Name
Thiepins
Accession Number
DBCAT001305
Description

Not Available

Drugs
DrugDrug Description
QuetiapineA psychotropic agent used for the management of bipolar disorder, schizophrenia, and major depressive disorder.
OmapatrilatFor the treatment of hypertension.
TemocaprilTemocapril is an ACE inhibitor primarily indicated in the treatment of hypertension and congestive heart failure, diabetic nephropathy, and improvement of prognosis for coronary artery diseases (including acute myocardial infarction).
DosulepinA tricyclic antidepressant commonly used only in patients for whom alternative therapies are ineffective due to its toxicity potential.
ZotepineZotepine, like other atypical antipsychotics, is considered as the first-line treatment in newly diagnosed schizophrenia. It is usually thought to be an option of choice for managing acute schizophrenic episodes...
TianeptineAn atypical tricyclic antidepressant with antidepressant and anxiolytic effects primarily used to treat major depressive disorder.
LinerixibatGSK2330672 has been investigated for the treatment of Diabetes Mellitus, Type 2.
ElobixibatElobixibat has been used in trials studying the treatment and basic science of Dyslipidemia, Constipation, Chronic Constipation, Functional Constipation, and Chronic Idiopathic Constipation.
TropatepineTropatepine has been used in France for its antiparkinsons activities .
ClothiapineAn atypical antipsychotic indicated in the treatment of acute psychosis, exacerbations of chronic psychosis, chronic psychosis, paranoid psychosis, and anxiety.
Baloxavir marboxilA polymerase acidic endonuclease inhibitor used to treat uncomplicated influenza.
ZiresovirZiresovir is under investigation in clinical trial NCT03699202 (Anti-RSV Study in Chinese Patients (ASCENT)).
BaloxavirBaloxavir is under investigation in clinical trial NCT04327791 (Combination Therapy With Baloxavir and Oseltamavir 1 for Hospitalized Patients With Influenza (The COMBO Trial 1)).
ClorotepineNot Annotated
Drugs & Drug Targets
DrugTargetType
Quetiapine5-hydroxytryptamine receptor 2Atarget
Quetiapine5-hydroxytryptamine receptor 2Ctarget
QuetiapineDopamine D2 receptortarget
Quetiapine5-hydroxytryptamine receptor 1Atarget
QuetiapineHistamine H1 receptortarget
QuetiapineCytochrome P450 3A4enzyme
QuetiapineAlpha-1 adrenergic receptorstarget
QuetiapineAlpha-2A adrenergic receptortarget
QuetiapineAlpha-2B adrenergic receptortarget
QuetiapineAlpha-2C adrenergic receptortarget
Quetiapine5-hydroxytryptamine receptor 1Dtarget
QuetiapineMuscarinic acetylcholine receptor M1target
QuetiapineMuscarinic acetylcholine receptor M2target
QuetiapineMuscarinic acetylcholine receptor M3target
QuetiapineMuscarinic acetylcholine receptor M4target
QuetiapineMuscarinic acetylcholine receptor M5target
Quetiapine5-hydroxytryptamine receptor 1Btarget
Quetiapine5-hydroxytryptamine receptor 1Etarget
Quetiapine5-hydroxytryptamine receptor 3Atarget
Quetiapine5-hydroxytryptamine receptor 6target
Quetiapine5-hydroxytryptamine receptor 7target
QuetiapineDopamine D5 receptortarget
QuetiapineDopamine D1 receptortarget
QuetiapineDopamine D3 receptortarget
QuetiapineDopamine D4 receptortarget
QuetiapineCytochrome P450 3A5enzyme
QuetiapineP-glycoprotein 1transporter
QuetiapineCytochrome P450 2C19enzyme
QuetiapineCytochrome P450 2D6enzyme
QuetiapineCytochrome P450 3A7enzyme
OmapatrilatNeprilysintarget
OmapatrilatAngiotensin-converting enzymetarget
TemocaprilSolute carrier family 15 member 1transporter
TemocaprilSolute carrier organic anion transporter family member 1A2transporter
TemocaprilAngiotensin-converting enzymetarget
Dosulepin5-hydroxytryptamine receptor 1Atarget
Dosulepin5-hydroxytryptamine receptor 2Atarget
DosulepinCytochrome P450 2D6enzyme
DosulepinCytochrome P450 1A2enzyme
DosulepinCytochrome P450 2C19enzyme
DosulepinCytochrome P450 2C9enzyme
DosulepinHistamine H1 receptortarget
DosulepinMuscarinic acetylcholine receptor M1target
DosulepinMuscarinic acetylcholine receptor M2target
DosulepinMuscarinic acetylcholine receptor M3target
DosulepinMuscarinic acetylcholine receptor M4target
DosulepinMuscarinic acetylcholine receptor M5target
DosulepinSodium-dependent noradrenaline transportertarget
DosulepinSodium-dependent serotonin transportertarget
DosulepinAlpha-1 adrenergic receptorstarget
DosulepinAlpha-2 adrenergic receptorstarget
ZotepineD(1) dopamine receptortarget
ZotepineDopamine D2 receptortarget
Zotepine5-hydroxytryptamine receptor 2Atarget
Zotepine5-hydroxytryptamine receptor 6target
Zotepine5-hydroxytryptamine receptor 7target
ZotepineSodium-dependent noradrenaline transportertarget
ZotepineSodium-dependent serotonin transportertarget
ZotepineCytochrome P450 1A2enzyme
ZotepineCytochrome P450 3A4enzyme
TianeptineGlutamate receptor 1target
TianeptineMu-type opioid receptortarget
Tianeptine5-hydroxytryptamine receptor 1Atarget
TianeptineDopamine D3 receptortarget
TianeptineCytochrome P450 3A4enzyme
Baloxavir marboxilUDP-glucuronosyltransferase 1-3enzyme
Baloxavir marboxilCytochrome P450 3A4enzyme
Baloxavir marboxilPolymerase acidic proteintarget
Baloxavir marboxilP-glycoprotein 1transporter
Baloxavir marboxilCytochrome P450 2B6enzyme
Baloxavir marboxilCytochrome P450 2C8enzyme
Baloxavir marboxilATP-binding cassette sub-family G member 2transporter