Acute Migraine

Also known as: Migraine - Acute / Acute Migraine Headache / Migraine, Acute / Acute migraine (disorder) / Migraine, unspecified / Migraine, unspecified, not intractable, without status migrainosus / Migraine NOS / Migraine headaches / Migraine headache / Migrainous headache / Migraine type headaches / Migraine Disorders / Migraine (disorder) / Migraine

DrugDrug NameDrug Description
DB01424AminophenazoneAn analgesic drug used to treat acute migraine attacks in combination with ergotamine and caffeine.
DB00586DiclofenacAn NSAID used to treat the signs and symptoms of osteoarthritis and rheumatoid arthritis.
DB00465KetorolacAn NSAID used to treat moderate to severe pain, rheumatoid arthritis, osteoarthritis, ankylosing spondylitis, menstrual disorders, and headaches.
DB00788NaproxenAn NSAID used to treat rheumatoid arthritis, osteoarthritis, ankylosing spondylitis, polyarticular juvenile idiopathic arthritis, tendinitis, bursitis, acute gout, primary dysmenorrhea, and mild to moderate pain.
DB00433ProchlorperazineA phenothiazine derivative used in the treatment of schizophrenia and anxiety and to relieve severe nausea and vomiting.
DB00669SumatriptanA serotonin receptor agonist used to treat migraines and cluster headaches.
DB15688ZavegepantA calcitonin gene-related peptide receptor antagonist indicated for the acute treatment of migraine with or without aura.
DrugDrug NameTargetType
DB01424AminophenazoneCytochrome P450 2C19enzyme
DB01424AminophenazoneCytochrome P450 1A2enzyme
DB01424AminophenazoneCytochrome P450 2C8enzyme
DB01424AminophenazoneSolute carrier family 22 member 6transporter
DB01424AminophenazoneCytochrome P450 2C9enzyme
DB01424AminophenazoneCytochrome P450 2D6enzyme
DB01424AminophenazoneCytochrome P450 3A4enzyme
DB01424AminophenazoneCytochrome P450 2C18enzyme
DB01424AminophenazoneSteroid 17-alpha-hydroxylase/17,20 lyaseenzyme
DB00586DiclofenacProstaglandin G/H synthase 1target
DB00586DiclofenacProstaglandin G/H synthase 2target
DB00586DiclofenacTransthyretincarrier
DB00586DiclofenacCytochrome P450 2C9enzyme
DB00586DiclofenacCytochrome P450 2C19enzyme
DB00586DiclofenacCytochrome P450 1A2enzyme
DB00586DiclofenacCytochrome P450 2C8enzyme
DB00586DiclofenacSerum albumincarrier
DB00586DiclofenacMultidrug resistance-associated protein 4transporter
DB00586DiclofenacMultidrug resistance-associated protein 1transporter
DB00586DiclofenacSolute carrier family 22 member 6transporter
DB00586DiclofenacSolute carrier family 22 member 8transporter
DB00586DiclofenacSolute carrier organic anion transporter family member 1C1transporter
DB00586DiclofenacSolute carrier family 22 member 11transporter
DB00586DiclofenacUDP-glucuronosyltransferase 2B7enzyme
DB00586DiclofenacCytochrome P450 3A4enzyme
DB00586DiclofenacCytochrome P450 2B6enzyme
DB00586DiclofenacCytochrome P450 2C18enzyme
DB00586DiclofenacCytochrome P450 2E1enzyme
DB00586DiclofenacSolute carrier organic anion transporter family member 1B1transporter
DB00586DiclofenacBile salt export pumptransporter
DB00586DiclofenacUDP-glucuronosyltransferase 1-3enzyme
DB00586DiclofenacUDP-glucuronosyltransferase 1-9enzyme
DB00586DiclofenacUDP-glucuronosyltransferase 2B4enzyme
DB00586DiclofenacArachidonate 5-lipoxygenaseenzyme
DB00586DiclofenacSodium channel protein type 4 subunit alphatransporter
DB00586DiclofenacAcid-sensing ion channel 1transporter
DB00586DiclofenacPotassium voltage-gated channel subfamily KQT member 2transporter
DB00586DiclofenacPotassium voltage-gated channel subfamily KQT member 3transporter
DB00586DiclofenacPhospholipase A2, membrane associatedenzyme
DB00586DiclofenacP-glycoprotein 1transporter
DB00465KetorolacProstaglandin G/H synthase 1target
DB00465KetorolacProstaglandin G/H synthase 2target
DB00465KetorolacUDP-glucuronosyltransferase 2B7enzyme
DB00465KetorolacCytochrome P450 2C8enzyme
DB00465KetorolacCytochrome P450 2C9enzyme
DB00788NaproxenProstaglandin G/H synthase 1target
DB00788NaproxenProstaglandin G/H synthase 2target
DB00788NaproxenSerum albumincarrier
DB00788NaproxenCytochrome P450 2C9enzyme
DB00788NaproxenCytochrome P450 1A2enzyme
DB00788NaproxenSolute carrier organic anion transporter family member 1A2transporter
DB00788NaproxenSolute carrier family 22 member 6transporter
DB00788NaproxenCytochrome P450 2C8enzyme
DB00788NaproxenUDP-glucuronosyltransferase 2B7enzyme
DB00788NaproxenPeptostreptococcal albumin-binding proteintarget
DB00788NaproxenBile salt export pumptransporter
DB00788NaproxenP-glycoprotein 1transporter
DB00788NaproxenUDP-glucuronosyltransferase 1-3enzyme
DB00788NaproxenUDP-glucuronosyltransferase 1-6enzyme
DB00788NaproxenUDP-glucuronosyltransferase 1-7enzyme
DB00788NaproxenUDP-glucuronosyltransferase 1-8enzyme
DB00788NaproxenUDP-glucuronosyltransferase 1-9enzyme
DB00788NaproxenUDP-glucuronosyltransferase 1-10enzyme
DB00788NaproxenSolute carrier family 22 member 8transporter
DB00433ProchlorperazineDopamine D2 receptortarget
DB00433ProchlorperazineCytochrome P450 2D6enzyme
DB00433ProchlorperazineHistamine H1 receptortarget
DB00433ProchlorperazineAlpha-1 adrenergic receptorstarget
DB00433ProchlorperazineAlpha-2 adrenergic receptorstarget
DB00669Sumatriptan5-hydroxytryptamine receptor 1Dtarget
DB00669Sumatriptan5-hydroxytryptamine receptor 1Btarget
DB00669Sumatriptan5-hydroxytryptamine receptor 1Ftarget
DB00669SumatriptanAmine oxidase [flavin-containing] Aenzyme
DB00669Sumatriptan5-hydroxytryptamine receptor 1Atarget
DB00669SumatriptanSolute carrier organic anion transporter family member 1A2transporter
DB00669SumatriptanP-glycoprotein 1transporter
DB00669SumatriptanATP-binding cassette sub-family G member 2transporter
DB00669SumatriptanSolute carrier organic anion transporter family member 1B1transporter
DB15688ZavegepantCalcitonin gene-related peptide type 1 receptortarget
DB15688ZavegepantCytochrome P450 3A4enzyme
DB15688ZavegepantCytochrome P450 2D6enzyme
DB15688ZavegepantSolute carrier organic anion transporter family member 1B3transporter
DB15688ZavegepantSodium/bile acid cotransportertransporter
DB15688ZavegepantP-glycoprotein 1transporter
DB15688ZavegepantMultidrug and toxin extrusion protein 1transporter
DB15688ZavegepantMultidrug and toxin extrusion protein 2transporter
DrugDrug NamePhaseStatusCount
DB00669Sumatriptan1Completed1
DB11883SB-7054982Completed1
DB15688Zavegepant2 / 3Completed1
DB00315Zolmitriptan2 / 3Completed1
DB00316Acetaminophen3Completed1
DB00945Acetylsalicylic acid3Completed1
DB00241Butalbital3Completed1
DB01009Ketoprofen3Unknown Status1
DB11732Lasmiditan3Completed2
DB00788Naproxen3Completed1
DB12457Rimegepant3Completed2
DB00953Rizatriptan3Completed2
DB00669Sumatriptan3Completed2
DB00316Acetaminophen4Completed2
DB09214Dexketoprofen4Completed1
DB00465Ketorolac4Completed1
DB01233Metoclopramide4Completed1
DB00313Valproic acid4Completed1
DB00315Zolmitriptan4Completed1
DB00216EletriptanNot AvailableCompleted1
DB01050IbuprofenNot AvailableNot Yet Recruiting1
DB00465KetorolacNot AvailableNot Yet Recruiting1
DB01233MetoclopramideNot AvailableNot Yet Recruiting1
DB00433ProchlorperazineNot AvailableCompleted1
DB00669SumatriptanNot AvailableCompleted1
DB00315ZolmitriptanNot AvailableCompleted1