Tranquilizing Agents

Name
Tranquilizing Agents
Accession Number
DBCAT000398
Description

A traditional grouping of drugs said to have a soothing or calming effect on mood, thought, or behavior. Included here are the ANTI-ANXIETY AGENTS (minor tranquilizers), ANTIMANIC AGENTS, and the ANTIPSYCHOTIC AGENTS (major tranquilizers). These drugs act by different mechanisms and are used for different therapeutic purposes.

Drugs
DrugDrug Description
LorazepamA short-acting benzodiazepine commonly used to treat panic disorders, severe anxiety, and seizures.
PregabalinAn anticonvulsant drug used to treat neuropathic pain conditions and fibromyalgia, and for the treatment of partial onset seizures in combination with other anticonvulsants.
TemazepamA short-acting benzodiazepine commonly used to treat panic disorders, severe anxiety, and insomnia.
ZiprasidoneAn atypical antipsychotic used to manage schizophrenia, bipolar mania, and agitation in patients with schizophrenia.
OlanzapineAn antipsychotic drug used in the management of schizophrenia, bipolar 1 disorder, and agitation associated with these disorders.
ClozapineAn atypical or second-generation antipsychotic drug used in treatment-resistant schizophrenia and to decrease suicide risk in schizophrenic patients.
MeprobamateAn anxiolytic drug used for the short-term management of anxiety symptoms.
SulpirideA selective D2 dopamine receptor antagonist indicated to treat chronic and acute schizophrenia.
AlprazolamA triazolobenzodiazepine with intermediate onset commonly used to treat panic disorders and generalized anxiety in addition to anxiety associated with depression.
LoxapineA antipsychotic used for the treatment of schizophrenia.
RemoxiprideAn discontinued atypical antipsychotic selective for dopamine D2 receptors.
PromazineA phenothiazine used to manage schizophrenia.
ProchlorperazineA phenothiazine derivative used in the treatment of schizophrenia and anxiety and to relieve severe nausea and vomiting.
ChlordiazepoxideA benzodiazepine used to treat the withdrawal symptoms of acute alcoholism, to treat preoperative anxiety, and to treat anxiety over a short term period.
ChlorpromazineA phenothiazine antipsychotic used to treat nausea, vomiting, preoperative anxiety, schizophrenia, bipolar disorder, and severe behavioral problems in children.
BuspironeAn anxiolytic agent used for short-term treatment of generalized anxiety and second-line treatment of depression.
HaloperidolAn antipsychotic agent used to treat schizophrenia and other psychoses, as well as symptoms of agitation, irritability, and delirium.
TriflupromazineUsed mainly in the management of psychoses. Also used to control nausea and vomiting.
FluphenazineA phenothiazine used to treat patients requiring long-term neuroleptic therapy.
Clorazepic acidA benzodiazepine used to treat anxiety, partial seizures, and alcohol withdrawal.
TrazodoneA serotonin uptake inhibitor used to treat major depressive disorder.
ThioridazineA phenothiazine antipsychotic used to treat schizophrenia and generalized anxiety disorder.
MidazolamA short-acting benzodiazepine with rapid onset that is commonly used in seizures, anesthesia and anxiety disorders.
FlurazepamA long-acting benzodiazepine with a rapid onset of action that is commonly used to treat insomnia.
RisperidoneA second-generation antipsychotic medication used to treat a number of mental health disorders including schizophrenia, bipolar mania, psychosis, or as an adjunct in severe depression.
HalazepamUsed to relieve anxiety, nervousness, and tension associated with anxiety disorders.
DiazepamA long-acting benzodiazepine with rapid onset commonly used to treat panic disorders, severe anxiety, alcohol withdrawal, and seizures.
TrifluoperazineA phenothiazine used to treat depression, anxiety, and agitation.
OxazepamAn intermediate-acting benzodiazepine with slow onset commonly used to treat panic disorders, severe anxiety, alcohol withdrawals, and insomnia.
PerphenazineA phenothiazine used to treat schizophrenia as well as nausea and vomiting.
FlupentixolA thioxanthene neuroleptic used to treat schizophrenia and depression.
TriazolamA benzodiazepine used for short term treatment of insomnia.
CyclobenzaprineA skeletal muscle relaxant that works on the brainstem to treat muscle spasms of local origin.
MesoridazineA phenothiazine antipsychotic used to treat schizophrenia, organic brain disorders, alcoholism, and psychoneuroses.
GabapentinAn anticonvulsant medication used in the management of peripheral neuropathic pains, postherpetic neuralgia, and partial-onset seizures.
PimozideAn antipsychotic used to manage debilitating motor and phonic tics in patients with Tourette's Disorder.
ChlormezanoneUsed in the management of anxiety and in the treatment of muscle spasm.
EstazolamA benzodiazepine used for the short-term management of insomnia.
QuetiapineA psychotropic agent used for the management of bipolar disorder, schizophrenia, and major depressive disorder.
AripiprazoleAn atypical antipsychotic used in the treatment of a wide variety of mood and psychotic disorders, such as schizophrenia, bipolar I, major depressive disorder, irritability associated with autism, and Tourette's syndrome.
ChlorprothixeneA thioxanthene antipsychotic.
PaliperidoneAn atypical antipsychotic used in the treatment of schizophrenia and other schizoaffective or delusional disorders.
MethotrimeprazineA phenothiazine used in the management of psychosis, particular those of schizophrenia, and manic phases of bipolar disorder.
FlunitrazepamA benzodiazepine used to manage anxiety disorders and insomnia.
BromazepamA short-acting benzodiazepine with intermediate onset commonly used to treat panic disorders and severe anxiety.
KetazolamA long-acting benzodiazepine used to manage anxiety and insomnia.
PrazepamA benzodiazepine used to manage more severe forms of anxiety disorders.
NitrazepamA long-acting benzodiazepine with intermediate onset commonly used to treat panic disorders, severe anxiety, insomnia, and seizures.
MolindoneAn antipsychotic used to treat schizophrenia.
ThiothixeneAn antipsychotic indicated for the management of schizophrenia.
ZuclopenthixolAn antipsychotic indicated for the management of schizophrenia. The acuphase formulation is indicated for initial treatment of acute psychosis or exacerbation of psychosis, while the depot formulation is best for maintenance.
FluspirileneAn antipsychotic agent used in the treatment of schizophrenia.
SertindoleAn atypical antipsychotic indicated in the treatment of schizophrenia.
AsenapineAn atypical antipsychotic used to treat patients with bipolar I disorder and patients with schizophrenia.
AmisulprideA dopamine D2 receptor antagonist used in the treatment of acute and chronic schizophrenia, and in the prevention and treatment of postoperative nausea and vomiting in adults.
LurasidoneAn atypical antipsychotic used to treat schizophrenia and depressive episodes associated with bipolar I disorder.
VortioxetineA serotonin modulating antidepressant indicated for the treatment of major depressive disorder (MDD).
EtizolamA thienodiazepine derivative used to treat anxiety and insomnia.
ZotepineZotepine, like other atypical antipsychotics, is considered as the first-line treatment in newly diagnosed schizophrenia. It is usually thought to be an option of choice for managing acute schizophrenic episodes...
BromperidolA first-generation butyrophenone antipsychotic used in the treatment of schizophrenia and other psychotic manifestations.
PerazineA phenothiazine antipsychotic used in the acute and chronic treatment of psychotic disorders.
BenperidolA neuroleptic butyrophenone derivative indicated in the treatment of psychoses, manic episodes, and psychomotor agitation.
ClothiapineAn atypical antipsychotic indicated in the treatment of acute psychosis, exacerbations of chronic psychosis, chronic psychosis, paranoid psychosis, and anxiety.
SultoprideSultopride is used in Japan, Hong Kong, and Europe to treat schizophrenia. It is of the drug class atypical antipsychotics .
Aripiprazole lauroxilAn antipsychotic used to treat schizophrenia in adults.
Lithium carbonateA medication used to treat manic episodes of bipolar disorder.
ClobazamA benzodiazepine used as adjunct treatment in seizures associated with Lennox-Gastaut syndrome.
LamotrigineA phenyltriazine antiepileptic used to treat some types of epilepsy and bipolar I disorder.
IloperidoneAn atypical antipsychotic agent used for the acute treatment of schizophrenia in adults.
CariprazineAn atypical antipsychotic used to treat schizophrenia and acute manic or mixed episodes due to bipolar I disorder.
RemimazolamAn ultra short-acting benzodiazepine used for the induction and maintenence of procedural sedation during short procedures.
PhenibutNot Annotated
FluvoxamineA selective serotonin-reuptake inhibitor used to treat obsessive-compulsive disorder.
ReserpineFor the treatment of hypertension
DapiprazoleUsed in the treatment of iatrogenically induced mydriasis produced by adrenergic (phenylephrine) or parasympatholytic (tropicamide) agents used in certain eye examinations.
Valproic acidAn anticonvulsant used to control complex partial seizures and both simple and complex absence seizures.
MirtazapineA tetracyclic antidepressant used in the treatment of major depression and is used off-label as a drug for insomnia and to increase appetite.
DroperidolA butyrophenone derivative and dopamine antagonist used to prevent and treat postoperative nausea and vomiting.
NabiloneA synthetic delta-9-THC used in the treatment of anorexia and weight loss in HIV patients as well as nausea and vomiting in cancer chemotherapy.
TranylcypromineA monoamine oxidase inhibitor used to treat major depressive disorder.
FencamfaminFor the the treatment of depressive fatigue in convalescence and other debilitated states as well as in the treatment of depressive day-time fatigue, lack of concentration and lethargy.
Ethyl loflazepateNot Available
FludiazepamUsed for the short-term treatment of anxiety disorders.
OxprenololA non-selective beta-adrenergic antagonist used to treat hypertension, angina pectoris, arrhythmias, and anxiety.
AcepromazineAcepromazine was first used in humans in the 1950s as an antipsychotic agent. It is now rarely used in humans. Acepromazine is frequently used in animals as a sedative and...
AceprometazineAceprometazine is often used in combination with meprobamate for the treatment of sleep disorders.
7-NitroindazoleNot Available
OsanetantPotential therapy for schizophrenia, depression and visceral pain.
DeramciclaneInvestigated for use/treatment in anxiety disorders.
AdipiplonInvestigated for use/treatment in insomnia and sleep disorders.
EsmirtazapineInvestigated for use/treatment in insomnia and sleep disorders.
PerospironeFor the treatment of schizophrenia and acute cases of bipolar mania.
AmperozideAmperozide is a diphenylbutylpiperazine atypical antipsychotic which antagonizes 5-HT2A receptors. It inhibits dopamine release and alters the firing of dopaminergic neurons. Investigations regarding the use of the agent revolved primarily...
EtifoxineA benzoxazine class drug primarily used as an anxiolytic, but that also possesses neuroprotective, neuroplastic, and anti-inflammatory properties; these effects are thought to arise due to modulation of GABAergic neurotransmission and neurosteroid synthesis.
ButriptylineButriptyline is a tricyclic antidepressant which has been used in Europe since 1974. It is the isobutyl side chain homologue of amitriptyline.
MelperoneAn atypical butyrophenone antipsychotic used to treat sleep disorders, confusion, and psychomotor dysfunction associated with geriatric, psychiatric, and alcohol-dependent patients.
BrilaroxazineInvestigated for the treatment of schizophrenia and schizoaffective disorder.
PipamperoneTreatment of chronic psychoses and states of aggressiveness of various origins .
AzaperoneAzaperone is a pyridinylpiperazine and butyrophenone agent that is capable of eliciting neuroleptic sedative and antiemetic effects. It is subsequently employed predominantly as a veterinary tranquilizer and mainly for pigs...
DoramectinDoramectin is a veterinary drug approved by the Food and Drug Administration for the treatment of parasites such as gastrointestinal roundworms, lungworms, eyeworms, grubs, sucking lice and mange mites in...
ZolazepamZolazepam is a pyrazolodiazepinone derivative used as an anaesthetic in veterinary medicine. Zolazepam is typically used in combination with the NMDA antagonist tiletamine or the α2 adrenoceptor agonist xylazine. It...
TetrahydropalmatineTetrahydropalmatine is under investigation in clinical trial NCT02118610 (Treatment of Schizophrenia With L-tetrahydropalmatine (l-THP): a Novel Dopamine Antagonist With Anti-inflammatory and Antiprotozoal Activity).
GepironeA serotonin receptor agonist used to treat major depressive disorder in adults
EcopipamEcopipam has been used in trials studying the treatment of Tourette's Syndrome, Lesch-Nyhan Disease, Pathological Gambling, and Self-injurious Behavior.
RacloprideRaclopride has been used in trials studying Parkinson Disease.
RitanserinRitanserin has been used in trials studying the treatment of Cocaine-Related Disorders.
TandospironeTandospirone has been used in trials studying the treatment of Schizophrenia.
TiaprideA dopamine D2 and D3 receptor antagonist indicated in the treatment of chorea in Huntington's disease, as well as agitation and anxiety in the elderly or with acute or chronic alcoholism.
PinazepamA benzodiazepine indicated in the treatment of anxiety and severe insomnia.
MedazepamA long-acting benzodiazepine used for its sedative and anxiolytic properties.
MebicarNot Annotated
VeraliprideNot Annotated
TrifluperidolNot Annotated
LoprazolamLoprazolam is an imidazobenzodiazepine with anxiolytic, anticonvulsant, hypnotic, sedative and skeletal muscle relaxant properties. It is indicated for the short-term treatment of insomnia including difficulty in falling asleep and/or frequent...
FluanisoneNot Annotated
DixyrazineNot Annotated
PenfluridolNot Annotated
ClopenthixolClopenthixol is a thioxanthene with therapeutic actions similar to the phenothiazine antipsychotics. It is an antagonist at D1 and D2 dopamine receptors.
NordazepamA benzodiazepine indicated in the treatment of insomnia.
Lithium chlorideAn injection indicated for cardiac output measurement.
NorclozapineInvestigated for use/treatment in schizophrenia and schizoaffective disorders.
SpiperoneSpiperone is a dopamine antagonist that binds dopamine and serotonin receptors.
ZK-93423ZK-93423 is a beta-carboline with muscle relaxant activity with agonistic properties at the benzodiazepine receptor.
Drugs & Drug Targets
DrugTargetType
LorazepamUDP-glucuronosyltransferase 2B15enzyme
LorazepamGABA(A) Receptortarget
LorazepamCytochrome P450 3A4enzyme
LorazepamGABA(A) Receptor Benzodiazepine Binding Sitetarget
PregabalinExcitatory amino acid transporter 3transporter
PregabalinVoltage-dependent calcium channel subunit alpha-2/delta-1target
PregabalinLarge neutral amino acids transporter small subunit 1transporter
TemazepamCytochrome P450 3A4enzyme
TemazepamCytochrome P450 2B6enzyme
TemazepamCytochrome P450 2C9enzyme
TemazepamGABA(A) Receptortarget
TemazepamGABA(A) Receptor Benzodiazepine Binding Sitetarget
ZiprasidoneAlpha-1A adrenergic receptortarget
ZiprasidoneDopamine D2 receptortarget
Ziprasidone5-hydroxytryptamine receptor 2Ctarget
ZiprasidoneDopamine D3 receptortarget
Ziprasidone5-hydroxytryptamine receptor 1Atarget
Ziprasidone5-hydroxytryptamine receptor 1Dtarget
ZiprasidoneHistamine H1 receptortarget
Ziprasidone5-hydroxytryptamine receptor 2Atarget
ZiprasidoneDopamine D4 receptortarget
Ziprasidone5-hydroxytryptamine receptor 7target
ZiprasidoneCytochrome P450 3A4enzyme
ZiprasidoneAlpha-2A adrenergic receptortarget
ZiprasidoneAlpha-1B adrenergic receptortarget
ZiprasidoneAlpha-2B adrenergic receptortarget
ZiprasidoneAlpha-2C adrenergic receptortarget
ZiprasidoneDopamine D1 receptortarget
ZiprasidoneDopamine D5 receptortarget
ZiprasidoneMuscarinic acetylcholine receptor M1target
ZiprasidoneMuscarinic acetylcholine receptor M2target
ZiprasidoneMuscarinic acetylcholine receptor M3target
ZiprasidoneMuscarinic acetylcholine receptor M4target
ZiprasidoneMuscarinic acetylcholine receptor M5target
Ziprasidone5-hydroxytryptamine receptor 1Btarget
Ziprasidone5-hydroxytryptamine receptor 1Etarget
Ziprasidone5-hydroxytryptamine receptor 6target
ZiprasidoneAldehyde oxidaseenzyme
ZiprasidoneSerum albumincarrier
ZiprasidoneP-glycoprotein 1transporter
ZiprasidoneAlpha-1-acid glycoprotein 1carrier
Ziprasidone5-hydroxytryptamine 3 receptortarget
Ziprasidone5-hydroxytryptamine receptor 5Atarget
OlanzapineDopamine D1 receptortarget
OlanzapineMuscarinic acetylcholine receptor M1target
OlanzapineMuscarinic acetylcholine receptor M3target
Olanzapine5-hydroxytryptamine receptor 2Atarget
OlanzapineDopamine D4 receptortarget
OlanzapineHistamine H1 receptortarget
OlanzapineMuscarinic acetylcholine receptor M4target
OlanzapineMuscarinic acetylcholine receptor M2target
OlanzapineDopamine D2 receptortarget
Olanzapine5-hydroxytryptamine receptor 2Ctarget
OlanzapineDopamine D3 receptortarget
OlanzapineAlpha-1B adrenergic receptortarget
OlanzapineCytochrome P450 1A2enzyme
Olanzapine5-hydroxytryptamine receptor 3Atarget
Olanzapine5-hydroxytryptamine receptor 6target
OlanzapineAlpha-1A adrenergic receptortarget
OlanzapineDopamine D5 receptortarget
OlanzapineSerum albumincarrier
OlanzapineAlpha-1-acid glycoprotein 1carrier
OlanzapineDimethylaniline monooxygenase [N-oxide-forming] 3enzyme
OlanzapineCytochrome P450 2D6enzyme
OlanzapineP-glycoprotein 1transporter
OlanzapineCytochrome P450 2C19enzyme
OlanzapineD(1) dopamine receptortarget
OlanzapineBeta adrenergic receptortarget
Olanzapine5-hydroxytryptamine receptor 1target
OlanzapineGABA(A) Receptor Benzodiazepine Binding Sitetarget
OlanzapineCytochrome P450 2C9enzyme
OlanzapineUDP-glucuronosyltransferase 1-4enzyme
OlanzapineCytochrome P450 3A4enzyme
OlanzapineCytochrome P450 3A Subfamilyenzyme
ClozapineDopamine D4 receptortarget
ClozapineHistamine H1 receptortarget
ClozapineDopamine D2 receptortarget
ClozapineNeuron-specific vesicular protein calcyontarget
ClozapineHistamine H4 receptortarget
Clozapine5-hydroxytryptamine receptor 2Atarget
Clozapine5-hydroxytryptamine receptor 1Atarget
Clozapine5-hydroxytryptamine receptor 2Ctarget
ClozapineDopamine D1 receptortarget
ClozapineCytochrome P450 1A2enzyme
ClozapineCytochrome P450 2D6enzyme
ClozapineDopamine D3 receptortarget
ClozapineMuscarinic acetylcholine receptor M1target
ClozapineMuscarinic acetylcholine receptor M2target
ClozapineMuscarinic acetylcholine receptor M3target
ClozapineMuscarinic acetylcholine receptor M4target
ClozapineMuscarinic acetylcholine receptor M5target
Clozapine5-hydroxytryptamine receptor 1Btarget
Clozapine5-hydroxytryptamine receptor 1Dtarget
Clozapine5-hydroxytryptamine receptor 1Etarget
Clozapine5-hydroxytryptamine receptor 3Atarget
Clozapine5-hydroxytryptamine receptor 6target
Clozapine5-hydroxytryptamine receptor 7target
ClozapineAlpha-1A adrenergic receptortarget
ClozapineAlpha-1B adrenergic receptortarget
ClozapineAlpha-2A adrenergic receptortarget
ClozapineAlpha-2B adrenergic receptortarget
ClozapineAlpha-2C adrenergic receptortarget
ClozapineCytochrome P450 2C9enzyme
ClozapineP-glycoprotein 1transporter
ClozapineCytochrome P450 3A4enzyme
ClozapineCytochrome P450 2C19enzyme
ClozapineDimethylaniline monooxygenase [N-oxide-forming] 3enzyme
ClozapineUDP-glucuronosyltransferase 1-4enzyme
ClozapineCytochrome P450 1A1enzyme
ClozapineCytochrome P450 2A6enzyme
ClozapineCytochrome P450 2C8enzyme
ClozapineGlutathione S-transferase Ptarget
ClozapineAlpha-1-acid glycoprotein 1carrier
ClozapineSerum albumincarrier
ClozapineDopamine D5 receptortarget
ClozapineGamma-aminobutyric acid type B receptor subunit 1target
ClozapineGamma-aminobutyric acid type B receptor subunit 2target
ClozapineSolute carrier family 22 member 1transporter
ClozapineSolute carrier family 22 member 2transporter
ClozapineSolute carrier family 22 member 3transporter
ClozapineGamma-aminobutyric acid receptor subunit alpha-1target
ClozapineGamma-aminobutyric acid receptor subunit beta-1target
ClozapineGamma-aminobutyric acid receptor subunit gamma-1target
MeprobamateGamma-aminobutyric acid receptor subunit alpha-1target
MeprobamateGamma-aminobutyric acid receptor subunit alpha-2target
MeprobamateGamma-aminobutyric acid receptor subunit alpha-3target
MeprobamateGamma-aminobutyric acid receptor subunit alpha-4target
MeprobamateGamma-aminobutyric acid receptor subunit alpha-5target
MeprobamateGamma-aminobutyric acid receptor subunit alpha-6target
MeprobamateGABA(A) Receptortarget
SulpirideDopamine D2 receptortarget
SulpirideDopamine D3 receptortarget
SulpirideCholinesteraseenzyme
SulpirideCarbonic anhydrase 2target
SulpirideCarbonic anhydrase 3target
SulpirideSerum albumincarrier
SulpirideSolute carrier family 22 member 1transporter
SulpirideSolute carrier family 22 member 2transporter
SulpirideMultidrug and toxin extrusion protein 1transporter
SulpirideMultidrug and toxin extrusion protein 2transporter
SulpirideDopamine D4 receptortarget
SulpirideSolute carrier family 22 member 3transporter
SulpirideP-glycoprotein 1transporter
SulpirideATP-binding cassette sub-family G member 2transporter
AlprazolamCytochrome P450 3A4enzyme
AlprazolamCytochrome P450 2C9enzyme
AlprazolamCytochrome P450 3A5enzyme
AlprazolamCytochrome P450 3A7enzyme
AlprazolamGABA(A) Receptortarget
AlprazolamSerum albumincarrier
Alprazolamalpha1-acid glycoproteincarrier
AlprazolamGABA(A) Receptor Benzodiazepine Binding Sitetarget
LoxapineDopamine D1 receptortarget
LoxapineDopamine D2 receptortarget
Loxapine5-hydroxytryptamine receptor 2Atarget
Loxapine5-hydroxytryptamine receptor 2Ctarget
Loxapine5-hydroxytryptamine receptor 1Atarget
Loxapine5-hydroxytryptamine receptor 1Btarget
Loxapine5-hydroxytryptamine receptor 1Dtarget
Loxapine5-hydroxytryptamine receptor 1Etarget
Loxapine5-hydroxytryptamine receptor 3Atarget
Loxapine5-hydroxytryptamine receptor 5Atarget
Loxapine5-hydroxytryptamine receptor 6target
Loxapine5-hydroxytryptamine receptor 7target
LoxapineAlpha-1A adrenergic receptortarget
LoxapineAlpha-1B adrenergic receptortarget
LoxapineAlpha-2A adrenergic receptortarget
LoxapineAlpha-2B adrenergic receptortarget
LoxapineAlpha-2C adrenergic receptortarget
LoxapineBeta-1 adrenergic receptortarget
LoxapineMuscarinic acetylcholine receptor M1target
LoxapineMuscarinic acetylcholine receptor M2target
LoxapineMuscarinic acetylcholine receptor M3target
LoxapineMuscarinic acetylcholine receptor M4target
LoxapineMuscarinic acetylcholine receptor M5target
LoxapineD(1) dopamine receptortarget
LoxapineDopamine D3 receptortarget
LoxapineDopamine D4 receptortarget
LoxapineDopamine D5 receptortarget
LoxapineHistamine H1 receptortarget
LoxapineHistamine H2 receptortarget
LoxapineHistamine H4 receptortarget
LoxapineSodium-dependent serotonin transportertarget
LoxapineSodium-dependent noradrenaline transportertarget
LoxapineSodium-dependent dopamine transportertarget
RemoxiprideDopamine D2 receptortarget
RemoxiprideDopamine D4 receptortarget
Remoxipride5-hydroxytryptamine receptor 2Atarget
RemoxiprideSigma non-opioid intracellular receptor 1target
RemoxiprideDopamine D3 receptortarget
RemoxiprideCytochrome P450 2D6enzyme
Remoxipridealpha1-acid glycoproteincarrier
RemoxiprideCytochrome P450 1A2enzyme
RemoxiprideCytochrome P450 2B1enzyme
RemoxiprideCytochrome P450 3A Subfamilyenzyme
PromazineDopamine D2 receptortarget
Promazine5-hydroxytryptamine receptor 2Atarget
Promazine5-hydroxytryptamine receptor 2Ctarget
PromazineAlpha-1A adrenergic receptortarget
PromazineMuscarinic acetylcholine receptor M1target
PromazineHistamine H1 receptortarget
PromazineCytochrome P450 2C19enzyme
PromazineCytochrome P450 1A2enzyme
PromazineCytochrome P450 3A4enzyme
PromazineCytochrome P450 2C9enzyme
PromazineCytochrome P450 2D6enzyme
ProchlorperazineDopamine D2 receptortarget
ProchlorperazineCytochrome P450 2D6enzyme
ProchlorperazineHistamine H1 receptortarget
ProchlorperazineAlpha-1 adrenergic receptorstarget
ProchlorperazineAlpha-2 adrenergic receptorstarget
ChlordiazepoxideGABA(A) Receptortarget
ChlordiazepoxideGABA(A) Receptor Benzodiazepine Binding Sitetarget
ChlordiazepoxideCytochrome P450 3A4enzyme
ChlorpromazineDopamine D2 receptortarget
Chlorpromazine5-hydroxytryptamine receptor 2Atarget
ChlorpromazineCytochrome P450 2D6enzyme
ChlorpromazineCholinesteraseenzyme
ChlorpromazineCytochrome P450 1A2enzyme
ChlorpromazineSerum albumincarrier
ChlorpromazineP-glycoprotein 1transporter
ChlorpromazineDopamine D1 receptortarget
Chlorpromazine5-hydroxytryptamine receptor 1Atarget
ChlorpromazineAlpha-1A adrenergic receptortarget
ChlorpromazineAlpha-1B adrenergic receptortarget
ChlorpromazineCytochrome P450 2E1enzyme
ChlorpromazineCytochrome P450 3A4enzyme
ChlorpromazineHistamine H1 receptortarget
ChlorpromazinePotassium voltage-gated channel subfamily H member 2target
ChlorpromazineD(1) dopamine receptortarget
ChlorpromazineDopamine D3 receptortarget
ChlorpromazineDopamine D4 receptortarget
ChlorpromazineDopamine D5 receptortarget
Chlorpromazine5-hydroxytryptamine receptor 2Ctarget
Chlorpromazine5-hydroxytryptamine 2 receptortarget
ChlorpromazineAlpha-1 adrenergic receptorstarget
ChlorpromazineAlpha-2 adrenergic receptorstarget
ChlorpromazineMuscarinic acetylcholine receptor M1target
ChlorpromazineMuscarinic acetylcholine receptor M3target
ChlorpromazineSphingomyelin phosphodiesterasetarget
ChlorpromazineCalmodulintarget
Chlorpromazinealpha1-acid glycoproteintarget
Chlorpromazine5-hydroxytryptamine receptor 6target
Chlorpromazine5-hydroxytryptamine receptor 7target
ChlorpromazineHistamine H4 receptortarget
ChlorpromazineBile salt export pumptransporter
Buspirone5-hydroxytryptamine receptor 1Atarget
BuspironeDopamine D2 receptortarget
BuspironeCytochrome P450 3A4enzyme
BuspironeCytochrome P450 3A5enzyme
BuspironeCytochrome P450 3A7enzyme
BuspironeP-glycoprotein 1transporter
BuspironeCytochrome P450 2D6enzyme
BuspironeSerum albumincarrier
BuspironeAlpha-1-acid glycoprotein 1carrier
BuspironeDopamine D3 receptortarget
BuspironeDopamine D4 receptortarget
BuspironeAlpha-1 adrenergic receptorstarget
HaloperidolDopamine D2 receptortarget
HaloperidolGlutamate receptor ionotropic, NMDA 2Btarget
HaloperidolDopamine D1 receptortarget
HaloperidolCytochrome P450 1A2enzyme
HaloperidolCytochrome P450 2D6enzyme
Haloperidol5-hydroxytryptamine receptor 2Atarget
HaloperidolDopamine D3 receptortarget
HaloperidolCytochrome P450 3A4enzyme
HaloperidolCytochrome P450 3A5enzyme
HaloperidolCytochrome P450 3A7enzyme
HaloperidolP-glycoprotein 1transporter
HaloperidolCarbonyl reductase [NADPH] 1enzyme
HaloperidolUDP-glucuronosyltransferase 1-9enzyme
HaloperidolCytochrome P450 2C19enzyme
HaloperidolCytochrome P450 2C9enzyme
HaloperidolMelanin-concentrating hormone receptor 1target
HaloperidolSynaptic vesicular amine transportertarget
Haloperidol5-hydroxytryptamine receptor 2Ctarget
HaloperidolSigma non-opioid intracellular receptor 1target
HaloperidolHistamine H1 receptortarget
HaloperidolMuscarinic acetylcholine receptor M3target
HaloperidolAlpha-1A adrenergic receptortarget
HaloperidolAlpha-2A adrenergic receptortarget
HaloperidolAlpha-2B adrenergic receptortarget
HaloperidolAlpha-2C adrenergic receptortarget
Haloperidol5-hydroxytryptamine receptor 1Atarget
Haloperidol5-hydroxytryptamine receptor 6target
Haloperidol5-hydroxytryptamine receptor 7target
HaloperidolCytochrome P450 1A1enzyme
TriflupromazineDopamine D1 receptortarget
TriflupromazineDopamine D2 receptortarget
TriflupromazineMuscarinic acetylcholine receptor M1target
TriflupromazineMuscarinic acetylcholine receptor M2target
Triflupromazine5-hydroxytryptamine receptor 2Btarget
TriflupromazineP-glycoprotein 1transporter
TriflupromazineCholinesteraseenzyme
FluphenazineDopamine D2 receptortarget
FluphenazineCalmodulintarget
FluphenazineDopamine D1 receptortarget
FluphenazineCytochrome P450 2D6enzyme
FluphenazineP-glycoprotein 1transporter
FluphenazineCytochrome P450 2E1enzyme
FluphenazineAndrogen receptortarget
Fluphenazine5-hydroxytryptamine receptor 2Atarget
Fluphenazine5-hydroxytryptamine receptor 2Ctarget
Clorazepic acidCytochrome P450 3A4enzyme
Clorazepic acidGABA(A) Receptortarget
Clorazepic acidGABA(A) Receptor Benzodiazepine Binding Sitetarget
Trazodone5-hydroxytryptamine receptor 2Atarget
TrazodoneSodium-dependent serotonin transportertarget
TrazodoneAlpha-1A adrenergic receptortarget
TrazodoneAlpha-2A adrenergic receptortarget
TrazodoneHistamine H1 receptortarget
Trazodone5-hydroxytryptamine receptor 1Atarget
TrazodoneCytochrome P450 2D6enzyme
TrazodoneCytochrome P450 3A4enzyme
Trazodone5-hydroxytryptamine receptor 2Ctarget
TrazodoneCytochrome P450 3A5enzyme
TrazodoneCytochrome P450 3A7enzyme
TrazodoneP-glycoprotein 1transporter
Trazodone5-hydroxytryptamine receptor 1Ctarget
ThioridazineAlpha-1A adrenergic receptortarget
ThioridazineDopamine D2 receptortarget
Thioridazine5-hydroxytryptamine receptor 2Atarget
ThioridazineDopamine D1 receptortarget
ThioridazineCytochrome P450 2C19enzyme
ThioridazineCytochrome P450 2D6enzyme
ThioridazineAlpha-1B adrenergic receptortarget
ThioridazinePotassium voltage-gated channel subfamily H member 2target
ThioridazineCytochrome P450 2E1enzyme
MidazolamCytochrome P450 3A4enzyme
MidazolamCytochrome P450 3A5enzyme
MidazolamUDP-glucuronosyltransferase 1-4enzyme
MidazolamCytochrome P450 3A7enzyme
MidazolamGABA(A) Receptortarget
MidazolamGABA(A) Receptor Benzodiazepine Binding Sitetarget
MidazolamP-glycoprotein 1transporter
MidazolamSerum albumincarrier
MidazolamAlpha-1-acid glycoprotein 1carrier
MidazolamAdenosine receptor A2atarget
MidazolamExcitatory amino acid transporter 2transporter
MidazolamUDP-glucuronosyltransferase 2B7enzyme
MidazolamUDP-glucuronosyltransferase 2B4enzyme
FlurazepamCytochrome P450 3A4enzyme
FlurazepamP-glycoprotein 1transporter
FlurazepamCytochrome P450 2E1enzyme
FlurazepamCytochrome P450 2A6enzyme
FlurazepamSolute carrier family 22 member 2transporter
FlurazepamGABA(A) Receptortarget
FlurazepamGABA(A) Receptor Benzodiazepine Binding Sitetarget
RisperidoneCytochrome P450 2D6enzyme
RisperidoneCytochrome P450 3A4enzyme
RisperidoneP-glycoprotein 1transporter
RisperidoneSerum albumincarrier
RisperidoneAlpha-1-acid glycoprotein 1carrier
Risperidone5-hydroxytryptamine receptor 2Atarget
RisperidoneDopamine D2 receptortarget
RisperidoneAlpha-1B adrenergic receptortarget
RisperidoneAlpha-2B adrenergic receptortarget
RisperidoneAlpha-1A adrenergic receptortarget
RisperidoneAlpha-2C adrenergic receptortarget
RisperidoneHistamine H1 receptortarget
Risperidone5-hydroxytryptamine receptor 2Ctarget
Risperidone5-hydroxytryptamine receptor 1Dtarget
Risperidone5-hydroxytryptamine receptor 1Atarget
Risperidone5-hydroxytryptamine receptor 7target
RisperidoneD(2L) dopamine receptortarget
RisperidoneDopamine D1 receptortarget
HalazepamGABA(A) Receptortarget
HalazepamGABA(A) Receptor Benzodiazepine Binding Sitetarget
DiazepamCytochrome P450 3A4enzyme
DiazepamSerum albumincarrier
DiazepamCytochrome P450 2C9enzyme
DiazepamCytochrome P450 2C19enzyme
DiazepamCytochrome P450 3A5enzyme
DiazepamCytochrome P450 3A7enzyme
DiazepamP-glycoprotein 1transporter
DiazepamCytochrome P450 2B6enzyme
DiazepamProstaglandin G/H synthase 1enzyme
DiazepamCytochrome P450 2C18enzyme
DiazepamCytochrome P450 2C8enzyme
DiazepamGABA(A) Receptortarget
DiazepamGABA(A) Receptor Benzodiazepine Binding Sitetarget
TrifluoperazineDopamine D2 receptortarget
TrifluoperazineAlpha-1A adrenergic receptortarget
TrifluoperazineNeuron-specific vesicular protein calcyontarget
TrifluoperazineXanthine dehydrogenase/oxidaseenzyme
TrifluoperazineUDP-glucuronosyltransferase 1-4enzyme
TrifluoperazineCytochrome P450 1A2enzyme
TrifluoperazineP-glycoprotein 1transporter
TrifluoperazineCalmodulintarget
TrifluoperazineTroponin C, slow skeletal and cardiac musclestarget
TrifluoperazineProtein S100-A4target
OxazepamUDP-glucuronosyltransferase 2B15enzyme
OxazepamUDP-glucuronosyltransferase 2B7enzyme
OxazepamUDP-glucuronosyltransferase 1-9enzyme
OxazepamGABA(A) Receptortarget
OxazepamGABA(A) Receptor Benzodiazepine Binding Sitetarget
OxazepamSerum albumincarrier
PerphenazineDopamine D1 receptortarget
PerphenazineDopamine D2 receptortarget
PerphenazineCalmodulintarget
PerphenazineCytochrome P450 2D6enzyme
PerphenazineCytochrome P450 1A2enzyme
PerphenazineCytochrome P450 2C18enzyme
PerphenazineCytochrome P450 2C19enzyme
PerphenazineCytochrome P450 2C8enzyme
PerphenazineCytochrome P450 2C9enzyme
PerphenazineCytochrome P450 3A4enzyme
PerphenazineSerum albumincarrier
FlupentixolAlpha-1A adrenergic receptortarget
FlupentixolDopamine D2 receptortarget
FlupentixolDopamine D1 receptortarget
FlupentixolAromatic-L-amino-acid decarboxylaseenzyme
Flupentixol5-hydroxytryptamine receptor 2Atarget
FlupentixolP-glycoprotein 1transporter
FlupentixolMuscarinic acetylcholine receptor M1target
FlupentixolLiver carboxylesterase 1enzyme
FlupentixolDopamine D3 receptortarget
FlupentixolDopamine D4 receptortarget
Flupentixol5-hydroxytryptamine receptor 2Ctarget
TriazolamCytochrome P450 3A4enzyme
TriazolamCytochrome P450 3A5enzyme
TriazolamCytochrome P450 3A7enzyme
TriazolamCytochrome P450 2C8enzyme
TriazolamGABA(A) Receptor Benzodiazepine Binding Sitetarget
TriazolamGABA(A) Receptortarget
Cyclobenzaprine5-hydroxytryptamine receptor 2Atarget
CyclobenzaprineCytochrome P450 1A2enzyme
CyclobenzaprineCytochrome P450 3A4enzyme
CyclobenzaprineCytochrome P450 2D6enzyme
CyclobenzaprineSerum albumincarrier
CyclobenzaprineUDP-glucuronosyltransferase 1-4enzyme
CyclobenzaprineUDP-glucuronosyltransferase 2B10enzyme
Cyclobenzaprine5-hydroxytryptamine receptor 2Btarget
Cyclobenzaprine5-hydroxytryptamine receptor 2Ctarget
Cyclobenzaprine5-hydroxytryptamine receptor 7target
Cyclobenzaprine5-hydroxytryptamine receptor 6target
CyclobenzaprineSodium-dependent serotonin transportertarget
CyclobenzaprineSodium-dependent noradrenaline transportertarget
CyclobenzaprineToll-like receptor 4target
CyclobenzaprineAldehyde oxidasetarget
MesoridazineDopamine D2 receptortarget
Mesoridazine5-hydroxytryptamine receptor 2Atarget
MesoridazineCytochrome P450 2D6enzyme
GabapentinAdenosine receptor A1target
GabapentinVoltage-dependent calcium channel subunit alpha-2/delta-1target
GabapentinVoltage-dependent calcium channel subunit alpha-2/delta-2target
GabapentinBranched-chain-amino-acid aminotransferase, cytosolicenzyme
GabapentinLarge neutral amino acids transporter small subunit 1transporter
GabapentinVoltage-dependent N-type calcium channeltarget
GabapentinPotassium voltage-gated channel subfamily KQT member 3target
GabapentinPotassium voltage-gated channel subfamily KQT member 5target
PimozideDopamine D2 receptortarget
PimozideCalmodulintarget
PimozidePotassium voltage-gated channel subfamily H member 2target
PimozideCytochrome P450 3A4enzyme
PimozideCytochrome P450 1A2enzyme
PimozideCytochrome P450 3A5enzyme
PimozideCytochrome P450 3A7enzyme
PimozideP-glycoprotein 1transporter
PimozideDopamine D3 receptortarget
PimozideCytochrome P450 2D6enzyme
ChlormezanoneTranslocator proteintarget
EstazolamCytochrome P450 3A4enzyme
EstazolamGABA(A) Receptortarget
EstazolamGABA(A) Receptor Benzodiazepine Binding Sitetarget
Quetiapine5-hydroxytryptamine receptor 2Atarget
Quetiapine5-hydroxytryptamine receptor 2Ctarget
QuetiapineDopamine D2 receptortarget
Quetiapine5-hydroxytryptamine receptor 1Atarget
QuetiapineHistamine H1 receptortarget
QuetiapineCytochrome P450 3A4enzyme
QuetiapineAlpha-1 adrenergic receptorstarget
QuetiapineAlpha-2A adrenergic receptortarget
QuetiapineAlpha-2B adrenergic receptortarget
QuetiapineAlpha-2C adrenergic receptortarget
Quetiapine5-hydroxytryptamine receptor 1Dtarget
QuetiapineMuscarinic acetylcholine receptor M1target
QuetiapineMuscarinic acetylcholine receptor M2target
QuetiapineMuscarinic acetylcholine receptor M3target
QuetiapineMuscarinic acetylcholine receptor M4target
QuetiapineMuscarinic acetylcholine receptor M5target
Quetiapine5-hydroxytryptamine receptor 1Btarget
Quetiapine5-hydroxytryptamine receptor 1Etarget
Quetiapine5-hydroxytryptamine receptor 3Atarget
Quetiapine5-hydroxytryptamine receptor 6target
Quetiapine5-hydroxytryptamine receptor 7target
QuetiapineDopamine D5 receptortarget
QuetiapineDopamine D1 receptortarget
QuetiapineDopamine D3 receptortarget
QuetiapineDopamine D4 receptortarget
QuetiapineCytochrome P450 3A5enzyme
QuetiapineP-glycoprotein 1transporter
QuetiapineCytochrome P450 2C19enzyme
QuetiapineCytochrome P450 2D6enzyme
QuetiapineCytochrome P450 3A7enzyme
AripiprazoleDopamine D2 receptortarget
Aripiprazole5-hydroxytryptamine receptor 1Atarget
Aripiprazole5-hydroxytryptamine receptor 2Atarget
AripiprazoleCytochrome P450 3A4enzyme
AripiprazoleCytochrome P450 2D6enzyme
Aripiprazole5-hydroxytryptamine receptor 1Btarget
Aripiprazole5-hydroxytryptamine receptor 1Dtarget
Aripiprazole5-hydroxytryptamine receptor 1Etarget
AripiprazoleDopamine D1 receptortarget
AripiprazoleDopamine D5 receptortarget
AripiprazoleDopamine D3 receptortarget
AripiprazoleDopamine D4 receptortarget
Aripiprazole5-hydroxytryptamine receptor 2Ctarget
Aripiprazole5-hydroxytryptamine receptor 3Atarget
Aripiprazole5-hydroxytryptamine receptor 6target
Aripiprazole5-hydroxytryptamine receptor 7target
AripiprazoleHistamine H1 receptortarget
AripiprazoleAlpha-1A adrenergic receptortarget
AripiprazoleAlpha-1B adrenergic receptortarget
AripiprazoleAlpha-2A adrenergic receptortarget
AripiprazoleAlpha-2B adrenergic receptortarget
AripiprazoleAlpha-2C adrenergic receptortarget
AripiprazoleCytochrome P450 3A5enzyme
AripiprazoleCytochrome P450 3A7enzyme
AripiprazoleSerum albumincarrier
Aripiprazole5-hydroxytryptamine receptor 2Btarget
Aripiprazole5-hydroxytryptamine receptor 5Atarget
AripiprazoleBeta-1 adrenergic receptortarget
AripiprazoleBeta-2 adrenergic receptortarget
AripiprazoleHistamine H2 receptortarget
AripiprazoleHistamine H3 receptortarget
AripiprazoleHistamine H4 receptortarget
AripiprazoleMuscarinic acetylcholine receptor M1target
AripiprazoleMuscarinic acetylcholine receptor M2target
AripiprazoleMuscarinic acetylcholine receptor M3target
AripiprazoleMuscarinic acetylcholine receptor M4target
AripiprazoleMuscarinic acetylcholine receptor M5target
AripiprazoleKappa-type opioid receptortarget
AripiprazoleMu-type opioid receptortarget
AripiprazoleDelta-type opioid receptortarget
AripiprazoleGlutamate (NMDA) receptortarget
AripiprazoleSodium-dependent dopamine transportertarget
AripiprazoleSodium-dependent serotonin transportertarget
AripiprazoleP-glycoprotein 1transporter
AripiprazoleATP-binding cassette sub-family G member 2transporter
ChlorprothixeneDopamine D1 receptortarget
ChlorprothixeneDopamine D2 receptortarget
ChlorprothixeneDopamine D3 receptortarget
Chlorprothixene5-hydroxytryptamine receptor 2Atarget
ChlorprothixeneHistamine H1 receptortarget
ChlorprothixeneMuscarinic acetylcholine receptor M1target
ChlorprothixeneMuscarinic acetylcholine receptor M2target
ChlorprothixeneMuscarinic acetylcholine receptor M3target
ChlorprothixeneMuscarinic acetylcholine receptor M4target
ChlorprothixeneMuscarinic acetylcholine receptor M5target
ChlorprothixeneP-glycoprotein 1transporter
ChlorprothixeneSerotonin Receptorstarget
PaliperidoneDopamine D2 receptortarget
Paliperidone5-hydroxytryptamine receptor 2Atarget
PaliperidoneHistamine H1 receptortarget
PaliperidoneAlpha-1A adrenergic receptortarget
PaliperidoneAlpha-1B adrenergic receptortarget
PaliperidoneDopamine D3 receptortarget
PaliperidoneDopamine D4 receptortarget
PaliperidoneDopamine D1 receptortarget
PaliperidoneAlpha-2A adrenergic receptortarget
PaliperidoneAlpha-2B adrenergic receptortarget
PaliperidoneAlpha-2C adrenergic receptortarget
Paliperidone5-hydroxytryptamine receptor 1Atarget
Paliperidone5-hydroxytryptamine receptor 1Dtarget
Paliperidone5-hydroxytryptamine receptor 2Ctarget
Paliperidone5-hydroxytryptamine receptor 7target
PaliperidoneCytochrome P450 3A4enzyme
PaliperidoneCytochrome P450 2D6enzyme
PaliperidoneCytochrome P450 3A5enzyme
PaliperidoneP-glycoprotein 1transporter
MethotrimeprazineDopamine D3 receptortarget
MethotrimeprazineHistamine H1 receptortarget
MethotrimeprazineMuscarinic acetylcholine receptor M1target
MethotrimeprazineMuscarinic acetylcholine receptor M2target
MethotrimeprazineMuscarinic acetylcholine receptor M3target
MethotrimeprazineMuscarinic acetylcholine receptor M4target
MethotrimeprazineMuscarinic acetylcholine receptor M5target
MethotrimeprazineAlpha-1A adrenergic receptortarget
MethotrimeprazineAlpha-1B adrenergic receptortarget
MethotrimeprazineAlpha-1D adrenergic receptortarget
MethotrimeprazineCytochrome P450 2D6enzyme
MethotrimeprazineDopamine D2 receptortarget
MethotrimeprazineDopamine D1 receptortarget
MethotrimeprazineDopamine D5 receptortarget
MethotrimeprazineDopamine D4 receptortarget
MethotrimeprazineAlpha-2A adrenergic receptortarget
MethotrimeprazineAlpha-2B adrenergic receptortarget
MethotrimeprazineAlpha-2C adrenergic receptortarget
Methotrimeprazine5-hydroxytryptamine receptor 2Atarget
Methotrimeprazine5-hydroxytryptamine receptor 2Ctarget
MethotrimeprazineCytochrome P450 2E1enzyme
FlunitrazepamCytochrome P450 2C19enzyme
FlunitrazepamUDP-glucuronosyltransferase 2B7enzyme
FlunitrazepamCytochrome P450 2A6enzyme
FlunitrazepamCytochrome P450 2B6enzyme
FlunitrazepamCytochrome P450 2C9enzyme
FlunitrazepamCytochrome P450 3A4enzyme
FlunitrazepamCytochrome P450 2E1enzyme
FlunitrazepamUDP-glucuronosyltransferase 1-1enzyme
FlunitrazepamUDP-glucuronosyltransferase 1-3enzyme
FlunitrazepamGABA(A) Receptortarget
FlunitrazepamGABA(A) Receptor Benzodiazepine Binding Sitetarget
BromazepamCytochrome P450 1A2enzyme
BromazepamCytochrome P450 2C19enzyme
BromazepamCytochrome P450 2E1enzyme
BromazepamGABA(A) Receptortarget
BromazepamGABA(A) Receptor Benzodiazepine Binding Sitetarget
KetazolamCytochrome P450 3A4enzyme
KetazolamP-glycoprotein 1transporter
KetazolamSerum albumincarrier
KetazolamGABA(A) Receptortarget
KetazolamGABA(A) Receptor Benzodiazepine Binding Sitetarget
PrazepamCytochrome P450 3A4enzyme
PrazepamGABA(A) Receptortarget
PrazepamGABA(A) Receptor Benzodiazepine Binding Sitetarget
NitrazepamSodium channel protein type 1 subunit alphatarget
NitrazepamCytochrome P450 3A4enzyme
NitrazepamCytochrome P450 2E1enzyme
NitrazepamGABA(A) Receptortarget
NitrazepamGABA(A) Receptor Benzodiazepine Binding Sitetarget
MolindoneDopamine D2 receptortarget
Molindone5-hydroxytryptamine receptor 1Atarget
Molindone5-hydroxytryptamine receptor 2Atarget
MolindoneMuscarinic acetylcholine receptor M1target
ThiothixeneCytochrome P450 1A2enzyme
ThiothixeneCytochrome P450 2D6enzyme
ThiothixeneDopamine D2 receptortarget
ThiothixeneDopamine D1 receptortarget
Thiothixene5-hydroxytryptamine receptor 2Atarget
ThiothixeneSolute carrier family 22 member 1transporter
ThiothixeneSerum albumincarrier
ZuclopenthixolDopamine D1 receptortarget
ZuclopenthixolDopamine D5 receptortarget
ZuclopenthixolDopamine D2 receptortarget
ZuclopenthixolCytochrome P450 2D6enzyme
ZuclopenthixolAlpha-1A adrenergic receptortarget
ZuclopenthixolAlpha-2A adrenergic receptortarget
Zuclopenthixol5-hydroxytryptamine receptor 2Atarget
ZuclopenthixolHistamine H1 receptortarget
ZuclopenthixolCytochrome P450 3A4enzyme
FluspirileneDopamine D2 receptortarget
Fluspirilene5-hydroxytryptamine receptor 2Atarget
FluspirileneVoltage-dependent calcium channel gamma-1 subunittarget
FluspirileneCytochrome P450 3A4enzyme
Sertindole5-hydroxytryptamine receptor 2Atarget
Sertindole5-hydroxytryptamine receptor 2Ctarget
SertindoleDopamine D2 receptortarget
SertindoleAlpha-1A adrenergic receptortarget
SertindoleAlpha-1B adrenergic receptortarget
SertindoleAlpha-1D adrenergic receptortarget
SertindolePotassium voltage-gated channel subfamily H member 2target
Sertindole5-hydroxytryptamine receptor 6target
SertindoleCytochrome P450 2D6enzyme
SertindoleCytochrome P450 3A4enzyme
Asenapine5-hydroxytryptamine receptor 1Atarget
Asenapine5-hydroxytryptamine receptor 1Btarget
Asenapine5-hydroxytryptamine receptor 2Atarget
Asenapine5-hydroxytryptamine receptor 2Btarget
Asenapine5-hydroxytryptamine receptor 2Ctarget
Asenapine5-hydroxytryptamine receptor 6target
Asenapine5-hydroxytryptamine receptor 7target
AsenapineAlpha-2A adrenergic receptortarget
AsenapineAlpha-2B adrenergic receptortarget
AsenapineAlpha-2C adrenergic receptortarget
AsenapineAlpha-1A adrenergic receptortarget
AsenapineDopamine D1 receptortarget
AsenapineDopamine D2 receptortarget
AsenapineDopamine D3 receptortarget
AsenapineDopamine D4 receptortarget
AsenapineHistamine H1 receptortarget
AsenapineHistamine H2 receptortarget
AsenapineCytochrome P450 1A2enzyme
AsenapineCytochrome P450 2D6enzyme
Asenapine5-hydroxytryptamine receptor 5Atarget
AsenapineUDP-glucuronosyltransferase 1-4enzyme
AsenapineCytochrome P450 3A4enzyme
AsenapineBeta-1 adrenergic receptortarget
AsenapineBeta-2 adrenergic receptortarget
AsenapineSerum albumincarrier
Asenapinealpha1-acid glycoproteincarrier
AmisulprideDopamine D2 receptortarget
AmisulprideDopamine D3 receptortarget
Amisulpride5-hydroxytryptamine receptor 7target
Amisulpride5-hydroxytryptamine receptor 2Atarget
AmisulprideErythrocytecarrier
AmisulprideMultidrug and toxin extrusion protein 1transporter
AmisulprideMultidrug and toxin extrusion protein 2transporter
AmisulprideP-glycoprotein 1transporter
AmisulprideATP-binding cassette sub-family G member 2transporter
AmisulprideSolute carrier family 22 member 1transporter
AmisulprideMu-type opioid receptortarget
AmisulprideDelta-type opioid receptortarget
AmisulprideKappa-type opioid receptortarget
LurasidoneCytochrome P450 3A4enzyme
LurasidoneDopamine D2 receptortarget
Lurasidone5-hydroxytryptamine receptor 2Atarget
Lurasidone5-hydroxytryptamine receptor 7target
Lurasidone5-hydroxytryptamine receptor 1Atarget
LurasidoneAlpha-2C adrenergic receptortarget
LurasidoneAlpha-2A adrenergic receptortarget
VortioxetineSodium-dependent serotonin transportertarget
Vortioxetine5-hydroxytryptamine receptor 3Atarget
Vortioxetine5-hydroxytryptamine receptor 7target
Vortioxetine5-hydroxytryptamine receptor 1Btarget
Vortioxetine5-hydroxytryptamine receptor 1Atarget
VortioxetineBeta-1 adrenergic receptortarget
VortioxetineSodium-dependent noradrenaline transportertarget
VortioxetineCytochrome P450 2D6enzyme
VortioxetineCytochrome P450 3A4enzyme
VortioxetineCytochrome P450 3A5enzyme
VortioxetineCytochrome P450 2C19enzyme
VortioxetineCytochrome P450 2C9enzyme
VortioxetineCytochrome P450 2A6enzyme
VortioxetineCytochrome P450 2C8enzyme
VortioxetineCytochrome P450 2B6enzyme
EtizolamCytochrome P450 3A4enzyme
EtizolamCytochrome P450 2C18enzyme
EtizolamCytochrome P450 2C19enzyme
EtizolamPlatelet-activating factor receptortarget
EtizolamGABA(A) Receptortarget
EtizolamGABA(A) Receptor Benzodiazepine Binding Sitetarget
ZotepineD(1) dopamine receptortarget
ZotepineDopamine D2 receptortarget
Zotepine5-hydroxytryptamine receptor 2Atarget
Zotepine5-hydroxytryptamine receptor 6target
Zotepine5-hydroxytryptamine receptor 7target
ZotepineSodium-dependent noradrenaline transportertarget
ZotepineSodium-dependent serotonin transportertarget
ZotepineCytochrome P450 1A2enzyme
ZotepineCytochrome P450 3A4enzyme
Aripiprazole lauroxilDopamine D2 receptortarget
Aripiprazole lauroxil5-hydroxytryptamine receptor 1Atarget
Aripiprazole lauroxil5-hydroxytryptamine receptor 2Atarget
Aripiprazole lauroxilCytochrome P450 3A4enzyme
Aripiprazole lauroxilCytochrome P450 2D6enzyme
Aripiprazole lauroxil5-hydroxytryptamine receptor 1Btarget
Aripiprazole lauroxil5-hydroxytryptamine receptor 1Dtarget
Aripiprazole lauroxil5-hydroxytryptamine receptor 1Etarget
Aripiprazole lauroxilDopamine D1 receptortarget
Aripiprazole lauroxilDopamine D5 receptortarget
Aripiprazole lauroxilDopamine D3 receptortarget
Aripiprazole lauroxilDopamine D4 receptortarget
Aripiprazole lauroxil5-hydroxytryptamine receptor 2Ctarget
Aripiprazole lauroxil5-hydroxytryptamine receptor 3Atarget
Aripiprazole lauroxil5-hydroxytryptamine receptor 6target
Aripiprazole lauroxil5-hydroxytryptamine receptor 7target
Aripiprazole lauroxilHistamine H1 receptortarget
Aripiprazole lauroxilAlpha-1A adrenergic receptortarget
Aripiprazole lauroxilAlpha-1B adrenergic receptortarget
Aripiprazole lauroxilAlpha-2A adrenergic receptortarget
Aripiprazole lauroxilAlpha-2B adrenergic receptortarget
Aripiprazole lauroxilAlpha-2C adrenergic receptortarget
Aripiprazole lauroxilMuscarinic acetylcholine receptor M1target
Aripiprazole lauroxilMuscarinic acetylcholine receptor M2target
Aripiprazole lauroxilMuscarinic acetylcholine receptor M3target
Aripiprazole lauroxilMuscarinic acetylcholine receptor M4target
Aripiprazole lauroxilMuscarinic acetylcholine receptor M5target
Aripiprazole lauroxilCytochrome P450 3A5enzyme
Aripiprazole lauroxilCytochrome P450 3A7enzyme
Aripiprazole lauroxilSerum albumincarrier
Lithium carbonateInositol monophosphatase 2target
Lithium carbonateInositol monophosphatase 1target
Lithium carbonateGlycogen synthase kinase-3 betatarget
Lithium carbonateGlutamate receptor 3target
Lithium carbonateAmiloride-sensitive sodium channel subunit alphatransporter
Lithium carbonateAmiloride-sensitive sodium channel subunit betatransporter
Lithium carbonateAmiloride-sensitive sodium channel subunit gammatransporter
ClobazamCytochrome P450 2C19enzyme
ClobazamCytochrome P450 3A4enzyme
ClobazamCytochrome P450 2B6enzyme
ClobazamCytochrome P450 2C18enzyme
ClobazamP-glycoprotein 1transporter
ClobazamGABA(A) Receptortarget
ClobazamCytochrome P450 2D6enzyme
ClobazamGABA(A) Receptor Benzodiazepine Binding Sitetarget
ClobazamSerum albumincarrier
ClobazamAlpha-1-acid glycoprotein 1carrier
ClobazamCytochrome P450 2C9enzyme
ClobazamUDP-glucuronosyltransferase 1-4enzyme
ClobazamUDP-glucuronosyltransferase 1-6enzyme
ClobazamUDP-glucuronosyltransferase 2B4enzyme
ClobazamUDP-glucuronosyltransferase 1-1enzyme
ClobazamCytochrome P450 1A2enzyme
ClobazamCytochrome P450 2C8enzyme
ClobazamCytochrome P450 3A5enzyme
ClobazamCytochrome P450 3A7enzyme
LamotrigineVoltage-gated sodium channel alpha subunittarget
LamotrigineUDP-glucuronosyltransferases (UGTs)enzyme
LamotrigineP-glycoprotein 1transporter
LamotrigineDihydrofolate reductaseenzyme
Lamotrigine5-hydroxytryptamine receptor 3Atarget
LamotrigineVoltage-dependent R-type calcium channel subunit alpha-1E (CACNA1E)target
LamotrigineAdenosine receptor A1target
LamotrigineAdenosine receptor A2atarget
LamotrigineAlpha-1A adrenergic receptortarget
LamotrigineAlpha-2A adrenergic receptortarget
LamotrigineBeta-1 adrenergic receptortarget
LamotrigineD(1) dopamine receptortarget
LamotrigineDopamine D2 receptortarget
LamotrigineGABA(A) Receptortarget
LamotrigineGABA(A) Receptor Benzodiazepine Binding Sitetarget
LamotrigineHistamine H1 receptortarget
LamotrigineKappa-type opioid receptortarget
LamotrigineAcetylcholine receptor subunit alphatarget
Lamotrigine5-hydroxytryptamine receptor 2Atarget
LamotrigineSolute carrier family 22 member 2transporter
LamotrigineSerum albumincarrier
LamotrigineSolute carrier family 22 member 1transporter
LamotrigineGlutamate receptor 1target
IloperidoneDopamine D2 receptortarget
Iloperidone5-hydroxytryptamine receptor 2Atarget
IloperidoneCytochrome P450 2D6enzyme
IloperidoneCytochrome P450 3A4enzyme
IloperidoneCytochrome P450 3A5enzyme
IloperidoneCytochrome P450 3A7enzyme
IloperidoneCytochrome P450 2E1enzyme
IloperidoneDopamine D3 receptortarget
IloperidoneAlpha-1A adrenergic receptortarget
IloperidoneDopamine D4 receptortarget
Iloperidone5-hydroxytryptamine receptor 6target
Iloperidone5-hydroxytryptamine receptor 7target
IloperidoneHistamine H1 receptortarget
IloperidoneDopamine D1 receptortarget
Iloperidone5-hydroxytryptamine receptor 1Atarget
IloperidoneAlpha-2C adrenergic receptortarget
CariprazineCytochrome P450 3A4enzyme
CariprazineCytochrome P450 2D6enzyme
CariprazineP-glycoprotein 1transporter
CariprazineCytochrome P450 3A5enzyme
CariprazineDopamine D3 receptortarget
CariprazineDopamine D2 receptortarget
Cariprazine5-hydroxytryptamine receptor 1Atarget
Cariprazine5-hydroxytryptamine receptor 2Btarget
Cariprazine5-hydroxytryptamine receptor 2Atarget
CariprazineHistamine H1 receptortarget
Cariprazine5-hydroxytryptamine receptor 2Ctarget
CariprazineAlpha-1A adrenergic receptortarget
CariprazineCytochrome P450 1A2enzyme
CariprazineCytochrome P450 2C9enzyme
CariprazineCytochrome P450 2C19enzyme
CariprazineCytochrome P450 2E1enzyme
RemimazolamLiver carboxylesterase 1enzyme
RemimazolamGABA(A) Receptor Benzodiazepine Binding Sitetarget
RemimazolamGABA(A) Receptortarget
RemimazolamSerum albumincarrier
FluvoxamineSodium-dependent serotonin transportertarget
FluvoxamineCytochrome P450 1A2enzyme
FluvoxamineCytochrome P450 2D6enzyme
FluvoxamineCytochrome P450 2C9enzyme
FluvoxamineCytochrome P450 2C19enzyme
FluvoxamineCytochrome P450 1A1enzyme
FluvoxamineCytochrome P450 3A4enzyme
FluvoxamineCytochrome P450 3A Subfamilyenzyme
FluvoxamineP-glycoprotein 1transporter
FluvoxamineCytochrome P450 2B6enzyme
FluvoxaminePotassium voltage-gated channel subfamily H member 2target
FluvoxamineBile salt export pumptransporter
ReserpineSynaptic vesicular amine transportertarget
ReserpineP-glycoprotein 1transporter
ReserpineSolute carrier family 22 member 1transporter
ReserpineBile salt export pumptransporter
ReserpineCanalicular multispecific organic anion transporter 1transporter
ReserpineSolute carrier family 22 member 2transporter
ReserpineCytochrome P450 3A5enzyme
ReserpineChromaffin granule amine transportertarget
ReserpineBaculoviral IAP repeat-containing protein 5target
ReserpineSolute carrier organic anion transporter family member 1B1transporter
ReserpineSolute carrier organic anion transporter family member 2B1transporter
DapiprazoleAlpha-1A adrenergic receptortarget
DapiprazoleAlpha-1D adrenergic receptortarget
DapiprazoleAlpha-1B adrenergic receptortarget
Valproic acidHistone deacetylase 9target
Valproic acidShort/branched chain specific acyl-CoA dehydrogenase, mitochondrialtarget
Valproic acidCytochrome P450 2A6enzyme
Valproic acidCytochrome P450 2B6enzyme
Valproic acidCytochrome P450 2C9enzyme
Valproic acidSolute carrier family 22 member 5transporter
Valproic acidSolute carrier family 22 member 6transporter
Valproic acidSolute carrier family 22 member 8transporter
Valproic acidMonocarboxylate transporter 1transporter
Valproic acidSolute carrier family 22 member 7transporter
Valproic acidCytochrome P450 3A5enzyme
Valproic acidUDP-glucuronosyltransferase 1-9enzyme
Valproic acidProstaglandin G/H synthase 1enzyme
Valproic acidCytochrome P450 1A2enzyme
Valproic acidCytochrome P450 2C19enzyme
Valproic acidCytochrome P450 3A4enzyme
Valproic acidUDP-glucuronosyltransferase 1-4enzyme
Valproic acidUDP-glucuronosyltransferase 1-8enzyme
Valproic acidUDP-glucuronosyltransferase 1-10enzyme
Valproic acidUDP-glucuronosyltransferase 1-6enzyme
Valproic acidUDP-glucuronosyltransferase 1-3enzyme
Valproic acidUDP-glucuronosyltransferase 2B7enzyme
Valproic acidUDP-glucuronosyltransferase 2B15enzyme
Valproic acid2-oxoglutarate dehydrogenase, mitochondrialtarget
Valproic acidSuccinate-semialdehyde dehydrogenase, mitochondrialtarget
Valproic acidSodium channel proteintarget
Valproic acidHistone deacetylase 2target
Valproic acidPeroxisome proliferator-activated receptor alphatarget
Valproic acidPeroxisome proliferator-activated receptor deltatarget
Valproic acidPeroxisome proliferator-activated receptor gammatarget
Valproic acidSerum albumincarrier
Valproic acidUDP-glucuronosyltransferase 1-1enzyme
Valproic acidSolute carrier organic anion transporter family member 2B1transporter
Valproic acidHistone deacetylasetarget
Valproic acidCyclin-dependent kinase inhibitor 1target
Valproic acidHepatocyte growth factortarget
Valproic acidOrnithine decarboxylasetarget
Valproic acidProgrammed cell death 1 ligand 1target
Mirtazapine5-hydroxytryptamine receptor 2Atarget
Mirtazapine5HT3 serotonin receptortarget
MirtazapineAlpha-2A adrenergic receptortarget
Mirtazapine5-hydroxytryptamine receptor 2Ctarget
MirtazapineKappa-type opioid receptortarget
MirtazapineHistamine H1 receptortarget
MirtazapineCytochrome P450 1A2enzyme
MirtazapineCytochrome P450 3A4enzyme
MirtazapineCytochrome P450 2D6enzyme
MirtazapineAlpha-1 adrenergic receptorstarget
MirtazapineSodium-dependent serotonin transportertransporter
DroperidolDopamine D2 receptortarget
DroperidolAlpha-1A adrenergic receptortarget
NabiloneCannabinoid receptor 2target
NabiloneCannabinoid receptor 1target
NabiloneCytochrome P450 2E1enzyme
NabiloneCytochrome P450 2C8enzyme
NabiloneCytochrome P450 2C9enzyme
NabiloneCytochrome P450 3A4enzyme
NabiloneCytochrome P450 2J2enzyme
TranylcypromineAmine oxidase [flavin-containing] Btarget
TranylcypromineAmine oxidase [flavin-containing] Atarget
TranylcypromineCytochrome P450 2C19enzyme
TranylcypromineCytochrome P450 2A6enzyme
TranylcypromineCytochrome P450 2D6enzyme
TranylcypromineCytochrome P450 1A2enzyme
TranylcypromineCytochrome P450 2C9enzyme
TranylcypromineCytochrome P450 3A4enzyme
FencamfaminSodium-dependent dopamine transportertarget
Ethyl loflazepateGABA(A) Receptortarget
Ethyl loflazepateGABA(A) Receptor Benzodiazepine Binding Sitetarget
FludiazepamGamma-aminobutyric acid receptor subunit alpha-2target
FludiazepamGamma-aminobutyric acid receptor subunit alpha-1target
FludiazepamGamma-aminobutyric acid receptor subunit alpha-3target
FludiazepamGamma-aminobutyric acid receptor subunit alpha-5target
FludiazepamGamma-aminobutyric acid receptor subunit gamma-1target
FludiazepamGamma-aminobutyric acid receptor subunit gamma-2target
FludiazepamGamma-aminobutyric acid receptor subunit gamma-3target
FludiazepamGamma-aminobutyric acid receptor subunit beta-1target
FludiazepamGamma-aminobutyric acid receptor subunit beta-2target
FludiazepamGamma-aminobutyric acid receptor subunit beta-3target
FludiazepamGamma-aminobutyric acid receptor subunit deltatarget
FludiazepamGamma-aminobutyric acid receptor subunit epsilontarget
FludiazepamGamma-aminobutyric acid receptor subunit pitarget
FludiazepamGamma-aminobutyric acid receptor subunit rho-1target
FludiazepamGamma-aminobutyric acid receptor subunit rho-2target
FludiazepamGamma-aminobutyric acid receptor subunit rho-3target
OxprenololBeta-1 adrenergic receptortarget
OxprenololBeta-2 adrenergic receptortarget
OxprenololSolute carrier family 22 member 2transporter
OxprenololCytochrome P450 2D6enzyme
OxprenololBeta-3 adrenergic receptortarget
AcepromazineDopamine D2 receptortarget
AcepromazineDopamine D1 receptortarget
Acepromazine5-hydroxytryptamine receptor 2Atarget
Acepromazine5-hydroxytryptamine receptor 1Atarget
AcepromazineAlpha-1A adrenergic receptortarget
AcepromazineAlpha-1B adrenergic receptortarget
AcepromazineSerum albumincarrier
AceprometazineHistamine H1 receptortarget
7-NitroindazoleNitric oxide synthase, endothelialtarget
7-NitroindazoleNitric oxide synthase, inducibletarget
7-NitroindazoleNitric oxide synthase, braintarget
OsanetantNeuromedin-K receptortarget
Deramciclane5-hydroxytryptamine receptor 2Atarget
Deramciclane5-hydroxytryptamine receptor 2Ctarget
DeramciclaneCytochrome P450 2D6enzyme
AdipiplonGABA(A) Receptor Benzodiazepine Binding Sitetarget
EsmirtazapineCytochrome P450 2D6enzyme
EsmirtazapineHistamine H1 receptortarget
Esmirtazapine5-hydroxytryptamine receptor 2target
EsmirtazapineAlpha-2 adrenergic receptorstarget
Perospirone5-hydroxytryptamine receptor 2Atarget
PerospironeDopamine D2 receptortarget
Perospirone5-hydroxytryptamine receptor 1Atarget
PerospironeCytochrome P450 3A4enzyme
PerospironeCytochrome P450 2D6enzyme
PerospironeCytochrome P450 2C8enzyme
PerospironeCytochrome P450 1A1enzyme
PerospironeHistamine H1 receptortarget
PerospironeDopamine D4 receptortarget
PerospironeAlpha-1 adrenergic receptorstarget
Amperozide5-hydroxytryptamine receptor 2Atarget
ButriptylineSodium-dependent serotonin transportertarget
ButriptylineHistamine H1 receptortarget
Butriptyline5-hydroxytryptamine receptor 2Atarget
MelperoneDopamine D2 receptortarget
MelperoneCytochrome P450 2D6enzyme
PipamperoneDopamine D2 receptortarget
Pipamperone5-hydroxytryptamine receptor 2Atarget
PipamperoneAlpha-1 adrenergic receptorstarget
PipamperoneDopamine D4 receptortarget
PipamperoneDopamine D1 receptortarget
PipamperoneDopamine D3 receptortarget
Pipamperone5-hydroxytryptamine receptor 2Btarget
PipamperoneAlpha-2A adrenergic receptortarget
DoramectinCytochrome P450 3A4enzyme
TetrahydropalmatineDopamine D1 receptortarget
TetrahydropalmatineDopamine D2 receptortarget
TetrahydropalmatineCytochrome P450 3A4enzyme
GepironeCytochrome P450 3A4enzyme
Gepirone5-hydroxytryptamine receptor 1Atarget
RacloprideDopamine D2 receptortarget
Ritanserin5-hydroxytryptamine receptor 2Atarget
RitanserinCytochrome P450 2D6enzyme
TiaprideDopamine D2 receptortarget
TiaprideDopamine D3 receptortarget
TiaprideSerotonin Receptorstarget
TiaprideAlpha-1 adrenergic receptorstarget
TiaprideAlpha-2 adrenergic receptorstarget
PinazepamGABA(A) Receptortarget
PinazepamGABA(A) Receptor Benzodiazepine Binding Sitetarget
MedazepamGABA(A) Receptortarget
MedazepamGABA(A) Receptor Benzodiazepine Binding Sitetarget
LoprazolamGABA(A) Receptortarget
LoprazolamGABA(A) Receptor Benzodiazepine Binding Sitetarget
PenfluridolCytochrome P450 3A4enzyme
NordazepamGABA(A) Receptortarget
NordazepamGABA(A) Receptor Benzodiazepine Binding Sitetarget
NorclozapineMuscarinic acetylcholine receptor M1target
NorclozapineDopamine D2 receptortarget
NorclozapineDopamine D3 receptortarget