Showing BioInteractions for Loxapine (DB00408)

BioInteractor utilizes data on drug-target, -enzyme and -transporter associations to provide insight on drug-drug interactions. It allows you to identify, for instance, which drugs act similarly on the same target. Such drugs may have additive pharmacodynamic effects if given concomitantly. Conversely, two drugs may antagonize the beneficial effects of each other by having opposite actions on a specific drug target. BioInteractor uses ranked drug-enzyme association information to predict enzyme-mediated drug interactions that may be clinically relevant.
Interacting GroupInteracting Drugs
Loxapine is a Dopamine D1 receptor antagonist
1Dopamine D1 receptor antagonistsAcepromazine, Amoxapine, Aripiprazole, Asenapine, Carphenazine, Chlorpromazine, Chlorprothixene, Clozapine, Flupentixol, Fluphenazine, Haloperidol, Iloperidone, Lisuride, Methotrimeprazine, Methylergometrine, Olanzapine, Paliperidone, Periciazine, Perphenazine, Pipamperone, Pipotiazine, Quetiapine, Risperidone, Tetrahydropalmatine, Thioproperazine, Thioridazine, Thiothixene, Triflupromazine, Ziprasidone, Zuclopenthixol
2Dopamine D1 receptor agonistsApomorphine, Bromocriptine, Cabergoline, Dopamine, Fenoldopam, Levodopa, Minaprine, Pergolide, Rotigotine
3Dopamine D1 receptor partial agonistsAripiprazole, Phenylpropanolamine
4Dopamine D1 receptor ligandsAripiprazole
Interacting GroupInteracting Drugs
Loxapine is a Dopamine D2 receptor antagonist
1Dopamine D2 receptor agonistsAmantadine, Apomorphine, Brexpiprazole, Bromocriptine, Cabergoline, Cariprazine, Dihydro-alpha-ergocryptine, Dopamine, Ergotamine, Ketamine, Lamotrigine, Levodopa, Lisuride, Memantine, Minaprine, Pergolide, Pramipexole, Quinagolide, Ropinirole, Rotigotine
2Dopamine D2 receptor antagonistsAcepromazine, Acetophenazine, Alizapride, Amisulpride, Amoxapine, Aripiprazole, AS-8112, Asenapine, Blonanserin, Bromopride, Buspirone, Carphenazine, Chlorpromazine, Chlorprothixene, Clozapine, Domperidone, Droperidol, Etoperidone, Flupentixol, Fluphenazine, Fluspirilene, Haloperidol, Iloperidone, JNJ-37822681, Lurasidone, Melperone, Memantine, Mesoridazine, Methotrimeprazine, Metoclopramide, Mianserin, Molindone, Nortriptyline, Olanzapine, Paliperidone, Perospirone, Perphenazine, Pimozide, Pipamperone, Pipotiazine, Prochlorperazine, Promazine, Promethazine, Propiomazine, Quetiapine, Raclopride, Remoxipride, Risperidone, Sertindole, Sulpiride, Tetrahydropalmatine, Thiethylperazine, Thioproperazine, Thioridazine, Thiothixene, Trifluoperazine, Triflupromazine, YKP-1358, Yohimbine, Ziprasidone, Zotepine, Zuclopenthixol
3Dopamine D2 receptor partial agonistsAripiprazole, Aripiprazole lauroxil, Brexpiprazole, Cariprazine, Ketamine, Lumateperone, Sarizotan
4Dopamine D2 receptor inhibitorsEscitalopram, Lamotrigine, Tetrabenazine
5Dopamine D2 receptor bindersAmphetamine, Desipramine, Imipramine, Maprotiline
6Dopamine D2 receptor blockersTiapride
Interacting GroupInteracting Drugs
Loxapine is a 5-hydroxytryptamine receptor 2A antagonist
15-hydroxytryptamine receptor 2A antagonistsAcepromazine, Amisulpride, Amitriptyline, Amoxapine, Amperozide, Aripiprazole, Aripiprazole lauroxil, Asenapine, Blonanserin, Brexpiprazole, Butriptyline, Cariprazine, Chlorpromazine, Chlorprothixene, Cinitapride, Clomipramine, Clozapine, Cyclobenzaprine, Cyproheptadine, Deramciclane, Desipramine, Dosulepin, Doxepin, Epinastine, Etoperidone, Flibanserin, Flupentixol, Fluspirilene, Iloperidone, Imipramine, Lorpiprazole, Lumateperone, Lurasidone, Mesoridazine, Methotrimeprazine, Methysergide, Mianserin, Minaprine, Mirtazapine, Molindone, Nefazodone, Nortriptyline, Olanzapine, Paliperidone, Pipotiazine, Pizotifen, Promazine, Propiomazine, Quetiapine, Risperidone, Sertindole, Tegaserod, Thioridazine, Thiothixene, Trazodone, Yohimbine, Ziprasidone, Zotepine, Zuclopenthixol
25-hydroxytryptamine receptor 2A partial agonists4-Bromo-2,5-dimethoxyphenethylamine, Aripiprazole
35-hydroxytryptamine receptor 2A agonists2,5-Dimethoxy-4-ethylthioamphetamine, 5-methoxy-N,N-dimethyltryptamine, Apomorphine, Bromocriptine, Cabergoline, Cannabidiol, Cisapride, Ergotamine, Fenfluramine, Lisuride, Midomafetamine, MMDA, N-(2-hydroxybenzyl)-2,5-dimethoxy-4-cyanophenylethylamine, Paroxetine, Pergolide, Pipamperone, Trimipramine, Zolmitriptan
45-hydroxytryptamine receptor 2A inducersDonepezil
55-hydroxytryptamine receptor 2A inverse agonistsKetanserin, Perospirone, Pimavanserin, Ritanserin, Sarpogrelate
65-hydroxytryptamine receptor 2A bindersMaprotiline
75-hydroxytryptamine receptor 2A inhibitorsEscitalopram, Lamotrigine
Interacting GroupInteracting Drugs
Loxapine is a 5-hydroxytryptamine receptor 2C antagonist
15-hydroxytryptamine receptor 2C agonists2,5-Dimethoxy-4-ethylthioamphetamine, Apomorphine, Bromocriptine, Cabergoline, Dexfenfluramine, Ergotamine, Etoperidone, Fenfluramine, Lisuride, Lofexidine, m-Chlorophenylpiperazine, Midomafetamine, Pergolide, Trazodone
25-hydroxytryptamine receptor 2C antagonistsAgomelatine, Amitriptyline, Amoxapine, Aripiprazole, Asenapine, Captodiame, Clomipramine, Clozapine, Cyclobenzaprine, Cyproheptadine, Doxepin, Fluoxetine, Flupentixol, Imipramine, Lorpiprazole, Methotrimeprazine, Methysergide, Mianserin, Minaprine, Mirtazapine, Nefazodone, Nortriptyline, Olanzapine, Paliperidone, Pizotifen, Promazine, Propiomazine, Risperidone, Sertindole, Tegaserod, Tramadol, Trimipramine, Yohimbine, Ziprasidone
35-hydroxytryptamine receptor 2C ligandsQuetiapine
45-hydroxytryptamine receptor 2C inverse agonistsDeramciclane
55-hydroxytryptamine receptor 2C partial agonists4-Bromo-2,5-dimethoxyphenethylamine, Aripiprazole
65-hydroxytryptamine receptor 2C bindersChlorpromazine, Desipramine, Imipramine, Maprotiline
75-hydroxytryptamine receptor 2C inhibitorsEscitalopram
Interacting GroupInteracting Drugs
Loxapine is a 5-hydroxytryptamine receptor 1A binder
15-hydroxytryptamine receptor 1A partial agonistsAripiprazole, Aripiprazole lauroxil, Brexpiprazole, Buspirone, Cariprazine, Perospirone, Quetiapine, Trazodone, Yohimbine
25-hydroxytryptamine receptor 1A agonists5-methoxy-N,N-dimethyltryptamine, Apomorphine, Brexpiprazole, Bromocriptine, Cabergoline, Cannabidiol, Cariprazine, Cinitapride, Eletriptan, Ergotamine, Fenfluramine, Flibanserin, Lisuride, Lofexidine, Methysergide, Naluzotan, Naratriptan, Oxymetazoline, Pergolide, Pramipexole, Rotigotine, SEP-363856, Sumatriptan, Tetrahydrocannabivarin, Vilazodone, Vortioxetine, Ziprasidone, Zolmitriptan
35-hydroxytryptamine receptor 1A antagonistsAcepromazine, Alprenolol, Alverine, Amoxapine, Asenapine, Chlorpromazine, Clozapine, Dosulepin, Doxepin, Iloperidone, Lurasidone, Molindone, Nefazodone, Nortriptyline, Paliperidone, Penbutolol, Pindolol, Pipotiazine, Pirlindole, Pizotifen, Quetiapine, Risperidone, Trazodone, Trimipramine
45-hydroxytryptamine receptor 1A inhibitorsAmitriptyline, Escitalopram, Tianeptine
55-hydroxytryptamine receptor 1A inducersAmitriptyline
65-hydroxytryptamine receptor 1A bindersDesipramine, Dopamine
75-hydroxytryptamine receptor 1A activatorsImipramine
85-hydroxytryptamine receptor 1A blockersMianserin
Interacting GroupInteracting Drugs
Loxapine is a 5-hydroxytryptamine receptor 1B binder
15-hydroxytryptamine receptor 1B agonistsAlmotriptan, Apomorphine, Bromocriptine, Cabergoline, Dihydroergotamine, Eletriptan, Ergotamine, Frovatriptan, Lisuride, Naratriptan, Oxymetazoline, Pergolide, Rizatriptan, Sumatriptan, Zolmitriptan
25-hydroxytryptamine receptor 1B antagonistsAmoxapine, Aripiprazole, Asenapine, Clozapine, Penbutolol, Pizotifen, Ziprasidone
35-hydroxytryptamine receptor 1B ligandsAripiprazole, Quetiapine
45-hydroxytryptamine receptor 1B partial agonistsVortioxetine, Yohimbine
55-hydroxytryptamine receptor 1B bindersAmitriptyline, Methysergide
Interacting GroupInteracting Drugs
Loxapine is a 5-hydroxytryptamine receptor 1D binder
15-hydroxytryptamine receptor 1D agonistsAlmotriptan, Apomorphine, Bromocriptine, Cabergoline, Dihydroergotamine, Eletriptan, Ergotamine, Fenfluramine, Frovatriptan, Lisuride, Lofexidine, Naratriptan, Oxymetazoline, Pergolide, Rizatriptan, Sumatriptan, Zolmitriptan
25-hydroxytryptamine receptor 1D antagonistsAripiprazole, Clozapine, Paliperidone, Pizotifen, Risperidone, Ziprasidone
35-hydroxytryptamine receptor 1D ligandsAripiprazole, Quetiapine
45-hydroxytryptamine receptor 1D partial agonistsYohimbine
55-hydroxytryptamine receptor 1D bindersAmitriptyline, Trimipramine
Interacting GroupInteracting Drugs
Loxapine is a 5-hydroxytryptamine receptor 1E binder
15-hydroxytryptamine receptor 1E antagonistsAripiprazole, Clozapine, Ziprasidone
25-hydroxytryptamine receptor 1E ligandsAripiprazole, Quetiapine
35-hydroxytryptamine receptor 1E bindersMethysergide
45-hydroxytryptamine receptor 1E agonistsZolmitriptan
Interacting GroupInteracting Drugs
Loxapine is a 5-hydroxytryptamine receptor 3A binder
15-hydroxytryptamine receptor 3A antagonistsAlosetron, Amoxapine, Aripiprazole, Cannabidiol, Clozapine, Dolasetron, Granisetron, Memantine, Methadone, Metoclopramide, Olanzapine, Ondansetron, Palonosetron, Procaine, Ramosetron, Rocuronium, Tropisetron, Tubocurarine, Vortioxetine
25-hydroxytryptamine receptor 3A agonistsCisapride
35-hydroxytryptamine receptor 3A ligandsQuetiapine
45-hydroxytryptamine receptor 3A bindersTrimipramine
55-hydroxytryptamine receptor 3A inhibitorsLamotrigine
65-hydroxytryptamine receptor 3A potentiatorsKetamine
75-hydroxytryptamine receptor 3A negative modulatorsBupropion
Interacting GroupInteracting Drugs
Loxapine is a 5-hydroxytryptamine receptor 5A binder
15-hydroxytryptamine receptor 5A antagonistsAsenapine, Ziprasidone
25-hydroxytryptamine receptor 5A ligandsAripiprazole
Interacting GroupInteracting Drugs
Loxapine is a 5-hydroxytryptamine receptor 6 binder
15-hydroxytryptamine receptor 6 antagonistsAmitriptyline, Amoxapine, Aripiprazole, Asenapine, Clozapine, Cyclobenzaprine, Iloperidone, Olanzapine, Quetiapine, Sertindole, Ziprasidone, Zotepine
25-hydroxytryptamine receptor 6 bindersChlorpromazine, Doxepin, Imipramine, Mianserin
Interacting GroupInteracting Drugs
Loxapine is a 5-hydroxytryptamine receptor 7 binder
15-hydroxytryptamine receptor 7 antagonistsAmisulpride, Amitriptyline, Amoxapine, Aripiprazole, Asenapine, Bromocriptine, Cabergoline, Clozapine, Cyclobenzaprine, Epinastine, Iloperidone, Imipramine, Lurasidone, Maprotiline, Methysergide, Mianserin, Risperidone, SB-269970, Vortioxetine, Ziprasidone, Zotepine
25-hydroxytryptamine receptor 7 partial agonistsAripiprazole
35-hydroxytryptamine receptor 7 ligandsQuetiapine
45-hydroxytryptamine receptor 7 bindersChlorpromazine, Dopamine
55-hydroxytryptamine receptor 7 agonistsLofexidine, Zolmitriptan
Interacting GroupInteracting Drugs
Loxapine is a Alpha-1A adrenergic receptor binder
1Alpha-1A adrenergic receptor agonists4-Methoxyamphetamine, Apraclonidine, Benzphetamine, Bromocriptine, Cirazoline, Clonidine, Dipivefrin, Droxidopa, Ephedrine, Epinephrine, Ergometrine, Isometheptene, Lofexidine, Metaraminol, Methoxamine, Midodrine, Naphazoline, Norepinephrine, Pergolide, Phendimetrazine, Phenylephrine, Pseudoephedrine, Racepinephrine, Tetryzoline, Xylometazoline
2Alpha-1A adrenergic receptor antagonistsAcepromazine, Alfuzosin, Amitriptyline, Amoxapine, Aripiprazole, Aripiprazole lauroxil, Asenapine, Bevantolol, Bromocriptine, Carvedilol, Chlorpromazine, Clozapine, Dapiprazole, Doxazosin, Doxepin, Dronedarone, Droperidol, Flupentixol, Iloperidone, Imipramine, Indoramin, Methotrimeprazine, Nefazodone, Nicardipine, Nicergoline, Niguldipine, Nortriptyline, Olanzapine, Paliperidone, Phenoxybenzamine, Phentolamine, Pizotifen, Prazosin, Promazine, Propiomazine, Propiverine, Quinidine, Risperidone, Silodosin, Tamsulosin, Terazosin, Thioproperazine, Thioridazine, Tolazoline, Trazodone, Trifluoperazine, Trimipramine, Verapamil, Ziprasidone, Zuclopenthixol
3Alpha-1A adrenergic receptor partial agonistsErgotamine, Oxymetazoline, Xylometazoline
4Alpha-1A adrenergic receptor potentiatorsCarvedilol
5Alpha-1A adrenergic receptor inhibitorsAmitriptyline, Fenoldopam, Lamotrigine
6Alpha-1A adrenergic receptor bindersCabergoline
Interacting GroupInteracting Drugs
Loxapine is a Alpha-1B adrenergic receptor binder
1Alpha-1B adrenergic receptor antagonistsAcepromazine, Alfuzosin, Amitriptyline, Aripiprazole, Aripiprazole lauroxil, Brexpiprazole, Bromocriptine, Carvedilol, Chlorpromazine, Clozapine, Dapiprazole, Dextroamphetamine, Doxepin, Dronedarone, Imipramine, Methotrimeprazine, Nicardipine, Nortriptyline, Olanzapine, Paliperidone, Periciazine, Phenoxybenzamine, Phentolamine, Pizotifen, Prazosin, Quinidine, Risperidone, Silodosin, Tamsulosin, Terazosin, Thioproperazine, Thioridazine, Trimipramine, Verapamil, Ziprasidone
2Alpha-1B adrenergic receptor partial agonistsCirazoline, Ergotamine, Modafinil
3Alpha-1B adrenergic receptor agonistsBromocriptine, Clonidine, Droxidopa, Epinephrine, Methoxamine, Midodrine, Norepinephrine, Oxymetazoline, Pergolide, Phendimetrazine, Phenylephrine, Racepinephrine, Xylometazoline
4Alpha-1B adrenergic receptor bindersCabergoline
5Alpha-1B adrenergic receptor inhibitorsFenoldopam
Interacting GroupInteracting Drugs
Loxapine is a Alpha-2A adrenergic receptor binder
1Alpha-2A adrenergic receptor agonists4-Methoxyamphetamine, Amitriptyline, Apomorphine, Apraclonidine, Benzphetamine, Brimonidine, Bromocriptine, Clonidine, Dexmedetomidine, Dihydroergotamine, Dipivefrin, DL-Methylephedrine, Droxidopa, Ephedra sinica root, Epinephrine, Guanabenz, Guanfacine, Lofexidine, Metamfetamine, Moxonidine, Naphazoline, Norepinephrine, Oxymetazoline, Pramipexole, Pseudoephedrine, Racepinephrine, Xylometazoline
2Alpha-2A adrenergic receptor antagonistsAmitriptyline, Amoxapine, Aripiprazole, Asenapine, Cabergoline, Carvedilol, Celiprolol, Clozapine, Dronedarone, Fenoldopam, Methotrimeprazine, Mianserin, Mirtazapine, Nefazodone, Paliperidone, Periciazine, Phenoxybenzamine, Phentolamine, Pipamperone, Pirlindole, Pizotifen, Quetiapine, Tolazoline, Trazodone, Yohimbine, Ziprasidone, Zuclopenthixol
3Alpha-2A adrenergic receptor partial agonistsErgotamine, Oxymetazoline
4Alpha-2A adrenergic receptor bindersPrazosin
5Alpha-2A adrenergic receptor inhibitorsLamotrigine
Interacting GroupInteracting Drugs
Loxapine is a Alpha-2B adrenergic receptor binder
1Alpha-2B adrenergic receptor antagonistsAripiprazole, Asenapine, Cabergoline, Carvedilol, Celiprolol, Clozapine, Dronedarone, Fenoldopam, Methotrimeprazine, Mianserin, Paliperidone, Phenoxybenzamine, Pizotifen, Quetiapine, Risperidone, Rotigotine, Yohimbine, Ziprasidone
2Alpha-2B adrenergic receptor agonistsApomorphine, Apraclonidine, Brimonidine, Bromocriptine, Clonidine, Droxidopa, Ephedra sinica root, Epinephrine, Etomidate, Metamfetamine, Norepinephrine, Oxymetazoline, Racepinephrine, Xylometazoline
3Alpha-2B adrenergic receptor ligandsAripiprazole
4Alpha-2B adrenergic receptor bindersGuanabenz, Guanfacine, Prazosin, Tolazoline
Interacting GroupInteracting Drugs
Loxapine is a Alpha-2C adrenergic receptor binder
1Alpha-2C adrenergic receptor antagonistsAripiprazole, Asenapine, Brexpiprazole, Cabergoline, Carvedilol, Celiprolol, Clozapine, Dronedarone, Fenoldopam, Iloperidone, Lurasidone, Methotrimeprazine, Mianserin, Phenoxybenzamine, Pizotifen, Quetiapine, Risperidone, Yohimbine, Ziprasidone
2Alpha-2C adrenergic receptor agonistsAgmatine, Apomorphine, Brimonidine, Bromocriptine, Clonidine, Droxidopa, Ephedra sinica root, Metamfetamine, Norepinephrine, Oxymetazoline, Paliperidone, Racepinephrine, Xylometazoline
3Alpha-2C adrenergic receptor bindersTolazoline
Interacting GroupInteracting Drugs
Loxapine is a Beta-1 adrenergic receptor binder
1Beta-1 adrenergic receptor antagonistsAlprenolol, Arotinolol, Asenapine, Atenolol, Betaxolol, Bevantolol, Bisoprolol, Bupranolol, Carvedilol, Celiprolol, Dronedarone, Esmolol, Labetalol, Levobetaxolol, Levobunolol, Metipranolol, Metoprolol, Nadolol, Nebivolol, Oxprenolol, Penbutolol, Practolol, Propafenone, Propranolol, Ranolazine, Sotalol, Terbutaline, Timolol
2Beta-1 adrenergic receptor agonistsArbutamine, Clenbuterol, DL-Methylephedrine, Dobutamine, Droxidopa, Ephedra sinica root, Ephedrine, Epinephrine, Fenoterol, Formoterol, Isoetharine, Isoprenaline, Norepinephrine, Phenylpropanolamine, Pirbuterol, Pseudoephedrine, Racepinephrine, Salbutamol
3Beta-1 adrenergic receptor partial agonistsAcebutolol, Bopindolol, Carteolol, Penbutolol, Pindolol, Pseudoephedrine, Xamoterol
4Beta-1 adrenergic receptor bindersCabergoline
5Beta-1 adrenergic receptor ligandsAripiprazole, Vortioxetine
6Beta-1 adrenergic receptor inverse agonistsSalmeterol
7Beta-1 adrenergic receptor inhibitorsLamotrigine
Interacting GroupInteracting Drugs
Loxapine is a Muscarinic acetylcholine receptor M1 binder
1Muscarinic acetylcholine receptor M1 agonistsCarbamoylcholine, Cevimeline, Methacholine, Metoclopramide, Minaprine, Pilocarpine, Pyrantel, Succinylcholine
2Muscarinic acetylcholine receptor M1 antagonistsAclidinium, Amoxapine, Anisotropine methylbromide, Atropine, Benzatropine, Benzquinamide, Biperiden, Brompheniramine, Buclizine, Chlorpromazine, Chlorprothixene, Clidinium, Clozapine, Cocaine, Cyclopentolate, Cycrimine, Cyproheptadine, Darifenacin, Desipramine, Dicyclomine, Diphenidol, Disopyramide, Dosulepin, Doxepin, Fesoterodine, Flavoxate, Flupentixol, Glycopyrronium, Hexocyclium, Homatropine, Homatropine methylbromide, Hyoscyamine, Imidafenacin, Imipramine, Ipratropium, Maprotiline, Mepenzolate, Methantheline, Methotrimeprazine, Methscopolamine bromide, Nicardipine, Olanzapine, Oxybutynin, Oxyphencyclimine, Oxyphenonium, Pirenzepine, Pizotifen, Procyclidine, Profenamine, Promazine, Promethazine, Propantheline, Propiverine, Pyrantel, Quetiapine, Rociverine, Scopolamine, Solifenacin, Thonzylamine, Tiotropium, Tolterodine, Tramadol, Tridihexethyl, Triflupromazine, Trihexyphenidyl, Trimebutine, Tropicamide, Trospium, Umeclidinium, Ziprasidone
3Muscarinic acetylcholine receptor M1 weak inhibitorsBuclizine
4Muscarinic acetylcholine receptor M1 inhibitorsEscitalopram
5Muscarinic acetylcholine receptor M1 bindersTerfenadine
6Muscarinic acetylcholine receptor M1 ligandsAripiprazole
Interacting GroupInteracting Drugs
Loxapine is a Muscarinic acetylcholine receptor M2 binder
1Muscarinic acetylcholine receptor M2 antagonistsAclidinium, Anisotropine methylbromide, Atropine, Benzquinamide, Brompheniramine, Butylscopolamine, Chlorprothixene, Clozapine, Cocaine, Cryptenamine, Cyproheptadine, Darifenacin, Desipramine, Dicyclomine, Dimetindene, Diphenhydramine, Diphenidol, Disopyramide, Dosulepin, Doxacurium, Doxepin, Fesoterodine, Flavoxate, Gallamine triethiodide, Hexocyclium, Homatropine, Homatropine methylbromide, Hyoscyamine, Imidafenacin, Imipramine, Ipratropium, Maprotiline, Methotrimeprazine, Methscopolamine bromide, Metocurine, Mivacurium, Nicardipine, Olanzapine, Oxybutynin, Oxyphencyclimine, Pancuronium, Pipecuronium, Pizotifen, Procyclidine, Profenamine, Promethazine, Propiverine, Rapacuronium, Rociverine, Rocuronium, Scopolamine, Solifenacin, Thonzylamine, Tiotropium, Tolterodine, Tridihexethyl, Triflupromazine, Trihexyphenidyl, Trimebutine, Tropicamide, Umeclidinium, Ziprasidone
2Muscarinic acetylcholine receptor M2 agonistsBethanechol, Carbamoylcholine, Methacholine, Pilocarpine, Succinylcholine
3Muscarinic acetylcholine receptor M2 partial agonistsMivacurium
4Muscarinic acetylcholine receptor M2 ligandsAripiprazole, Quetiapine
5Muscarinic acetylcholine receptor M2 bindersGlycopyrronium, Terfenadine
Interacting GroupInteracting Drugs
Loxapine is a Muscarinic acetylcholine receptor M3 binder
1Muscarinic acetylcholine receptor M3 antagonistsAclidinium, Anisotropine methylbromide, Atropine, Benzquinamide, Brompheniramine, Butylscopolamine, Chlorpromazine, Chlorprothixene, Clozapine, Cyproheptadine, Darifenacin, Desipramine, Diphemanil, Diphenidol, Disopyramide, Dosulepin, Doxepin, Fesoterodine, Glycopyrronium, Hexocyclium, Homatropine, Homatropine methylbromide, Hyoscyamine, Imidafenacin, Imipramine, Ipratropium, Isopropamide, Maprotiline, Mepenzolate, Methotrimeprazine, Methscopolamine bromide, Mivacurium, Nicardipine, Olanzapine, Oxybutynin, Oxyphencyclimine, Pancuronium, Pipecuronium, Pizotifen, Procyclidine, Promethazine, Propiverine, Quetiapine, Rociverine, Scopolamine, Solifenacin, Terfenadine, Thonzylamine, Tiotropium, Tolterodine, Tramadol, Tridihexethyl, Trihexyphenidyl, Trimebutine, Tropicamide, Umeclidinium, Ziprasidone
2Muscarinic acetylcholine receptor M3 agonistsCarbamoylcholine, Cevimeline, Methacholine, Pilocarpine, Succinylcholine
3Muscarinic acetylcholine receptor M3 ligandsAripiprazole
Interacting GroupInteracting Drugs
Loxapine is a Muscarinic acetylcholine receptor M4 binder
1Muscarinic acetylcholine receptor M4 antagonistsAclidinium, Atropine, Benzquinamide, Brompheniramine, Chlorprothixene, Clozapine, Darifenacin, Desipramine, Dosulepin, Doxepin, Fesoterodine, Hexocyclium, Homatropine, Homatropine methylbromide, Hyoscyamine, Imipramine, Isopropamide, Maprotiline, Methotrimeprazine, Nicardipine, Olanzapine, Procyclidine, Promethazine, Propiverine, Rociverine, Scopolamine, Solifenacin, Thonzylamine, Tolterodine, Trihexyphenidyl, Trimebutine, Tropicamide, Umeclidinium, Ziprasidone
2Muscarinic acetylcholine receptor M4 ligandsAripiprazole, Quetiapine
3Muscarinic acetylcholine receptor M4 bindersTerfenadine
4Muscarinic acetylcholine receptor M4 agonistsCarbamoylcholine, Methacholine
5Muscarinic acetylcholine receptor M4 partial agonistsPilocarpine
Interacting GroupInteracting Drugs
Loxapine is a Muscarinic acetylcholine receptor M5 binder
1Muscarinic acetylcholine receptor M5 antagonistsAclidinium, Atropine, Benzquinamide, Brompheniramine, Chlorprothixene, Clozapine, Darifenacin, Desipramine, Dosulepin, Doxepin, Fesoterodine, Homatropine, Homatropine methylbromide, Imipramine, Maprotiline, Methotrimeprazine, Nicardipine, Promethazine, Rociverine, Scopolamine, Solifenacin, Thonzylamine, Tolterodine, Trihexyphenidyl, Umeclidinium, Ziprasidone
2Muscarinic acetylcholine receptor M5 ligandsAripiprazole, Quetiapine
3Muscarinic acetylcholine receptor M5 bindersTerfenadine
4Muscarinic acetylcholine receptor M5 agonistsMethacholine
Interacting GroupInteracting Drugs
Loxapine is a D(1) dopamine receptor binder
1D(1) dopamine receptor inhibitorsChlorpromazine, Lamotrigine
2D(1) dopamine receptor bindersCinnarizine, Imipramine, Mianserin, Trimipramine
3D(1) dopamine receptor agonistsCabergoline, Dopamine, Ergotamine, Pipradrol, Quinagolide
4D(1) dopamine receptor antagonistsOlanzapine, Zotepine
5D(1) dopamine receptor partial agonistsDihydro-alpha-ergocryptine
Interacting GroupInteracting Drugs
Loxapine is a Dopamine D3 receptor binder
1Dopamine D3 receptor antagonistsAmisulpride, Amoxapine, Aripiprazole, AS-8112, Asenapine, Blonanserin, Buspirone, Chlorprothixene, Clozapine, Domperidone, Flupentixol, Iloperidone, Methotrimeprazine, Olanzapine, Paliperidone, Pimozide, Remoxipride, Sulpiride, Yohimbine, Ziprasidone
2Dopamine D3 receptor agonistsApomorphine, Bromocriptine, Cabergoline, Captodiame, Cariprazine, Dopamine, Levodopa, Lisuride, Pergolide, Pramipexole, Ropinirole, Rotigotine, Tianeptine
3Dopamine D3 receptor partial agonistsAripiprazole, Cariprazine, Dihydro-alpha-ergocryptine
4Dopamine D3 receptor inverse agonistsHaloperidol
5Dopamine D3 receptor ligandsQuetiapine, Sarizotan
6Dopamine D3 receptor inhibitorsChlorpromazine
7Dopamine D3 receptor bindersMianserin
8Dopamine D3 receptor blockersTiapride
Interacting GroupInteracting Drugs
Loxapine is a Dopamine D4 receptor binder
1Dopamine D4 receptor antagonistsAmoxapine, Aripiprazole, Asenapine, Bromocriptine, Buspirone, Clozapine, Flibanserin, Flupentixol, Iloperidone, Methotrimeprazine, Olanzapine, Paliperidone, Perospirone, Pipamperone, Remoxipride, Sulpiride, Ziprasidone
2Dopamine D4 receptor agonistsApomorphine, Cabergoline, Dopamine, Flibanserin, Levodopa, Lisuride, Pergolide, Pramipexole, Ropinirole, Rotigotine
3Dopamine D4 receptor partial agonistsAripiprazole
4Dopamine D4 receptor ligandsQuetiapine
5Dopamine D4 receptor bindersChlorpromazine
Interacting GroupInteracting Drugs
Loxapine is a Dopamine D5 receptor binder
1Dopamine D5 receptor agonistsApomorphine, Bromocriptine, Cabergoline, Dopamine, Fenoldopam, Levodopa, Pergolide, Rotigotine
2Dopamine D5 receptor antagonistsAripiprazole, Carphenazine, Lisuride, Methotrimeprazine, Olanzapine, Ziprasidone, Zuclopenthixol
3Dopamine D5 receptor partial agonistsAripiprazole
4Dopamine D5 receptor ligandsAripiprazole, Quetiapine
5Dopamine D5 receptor inhibitorsChlorpromazine
Interacting GroupInteracting Drugs
Loxapine is a Histamine H1 receptor binder
1Histamine H1 receptor antagonistsAceprometazine, Acrivastine, Alcaftadine, Alimemazine, Amitriptyline, Amoxapine, Antazoline, Aripiprazole, Aripiprazole lauroxil, Asenapine, Astemizole, Azatadine, Azelastine, Benzatropine, Benzquinamide, Bepotastine, Bilastine, Bromodiphenhydramine, Brompheniramine, Buclizine, Butriptyline, Carbinoxamine, Cariprazine, Cetirizine, Chlorcyclizine, Chloropyramine, Chlorpheniramine, Chlorpromazine, Chlorprothixene, Cinnarizine, Clemastine, Clofedanol, Clozapine, Cyclizine, Cyproheptadine, Desipramine, Desloratadine, Dexbrompheniramine, Dexchlorpheniramine maleate, Dimenhydrinate, Dimetindene, Diphenhydramine, Diphenylpyraline, Dosulepin, Doxepin, Doxylamine, Emedastine, Epinastine, Fexofenadine, Flunarizine, Iloperidone, Imipramine, Isothipendyl, Ketotifen, Lamotrigine, Levocabastine, Levocetirizine, Loratadine, Lorpiprazole, Maprotiline, Meclizine, Mepyramine, Mequitazine, Methdilazine, Methotrimeprazine, Mianserin, Mirtazapine, Nortriptyline, Olanzapine, Olopatadine, Orphenadrine, Paliperidone, Phenindamine, Pizotifen, Prochlorperazine, Promazine, Promethazine, Propiomazine, Quetiapine, Risperidone, Rupatadine, Terfenadine, Tesmilifene, Thonzylamine, Trazodone, Trimipramine, Tripelennamine, Triprolidine, Ziprasidone, Zuclopenthixol
2Histamine H1 receptor inverse agonistsEsmirtazapine, Hydroxyzine, Perospirone, Pheniramine
3Histamine H1 receptor agonistsBetahistine, Histamine, Tolazoline
4Histamine H1 receptor inhibitorsEscitalopram, Levocetirizine, Paroxetine
5Histamine H1 receptor bindersCitalopram
Interacting GroupInteracting Drugs
Loxapine is a Histamine H2 receptor binder
1Histamine H2 receptor agonistsBetazole, Histamine, Tolazoline
2Histamine H2 receptor antagonistsAsenapine, Cimetidine, Doxepin, Epinastine, Famotidine, Methantheline, Metiamide, Nizatidine, Olopatadine, Promethazine, Ranitidine, Roxatidine acetate
3Histamine H2 receptor blockersAmitriptyline
4Histamine H2 receptor inhibitorsAzelastine
5Histamine H2 receptor ligandsAripiprazole
Interacting GroupInteracting Drugs
Loxapine is a Histamine H4 receptor binder
1Histamine H4 receptor antagonistsClozapine
2Histamine H4 receptor agonistsHistamine
3Histamine H4 receptor bindersAmitriptyline, Amoxapine, Chlorpromazine, Doxepin, Mianserin
4Histamine H4 receptor inverse agonistsPheniramine
5Histamine H4 receptor ligandsAripiprazole
Interacting GroupInteracting Drugs
Loxapine is a Sodium-dependent serotonin transporter binder
1Sodium-dependent serotonin transporter inhibitors4-Methoxyamphetamine, Amitriptyline, Amoxapine, Benzatropine, Butriptyline, Chlorpheniramine, Citalopram, Clomipramine, Cocaine, Cyclobenzaprine, Desipramine, Desvenlafaxine, Dexfenfluramine, Dexmethylphenidate, Dextromethorphan, Dopamine, Dosulepin, Doxepin, Duloxetine, Escitalopram, Etoperidone, Fenfluramine, Fluoxetine, Fluvoxamine, Imipramine, Levomilnacipran, Lumateperone, Mazindol, Mianserin, Milnacipran, Minaprine, Mirtazapine, Nefazodone, Nortriptyline, Paroxetine, Phentermine, Procaine, Protriptyline, Pseudoephedrine, Sertraline, Sibutramine, Tapentadol, Tegaserod, Tramadol, Trazodone, Trimipramine, Venlafaxine, Vilazodone, Vortioxetine
2Sodium-dependent serotonin transporter bindersAmphetamine, Atomoxetine, Sertraline
3Sodium-dependent serotonin transporter negative modulatorsEphedra sinica root, Metamfetamine, Midomafetamine, MMDA
4Sodium-dependent serotonin transporter substratesFenfluramine, Mirtazapine, Tegaserod
5Sodium-dependent serotonin transporter bindingsMeperidine
6Sodium-dependent serotonin transporter antagonistsButriptyline, Lorpiprazole, Zotepine
7Sodium-dependent serotonin transporter modulatorsAripiprazole
Interacting GroupInteracting Drugs
Loxapine is a Sodium-dependent noradrenaline transporter binder
1Sodium-dependent noradrenaline transporter inhibitorsAmitriptyline, Amoxapine, Atomoxetine, Benzatropine, Bupropion, Chlorpheniramine, Clomipramine, Cocaine, Cyclobenzaprine, Desipramine, Desvenlafaxine, Dexmethylphenidate, Dextromethorphan, Diethylpropion, Dopamine, Dosulepin, Doxepin, Duloxetine, Escitalopram, Etoperidone, Ginkgo biloba, Imipramine, Ketamine, Levomilnacipran, Maprotiline, Mazindol, Meperidine, Methylphenidate, Mianserin, Milnacipran, Nefazodone, Netarsudil, Nortriptyline, Orphenadrine, Paroxetine, Phenmetrazine, Phentermine, Procaine, Protriptyline, Pseudoephedrine, Rauwolfia serpentina root, Reboxetine, Sertraline, Sibutramine, Tapentadol, Tramadol, Trimipramine, Venlafaxine, Viloxazine
2Sodium-dependent noradrenaline transporter partial agonistsGuanadrel
3Sodium-dependent noradrenaline transporter inducersDebrisoquine, Guanethidine
4Sodium-dependent noradrenaline transporter negative modulatorsDextroamphetamine, Ephedra sinica root, Metamfetamine, Midomafetamine, MMDA, Phendimetrazine
5Sodium-dependent noradrenaline transporter inverse agonistsEphedrine
6Sodium-dependent noradrenaline transporter substratesDroxidopa, Iobenguane, Iobenguane sulfate I-123, Norepinephrine, Nortriptyline
7Sodium-dependent noradrenaline transporter stimulatorsAmphetamine
8Sodium-dependent noradrenaline transporter blockersVortioxetine
9Sodium-dependent noradrenaline transporter antagonistsZotepine
Interacting GroupInteracting Drugs
Loxapine is a Sodium-dependent dopamine transporter binder
1Sodium-dependent dopamine transporter inhibitors4-Methoxyamphetamine, Armodafinil, Benzatropine, Benzphetamine, Bupropion, Chloroprocaine, Chlorpheniramine, Cocaine, Desvenlafaxine, Dexmethylphenidate, Diethylpropion, Diphenylpyraline, Duloxetine, Escitalopram, Etoperidone, Fencamfamin, Imipramine, Mazindol, Meperidine, Methylphenidate, Modafinil, Nefazodone, Phenmetrazine, Phentermine, Procaine, Pseudoephedrine, Sertraline, Sibutramine, Trimipramine, Venlafaxine
2Sodium-dependent dopamine transporter negative modulatorsAmphetamine, Dextroamphetamine, Ephedra sinica root, Metamfetamine, Midomafetamine, MMDA
3Sodium-dependent dopamine transporter bindersAmoxapine, Mianserin, Sertraline
4Sodium-dependent dopamine transporter inducersDopamine
5Sodium-dependent dopamine transporter antagonistsArmodafinil
6Sodium-dependent dopamine transporter modulatorsAripiprazole