Acne Vulgaris

Also known as: Acne vulgaris (disorder) / Acne, unspecified / Acne / Acne NOS / Acnes

DrugDrug NameDrug Description
DB00210AdapaleneA third-generation topical retinoid with anti-comedogenic, comedolytic, and anti-inflammatory properties used to treat acne vulgaris in adolescents and adults.
DB00548Azelaic acidA saturated dicarboxylic acid used to treat mild to moderate acne vulgaris.
DB09096Benzoyl peroxideAn antibacterial and anti-inflammatory agent used for the symptomatic treatment of mild to moderate acne vulgaris and rosacea.
DB12499ClascoteroneAn androgen receptor antagonist used for the topical treatment of acne vulgaris in patients 12 years of age and older.
DB01190ClindamycinA lincosamide antibiotic used to treat serious infections caused by susceptible anaerobic, streptococcal, staphylococcal, and pneumococcal bacteria.
DB00250DapsoneA sulfone drug used to treat acne vulgaris, Hansen's disease, and dermatitis herpetiformis.
DB00199ErythromycinA macrolide antibiotic used to treat and prevent a variety of bacterial infections.
DB09526HydroquinoneA topical brightening agent used for the treatment of skin disorders associated with hyperpigmentation including melasma, post-inflammatory hyperpigmentation, sunspots, and freckles.
DB00256LymecyclineA tetracycline antibiotic used for the treatment of acne vulgaris and other susceptible infections.
DB01110MiconazoleAn azole antifungal with broad-spectrum activity used to treat fungal infections affecting the vagina, mouth and skin, including candidiasis.
DB12447NadifloxacinA topical fluoroquinolone used in the treatment of acne and topical bacterial skin infections.
DB00635PrednisoneA corticosteroid used to treat inflammation or immune-mediated reactions and to treat endocrine or neoplastic diseases.
DB11085ResorcinolContemporary therapeutic uses for resorcinol primarily revolve around the use of the phenol derivative as an active ingredient in topical antiseptics [L2745, L2744, L40069, F61] or as topical antibacterial skin...
DB00634SulfacetamideA sulfonamide used to treat inflammatory ocular conditions and acne vulgaris.
DB00755TretinoinA vitamin A derivative used to treat acne vulgaris and certain types of promyelocytic leukemia, as well as various skin conditions in over-the-counter medications.
DB00620TriamcinoloneA glucocorticoid used to treat a wide variety of inflammatory conditions of organ systems and tissues.
DB12808TrifaroteneA topical retinoid indicated for the treatment of acne vulgaris.
DrugDrug NameTargetType
DB00210AdapaleneRetinoic acid receptor betatarget
DB00210AdapaleneRetinoic acid receptor gammatarget
DB00210AdapaleneRetinoic acid receptor RXR-alphatarget
DB00210AdapaleneRetinoic acid receptor RXR-betatarget
DB00210AdapaleneRetinoic acid receptor RXR-gammatarget
DB00210AdapaleneTranscription factor AP-1target
DB00210AdapaleneRetinoic acid receptor alphatarget
DB00210AdapaleneAspartate aminotransferase, cytoplasmictarget
DB00210AdapaleneToll-like receptor 2target
DB00548Azelaic acid3-oxo-5-alpha-steroid 4-dehydrogenase 2target
DB00548Azelaic acidDNA polymerase Itarget
DB00548Azelaic acidThioredoxin reductasetarget
DB00548Azelaic acidTyrosinasetarget
DB00548Azelaic acid3-oxo-5-beta-steroid 4-dehydrogenasetarget
DB09096Benzoyl peroxideCatalaseenzyme
DB09096Benzoyl peroxideCatalasetarget
DB09096Benzoyl peroxideArginine decarboxylasetarget
DB09096Benzoyl peroxideProtein kinase Ctarget
DB09096Benzoyl peroxideGlutathione peroxidasetarget
DB09096Benzoyl peroxideSuperoxide Dismutasestarget
DB12499ClascoteroneAndrogen receptortarget
DB12499ClascoteroneCytochrome P450 1A2enzyme
DB12499ClascoteroneCytochrome P450 2B6enzyme
DB12499ClascoteroneCytochrome P450 2C8enzyme
DB12499ClascoteroneCytochrome P450 2C9enzyme
DB12499ClascoteroneCytochrome P450 2C19enzyme
DB12499ClascoteroneCytochrome P450 2D6enzyme
DB12499ClascoteroneCytochrome P450 2E1enzyme
DB12499ClascoteroneCytochrome P450 3A4enzyme
DB01190ClindamycinCytochrome P450 3A4enzyme
DB01190ClindamycinCytochrome P450 3A5enzyme
DB01190ClindamycinAlpha-1-acid glycoprotein 1carrier
DB01190ClindamycinP-glycoprotein 1transporter
DB01190Clindamycin50S ribosomal protein L1target
DB00250DapsoneInactive dihydropteroate synthase 2target
DB00250DapsoneDihydropteroate synthase 1target
DB00250DapsoneCytochrome P450 2C9enzyme
DB00250DapsoneCytochrome P450 2E1enzyme
DB00250DapsoneCytochrome P450 3A4enzyme
DB00250DapsoneDimethylaniline monooxygenase [N-oxide-forming] 3enzyme
DB00250DapsoneProstaglandin G/H synthase 1enzyme
DB00250DapsoneProstaglandin G/H synthase 2enzyme
DB00250DapsoneCytochrome P450 2C8enzyme
DB00250DapsoneCytochrome P450 2C19enzyme
DB00250DapsoneArylamine N-acetyltransferase 2enzyme
DB00250DapsoneCytochrome P450 3A5enzyme
DB00250DapsoneCytochrome P450 3A7enzyme
DB00250DapsoneMyeloperoxidaseenzyme
DB00250DapsoneCytochrome P450 2C18enzyme
DB00199Erythromycin23S ribosomal RNAtarget
DB00199ErythromycinCytochrome P450 3A4enzyme
DB00199ErythromycinCytochrome P450 3A7enzyme
DB00199ErythromycinP-glycoprotein 1transporter
DB00199ErythromycinSolute carrier organic anion transporter family member 1B1transporter
DB00199ErythromycinMotilin receptortarget
DB00199ErythromycinPotassium voltage-gated channel subfamily H member 2target
DB00199ErythromycinCytochrome P450 3A5enzyme
DB00199ErythromycinSolute carrier organic anion transporter family member 1B3transporter
DB00199ErythromycinBile salt export pumptransporter
DB00199ErythromycinCanalicular multispecific organic anion transporter 1transporter
DB00199ErythromycinSolute carrier organic anion transporter family member 1A2transporter
DB09526HydroquinoneTyrosinasetarget
DB09526HydroquinoneSerum albumincarrier
DB09526HydroquinoneLysosomal alpha-glucosidaseenzyme
DB09526HydroquinoneCysteinyl leukotriene receptor 1target
DB00256Lymecycline30S ribosomal protein S4target
DB01110MiconazoleCytochrome P450 2C9enzyme
DB01110MiconazoleCytochrome P450 2D6enzyme
DB01110MiconazoleCytochrome P450 3A4enzyme
DB01110MiconazoleP-glycoprotein 1transporter
DB01110MiconazoleCytochrome P450 51target
DB01110MiconazoleNitric oxide synthase, endothelialtarget
DB01110MiconazoleNitric oxide synthase, inducibletarget
DB01110MiconazoleCytochrome P450 11B1, mitochondrialenzyme
DB01110MiconazoleCytochrome P450 2A6enzyme
DB01110MiconazoleCytochrome P450 2B6enzyme
DB01110MiconazoleCytochrome P450 2C19enzyme
DB01110MiconazoleCytochrome P450 2E1enzyme
DB01110MiconazoleNuclear receptor subfamily 1 group I member 2target
DB01110MiconazoleLanosterol 14-alpha demethylaseenzyme
DB01110MiconazoleCytochrome P450 19A1enzyme
DB01110MiconazoleCalcium-activated potassium channeltarget
DB01110MiconazoleVoltage-gated Potassium Channelstarget
DB01110MiconazoleInward rectifier potassium channeltarget
DB01110MiconazoleVoltage gated L-type calcium channeltarget
DB01110MiconazoleSerum albumincarrier
DB01110MiconazoleCytochrome P450 2C8enzyme
DB00635PrednisoneGlucocorticoid receptortarget
DB00635PrednisoneCytochrome P450 3A4enzyme
DB00635PrednisoneP-glycoprotein 1transporter
DB00635PrednisoneSolute carrier organic anion transporter family member 1A2transporter
DB00635PrednisoneCytochrome P450 2C19enzyme
DB00635PrednisoneSerum albumincarrier
DB00635PrednisoneCytochrome P450 3A5enzyme
DB00635PrednisoneCorticosteroid-binding globulincarrier
DB00635PrednisoneCytochrome P450 3A Subfamilyenzyme
DB00635PrednisoneCytochrome P450 2A6enzyme
DB00635PrednisoneCytochrome P450 1B1enzyme
DB00635PrednisoneCytochrome P450 2B6enzyme
DB00635PrednisoneCytochrome P450 2C8enzyme
DB00635PrednisoneCytochrome P450 2C9enzyme
DB00635PrednisoneCorticosteroid 11-beta-dehydrogenase isozyme 1enzyme
DB11085ResorcinolThyroid peroxidasetarget
DB00634SulfacetamideDihydropteroate synthasetarget
DB00634SulfacetamideDihydropteroate synthase type-1target
DB00634SulfacetamideFolic acid synthesis protein FOL1target
DB00755TretinoinRetinoic acid receptor gammatarget
DB00755TretinoinRetinoic acid receptor RXR-betatarget
DB00755TretinoinRetinal dehydrogenase 1target
DB00755TretinoinRetinoic acid-induced protein 3target
DB00755TretinoinRetinoic acid receptor RXR-gammatarget
DB00755TretinoinRetinal dehydrogenase 2target
DB00755TretinoinRetinoic acid receptor responder protein 1target
DB00755TretinoinCytochrome P450 2C8enzyme
DB00755TretinoinCellular retinoic acid-binding protein 1transporter
DB00755TretinoinCellular retinoic acid-binding protein 2transporter
DB00755TretinoinCytochrome P450 2B6enzyme
DB00755TretinoinCytochrome P450 3A4enzyme
DB00755TretinoinCytochrome P450 3A5enzyme
DB00755TretinoinCytochrome P450 2A6enzyme
DB00755TretinoinCytochrome P450 3A7enzyme
DB00755TretinoinCytochrome P450 2C18enzyme
DB00755TretinoinCytochrome P450 2C9enzyme
DB00755TretinoinCytochrome P450 4A11enzyme
DB00755TretinoinCytochrome P450 1A1enzyme
DB00755TretinoinRetinoic acid receptor alphatarget
DB00755TretinoinRetinoic acid receptor betatarget
DB00755TretinoinLipocalin-1target
DB00755TretinoinOdorant-binding protein 2atarget
DB00755TretinoinRetinol-binding protein 4target
DB00755TretinoinSerum albumincarrier
DB00755Tretinoin[Pyruvate dehydrogenase [lipoamide]] kinase isozyme 4, mitochondrialtarget
DB00755TretinoinRetinoic acid receptor RXR-alphatarget
DB00755TretinoinCarcinoembryonic antigentarget
DB00755TretinoinUDP-glucuronosyltransferase 2B7enzyme
DB00755TretinoinCytochrome P450 2E1enzyme
DB00755TretinoinCytochrome P450 26A1enzyme
DB00755TretinoinCellular retinoic acid-binding protein 1target
DB00620TriamcinoloneCorticosteroid-binding globulincarrier
DB00620TriamcinoloneGlucocorticoid receptortarget
DB00620TriamcinoloneCytochrome P450 3A4enzyme
DB00620TriamcinoloneProstaglandin G/H synthase 2enzyme
DB00620TriamcinoloneCholinesteraseenzyme
DB00620TriamcinoloneCytochrome P450 3A5enzyme
DB00620TriamcinoloneCytochrome P450 3A7enzyme
DB00620TriamcinoloneSerum albumincarrier
DB12808TrifaroteneCytochrome P450 2C9enzyme
DB12808TrifaroteneCytochrome P450 3A4enzyme
DB12808TrifaroteneCytochrome P450 2C8enzyme
DB12808TrifaroteneCytochrome P450 2B6enzyme
DB12808TrifaroteneRetinoic acid receptor gammatarget
DB12808TrifaroteneRetinoic acid receptor alphatarget
DB12808TrifaroteneRetinoic acid receptor betatarget
DrugDrug NamePhaseStatusCount
DB00210Adapalene0Completed1
DB00207Azithromycin0Not Yet Recruiting1
DB00982Isotretinoin0Completed1
DB00982Isotretinoin0Not Yet Recruiting1
DB00759Tetracycline0Not Yet Recruiting1
DB00755Tretinoin0Completed5
DB00162Vitamin A0Not Yet Recruiting1
DB00210Adapalene1Active Not Recruiting1
DB00210Adapalene1Completed4
DB00210Adapalene1Withdrawn1
DB00855Aminolevulinic acid1Completed1
DB09495Avobenzone1Completed1
DB09096Benzoyl peroxide1Completed8
DB01373Calcium1Completed1
DB01190Clindamycin1Completed8
DB00250Dapsone1Completed3
DB00250Dapsone1Withdrawn2
DB00254Doxycycline1Completed1
DB00158Folic acid1Completed1
DB10344Ginger1Completed1
DB11064Homosalate1Completed1
DB00982Isotretinoin1Completed1
DB11062Octisalate1Completed1
DB09535Octocrylene1Completed1
DB01428Oxybenzone1Completed1
DB00935Oxymetazoline1Completed1
DB01783Pantothenic acid1Completed1
DB00165Pyridoxine1Completed1
DB00936Salicylic acid1Completed1
DB14546Sulfate ion1Completed1
DB00799Tazarotene1Completed7
DB00373Timolol1Completed1
DB00755Tretinoin1Completed3
DB12808Trifarotene1Completed1
DB00126Ascorbic acid1 / 2Completed1
DB09096Benzoyl peroxide1 / 2Completed1
DB12499Clascoterone1 / 2Not Yet Recruiting1
DB01190Clindamycin1 / 2Completed1
DB00254Doxycycline1 / 2Active Not Recruiting1
DB00254Doxycycline1 / 2Unknown Status1
DB11674Equol1 / 2Unknown Status1
DB00982Isotretinoin1 / 2Completed1
DB00350Minoxidil1 / 2Recruiting1
DB00435Nitric Oxide1 / 2Completed1
DB12642Olumacostat glasaretil1 / 2Completed1
DB00936Salicylic acid1 / 2Completed2
DB15385Acebilustat2Completed1
DB00210Adapalene2Completed2
DB00210Adapalene2Not Yet Recruiting1
DB04931Afamelanotide2Completed1
DB00855Aminolevulinic acid2Completed1
DB00855Aminolevulinic acid2Recruiting1
DB09096Benzoyl peroxide2Completed3
DB14947Bermekimab2Completed1
DB00083Botulinum toxin type A2Completed1
DB00083Botulinum toxin type A2Terminated1
DB12499Clascoterone2Completed3
DB01190Clindamycin2Completed2
DB00250Dapsone2Completed1
DB17576Denifanstat2Completed1
DB06133Dimethylcurcumin2Completed1
DB00254Doxycycline2Completed2
DB00254Doxycycline2Recruiting1
DB00898Ethanol2Completed1
DB12119Gevokizumab2Completed1
DB11091Hydrogen peroxide2Completed1
DB16658Imsidolimab2Completed1
DB15109Ingenol disoxate2Completed1
DB00982Isotretinoin2Active Not Recruiting1
DB00982Isotretinoin2Completed1
DB00331Metformin2Recruiting1
DB00992Methyl aminolevulinate2Completed2
DB01017Minocycline2Completed4
DB12642Olumacostat glasaretil2Completed1
DB06574Omiganan2Completed2
DB06610Omiganan2Completed3
DB12096PF-051751572Withdrawn1
DB12035Sarecycline2Completed1
DB00799Tazarotene2Completed5
DB00799Tazarotene2Unknown Status1
DB00755Tretinoin2Completed1
DB12808Trifarotene2Completed1
DB00744Zileuton2Unknown Status1
DB02300Calcipotriol2 / 3Completed1
DB11094Vitamin D2 / 3Completed1
DB00210Adapalene3Completed14
DB00210Adapalene3Withdrawn2
DB13906Aloe vera leaf3Not Yet Recruiting1
DB00126Ascorbic acid3Not Yet Recruiting1
DB00548Azelaic acid3Completed1
DB00207Azithromycin3Completed1
DB00207Azithromycin3Terminated1
DB09096Benzoyl peroxide3Completed21
DB09096Benzoyl peroxide3Unknown Status2
DB09096Benzoyl peroxide3Withdrawn1
DB12499Clascoterone3Completed3
DB01190Clindamycin3Completed14
DB00250Dapsone3Completed5
DB01075Diphenhydramine3Completed2
DB00254Doxycycline3Completed1
DB01395Drospirenone3Completed4
DB00977Ethinylestradiol3Completed1
DB09462Glycerin3Not Yet Recruiting1
DB00756Hexachlorophene3Unknown Status1
DB00982Isotretinoin3Recruiting1
DB00256Lymecycline3Completed1
DB01017Minocycline3Completed3
DB01017Minocycline3Terminated1
DB00471Montelukast3Not Yet Recruiting1
DB12447Nadifloxacin3Unknown Status1
DB02701Nicotinamide3Not Yet Recruiting1
DB12642Olumacostat glasaretil3Completed3
DB14556Peracetic acid3Completed1
DB00936Salicylic acid3Completed1
DB12035Sarecycline3Completed3
DB12035Sarecycline3Withdrawn1
DB00421Spironolactone3Completed1
DB00799Tazarotene3Completed7
DB00755Tretinoin3Completed5
DB11152Trichloroacetate3Completed1
DB12808Trifarotene3Completed5
DB00162Vitamin A3Not Yet Recruiting1
DB00210Adapalene4Active Not Recruiting1
DB00210Adapalene4Completed28
DB00210Adapalene4Terminated2
DB00210Adapalene4Unknown Status1
DB13906Aloe vera leaf4Completed1
DB00548Azelaic acid4Completed3
DB09096Benzoyl peroxide4Active Not Recruiting1
DB09096Benzoyl peroxide4Completed30
DB09096Benzoyl peroxide4Terminated1
DB09096Benzoyl peroxide4Unknown Status2
DB00169Cholecalciferol4Enrolling by Invitation1
DB12499Clascoterone4Active Not Recruiting2
DB01190Clindamycin4Active Not Recruiting1
DB01190Clindamycin4Completed19
DB01190Clindamycin4Recruiting1
DB01190Clindamycin4Unknown Status2
DB14322Coconut oil4Completed1
DB04839Cyproterone acetate4Completed1
DB00250Dapsone4Completed10
DB00250Dapsone4Not Yet Recruiting1
DB00304Desogestrel4Completed1
DB00254Doxycycline4Completed5
DB00199Erythromycin4Recruiting1
DB00783Estradiol4Completed1
DB00898Ethanol4Recruiting1
DB00977Ethinylestradiol4Completed1
DB08818Hyaluronic acid4Completed1
DB00982Isotretinoin4Active Not Recruiting1
DB00982Isotretinoin4Completed3
DB00982Isotretinoin4Not Yet Recruiting2
DB00331Metformin4Not Yet Recruiting1
DB01017Minocycline4Completed1
DB01017Minocycline4Terminated1
DB12447Nadifloxacin4Completed1
DB02701Nicotinamide4Completed1
DB00957Norgestimate4Completed1
DB01839Propylene glycol4Completed1
DB14272Rosemary4Completed1
DB00936Salicylic acid4Completed1
DB00936Salicylic acid4Not Yet Recruiting2
DB09298Silibinin4Not Yet Recruiting2
DB00799Tazarotene4Completed5
DB00799Tazarotene4Terminated1
DB00755Tretinoin4Completed9
DB00755Tretinoin4Terminated1
DB00755Tretinoin4Unknown Status2
DB11152Trichloroacetate4Not Yet Recruiting1
DB12808Trifarotene4Completed3
DB11094Vitamin D4Enrolling by Invitation1
DB11094Vitamin D4Unknown Status1
DB01593Zinc4Completed1
DB00210AdapaleneNot AvailableActive Not Recruiting1
DB00210AdapaleneNot AvailableCompleted7
DB00210AdapaleneNot AvailableNot Yet Recruiting1
DB00855Aminolevulinic acidNot AvailableCompleted1
DB00855Aminolevulinic acidNot AvailableWithdrawn1
DB00207AzithromycinNot AvailableNot Yet Recruiting1
DB03793Benzoic acidNot AvailableCompleted1
DB09096Benzoyl peroxideNot AvailableActive Not Recruiting1
DB09096Benzoyl peroxideNot AvailableCompleted12
DB01190ClindamycinNot AvailableCompleted3
DB04839Cyproterone acetateNot AvailableCompleted2
DB00254DoxycyclineNot AvailableCompleted1
DB00977EthinylestradiolNot AvailableCompleted2
DB00982IsotretinoinNot AvailableCompleted2
DB00982IsotretinoinNot AvailableNot Yet Recruiting1
DB00982IsotretinoinNot AvailableRecruiting1
DB01017MinocyclineNot AvailableEnrolling by Invitation1
DB00936Salicylic acidNot AvailableCompleted1
DB12035SarecyclineNot AvailableCompleted2
DB00755TretinoinNot AvailableActive Not Recruiting1
DB00620TriamcinoloneNot AvailableCompleted1
DB11152TrichloroacetateNot AvailableCompleted1