Bronchoconstriction

Also known as: Spasm bronchial / Bronchial Spasm / Bronchospasm (finding) / Bronchospasm / Bronchospasm NOS

DrugDrug NameDrug Description
DB01001AlbuterolA beta-2 adrenergic receptor agonist used to treat asthma, bronchitis, COPD, as well as prevent exercise induced bronchospasms.
DB01274ArformoterolA beta-2 adrenergic agonist and bronchodilator used for long-term, symptomatic treatment of reversible bronchoconstriction in patients with chronic obstructive pulmonary disease (COPD), including chronic bronchitis and emphysema.
DB01222BudesonideA corticosteroid used to treat Crohn's disease, asthma, COPD, hay fever and allergies, and ulcerative colitis.
DB15784CarmoterolA long acting beta-2 agonist indicated in the treatment of COPD, asthma, and chronic bronchitis.
DB01410CiclesonideA glucocorticoid used in the symptomatic relief of nasal symptoms associated with seasonal and perennial allergic rhinitis in adults and adolescents.
DB00983FormoterolAn inhaled long-acting beta2-adrenergic receptor agonist used as a bronchodilator in the management of asthma and COPD.
DB01303OxtriphyllineA bronchodilator used for the treatment of asthma, bronchitis, COPD, and emphysema.
DB00277TheophyllineA xanthine used to manage the symptoms of asthma, COPD, and other lung conditions caused by reversible airflow obstruction.
DB01409TiotropiumA long-acting bronchodilator used in the management of chronic obstructive pulmonary disease (COPD).
DrugDrug NameTargetType
DB01001AlbuterolBeta-2 adrenergic receptortarget
DB01001AlbuterolBeta-1 adrenergic receptortarget
DB01001AlbuterolCytochrome P450 3A4enzyme
DB01001AlbuterolBeta-3 adrenergic receptortarget
DB01274ArformoterolBeta-2 adrenergic receptortarget
DB01274ArformoterolCytochrome P450 2D6enzyme
DB01274ArformoterolCytochrome P450 2C19enzyme
DB01274ArformoterolCytochrome P450 2A6enzyme
DB01274ArformoterolCytochrome P450 2C9enzyme
DB01222BudesonideGlucocorticoid receptortarget
DB01222BudesonideCytochrome P450 3A4enzyme
DB01222BudesonideCytochrome P450 3A5enzyme
DB01222BudesonideBile salt export pumptransporter
DB01222BudesonideP-glycoprotein 1transporter
DB01222BudesonideAnnexin A1target
DB01222BudesonideCytochrome P450 3A Subfamilyenzyme
DB01222BudesonideCytochrome P450 2A6enzyme
DB01222BudesonideCytochrome P450 1B1enzyme
DB01222BudesonideCytochrome P450 2B6enzyme
DB01222BudesonideCytochrome P450 2C8enzyme
DB01222BudesonideCytochrome P450 2C9enzyme
DB01222BudesonideCytochrome P450 2C19enzyme
DB01222BudesonideCorticosteroid-binding globulincarrier
DB01222BudesonideSolute carrier organic anion transporter family member 1A2transporter
DB01222BudesonideSolute carrier family 22 member 8transporter
DB01222BudesonideSerum albumincarrier
DB01410CiclesonideCorticosteroid-binding globulincarrier
DB01410CiclesonideCytochrome P450 3A4enzyme
DB01410CiclesonideCytochrome P450 2D6enzyme
DB01410CiclesonideGlucocorticoid receptortarget
DB01410CiclesonideLiver carboxylesterase 1enzyme
DB00983FormoterolBeta-2 adrenergic receptortarget
DB00983FormoterolBeta-1 adrenergic receptortarget
DB00983FormoterolBeta-3 adrenergic receptortarget
DB00983FormoterolCytochrome P450 2D6enzyme
DB00983FormoterolCytochrome P450 2C19enzyme
DB00983FormoterolCytochrome P450 2C9enzyme
DB00983FormoterolCytochrome P450 2A6enzyme
DB00983FormoterolUDP-glucuronosyltransferase 1A1enzyme
DB00983FormoterolUDP-glucuronosyltransferase 1-8enzyme
DB00983FormoterolUDP-glucuronosyltransferase 1-9enzyme
DB00983FormoterolUDP-glucuronosyltransferase 2B7enzyme
DB00983FormoterolUDP-glucuronosyltransferase 2B15enzyme
DB00983FormoterolSolute carrier family 22 member 1transporter
DB00983FormoterolSolute carrier family 22 member 4transporter
DB00983FormoterolSolute carrier family 22 member 5transporter
DB00983FormoterolSolute carrier family 22 member 3transporter
DB00983FormoterolSerum albumincarrier
DB01303OxtriphyllinecGMP-inhibited 3',5'-cyclic phosphodiesterase Atarget
DB01303OxtriphyllinecAMP-specific 3',5'-cyclic phosphodiesterase 4Atarget
DB01303OxtriphyllineAdenosine receptor A2atarget
DB01303OxtriphyllineAdenosine receptor A1target
DB01303OxtriphyllineCytochrome P450 1A2enzyme
DB01303OxtriphyllineSolute carrier family 22 member 7transporter
DB01303OxtriphyllineHistone deacetylase 2target
DB00277TheophyllinecGMP-inhibited 3',5'-cyclic phosphodiesterase Atarget
DB00277TheophyllinecAMP-specific 3',5'-cyclic phosphodiesterase 4Btarget
DB00277TheophyllineAdenosine receptor A2btarget
DB00277TheophyllinecAMP-specific 3',5'-cyclic phosphodiesterase 4Atarget
DB00277TheophyllinecGMP-specific 3',5'-cyclic phosphodiesterasetarget
DB00277TheophyllineAdenosine receptor A1target
DB00277TheophyllineAdenosine receptor A2atarget
DB00277TheophyllineCytochrome P450 1A2enzyme
DB00277TheophyllineAdenosine deaminaseenzyme
DB00277TheophyllineCytochrome P450 2E1enzyme
DB00277TheophyllineCytochrome P450 3A4enzyme
DB00277TheophyllineSolute carrier family 22 member 7transporter
DB00277TheophyllineCytochrome P450 1A1enzyme
DB00277TheophyllineCytochrome P450 1B1enzyme
DB00277TheophyllineCytochrome P450 2D6enzyme
DB00277TheophyllineHistone deacetylase 2target
DB00277TheophyllineCopine-1target
DB00277TheophyllineMinor histocompatibility antigen H13target
DB00277TheophyllineNodal modulator 1target
DB00277TheophyllinePoly [ADP-ribose] polymerase 1target
DB00277TheophyllineProtein RIC-3target
DB00277TheophyllineTubulin monoglycylase TTLL3target
DB01409TiotropiumMuscarinic acetylcholine receptor M3target
DB01409TiotropiumCytochrome P450 2D6enzyme
DB01409TiotropiumCytochrome P450 3A4enzyme
DB01409TiotropiumMuscarinic acetylcholine receptor M1target
DB01409TiotropiumMuscarinic acetylcholine receptor M2target
DB01409TiotropiumSolute carrier family 22 member 5transporter
DB01409TiotropiumSolute carrier family 22 member 4transporter
DB01409TiotropiumMuscarinic acetylcholine receptor M4target
DB01409TiotropiumMuscarinic acetylcholine receptor M5target
DrugDrug NamePhaseStatusCount
DB01001Albuterol2Completed1
DB13139Levosalbutamol2Completed1
DB01001Albuterol3Completed1
DB13139Levosalbutamol3Completed1
DB01001Albuterol4Completed1