Showing BioInteractions for Crofelemer (DB04941)

BioInteractor utilizes data on drug-target, -enzyme and -transporter associations to provide insight on drug-drug interactions. It allows you to identify, for instance, which drugs act similarly on the same target. Such drugs may have additive pharmacodynamic effects if given concomitantly. Conversely, two drugs may antagonize the beneficial effects of each other by having opposite actions on a specific drug target. BioInteractor uses ranked drug-enzyme association information to predict enzyme-mediated drug interactions that may be clinically relevant.
Interacting GroupInteracting Drugs
Crofelemer is a Cystic fibrosis transmembrane conductance regulator antagonist
1Cystic fibrosis transmembrane conductance regulator antagonistsBumetanide, Glyburide
2Cystic fibrosis transmembrane conductance regulator potentiatorsIvacaftor
3Cystic fibrosis transmembrane conductance regulator inhibitorsColforsin, Dexibuprofen, Ibuprofen
4Cystic fibrosis transmembrane conductance regulator modulatorsElexacaftor, Lumacaftor
5Cystic fibrosis transmembrane conductance regulator cofactorsATP
6Cystic fibrosis transmembrane conductance regulator activatorsTezacaftor
Interacting GroupInteracting Drugs
Crofelemer is a Anoctamin-1 antagonist