Anabolic Agents for Systemic Use

Name
Anabolic Agents for Systemic Use
Accession Number
DBCAT002428
Description

Not Available

ATC Classification
Drugs
DrugDrug Description
OxandroloneAn androgenic hormone used to treat muscle loss from prolonged corticosteroid treatment and to treat bone pain associated with osteoporosis.
EthylestrenolAn anabolic steroid with some progestational activity and little androgenic effect. [PubChem]
OxymetholoneAn anabolic steroid used for the treatment of types of anemia, such as acquired aplastic anemia, congenital aplastic anemia, myelofibrosis, and the hypoplastic anemias.
StanozololAn anabolic steroid used to manage hereditary angioedema.
NorethandroloneNorethandrolone is under investigation in clinical trial NCT00700544 (Treatment Outcome in Elderly Patients).
NandroloneAn anabolic steroid indicated to increase bone density and muscle mass in patients with osteoporosis.
Oxabolone cipionateUsed as a performance enhancing drug illicitly in athletes.
QuinboloneNot Annotated
MetandienoneAn anabolic steroid indicated for appetite stimulation in patients with anorexia.
MetenoloneAn anabolic steroid indicated in the treatment and prevention of muscle wasting due to diseases, drug treatments, or other catabolic processes.
PrasteroneA steroid formulated as a vaginal insert indicated for the treatment of moderate to severe dyspareunia associated with menopausal vulvar and vaginal atrophy.
StanoloneA potent androgenic metabolite of testosterone. Dihydrotestosterone (DHT) is generated by a 5-alpha reduction of testosterone. Unlike testosterone, DHT cannot be aromatized to estradiol therefore DHT is considered a pure...
Drugs & Drug Targets
DrugTargetType
OxandroloneAndrogen receptortarget
OxandroloneCytochrome P450 2C9enzyme
OxymetholoneAndrogen receptortarget
OxymetholoneSerum albumincarrier
OxymetholoneSex hormone-binding globulincarrier
OxymetholoneNatriuretic peptides Btarget
OxymetholoneAmine oxidase [flavin-containing] Aenzyme
OxymetholoneCytochrome P450 2D6enzyme
Oxymetholone3-oxo-5-alpha-steroid 4-dehydrogenase 1enzyme
OxymetholoneCytochrome P450 3A4enzyme
OxymetholoneCytochrome P450 3A5enzyme
OxymetholoneCytochrome P450 3A7enzyme
OxymetholoneCytochrome P450 3A43enzyme
StanozololGlucocorticoid binding proteinstarget
StanozololAndrogen receptortarget
PrasteroneCytochrome P450 3A7enzyme
PrasteronePeroxisome proliferator-activated receptor alphatarget
PrasteroneEstrogen receptor alphatarget
PrasteroneSigma non-opioid intracellular receptor 1target
PrasteroneEstrogen receptor betatarget
PrasteroneNuclear receptor subfamily 1 group I member 2target
PrasteroneNuclear receptor subfamily 1 group I member 3target
PrasteroneGABA(A) Receptortarget
PrasteroneNMDA receptortarget
PrasteroneAndrogen receptortarget
PrasteroneEstradiol 17-beta-dehydrogenase 1enzyme
PrasteroneBile salt sulfotransferaseenzyme
PrasteroneSulfotransferase family cytosolic 2B member 1enzyme
Prasterone3 beta-hydroxysteroid dehydrogenase/Delta 5-->4-isomerase type 1enzyme
PrasteroneCholesterol oxidaseenzyme
PrasteroneSteroid 17-alpha-hydroxylase/17,20 lyaseenzyme
PrasteroneSolute carrier organic anion transporter family member 1B3transporter
PrasteroneSolute carrier organic anion transporter family member 2B1transporter
PrasteroneSolute carrier organic anion transporter family member 1B1transporter
PrasteroneSolute carrier organic anion transporter family member 1A2transporter
PrasteroneMultidrug resistance-associated protein 1transporter
PrasteroneATP-binding cassette sub-family G member 2transporter
PrasteroneMultidrug resistance-associated protein 4transporter
StanoloneSex hormone-binding globulincarrier
StanoloneAndrogen receptortarget
StanoloneEstradiol 17-beta-dehydrogenase 1target
StanoloneP-glycoprotein 1transporter
StanoloneCholesterol side-chain cleavage enzyme, mitochondrialenzyme
StanoloneSteroid 17-alpha-hydroxylase/17,20 lyaseenzyme
StanoloneCytochrome P450 19A1enzyme
StanoloneEstrogen receptor alphatarget
StanoloneMineralocorticoid receptortarget
StanoloneAldo-keto reductase family 1 member C3enzyme