Showing BioInteractions for Loxapine (DB00408)
BioInteractor utilizes data on drug-target, -enzyme and -transporter associations to provide insight on drug-drug interactions. It allows you to identify, for instance, which drugs act similarly on the same target. Such drugs may have additive pharmacodynamic effects if given concomitantly. Conversely, two drugs may antagonize the beneficial effects of each other by having opposite actions on a specific drug target. BioInteractor uses ranked drug-enzyme association information to predict enzyme-mediated drug interactions that may be clinically relevant.
Interacting Group | Interacting Drugs | |
---|---|---|
Loxapine is a Dopamine D1 receptor antagonist | ||
1 | Dopamine D1 receptor antagonists | Acepromazine, Amoxapine, Aripiprazole, Asenapine, Carphenazine, Chlorpromazine, Chlorprothixene, Clozapine, Flupentixol, Fluphenazine, Haloperidol, Iloperidone, Lisuride, Methotrimeprazine, Methylergometrine, Olanzapine, Paliperidone, Periciazine, Perphenazine, Pipamperone, Pipotiazine, Quetiapine, Risperidone, Tetrahydropalmatine, Thioproperazine, Thioridazine, Thiothixene, Triflupromazine, Ziprasidone, Zuclopenthixol |
2 | Dopamine D1 receptor agonists | Apomorphine, Bromocriptine, Cabergoline, Dopamine, Fenoldopam, Levodopa, Minaprine, Pergolide, Rotigotine |
3 | Dopamine D1 receptor partial agonists | Aripiprazole, Phenylpropanolamine |
4 | Dopamine D1 receptor ligands | Aripiprazole |
Interacting Group | Interacting Drugs | |
---|---|---|
Loxapine is a 5-hydroxytryptamine receptor 1B binder | ||
1 | 5-hydroxytryptamine receptor 1B agonists | Almotriptan, Apomorphine, Bromocriptine, Cabergoline, Dihydroergotamine, Eletriptan, Ergotamine, Frovatriptan, Lisuride, Naratriptan, Oxymetazoline, Pergolide, Rizatriptan, Sumatriptan, Zolmitriptan |
2 | 5-hydroxytryptamine receptor 1B antagonists | Amoxapine, Aripiprazole, Asenapine, Clozapine, Penbutolol, Pizotifen, Ziprasidone |
3 | 5-hydroxytryptamine receptor 1B ligands | Aripiprazole, Quetiapine |
4 | 5-hydroxytryptamine receptor 1B partial agonists | Vortioxetine, Yohimbine |
5 | 5-hydroxytryptamine receptor 1B binders | Amitriptyline, Methysergide |
Interacting Group | Interacting Drugs | |
---|---|---|
Loxapine is a 5-hydroxytryptamine receptor 1D binder | ||
1 | 5-hydroxytryptamine receptor 1D agonists | Almotriptan, Apomorphine, Bromocriptine, Cabergoline, Dihydroergotamine, Eletriptan, Ergotamine, Fenfluramine, Frovatriptan, Lisuride, Lofexidine, Naratriptan, Oxymetazoline, Pergolide, Rizatriptan, Sumatriptan, Zolmitriptan |
2 | 5-hydroxytryptamine receptor 1D antagonists | Aripiprazole, Clozapine, Paliperidone, Pizotifen, Risperidone, Ziprasidone |
3 | 5-hydroxytryptamine receptor 1D ligands | Aripiprazole, Quetiapine |
4 | 5-hydroxytryptamine receptor 1D partial agonists | Yohimbine |
5 | 5-hydroxytryptamine receptor 1D binders | Amitriptyline, Trimipramine |
Interacting Group | Interacting Drugs | |
---|---|---|
Loxapine is a 5-hydroxytryptamine receptor 1E binder | ||
1 | 5-hydroxytryptamine receptor 1E antagonists | Aripiprazole, Clozapine, Ziprasidone |
2 | 5-hydroxytryptamine receptor 1E ligands | Aripiprazole, Quetiapine |
3 | 5-hydroxytryptamine receptor 1E binders | Methysergide |
4 | 5-hydroxytryptamine receptor 1E agonists | Zolmitriptan |
Interacting Group | Interacting Drugs | |
---|---|---|
Loxapine is a 5-hydroxytryptamine receptor 3A binder | ||
1 | 5-hydroxytryptamine receptor 3A antagonists | Alosetron, Amoxapine, Aripiprazole, Cannabidiol, Clozapine, Dolasetron, Granisetron, Memantine, Methadone, Metoclopramide, Olanzapine, Ondansetron, Palonosetron, Procaine, Ramosetron, Rocuronium, Tropisetron, Tubocurarine, Vortioxetine |
2 | 5-hydroxytryptamine receptor 3A agonists | Cisapride |
3 | 5-hydroxytryptamine receptor 3A ligands | Quetiapine |
4 | 5-hydroxytryptamine receptor 3A binders | Trimipramine |
5 | 5-hydroxytryptamine receptor 3A inhibitors | Lamotrigine |
6 | 5-hydroxytryptamine receptor 3A potentiators | Ketamine |
7 | 5-hydroxytryptamine receptor 3A negative modulators | Bupropion |
Interacting Group | Interacting Drugs | |
---|---|---|
Loxapine is a 5-hydroxytryptamine receptor 5A binder | ||
1 | 5-hydroxytryptamine receptor 5A antagonists | Asenapine, Ziprasidone |
2 | 5-hydroxytryptamine receptor 5A ligands | Aripiprazole |
Interacting Group | Interacting Drugs | |
---|---|---|
Loxapine is a 5-hydroxytryptamine receptor 6 binder | ||
1 | 5-hydroxytryptamine receptor 6 antagonists | Amitriptyline, Amoxapine, Aripiprazole, Asenapine, Clozapine, Cyclobenzaprine, Iloperidone, Olanzapine, Quetiapine, Sertindole, Ziprasidone, Zotepine |
2 | 5-hydroxytryptamine receptor 6 binders | Chlorpromazine, Doxepin, Imipramine, Mianserin |
Interacting Group | Interacting Drugs | |
---|---|---|
Loxapine is a 5-hydroxytryptamine receptor 7 binder | ||
1 | 5-hydroxytryptamine receptor 7 antagonists | Amisulpride, Amitriptyline, Amoxapine, Aripiprazole, Asenapine, Bromocriptine, Cabergoline, Clozapine, Cyclobenzaprine, Epinastine, Iloperidone, Imipramine, Lurasidone, Maprotiline, Methysergide, Mianserin, Risperidone, SB-269970, Vortioxetine, Ziprasidone, Zotepine |
2 | 5-hydroxytryptamine receptor 7 partial agonists | Aripiprazole |
3 | 5-hydroxytryptamine receptor 7 ligands | Quetiapine |
4 | 5-hydroxytryptamine receptor 7 binders | Chlorpromazine, Dopamine |
5 | 5-hydroxytryptamine receptor 7 agonists | Lofexidine, Zolmitriptan |
Interacting Group | Interacting Drugs | |
---|---|---|
Loxapine is a Alpha-1B adrenergic receptor binder | ||
1 | Alpha-1B adrenergic receptor antagonists | Acepromazine, Alfuzosin, Amitriptyline, Aripiprazole, Aripiprazole lauroxil, Brexpiprazole, Bromocriptine, Carvedilol, Chlorpromazine, Clozapine, Dapiprazole, Dextroamphetamine, Doxepin, Dronedarone, Imipramine, Methotrimeprazine, Nicardipine, Nortriptyline, Olanzapine, Paliperidone, Periciazine, Phenoxybenzamine, Phentolamine, Pizotifen, Prazosin, Quinidine, Risperidone, Silodosin, Tamsulosin, Terazosin, Thioproperazine, Thioridazine, Trimipramine, Verapamil, Ziprasidone |
2 | Alpha-1B adrenergic receptor partial agonists | Cirazoline, Ergotamine, Modafinil |
3 | Alpha-1B adrenergic receptor agonists | Bromocriptine, Clonidine, Droxidopa, Epinephrine, Methoxamine, Midodrine, Norepinephrine, Oxymetazoline, Pergolide, Phendimetrazine, Phenylephrine, Racepinephrine, Xylometazoline |
4 | Alpha-1B adrenergic receptor binders | Cabergoline |
5 | Alpha-1B adrenergic receptor inhibitors | Fenoldopam |
Interacting Group | Interacting Drugs | |
---|---|---|
Loxapine is a Alpha-2B adrenergic receptor binder | ||
1 | Alpha-2B adrenergic receptor antagonists | Aripiprazole, Asenapine, Cabergoline, Carvedilol, Celiprolol, Clozapine, Dronedarone, Fenoldopam, Methotrimeprazine, Mianserin, Paliperidone, Phenoxybenzamine, Pizotifen, Quetiapine, Risperidone, Rotigotine, Yohimbine, Ziprasidone |
2 | Alpha-2B adrenergic receptor agonists | Apomorphine, Apraclonidine, Brimonidine, Bromocriptine, Clonidine, Droxidopa, Ephedra sinica root, Epinephrine, Etomidate, Metamfetamine, Norepinephrine, Oxymetazoline, Racepinephrine, Xylometazoline |
3 | Alpha-2B adrenergic receptor ligands | Aripiprazole |
4 | Alpha-2B adrenergic receptor binders | Guanabenz, Guanfacine, Prazosin, Tolazoline |
Interacting Group | Interacting Drugs | |
---|---|---|
Loxapine is a Alpha-2C adrenergic receptor binder | ||
1 | Alpha-2C adrenergic receptor antagonists | Aripiprazole, Asenapine, Brexpiprazole, Cabergoline, Carvedilol, Celiprolol, Clozapine, Dronedarone, Fenoldopam, Iloperidone, Lurasidone, Methotrimeprazine, Mianserin, Phenoxybenzamine, Pizotifen, Quetiapine, Risperidone, Yohimbine, Ziprasidone |
2 | Alpha-2C adrenergic receptor agonists | Agmatine, Apomorphine, Brimonidine, Bromocriptine, Clonidine, Droxidopa, Ephedra sinica root, Metamfetamine, Norepinephrine, Oxymetazoline, Paliperidone, Racepinephrine, Xylometazoline |
3 | Alpha-2C adrenergic receptor binders | Tolazoline |
Interacting Group | Interacting Drugs | |
---|---|---|
Loxapine is a Muscarinic acetylcholine receptor M4 binder | ||
1 | Muscarinic acetylcholine receptor M4 antagonists | Aclidinium, Atropine, Benzquinamide, Brompheniramine, Chlorprothixene, Clozapine, Darifenacin, Desipramine, Dosulepin, Doxepin, Fesoterodine, Hexocyclium, Homatropine, Homatropine methylbromide, Hyoscyamine, Imipramine, Isopropamide, Maprotiline, Methotrimeprazine, Nicardipine, Olanzapine, Procyclidine, Promethazine, Propiverine, Rociverine, Scopolamine, Solifenacin, Thonzylamine, Tolterodine, Trihexyphenidyl, Trimebutine, Tropicamide, Umeclidinium, Ziprasidone |
2 | Muscarinic acetylcholine receptor M4 ligands | Aripiprazole, Quetiapine |
3 | Muscarinic acetylcholine receptor M4 binders | Terfenadine |
4 | Muscarinic acetylcholine receptor M4 agonists | Carbamoylcholine, Methacholine |
5 | Muscarinic acetylcholine receptor M4 partial agonists | Pilocarpine |
Interacting Group | Interacting Drugs | |
---|---|---|
Loxapine is a Muscarinic acetylcholine receptor M5 binder | ||
1 | Muscarinic acetylcholine receptor M5 antagonists | Aclidinium, Atropine, Benzquinamide, Brompheniramine, Chlorprothixene, Clozapine, Darifenacin, Desipramine, Dosulepin, Doxepin, Fesoterodine, Homatropine, Homatropine methylbromide, Imipramine, Maprotiline, Methotrimeprazine, Nicardipine, Promethazine, Rociverine, Scopolamine, Solifenacin, Thonzylamine, Tolterodine, Trihexyphenidyl, Umeclidinium, Ziprasidone |
2 | Muscarinic acetylcholine receptor M5 ligands | Aripiprazole, Quetiapine |
3 | Muscarinic acetylcholine receptor M5 binders | Terfenadine |
4 | Muscarinic acetylcholine receptor M5 agonists | Methacholine |
Interacting Group | Interacting Drugs | |
---|---|---|
Loxapine is a D(1) dopamine receptor binder | ||
1 | D(1) dopamine receptor inhibitors | Chlorpromazine, Lamotrigine |
2 | D(1) dopamine receptor binders | Cinnarizine, Imipramine, Mianserin, Trimipramine |
3 | D(1) dopamine receptor agonists | Cabergoline, Dopamine, Ergotamine, Pipradrol, Quinagolide |
4 | D(1) dopamine receptor antagonists | Olanzapine, Zotepine |
5 | D(1) dopamine receptor partial agonists | Dihydro-alpha-ergocryptine |
Interacting Group | Interacting Drugs | |
---|---|---|
Loxapine is a Dopamine D3 receptor binder | ||
1 | Dopamine D3 receptor antagonists | Amisulpride, Amoxapine, Aripiprazole, AS-8112, Asenapine, Blonanserin, Buspirone, Chlorprothixene, Clozapine, Domperidone, Flupentixol, Iloperidone, Methotrimeprazine, Olanzapine, Paliperidone, Pimozide, Remoxipride, Sulpiride, Yohimbine, Ziprasidone |
2 | Dopamine D3 receptor agonists | Apomorphine, Bromocriptine, Cabergoline, Captodiame, Cariprazine, Dopamine, Levodopa, Lisuride, Pergolide, Pramipexole, Ropinirole, Rotigotine, Tianeptine |
3 | Dopamine D3 receptor partial agonists | Aripiprazole, Cariprazine, Dihydro-alpha-ergocryptine |
4 | Dopamine D3 receptor inverse agonists | Haloperidol |
5 | Dopamine D3 receptor ligands | Quetiapine, Sarizotan |
6 | Dopamine D3 receptor inhibitors | Chlorpromazine |
7 | Dopamine D3 receptor binders | Mianserin |
8 | Dopamine D3 receptor blockers | Tiapride |
Interacting Group | Interacting Drugs | |
---|---|---|
Loxapine is a Dopamine D4 receptor binder | ||
1 | Dopamine D4 receptor antagonists | Amoxapine, Aripiprazole, Asenapine, Bromocriptine, Buspirone, Clozapine, Flibanserin, Flupentixol, Iloperidone, Methotrimeprazine, Olanzapine, Paliperidone, Perospirone, Pipamperone, Remoxipride, Sulpiride, Ziprasidone |
2 | Dopamine D4 receptor agonists | Apomorphine, Cabergoline, Dopamine, Flibanserin, Levodopa, Lisuride, Pergolide, Pramipexole, Ropinirole, Rotigotine |
3 | Dopamine D4 receptor partial agonists | Aripiprazole |
4 | Dopamine D4 receptor ligands | Quetiapine |
5 | Dopamine D4 receptor binders | Chlorpromazine |
Interacting Group | Interacting Drugs | |
---|---|---|
Loxapine is a Dopamine D5 receptor binder | ||
1 | Dopamine D5 receptor agonists | Apomorphine, Bromocriptine, Cabergoline, Dopamine, Fenoldopam, Levodopa, Pergolide, Rotigotine |
2 | Dopamine D5 receptor antagonists | Aripiprazole, Carphenazine, Lisuride, Methotrimeprazine, Olanzapine, Ziprasidone, Zuclopenthixol |
3 | Dopamine D5 receptor partial agonists | Aripiprazole |
4 | Dopamine D5 receptor ligands | Aripiprazole, Quetiapine |
5 | Dopamine D5 receptor inhibitors | Chlorpromazine |
Interacting Group | Interacting Drugs | |
---|---|---|
Loxapine is a Histamine H2 receptor binder | ||
1 | Histamine H2 receptor agonists | Betazole, Histamine, Tolazoline |
2 | Histamine H2 receptor antagonists | Asenapine, Cimetidine, Doxepin, Epinastine, Famotidine, Methantheline, Metiamide, Nizatidine, Olopatadine, Promethazine, Ranitidine, Roxatidine acetate |
3 | Histamine H2 receptor blockers | Amitriptyline |
4 | Histamine H2 receptor inhibitors | Azelastine |
5 | Histamine H2 receptor ligands | Aripiprazole |
Interacting Group | Interacting Drugs | |
---|---|---|
Loxapine is a Histamine H4 receptor binder | ||
1 | Histamine H4 receptor antagonists | Clozapine |
2 | Histamine H4 receptor agonists | Histamine |
3 | Histamine H4 receptor binders | Amitriptyline, Amoxapine, Chlorpromazine, Doxepin, Mianserin |
4 | Histamine H4 receptor inverse agonists | Pheniramine |
5 | Histamine H4 receptor ligands | Aripiprazole |
Interacting Group | Interacting Drugs | |
---|---|---|
Loxapine is a Sodium-dependent dopamine transporter binder | ||
1 | Sodium-dependent dopamine transporter inhibitors | 4-Methoxyamphetamine, Armodafinil, Benzatropine, Benzphetamine, Bupropion, Chloroprocaine, Chlorpheniramine, Cocaine, Desvenlafaxine, Dexmethylphenidate, Diethylpropion, Diphenylpyraline, Duloxetine, Escitalopram, Etoperidone, Fencamfamin, Imipramine, Mazindol, Meperidine, Methylphenidate, Modafinil, Nefazodone, Phenmetrazine, Phentermine, Procaine, Pseudoephedrine, Sertraline, Sibutramine, Trimipramine, Venlafaxine |
2 | Sodium-dependent dopamine transporter negative modulators | Amphetamine, Dextroamphetamine, Ephedra sinica root, Metamfetamine, Midomafetamine, MMDA |
3 | Sodium-dependent dopamine transporter binders | Amoxapine, Mianserin, Sertraline |
4 | Sodium-dependent dopamine transporter inducers | Dopamine |
5 | Sodium-dependent dopamine transporter antagonists | Armodafinil |
6 | Sodium-dependent dopamine transporter modulators | Aripiprazole |