Moderate Vulvovaginal atrophy

DrugDrug NameDrug Description
DB09381Esterified estrogensA female hormone used to treat conditions related to estrogen deficiency and moderate to severe vasomotor menopausal symptoms in women.
DB04574Estrone sulfateAn estrogen used as monotherapy or in several combination hormone replacement products for managing menopause symptoms and hormone disorders.
DB00957NorgestimateA progesterone used as a contraceptive and to treat acne vulgaris.
DB09317Synthetic Conjugated Estrogens, AA mixture of estrogens used to treat a variety of postmenopausal symptoms, including vaginal atrophy and dyspareunia.
DB09318Synthetic Conjugated Estrogens, BA mixture of estrogens used to treat a variety of postmenopausal symptoms, including vaginal dryness.
DrugDrug NameTargetType
DB09381Esterified estrogensCytochrome P450 3A4enzyme
DB09381Esterified estrogensThyroxine-binding globulincarrier
DB04574Estrone sulfateCytochrome P450 1A2enzyme
DB04574Estrone sulfateCytochrome P450 3A4enzyme
DB04574Estrone sulfateEstrogen receptor alphatarget
DB04574Estrone sulfateEstrogen receptor betatarget
DB04574Estrone sulfateSex hormone-binding globulincarrier
DB04574Estrone sulfateSerum albumincarrier
DB04574Estrone sulfateCytochrome P450 2C9enzyme
DB04574Estrone sulfateMultidrug and toxin extrusion protein 1transporter
DB04574Estrone sulfateMultidrug and toxin extrusion protein 2transporter
DB04574Estrone sulfateSodium/bile acid cotransportertransporter
DB00957NorgestimateProgesterone receptortarget
DB00957NorgestimateEstrogen receptor alphatarget
DB00957NorgestimateCanalicular multispecific organic anion transporter 1transporter
DB00957NorgestimateCytochrome P450 3A4enzyme
DB00957NorgestimateAndrogen receptortarget
DB00957NorgestimateCytochrome P450 2B6enzyme
DB00957NorgestimateCytochrome P450 2C9enzyme
DB00957NorgestimateUDP-glucuronosyltransferase 1-1enzyme
DB00957NorgestimateSerum albumincarrier
DB00957NorgestimateSex hormone-binding globulincarrier
DB00957NorgestimateP-glycoprotein 1transporter
DB09317Synthetic Conjugated Estrogens, ACytochrome P450 3A4enzyme
DB09317Synthetic Conjugated Estrogens, AEstrogen receptor alphatarget
DB09317Synthetic Conjugated Estrogens, AThyroxine-binding globulincarrier
DB09318Synthetic Conjugated Estrogens, BEstrogen receptor alphatarget
DB09318Synthetic Conjugated Estrogens, BCytochrome P450 3A4enzyme
DB09318Synthetic Conjugated Estrogens, BThyroxine-binding globulincarrier
DrugDrug NamePhaseStatusCount