
SolithromycinCytochrome P450 3A4enzyme
FlurithromycinCytochrome P450 3A4enzyme
RokitamycinCytochrome P450 3A4enzyme
EverolimusSerine/threonine-protein kinase mTORtarget
EverolimusCytochrome P450 3A4enzyme
EverolimusSolute carrier organic anion transporter family member 1B1transporter
EverolimusSolute carrier organic anion transporter family member 1B3transporter
EverolimusSolute carrier organic anion transporter family member 1A2transporter
EverolimusCytochrome P450 2D6enzyme
EverolimusP-glycoprotein 1transporter
Epothilone DTubulin alpha 3C/D chaintarget
Epothilone DTubulin beta chaintarget
Epothilone DTubulin beta-1 chaintarget
Epothilone DTubulin beta-4B chaintarget
Epothilone DTubulin beta-4A chaintarget
Epothilone DTubulin alpha-4A chaintarget
Epothilone DTubulin beta-3 chaintarget
Epothilone DTubulin alpha-1C chaintarget
Epothilone DTubulin alpha-8 chaintarget
Epothilone DTubulin alpha-1B chaintarget
Epothilone DTubulin alpha-1A chaintarget
Epothilone DCytochrome P450 3A4enzyme
PatupiloneTubulin alpha 3C/D chaintarget
PatupiloneTubulin beta chaintarget
PatupiloneTubulin beta-1 chaintarget
PatupiloneTubulin beta-4B chaintarget
PatupiloneTubulin beta-4A chaintarget
PatupiloneTubulin alpha-4A chaintarget
PatupiloneTubulin beta-3 chaintarget
PatupiloneTubulin alpha-1C chaintarget
PatupiloneTubulin alpha-8 chaintarget
PatupiloneTubulin alpha-1B chaintarget
PatupiloneTubulin alpha-1A chaintarget
PatupiloneCytochrome P450 3A4enzyme
6-Deoxyerythronolide B6-deoxyerythronolide B hydroxylasetarget
6-Deoxyerythronolide BCytochrome P450 3A4enzyme
IxabepiloneTubulin beta-3 chaintarget
IxabepiloneCytochrome P450 3A4enzyme
IxabepiloneP-glycoprotein 1transporter
KOS-1584Cytochrome P450 3A4enzyme
RidaforolimusSerine/threonine-protein kinase mTORtarget
RidaforolimusCytochrome P450 3A4enzyme
TemsirolimusSerine/threonine-protein kinase mTORtarget
TemsirolimusCytochrome P450 3A4enzyme
TemsirolimusCytochrome P450 3A5enzyme
TemsirolimusCytochrome P450 3A7enzyme
TemsirolimusCytochrome P450 2D6enzyme
TemsirolimusP-glycoprotein 1transporter
AVE9633Myeloid cell surface antigen CD33target
AVE9633Cytochrome P450 3A4enzyme
Coltuximab ravtansineB-lymphocyte antigen CD19target
Coltuximab ravtansineCytochrome P450 3A4enzyme
MitemcinalMotilin receptortarget
MitemcinalCytochrome P450 3A4enzyme
CarbomycinCytochrome P450 3A4enzyme
DoramectinCytochrome P450 3A4enzyme
EprinomectinCytochrome P450 3A4enzyme
SelamectinCytochrome P450 3A4enzyme
TildipirosinCytochrome P450 3A4enzyme
Bryostatin 1Cytochrome P450 3A4enzyme
Bryostatin 1Protein kinase C alpha typetarget
Bryostatin 1Protein kinase C epsilon typetarget
Bryostatin 1Caspase-8target
Bryostatin 1Protein unc-13 homolog Btarget
Bryostatin 1Serine/threonine-protein kinase D1target
Bryostatin 1T-lymphocyte activation antigen CD86target
Bryostatin 1Prostaglandin G/H synthase 2target
Bryostatin 1G1/S-specific cyclin-D1target
Bryostatin 1Tumor necrosis factortarget
Lorvotuzumab mertansineCytochrome P450 3A4enzyme
EpofolateCytochrome P450 3A4enzyme
SagopiloneCytochrome P450 3A4enzyme
CefroxadineBeta-lactamaseenzyme
CefroxadinePenicillin-binding protein 1Btarget
Benzylpenicilloyl polylysineHigh affinity immunoglobulin epsilon receptor subunit gammatarget
Benzylpenicilloyl polylysineHigh affinity immunoglobulin epsilon receptor subunit alphatarget
AzidocillinPenicillin-binding protein 2atarget
AzidocillinPenicillin-binding protein 1btarget
AzidocillinPenicillin-binding protein 3target
AzidocillinPenicillin-binding protein 1Atarget
AzidocillinPenicillin-binding protein 2Btarget
AzidocillinSolute carrier family 22 member 5transporter
AzidocillinSolute carrier family 15 member 1transporter
AzidocillinSolute carrier family 15 member 2transporter
DoripenemDipeptidase 1enzyme
DoripenemPenicillin-binding protein 1Atarget
DoripenemPenicillin-binding protein 1Btarget
DoripenemPenicillin-binding protein 2target
DoripenemPenicillin-binding protein 3target
DoripenemPenicillin-binding protein 4target
DoripenemSolute carrier family 22 member 8transporter
Technetium Tc-99m ciprofloxacinDNA gyrase subunit Btarget
Technetium Tc-99m ciprofloxacinDNA topoisomerase 2-betatarget
Technetium Tc-99m ciprofloxacinCytochrome P450 1A2enzyme
OrbifloxacinCytochrome P450 1A2enzyme
SarafloxacinCytochrome P450 1A2enzyme
DifloxacinCytochrome P450 1A2enzyme
DifloxacinCytochrome P450 1A1enzyme
TrovafloxacinDNA gyrase subunit Atarget
TrovafloxacinDNA topoisomerase 4 subunit Atarget
TrovafloxacinDNA topoisomerase 2-alphatarget
TrovafloxacinCytochrome P450 1A2enzyme
RosoxacinDNA topoisomerase 4 subunit Atarget
RosoxacinDNA gyrase subunit Btarget
RosoxacinCytochrome P450 1A2enzyme
CinoxacinDNAtarget
CinoxacinDNA gyrase subunit Atarget
CinoxacinSolute carrier family 22 member 6transporter
CinoxacinCytochrome P450 1A2enzyme
FleroxacinDNA topoisomerase 2-alphatarget
FleroxacinDNA gyrase subunit Atarget
FleroxacinDNA topoisomerase 4 subunit Atarget
NemonoxacinCytochrome P450 1A2enzyme
FlumequineCytochrome P450 1A2enzyme
RufloxacinCytochrome P450 1A2enzyme
SulfamethoxazoleCytochrome P450 2C9enzyme
SulfamethoxazoleSerum albumincarrier
SulfamethoxazoleArylamine N-acetyltransferase 1enzyme
SulfamethoxazoleArylamine N-acetyltransferase 2enzyme
SulfamethoxazoleDihydropteroate synthasetarget
SulfamethoxazoleCytochrome P450 3A4enzyme
SulfamethoxazoleBile salt export pumptransporter
SulfisoxazoleDihydropteroate synthasetarget
SulfisoxazoleCytochrome P450 2C9enzyme
SulfadiazineCytochrome P450 2C9enzyme
SulfadiazineDihydropteroate synthetasetarget
SulfadiazineCytochrome P450 2C8enzyme
SulfadiazineCytochrome P450 3A4enzyme
Silver sulfadiazineDNAtarget
IsoniazidCatalase-peroxidasetarget
IsoniazidEnoyl-[acyl-carrier-protein] reductase [NADH]target
IsoniazidCytochrome P450 2E1enzyme
IsoniazidCytochrome P450 1A2enzyme
IsoniazidCytochrome P450 2C9enzyme
IsoniazidCytochrome P450 2D6enzyme
IsoniazidCytochrome P450 2C19enzyme
IsoniazidArylamine N-acetyltransferase 2enzyme
IsoniazidArylamine N-acetyltransferaseenzyme
IsoniazidCytochrome P450 2A6enzyme
IsoniazidCytochrome P450 2C8enzyme
IsoniazidCytochrome P450 2C8target
IsoniazidCytochrome P450 1A2target
IsoniazidCytochrome P450 3A4target
IsoniazidCytochrome P450 2C19target
IsoniazidDihydrofolate reductasetarget
IsoniazidSerum albumincarrier
IsoniazidCytochrome P450 3A4enzyme
GeneticinOrnithine decarboxylasetarget
Gentamicin C1a30S ribosomal protein S12target
Gentamicin C1a16S ribosomal RNAtarget
Arbekacin30S ribosomal protein S12target
Puromycin60S ribosomal protein L10-liketarget
Puromycin60S ribosomal protein L13atarget
Puromycin60S ribosomal protein L23target
Puromycin60S ribosomal protein L15target
Puromycin60S ribosomal protein L19target
Puromycin60S ribosomal protein L23atarget
PuromycinProbable ribosome biogenesis protein RLP24target
Puromycin60S ribosomal protein L26-like 1target
Puromycin60S ribosomal protein L8target
Puromycin60S ribosomal protein L37target
Puromycin60S ribosomal protein L3target
Puromycin60S ribosomal protein L11target
PuromycinLeucyl/phenylalanyl-tRNA--protein transferasetarget
PlazomicinMultidrug and toxin extrusion protein 1transporter
PlazomicinMultidrug and toxin extrusion protein 2transporter
Plazomicin30S ribosomal protein S14target
Plazomicin30S ribosomal protein S11target
SulfamerazineDihydropteroate synthasetarget
SulfamerazineSerum albumincarrier
SulfameterDihydropteroate synthasetarget
ValinomycinBile salt export pumptransporter
ValinomycinP-glycoprotein 1transporter
MafenideCarbonic anhydrase 6target
DoxycyclineSolute carrier family 22 member 6transporter
DoxycyclineCytochrome P450 3A4enzyme
DoxycyclineATP-binding cassette sub-family B member 5transporter
DoxycyclineSerum albumincarrier
Doxycycline30S ribosomal proteintarget
Lymecycline30S ribosomal protein S4target
Tigecycline30S ribosomal protein S9target
Tigecycline16S ribosomal RNAtarget
Tigecycline30S ribosomal protein S14target
Tigecycline30S ribosomal protein S13target
Tigecycline30S ribosomal protein S19target
Tigecycline30S ribosomal protein S12target
Demeclocycline30S ribosomal proteintarget
DemeclocyclineVasopressin V2 receptortarget
MetacyclineSerum albumincarrier
Metacycline16S ribosomal RNAtarget
Rolitetracycline30S ribosomal protein S9target
Rolitetracycline16S ribosomal RNAtarget
Tedizolid23S ribosomal RNAtarget
TedizolidAmine oxidase [flavin-containing] Aenzyme
TedizolidAmine oxidase [flavin-containing] Benzyme
RifamycinCytochrome P450 3A4enzyme
RifamycinCytochrome P450 2C19enzyme
RifamycinCytochrome P450 2B6enzyme
RifamycinCytochrome P450 2C8enzyme
RifamycinCytochrome P450 2C9enzyme
RifamycinSolute carrier organic anion transporter family member 1A2transporter
RifamycinSolute carrier organic anion transporter family member 1B1transporter
RifamycinSolute carrier organic anion transporter family member 1B3transporter
RifamycinSolute carrier organic anion transporter family member 2A1transporter
RifamycinSolute carrier organic anion transporter family member 2B1transporter
RifamycinSerum albumincarrier
RifamycinDNA-directed RNA polymerase subunit betatarget
RifamycinDNA-directed RNA polymerase subunit alphatarget
RifamycinDNA-directed RNA polymerase subunit beta'target
RifamycinMultidrug and toxin extrusion protein 1transporter
RifamycinCytochrome P450 1A2enzyme
RifamycinP-glycoprotein 1transporter
RifamycinCytochrome P450 2D6enzyme
CeftolozanePenicillin-binding protein 1Btarget
CeftolozanePenicillin-binding protein 3target
CeftolozanePenicillin-binding proteintarget
CeftolozanePenicillin-binding protein 1Ctarget
CeftolozanePenicillin-binding protein 2target
Acetyl sulfisoxazoleDihydropteroate synthasetarget
Acetyl sulfisoxazoleCytochrome P450 2C9enzyme
DelafloxacinUDP-glucuronosyltransferase 1-1enzyme
DelafloxacinUDP-glucuronosyltransferase 1-3enzyme
DelafloxacinUDP-glucuronosyltransferase 2B15enzyme
DelafloxacinDNA topoisomerase 4 subunit Atarget
DelafloxacinDNA gyrase subunit Atarget
DelafloxacinCytochrome P450 2E1enzyme
DelafloxacinCytochrome P450 2C9enzyme
DelafloxacinCytochrome P450 3A4enzyme
DelafloxacinATP-binding cassette sub-family B member 5transporter
DelafloxacinATP-binding cassette sub-family G member 2transporter
DelafloxacinSerum albumincarrier
Clomocycline30S ribosomal protein S4target
Clomocycline30S ribosomal protein S9target
Clomocycline16S ribosomal RNAtarget
SarecyclineP-glycoprotein 1transporter
OmadacyclineP-glycoprotein 1transporter
Omadacycline30S ribosomal protein S3target
Omadacycline30S ribosomal protein S7target
Omadacycline30S ribosomal protein S8target
Omadacycline30S ribosomal protein S19target
Omadacycline30S ribosomal protein S14target
Omadacycline16S ribosomal RNAtarget
OmadacyclineSerum albumincarrier
RadezolidRibosome-binding protein 1target
Radezolid50S ribosomal protein L1target
MeclocyclineOuter membrane protein Ftransporter
MeclocyclineOuter membrane porin Ctransporter
Meclocycline30S ribosomal protein S7target
MeclocyclineTetX family tetracycline inactivation enzymeenzyme
Polymyxin BBacterial outer membranetarget
Polymyxin BSolute carrier family 15 member 2transporter
EravacyclineCytochrome P450 3A4enzyme
EravacyclineAmine oxidase [flavin-containing] Aenzyme
Eravacycline30S ribosomal protein S4target
HetacillinPenicillin-binding protein 2atarget
HetacillinPenicillin-binding protein 1btarget
HetacillinPenicillin-binding protein 3target
HetacillinPenicillin-binding protein 1Atarget
HetacillinPenicillin-binding protein 2Btarget
Mycophenolate mofetilInosine-5'-monophosphate dehydrogenase 2target
Mycophenolate mofetilInosine-5'-monophosphate dehydrogenase 1target
Mycophenolate mofetilUDP-glucuronosyltransferase 1-1enzyme
Mycophenolate mofetilUDP-glucuronosyltransferase 1-7enzyme
Mycophenolate mofetilUDP-glucuronosyltransferase 1-6enzyme
Mycophenolate mofetilUDP-glucuronosyltransferase 1-9enzyme
Mycophenolate mofetilUDP-glucuronosyltransferase 2B7enzyme
Mycophenolate mofetilUDP-glucuronosyltransferase 1-8enzyme
Mycophenolate mofetilUDP-glucuronosyltransferase 1-10enzyme
Mycophenolate mofetilLiver carboxylesterase 1enzyme
Mycophenolate mofetilCytochrome P450 3A4enzyme
Mycophenolate mofetilCytochrome P450 3A5enzyme
Mycophenolate mofetilCytochrome P450 2C8enzyme
Mycophenolate mofetilSolute carrier organic anion transporter family member 1B1transporter
Mycophenolate mofetilSolute carrier organic anion transporter family member 1B3transporter
Mycophenolate mofetilATP-binding cassette sub-family G member 2transporter
Mycophenolate mofetilP-glycoprotein 1transporter
Mycophenolate mofetil6-pyruvoyl tetrahydrobiopterin synthasetarget
Mycophenolate mofetilCarboxylic ester hydrolaseenzyme
Mycophenolate mofetilCanalicular multispecific organic anion transporter 1transporter
Nitrofurantoin30S ribosomal protein S10target
NitrofurantoinOxygen-insensitive NADPH nitroreductasetarget
NitrofurantoinProbable pyruvate-flavodoxin oxidoreductasetarget
NitrofurantoinATP-binding cassette sub-family G member 2transporter
NitrofurantoinNADPH--cytochrome P450 reductaseenzyme
NitrofurantoinBile salt export pumptransporter
NitrofurantoinP-glycoprotein 1transporter
NitrofurantoinCanalicular multispecific organic anion transporter 1transporter
TinidazoleCytochrome P450 3A4enzyme
TinidazoleDNAtarget
TinidazoleBile salt export pumptransporter
Mycophenolic acidInosine-5'-monophosphate dehydrogenase 2target
Mycophenolic acidInosine-5'-monophosphate dehydrogenase 1target
Mycophenolic acidUDP-glucuronosyltransferase 1-1enzyme
Mycophenolic acidUDP-glucuronosyltransferase 1-9enzyme
Mycophenolic acidUDP-glucuronosyltransferase 2B7enzyme
Mycophenolic acidUDP-glucuronosyltransferase 1-7enzyme
Mycophenolic acidUDP-glucuronosyltransferase 1-6enzyme
Mycophenolic acidSerum albumincarrier
Mycophenolic acidUDP-glucuronosyltransferase 1-8enzyme
Mycophenolic acidUDP-glucuronosyltransferase 1-10enzyme
Mycophenolic acidCytochrome P450 3A4enzyme
Mycophenolic acidCytochrome P450 3A5enzyme
Mycophenolic acidCytochrome P450 2C8enzyme
Fosmidomycin1-deoxy-D-xylulose 5-phosphate reductoisomerasetarget
Acetic acidSolute carrier organic anion transporter family member 2B1transporter
Acetic acidMonocarboxylate transporter 1transporter
EnrofloxacinCytochrome P450 1A2enzyme
Malacidin ANAM/NAG peptide subunits of peptidoglycantarget
Malacidin BNAM/NAG peptide subunits of peptidoglycantarget
CefiderocolPenicillin-binding protein 3target
CefiderocolPenicillin-binding protein 1Atarget
CefiderocolPenicillin-binding protein 1Btarget
CefiderocolPenicillin-binding protein 2target
CefiderocolD-alanyl-D-alanine carboxypeptidase DacBtarget
CefiderocolMexAB-OprM efflux systemtransporter
CefiderocolSerum albumincarrier
CefiderocolCatecholate siderophore receptor Fiutransporter
CefiderocolColicin I receptortransporter
CefiderocolPutative outer membrane ferric siderophore receptortransporter
DurlobactamSolute carrier family 22 member 6transporter
DequaliniumE3 ubiquitin-protein ligase XIAPtarget
DequaliniumcGMP-gated cation channel alpha-1target
DequaliniumCalcium-activated potassium channel subunit alpha-1target
DequaliniumHTH-type transcriptional regulator QacRtarget
DequaliniumResponse regulator RamRtarget
DequaliniumAcriflavine resistance protein Btransporter
DequaliniumCalmodulintarget
DequaliniumSmall conductance calcium-activated potassium channel protein 3target
DequaliniumProtein kinase Ctarget
DequaliniumAlpha-synucleintarget
DequaliniumL-cysteine:1D-myo-inositol 2-amino-2-deoxy-alpha-D-glucopyranoside ligasetarget
SulfamethizoleDihydropteroate synthasetarget
SulfamethizoleSerum albumincarrier
SulfamethizoleCytochrome P450 2C9enzyme
LefamulinCytochrome P450 3A4enzyme
Lefamulin50S ribosomal protein L22target
LefamulinP-glycoprotein 1transporter
EnmetazobactamCytochrome P450 2E1enzyme
EnmetazobactamExtended-spectrum beta-lactamase PER-1target