Showing BioInteractions for Etomidate (DB00292)
BioInteractor utilizes data on drug-target, -enzyme and -transporter associations to provide insight on drug-drug interactions. It allows you to identify, for instance, which drugs act similarly on the same target. Such drugs may have additive pharmacodynamic effects if given concomitantly. Conversely, two drugs may antagonize the beneficial effects of each other by having opposite actions on a specific drug target. BioInteractor uses ranked drug-enzyme association information to predict enzyme-mediated drug interactions that may be clinically relevant.
Interacting Group | Interacting Drugs | |
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Etomidate is a Alpha-2B adrenergic receptor agonist | ||
1 | Alpha-2B adrenergic receptor antagonists | Aripiprazole, Asenapine, Cabergoline, Carvedilol, Celiprolol, Clozapine, Dronedarone, Fenoldopam, Methotrimeprazine, Mianserin, Paliperidone, Phenoxybenzamine, Pizotifen, Quetiapine, Risperidone, Rotigotine, Yohimbine, Ziprasidone |
2 | Alpha-2B adrenergic receptor agonists | Apomorphine, Apraclonidine, Brimonidine, Bromocriptine, Clonidine, Droxidopa, Ephedra sinica root, Epinephrine, Metamfetamine, Norepinephrine, Oxymetazoline, Racepinephrine, Xylometazoline |
3 | Alpha-2B adrenergic receptor ligands | Aripiprazole |
4 | Alpha-2B adrenergic receptor binders | Guanabenz, Guanfacine, Loxapine, Prazosin, Tolazoline |
Interacting Group | Interacting Drugs | |
---|---|---|
Etomidate is a Cytochrome P450 11B1, mitochondrial inhibitor | ||
1 | Cytochrome P450 11B1, mitochondrial inducers | Mitotane, Spironolactone |
2 | Cytochrome P450 11B1, mitochondrial inhibitors | Cimetidine, Dexamethasone, Dexamethasone acetate, Ketoconazole, Levoketoconazole, Metyrapone, Mibefradil, Miconazole, Osilodrostat, Phenytoin |
3 | Cytochrome P450 11B1, mitochondrial substrates | Aldosterone, Hydrocortisone, Hydrocortisone acetate, Hydrocortisone butyrate, Hydrocortisone probutate, Hydrocortisone succinate, Hydrocortisone valerate |
Interacting Group | Interacting Drugs | |
---|---|---|
Etomidate is a Cytochrome P450 11B2, mitochondrial inhibitor | ||
1 | Cytochrome P450 11B2, mitochondrial inhibitors | Eplerenone, Metyrapone, Mibefradil, Osilodrostat |
2 | Cytochrome P450 11B2, mitochondrial substrates | Aldosterone, Hydrocortisone, Hydrocortisone acetate, Hydrocortisone butyrate, Hydrocortisone probutate, Hydrocortisone succinate, Hydrocortisone valerate |
3 | Cytochrome P450 11B2, mitochondrial inducers | Torcetrapib |
4 | Cytochrome P450 11B2, mitochondrial antagonists | Spironolactone |