Endothelin B Receptor Antagonists
- Name
- Endothelin B Receptor Antagonists
- Accession Number
- DBCAT001699
- Description
Compounds and drugs that bind to and inhibit or block the activation of ENDOTHELIN B RECEPTORS.
- Drugs
Drug Drug Description Actelion-1 Investigated for use/treatment in cardiovascular disorders, hypertension, and pulmonary hypertension. Macitentan An endothelin receptor antagonist used to manage pulmonary arterial hypertension to delay disease progression. BQ-788 Not Annotated - Drugs & Drug Targets
Drug Target Type Actelion-1 Endothelin-1 receptor target Macitentan Cytochrome P450 3A4 enzyme Macitentan Cytochrome P450 2C19 enzyme Macitentan Endothelin-1 receptor target Macitentan Endothelin B receptor target Macitentan Serum albumin carrier Macitentan Cytochrome P450 2C9 enzyme Macitentan Cytochrome P450 2C8 enzyme Macitentan alpha1-acid glycoprotein carrier