Showing BioInteractions for Rizatriptan (DB00953)

BioInteractor utilizes data on drug-target, -enzyme and -transporter associations to provide insight on drug-drug interactions. It allows you to identify, for instance, which drugs act similarly on the same target. Such drugs may have additive pharmacodynamic effects if given concomitantly. Conversely, two drugs may antagonize the beneficial effects of each other by having opposite actions on a specific drug target. BioInteractor uses ranked drug-enzyme association information to predict enzyme-mediated drug interactions that may be clinically relevant.
Interacting GroupInteracting Drugs
Rizatriptan is a 5-hydroxytryptamine receptor 1D agonist
15-hydroxytryptamine receptor 1D agonistsAlmotriptan, Apomorphine, Bromocriptine, Cabergoline, Dihydroergotamine, Eletriptan, Ergotamine, Fenfluramine, Frovatriptan, Lisuride, Lofexidine, Naratriptan, Oxymetazoline, Pergolide, Sumatriptan, Zolmitriptan
25-hydroxytryptamine receptor 1D antagonistsAripiprazole, Clozapine, Paliperidone, Pizotifen, Risperidone, Ziprasidone
35-hydroxytryptamine receptor 1D ligandsAripiprazole, Quetiapine
45-hydroxytryptamine receptor 1D partial agonistsYohimbine
55-hydroxytryptamine receptor 1D bindersAmitriptyline, Loxapine, Trimipramine
Interacting GroupInteracting Drugs
Rizatriptan is a 5-hydroxytryptamine receptor 1B agonist
15-hydroxytryptamine receptor 1B agonistsAlmotriptan, Apomorphine, Bromocriptine, Cabergoline, Dihydroergotamine, Eletriptan, Ergotamine, Frovatriptan, Lisuride, Naratriptan, Oxymetazoline, Pergolide, Sumatriptan, Zolmitriptan
25-hydroxytryptamine receptor 1B antagonistsAmoxapine, Aripiprazole, Asenapine, Clozapine, Penbutolol, Pizotifen, Ziprasidone
35-hydroxytryptamine receptor 1B ligandsAripiprazole, Quetiapine
45-hydroxytryptamine receptor 1B partial agonistsVortioxetine, Yohimbine
55-hydroxytryptamine receptor 1B bindersAmitriptyline, Loxapine, Methysergide
Interacting GroupInteracting Drugs
Rizatriptan is a 5-hydroxytryptamine receptor 1F agonist
15-hydroxytryptamine receptor 1F agonistsEletriptan, Ergotamine, Lasmiditan, Naratriptan, Sumatriptan, Zolmitriptan
25-hydroxytryptamine receptor 1F bindersMethysergide, Mianserin