Showing BioInteractions for Chlorprothixene (DB01239)

BioInteractor utilizes data on drug-target, -enzyme and -transporter associations to provide insight on drug-drug interactions. It allows you to identify, for instance, which drugs act similarly on the same target. Such drugs may have additive pharmacodynamic effects if given concomitantly. Conversely, two drugs may antagonize the beneficial effects of each other by having opposite actions on a specific drug target. BioInteractor uses ranked drug-enzyme association information to predict enzyme-mediated drug interactions that may be clinically relevant.
Interacting GroupInteracting Drugs
Chlorprothixene is a Dopamine D1 receptor antagonist
1Dopamine D1 receptor antagonistsAcepromazine, Amoxapine, Aripiprazole, Asenapine, Carphenazine, Chlorpromazine, Clozapine, Flupentixol, Fluphenazine, Haloperidol, Iloperidone, Lisuride, Loxapine, Methotrimeprazine, Methylergometrine, Olanzapine, Paliperidone, Periciazine, Perphenazine, Pipamperone, Pipotiazine, Quetiapine, Risperidone, Tetrahydropalmatine, Thioproperazine, Thioridazine, Thiothixene, Triflupromazine, Ziprasidone, Zuclopenthixol
2Dopamine D1 receptor agonistsApomorphine, Bromocriptine, Cabergoline, Dopamine, Fenoldopam, Levodopa, Minaprine, Pergolide, Rotigotine
3Dopamine D1 receptor partial agonistsAripiprazole, Phenylpropanolamine
4Dopamine D1 receptor ligandsAripiprazole
Interacting GroupInteracting Drugs
Chlorprothixene is a Dopamine D2 receptor antagonist
1Dopamine D2 receptor agonistsAmantadine, Apomorphine, Brexpiprazole, Bromocriptine, Cabergoline, Cariprazine, Dihydro-alpha-ergocryptine, Dopamine, Ergotamine, Ketamine, Lamotrigine, Levodopa, Lisuride, Memantine, Minaprine, Pergolide, Pramipexole, Quinagolide, Ropinirole, Rotigotine
2Dopamine D2 receptor antagonistsAcepromazine, Acetophenazine, Alizapride, Amisulpride, Amoxapine, Aripiprazole, AS-8112, Asenapine, Blonanserin, Bromopride, Buspirone, Carphenazine, Chlorpromazine, Clozapine, Domperidone, Droperidol, Etoperidone, Flupentixol, Fluphenazine, Fluspirilene, Haloperidol, Iloperidone, JNJ-37822681, Loxapine, Lurasidone, Melperone, Memantine, Mesoridazine, Methotrimeprazine, Metoclopramide, Mianserin, Molindone, Nortriptyline, Olanzapine, Paliperidone, Perospirone, Perphenazine, Pimozide, Pipamperone, Pipotiazine, Prochlorperazine, Promazine, Promethazine, Propiomazine, Quetiapine, Raclopride, Remoxipride, Risperidone, Sertindole, Sulpiride, Tetrahydropalmatine, Thiethylperazine, Thioproperazine, Thioridazine, Thiothixene, Trifluoperazine, Triflupromazine, YKP-1358, Yohimbine, Ziprasidone, Zotepine, Zuclopenthixol
3Dopamine D2 receptor partial agonistsAripiprazole, Aripiprazole lauroxil, Brexpiprazole, Cariprazine, Ketamine, Lumateperone, Sarizotan
4Dopamine D2 receptor inhibitorsEscitalopram, Lamotrigine, Tetrabenazine
5Dopamine D2 receptor bindersAmphetamine, Desipramine, Imipramine, Maprotiline
6Dopamine D2 receptor blockersTiapride
Interacting GroupInteracting Drugs
Chlorprothixene is a Dopamine D3 receptor antagonist
1Dopamine D3 receptor antagonistsAmisulpride, Amoxapine, Aripiprazole, AS-8112, Asenapine, Blonanserin, Buspirone, Clozapine, Domperidone, Flupentixol, Iloperidone, Methotrimeprazine, Olanzapine, Paliperidone, Pimozide, Remoxipride, Sulpiride, Yohimbine, Ziprasidone
2Dopamine D3 receptor agonistsApomorphine, Bromocriptine, Cabergoline, Captodiame, Cariprazine, Dopamine, Levodopa, Lisuride, Pergolide, Pramipexole, Ropinirole, Rotigotine, Tianeptine
3Dopamine D3 receptor partial agonistsAripiprazole, Cariprazine, Dihydro-alpha-ergocryptine
4Dopamine D3 receptor inverse agonistsHaloperidol
5Dopamine D3 receptor ligandsQuetiapine, Sarizotan
6Dopamine D3 receptor inhibitorsChlorpromazine
7Dopamine D3 receptor bindersLoxapine, Mianserin
8Dopamine D3 receptor blockersTiapride
Interacting GroupInteracting Drugs
Chlorprothixene is a 5-hydroxytryptamine receptor 2A antagonist
15-hydroxytryptamine receptor 2A antagonistsAcepromazine, Amisulpride, Amitriptyline, Amoxapine, Amperozide, Aripiprazole, Aripiprazole lauroxil, Asenapine, Blonanserin, Brexpiprazole, Butriptyline, Cariprazine, Chlorpromazine, Cinitapride, Clomipramine, Clozapine, Cyclobenzaprine, Cyproheptadine, Deramciclane, Desipramine, Dosulepin, Doxepin, Epinastine, Etoperidone, Flibanserin, Flupentixol, Fluspirilene, Iloperidone, Imipramine, Lorpiprazole, Loxapine, Lumateperone, Lurasidone, Mesoridazine, Methotrimeprazine, Methysergide, Mianserin, Minaprine, Mirtazapine, Molindone, Nefazodone, Nortriptyline, Olanzapine, Paliperidone, Pipotiazine, Pizotifen, Promazine, Propiomazine, Quetiapine, Risperidone, Sertindole, Tegaserod, Thioridazine, Thiothixene, Trazodone, Yohimbine, Ziprasidone, Zotepine, Zuclopenthixol
25-hydroxytryptamine receptor 2A partial agonists4-Bromo-2,5-dimethoxyphenethylamine, Aripiprazole
35-hydroxytryptamine receptor 2A agonists2,5-Dimethoxy-4-ethylthioamphetamine, 5-methoxy-N,N-dimethyltryptamine, Apomorphine, Bromocriptine, Cabergoline, Cannabidiol, Cisapride, Ergotamine, Fenfluramine, Lisuride, Midomafetamine, MMDA, N-(2-hydroxybenzyl)-2,5-dimethoxy-4-cyanophenylethylamine, Paroxetine, Pergolide, Pipamperone, Trimipramine, Zolmitriptan
45-hydroxytryptamine receptor 2A inducersDonepezil
55-hydroxytryptamine receptor 2A inverse agonistsKetanserin, Perospirone, Pimavanserin, Ritanserin, Sarpogrelate
65-hydroxytryptamine receptor 2A bindersMaprotiline
75-hydroxytryptamine receptor 2A inhibitorsEscitalopram, Lamotrigine
Interacting GroupInteracting Drugs
Chlorprothixene is a Histamine H1 receptor antagonist
1Histamine H1 receptor antagonistsAceprometazine, Acrivastine, Alcaftadine, Alimemazine, Amitriptyline, Amoxapine, Antazoline, Aripiprazole, Aripiprazole lauroxil, Asenapine, Astemizole, Azatadine, Azelastine, Benzatropine, Benzquinamide, Bepotastine, Bilastine, Bromodiphenhydramine, Brompheniramine, Buclizine, Butriptyline, Carbinoxamine, Cariprazine, Cetirizine, Chlorcyclizine, Chloropyramine, Chlorpheniramine, Chlorpromazine, Cinnarizine, Clemastine, Clofedanol, Clozapine, Cyclizine, Cyproheptadine, Desipramine, Desloratadine, Dexbrompheniramine, Dexchlorpheniramine maleate, Dimenhydrinate, Dimetindene, Diphenhydramine, Diphenylpyraline, Dosulepin, Doxepin, Doxylamine, Emedastine, Epinastine, Fexofenadine, Flunarizine, Iloperidone, Imipramine, Isothipendyl, Ketotifen, Lamotrigine, Levocabastine, Levocetirizine, Loratadine, Lorpiprazole, Maprotiline, Meclizine, Mepyramine, Mequitazine, Methdilazine, Methotrimeprazine, Mianserin, Mirtazapine, Nortriptyline, Olanzapine, Olopatadine, Orphenadrine, Paliperidone, Phenindamine, Pizotifen, Prochlorperazine, Promazine, Promethazine, Propiomazine, Quetiapine, Risperidone, Rupatadine, Terfenadine, Tesmilifene, Thonzylamine, Trazodone, Trimipramine, Tripelennamine, Triprolidine, Ziprasidone, Zuclopenthixol
2Histamine H1 receptor inverse agonistsEsmirtazapine, Hydroxyzine, Perospirone, Pheniramine
3Histamine H1 receptor agonistsBetahistine, Histamine, Tolazoline
4Histamine H1 receptor inhibitorsEscitalopram, Levocetirizine, Paroxetine
5Histamine H1 receptor bindersCitalopram, Loxapine
Interacting GroupInteracting Drugs
Chlorprothixene is a Muscarinic acetylcholine receptor M1 antagonist
1Muscarinic acetylcholine receptor M1 agonistsCarbamoylcholine, Cevimeline, Methacholine, Metoclopramide, Minaprine, Pilocarpine, Pyrantel, Succinylcholine
2Muscarinic acetylcholine receptor M1 antagonistsAclidinium, Amoxapine, Anisotropine methylbromide, Atropine, Benzatropine, Benzquinamide, Biperiden, Brompheniramine, Buclizine, Chlorpromazine, Clidinium, Clozapine, Cocaine, Cyclopentolate, Cycrimine, Cyproheptadine, Darifenacin, Desipramine, Dicyclomine, Diphenidol, Disopyramide, Dosulepin, Doxepin, Fesoterodine, Flavoxate, Flupentixol, Glycopyrronium, Hexocyclium, Homatropine, Homatropine methylbromide, Hyoscyamine, Imidafenacin, Imipramine, Ipratropium, Maprotiline, Mepenzolate, Methantheline, Methotrimeprazine, Methscopolamine bromide, Nicardipine, Olanzapine, Oxybutynin, Oxyphencyclimine, Oxyphenonium, Pirenzepine, Pizotifen, Procyclidine, Profenamine, Promazine, Promethazine, Propantheline, Propiverine, Pyrantel, Quetiapine, Rociverine, Scopolamine, Solifenacin, Thonzylamine, Tiotropium, Tolterodine, Tramadol, Tridihexethyl, Triflupromazine, Trihexyphenidyl, Trimebutine, Tropicamide, Trospium, Umeclidinium, Ziprasidone
3Muscarinic acetylcholine receptor M1 weak inhibitorsBuclizine
4Muscarinic acetylcholine receptor M1 inhibitorsEscitalopram
5Muscarinic acetylcholine receptor M1 bindersLoxapine, Terfenadine
6Muscarinic acetylcholine receptor M1 ligandsAripiprazole
Interacting GroupInteracting Drugs
Chlorprothixene is a Muscarinic acetylcholine receptor M2 antagonist
1Muscarinic acetylcholine receptor M2 antagonistsAclidinium, Anisotropine methylbromide, Atropine, Benzquinamide, Brompheniramine, Butylscopolamine, Clozapine, Cocaine, Cryptenamine, Cyproheptadine, Darifenacin, Desipramine, Dicyclomine, Dimetindene, Diphenhydramine, Diphenidol, Disopyramide, Dosulepin, Doxacurium, Doxepin, Fesoterodine, Flavoxate, Gallamine triethiodide, Hexocyclium, Homatropine, Homatropine methylbromide, Hyoscyamine, Imidafenacin, Imipramine, Ipratropium, Maprotiline, Methotrimeprazine, Methscopolamine bromide, Metocurine, Mivacurium, Nicardipine, Olanzapine, Oxybutynin, Oxyphencyclimine, Pancuronium, Pipecuronium, Pizotifen, Procyclidine, Profenamine, Promethazine, Propiverine, Rapacuronium, Rociverine, Rocuronium, Scopolamine, Solifenacin, Thonzylamine, Tiotropium, Tolterodine, Tridihexethyl, Triflupromazine, Trihexyphenidyl, Trimebutine, Tropicamide, Umeclidinium, Ziprasidone
2Muscarinic acetylcholine receptor M2 agonistsBethanechol, Carbamoylcholine, Methacholine, Pilocarpine, Succinylcholine
3Muscarinic acetylcholine receptor M2 partial agonistsMivacurium
4Muscarinic acetylcholine receptor M2 ligandsAripiprazole, Quetiapine
5Muscarinic acetylcholine receptor M2 bindersGlycopyrronium, Loxapine, Terfenadine
Interacting GroupInteracting Drugs
Chlorprothixene is a Muscarinic acetylcholine receptor M3 antagonist
1Muscarinic acetylcholine receptor M3 antagonistsAclidinium, Anisotropine methylbromide, Atropine, Benzquinamide, Brompheniramine, Butylscopolamine, Chlorpromazine, Clozapine, Cyproheptadine, Darifenacin, Desipramine, Diphemanil, Diphenidol, Disopyramide, Dosulepin, Doxepin, Fesoterodine, Glycopyrronium, Hexocyclium, Homatropine, Homatropine methylbromide, Hyoscyamine, Imidafenacin, Imipramine, Ipratropium, Isopropamide, Maprotiline, Mepenzolate, Methotrimeprazine, Methscopolamine bromide, Mivacurium, Nicardipine, Olanzapine, Oxybutynin, Oxyphencyclimine, Pancuronium, Pipecuronium, Pizotifen, Procyclidine, Promethazine, Propiverine, Quetiapine, Rociverine, Scopolamine, Solifenacin, Terfenadine, Thonzylamine, Tiotropium, Tolterodine, Tramadol, Tridihexethyl, Trihexyphenidyl, Trimebutine, Tropicamide, Umeclidinium, Ziprasidone
2Muscarinic acetylcholine receptor M3 agonistsCarbamoylcholine, Cevimeline, Methacholine, Pilocarpine, Succinylcholine
3Muscarinic acetylcholine receptor M3 bindersLoxapine
4Muscarinic acetylcholine receptor M3 ligandsAripiprazole
Interacting GroupInteracting Drugs
Chlorprothixene is a Muscarinic acetylcholine receptor M4 antagonist
1Muscarinic acetylcholine receptor M4 antagonistsAclidinium, Atropine, Benzquinamide, Brompheniramine, Clozapine, Darifenacin, Desipramine, Dosulepin, Doxepin, Fesoterodine, Hexocyclium, Homatropine, Homatropine methylbromide, Hyoscyamine, Imipramine, Isopropamide, Maprotiline, Methotrimeprazine, Nicardipine, Olanzapine, Procyclidine, Promethazine, Propiverine, Rociverine, Scopolamine, Solifenacin, Thonzylamine, Tolterodine, Trihexyphenidyl, Trimebutine, Tropicamide, Umeclidinium, Ziprasidone
2Muscarinic acetylcholine receptor M4 ligandsAripiprazole, Quetiapine
3Muscarinic acetylcholine receptor M4 bindersLoxapine, Terfenadine
4Muscarinic acetylcholine receptor M4 agonistsCarbamoylcholine, Methacholine
5Muscarinic acetylcholine receptor M4 partial agonistsPilocarpine
Interacting GroupInteracting Drugs
Chlorprothixene is a Muscarinic acetylcholine receptor M5 antagonist
1Muscarinic acetylcholine receptor M5 antagonistsAclidinium, Atropine, Benzquinamide, Brompheniramine, Clozapine, Darifenacin, Desipramine, Dosulepin, Doxepin, Fesoterodine, Homatropine, Homatropine methylbromide, Imipramine, Maprotiline, Methotrimeprazine, Nicardipine, Promethazine, Rociverine, Scopolamine, Solifenacin, Thonzylamine, Tolterodine, Trihexyphenidyl, Umeclidinium, Ziprasidone
2Muscarinic acetylcholine receptor M5 ligandsAripiprazole, Quetiapine
3Muscarinic acetylcholine receptor M5 bindersLoxapine, Terfenadine
4Muscarinic acetylcholine receptor M5 agonistsMethacholine
Interacting GroupInteracting Drugs
Chlorprothixene is a Serotonin Receptors inhibitor
1Serotonin Receptors antagonistsDihydroergocornine, Dihydroergocristine, Ergoloid mesylate, Setiptiline, Tiapride
2Serotonin Receptors agonistsDihydroergocornine, Ergoloid mesylate
3Serotonin Receptors inhibitorsGilteritinib
Interacting GroupInteracting Drugs
Chlorprothixene is a P-glycoprotein 1 inhibitor
1P-glycoprotein 1 inducersAcetylsalicylic acid, Aldosterone, Amiodarone, Amprenavir, Apalutamide, Atazanavir, Beclomethasone dipropionate, Betamethasone phosphate, Carbamazepine, Cholic Acid, Cimetidine, Clotrimazole, Colchicine, Cortisone acetate, Darunavir, Daunorubicin, Dexamethasone, Dexamethasone acetate, Diclofenac, Digoxin, Doxorubicin, Estriol, Estrone, Etravirine, Hydrocortisone, Indinavir, Ivermectin, Levothyroxine, Liothyronine, Liotrix, Lopinavir, Lumacaftor, Methylprednisolone, Mifepristone, Mitoxantrone, Nefazodone, Nelfinavir, Nifedipine, Phenobarbital, Platelet Activating Factor, Prednisolone phosphate, Prednisone, Progesterone, Propofol, Reserpine, Rifabutin, Rifampicin, Ritonavir, Saquinavir, Sirolimus, Spironolactone, St. John's Wort, Streptozocin, Tacrolimus, Tamoxifen, Tesmilifene, Tipranavir, Trazodone, Vinblastine, Vincristine
2P-glycoprotein 1 inhibitorsAbemaciclib, Acetaminophen, Afatinib, Alectinib, Alfentanil, Alpelisib, Amiodarone, Amlodipine, Amodiaquine, Amsacrine, Arsenic trioxide, Astemizole, Asunaprevir, Atazanavir, Atorvastatin, Atovaquone, Axitinib, Azelastine, Azithromycin, Benzocaine, Bepridil, Berotralstat, Bicalutamide, Biricodar, Bisoprolol, Boceprevir, Bromocriptine, Buprenorphine, Buspirone, Cabazitaxel, Canagliflozin, Candesartan, Candesartan cilexetil, Captopril, Carfilzomib, Carvedilol, Caspofungin, Ceftriaxone, Cethromycin, Cetirizine, Chloroquine, Chlorpromazine, Cholesterol, Cilazapril, Citalopram, Clarithromycin, Clofazimine, Clomipramine, Clotrimazole, Cobicistat, Colforsin, Concanamycin A, Conivaptan, Crizotinib, Curcumin, Cyclosporine, Daclatasvir, Dacomitinib, Dactinomycin, Darunavir, Dasatinib, Daunorubicin, Desipramine, Desloratadine, Desmethylsertraline, Dexamethasone, Dexamethasone acetate, Dexniguldipine, Dexverapamil, Digoxin, Dihydroergotamine, Diltiazem, Dipyridamole, Dofequidar, Dovitinib, Doxazosin, Doxorubicin, Dronabinol, Dronedarone, Duloxetine, Elacridar, Elagolix, Elbasvir, Elexacaftor, Emopamil, Enalapril, Enasidenib, Entrectinib, Enzalutamide, Erdafitinib, Ergometrine, Ergotamine, Erlotinib, Erythromycin, Esomeprazole, Estramustine, Etoposide, Everolimus, Favipiravir, Fedratinib, Felodipine, Fentanyl, Fingolimod, Flibanserin, Fluconazole, Fluoxetine, Flupentixol, Fluphenazine, Flurazepam, Fluvoxamine, Galantamine, Gallopamil, Gefitinib, Genistein, Glasdegib, Glecaprevir, Glyburide, Gramicidin D, Grepafloxacin, Haloperidol, HM-30181, Hycanthone, Hydroxychloroquine, Idelalisib, Imatinib, Indinavir, Indomethacin, Isavuconazole, Isavuconazonium, Istradefylline, Itraconazole, Ivacaftor, Ivermectin, Ivosidenib, Ixabepilone, Ketoconazole, Lamotrigine, Laniquidar, Lansoprazole, Lapatinib, Lasmiditan, Lenvatinib, Letermovir, Levofloxacin, Lidocaine, Lomerizine, Lomitapide, Lonafarnib, Lopinavir, Loratadine, Losartan, Lovastatin, Lumacaftor, Lurbinectedin, Medroxyprogesterone acetate, Mefloquine, Megestrol acetate, Methadone, Methylene blue, Metronidazole, Mibefradil, Miconazole, Mifepristone, Mirabegron, Mitotane, Mitoxantrone, Naproxen, Nefazodone, Nelfinavir, Neratinib, Netupitant, Nicardipine, Niguldipine, Nilotinib, Nintedanib, Nisoldipine, Nitrendipine, Norethisterone, Norgestimate, Olaparib, Omeprazole, ONT-093, Paclitaxel, Palbociclib, Paliperidone, Pantoprazole, Paroxetine, Pemigatinib, Pibrentasvir, Pimozide, Piperine, Polyethylene glycol, Polyethylene glycol 400, Ponatinib, Posaconazole, Pralsetinib, Prazosin, Primaquine, Progesterone, Promethazine, Propafenone, Protriptyline, Quercetin, Quinacrine, Quinidine, Quinine, Ranitidine, Ranolazine, Reboxetine, Regorafenib, Relugolix, Reserpine, Reversin 121, Rifamycin, Rilpivirine, Ripretinib, Ritonavir, Rolapitant, Rucaparib, Salinomycin, Saquinavir, Sarecycline, Selegiline, Selpercatinib, Sertraline, Sildenafil, Simeprevir, Simvastatin, Sirolimus, Sorafenib, Staurosporine, Sunitinib, Tacrolimus, Tamoxifen, Tariquidar, Taurocholic acid, Telaprevir, Telmisartan, Temsirolimus, Tenofovir disoproxil, Tepotinib, Terazosin, Terfenadine, Testosterone cypionate, Testosterone enanthate, Testosterone undecanoate, Tetrandrine, Tezacaftor, Ticagrelor, Tipifarnib, Tipranavir, Tolvaptan, Trifluoperazine, Triflupromazine, Troleandomycin, Umbralisib, Upadacitinib, Valinomycin, Valspodar, Vandetanib, Vardenafil, Velpatasvir, Vemurafenib, Venetoclax, Venlafaxine, Verapamil, Vinblastine, Vincristine, Voacamine, Voclosporin, Voxilaprevir, Zimelidine, Zonisamide, Zosuquidar
3P-glycoprotein 1 substratesAbemaciclib, Acebutolol, Acenocoumarol, Acetaminophen, Acetylsalicylic acid, Afatinib, Albendazole, Aldosterone, Alfuzosin, Aliskiren, Alitretinoin, alpha-Tocopherol acetate, Ambrisentan, Amitriptyline, Amlodipine, Amprenavir, Anastrozole, Apixaban, Apremilast, Artesunate, Asunaprevir, Atazanavir, Atorvastatin, Avanafil, Avatrombopag, Axitinib, Azathioprine, Azithromycin, Baricitinib, Beclomethasone dipropionate, Belantamab mafodotin, Belinostat, Berotralstat, Betamethasone, Betamethasone phosphate, Betrixaban, Bisoprolol, Bortezomib, Bosutinib, Bromocriptine, Budesonide, Cabazitaxel, Cabergoline, Cabotegravir, Camptothecin, Canagliflozin, Capmatinib, Carfilzomib, Celecoxib, Ceritinib, Cerivastatin, Cethromycin, Cetirizine, Chloramphenicol succinate, Chloroquine, Chlorpromazine, Cimetidine, Ciprofloxacin, Citalopram, Clarithromycin, Clindamycin, Clobazam, Clofazimine, Clomifene, Clopidogrel, Clozapine, Cobimetinib, Colchicine, Conjugated estrogens, Copanlisib, Cortisone acetate, Crizotinib, Cyclosporine, Dabigatran etexilate, Dabrafenib, Daclatasvir, Dacomitinib, Dactinomycin, Dapagliflozin, Darolutamide, Darunavir, Dasabuvir, Dasatinib, Daunorubicin, Debrisoquine, Dexamethasone, Dexamethasone acetate, Diazepam, Diethylstilbestrol, Digitoxin, Digoxin, Diltiazem, Dipyridamole, Docetaxel, Dolutegravir, Domperidone, Doxepin, Doxorubicin, Duvelisib, Edoxaban, Elagolix, Elbasvir, Eletriptan, Elexacaftor, Eliglustat, Empagliflozin, Enasidenib, Enfortumab vedotin, Entrectinib, Epinastine, Erdafitinib, Erlotinib, Ertugliflozin, Erythromycin, Escitalopram, Esomeprazole, Estradiol, Estradiol acetate, Estradiol benzoate, Estradiol cypionate, Estradiol dienanthate, Estradiol valerate, Estriol, Estrone, Ethinylestradiol, Etoposide, Everolimus, Ezetimibe, Fedratinib, Fesoterodine, Fexofenadine, Fidaxomicin, Filgotinib, Flecainide, Fluticasone, Fluticasone furoate, Fluticasone propionate, Fostemsavir, Gefitinib, Gemcitabine, Gilteritinib, Glasdegib, Glecaprevir, Gramicidin D, Grapiprant, Grazoprevir, Grepafloxacin, Haloperidol, Hydrocortisone, Hydroxyzine, Ibuprofen, Idelalisib, Imatinib, Imipramine, Indacaterol, Indinavir, Indomethacin, Inotuzumab ozogamicin, Irinotecan, Ivermectin, Ivosidenib, Ixabepilone, Ketazolam, Lamivudine, Lamotrigine, Lansoprazole, Larotrectinib, Lasmiditan, Ledipasvir, Lefamulin, Lemborexant, Lenalidomide, Lenvatinib, Letermovir, Letrozole, Levamlodipine, Levetiracetam, Levofloxacin, Levomilnacipran, Linagliptin, Lonafarnib, Loperamide, Loratadine, Losartan, Lurbinectedin, Lusutrombopag, Medrysone, Mefloquine, Meperidine, Methotrexate, Methylene blue, Methylprednisolone, Metoclopramide, Mibefradil, Mirabegron, Mitoxantrone, Monensin, Morphine, Mycophenolate mofetil, Nadolol, Naloxone, Nelfinavir, Nicardipine, Nifedipine, Nilotinib, Nintedanib, Nitrofurantoin, Nizatidine, Nortriptyline, Octreotide, Odanacatib, Olanzapine, Olaparib, Olopatadine, Omadacycline, Ombitasvir, Omeprazole, Opicapone, Osimertinib, Oxcarbazepine, Ozanimod, Paclitaxel, Palbociclib, Paliperidone, Panobinostat, Pantoprazole, Paritaprevir, Pazopanib, Pemigatinib, Pentazocine, Phenobarbital, Phenytoin, Pibrentasvir, Pitavastatin, Platelet Activating Factor, Pomalidomide, Ponatinib, Posaconazole, Pralsetinib, Pravastatin, Prazosin, Prednisolone, Prednisolone acetate, Prednisolone phosphate, Prednisone, Progesterone, Propranolol, Prucalopride, Quetiapine, Quinidine, Quinine, Raloxifene, Ranitidine, Ranolazine, Regorafenib, Relugolix, Remdesivir, Reserpine, Revefenacin, Rhodamine 6G, Rifamycin, Rimegepant, Ripretinib, Risdiplam, Risperidone, Ritonavir, Rivaroxaban, Romidepsin, Rucaparib, Saquinavir, Selexipag, Selpercatinib, Selumetinib, Sildenafil, Silodosin, Simeprevir, Sitagliptin, Sofosbuvir, Somatostatin, Somatotropin, Sorafenib, Sparfloxacin, Sphingosine, Stanolone, Stanolone acetate, Sulpiride, Sumatriptan, Tacrine, Tacrolimus, Talazoparib, Talinolol, Tamoxifen, Taurocholic acid, Tazemetostat, Technetium Tc-99m sestamibi, Tegaserod, Telaprevir, Temozolomide, Temsirolimus, Tenofovir, Tenofovir alafenamide, Tenofovir disoproxil, Tepotinib, Testosterone propionate, Tezacaftor, Ticagrelor, Timolol, Tipranavir, Tolvaptan, Topiramate, Topotecan, Toremifene, Trastuzumab deruxtecan, Trastuzumab emtansine, Trilaciclib, Trimethoprim, Trimipramine, Tucatinib, Ubidecarenone, Ubrogepant, Umeclidinium, Upadacitinib, Valinomycin, Vardenafil, Vecuronium, Velpatasvir, Vemurafenib, Venetoclax, Venlafaxine, Verapamil, Vericiguat, Vibegron, Vinblastine, Vincristine, Vinflunine, Vismodegib, Voclosporin, Voxilaprevir, Zanubrutinib, Zidovudine
4P-glycoprotein 1 modulatorsAcetylsalicylic acid, Avapritinib, Prazosin
5P-glycoprotein 1 transportersLedipasvir, Tocopherol
6P-glycoprotein 1 bindersTechnetium Tc-99m tetrofosmin
7P-glycoprotein 1 antagonistsTocofersolan