Seizures

Also known as: Seizure / Convulsions / Convulsion / Seizure (finding) / Convulsions NOS

DrugDrug NameDrug Description
DB09061CannabidiolAn active cannabinoid used as an adjunctive treatment for the management of seizures associated with Lennox-Gastaut syndrome or Dravet syndrome and symptomatic relief of moderate to severe neuropathic pain or other painful conditions, like cancer.
DB00349ClobazamA benzodiazepine used as adjunct treatment in seizures associated with Lennox-Gastaut syndrome.
DB00574FenfluramineFenfluramine is a phenethylamine that is structurally similar to serotonin. Due to its ability to increase extracellular serotonin levels, modulate serotonergic and other neurologic receptors, and control neurotransmission, it is effective in treating pharmacoresistant seizures.
DB01320FosphenytoinAn antiepileptic agent used for the management of generalized convulsive status epilepticus and prevention and treatment of seizures occurring during neurosurgery.
DB05087GanaxoloneA neuroactive steroid GABA-A receptor modulator used for the treatment of seizures associated with CDKL5 deficiency disorder (CDD).
DB00252PhenytoinAn anticonvulsant drug used in the prophylaxis and control of various types of seizures.
DB09118StiripentolAn antiepileptic agent used in combination with other anticonvulsants to treat seizures associated with Dravet syndrome.
DB00599ThiopentalA barbiturate used to induce general anesthesia, treat convulsions, and reduce intracranial pressure.
DB00697TizanidineAn alpha-2 adrenergic agonist used for the short-term treatment of muscle spasticity.
DB00273TopiramateAn anticonvulsant drug used in the control of epilepsy and in the prophylaxis and treatment of migraines.
DrugDrug NameTargetType
DB09061CannabidiolCytochrome P450 2C9enzyme
DB09061CannabidiolCytochrome P450 2C19enzyme
DB09061CannabidiolCytochrome P450 2D6enzyme
DB09061CannabidiolCytochrome P450 3A4enzyme
DB09061CannabidiolCannabinoid receptor 1target
DB09061CannabidiolCannabinoid receptor 2target
DB09061CannabidiolG-protein coupled receptor 12target
DB09061CannabidiolGlycine receptor subunit alpha-1target
DB09061CannabidiolGlycine receptor (alpha-1/beta)target
DB09061CannabidiolGlycine receptor subunit alpha-3target
DB09061CannabidiolN-arachidonyl glycine receptortarget
DB09061CannabidiolG-protein coupled receptor 55target
DB09061Cannabidiol5-hydroxytryptamine receptor 1Atarget
DB09061Cannabidiol5-hydroxytryptamine receptor 2Atarget
DB09061CannabidiolNeuronal acetylcholine receptor subunit alpha-7target
DB09061CannabidiolDelta-type opioid receptortarget
DB09061CannabidiolMu-type opioid receptortarget
DB09061CannabidiolPeroxisome proliferator-activated receptor gammatarget
DB09061CannabidiolCytochrome P450 3A5enzyme
DB09061CannabidiolSerotonin N-acetyltransferaseenzyme
DB09061CannabidiolCytochrome P450 1A1enzyme
DB09061CannabidiolFatty-acid amide hydrolase 1enzyme
DB09061CannabidiolArachidonate 5-lipoxygenaseenzyme
DB09061CannabidiolArachidonate 15-lipoxygenaseenzyme
DB09061CannabidiolQuinone oxidoreductaseenzyme
DB09061CannabidiolMultidrug resistance-associated protein 1transporter
DB09061CannabidiolATP-binding cassette sub-family G member 2transporter
DB09061CannabidiolEquilibrative nucleoside transporter 1transporter
DB09061CannabidiolTransient receptor potential cation channel subfamily V member 1target
DB09061CannabidiolVoltage-dependent T-type calcium channel subunit alpha-1Gtarget
DB09061CannabidiolVoltage-dependent T-type calcium channel subunit alpha-1Htarget
DB09061CannabidiolVoltage-dependent T-type calcium channel subunit alpha-1Itarget
DB09061CannabidiolTransient receptor potential cation channel subfamily A member 1target
DB09061CannabidiolTransient receptor potential cation channel subfamily M member 8target
DB09061CannabidiolTransient receptor potential cation channel subfamily V member 2target
DB09061CannabidiolTransient receptor potential cation channel subfamily V member 3target
DB09061CannabidiolTransient receptor potential cation channel subfamily V member 4target
DB09061CannabidiolVoltage-dependent anion-selective channel protein 1target
DB09061Cannabidiol5-hydroxytryptamine receptor 3Atarget
DB09061CannabidiolAdenosine receptor A1target
DB09061CannabidiolProstaglandin G/H synthase 1target
DB09061CannabidiolProstaglandin G/H synthase 2target
DB09061CannabidiolAcetyl-CoA acetyltransferase, mitochondrialtarget
DB09061CannabidiolSteroid 17-alpha-hydroxylase/17,20 lyasetarget
DB09061Cannabidiol3-hydroxy-3-methylglutaryl-coenzyme A reductasetarget
DB09061CannabidiolGlutathione reductase, mitochondrialtarget
DB09061CannabidiolGlutathione peroxidase 1target
DB09061CannabidiolIndoleamine 2,3-dioxygenase 1target
DB09061CannabidiolCytochrome P450 1B1target
DB09061CannabidiolNAD(P)H dehydrogenase [quinone] 1target
DB09061CannabidiolCatalasetarget
DB09061CannabidiolCytochrome P450 3A5target
DB09061CannabidiolCytochrome P450 2D6target
DB09061CannabidiolSuperoxide dismutase [Cu-Zn]target
DB09061CannabidiolCytochrome P450 1A2target
DB09061CannabidiolCytochrome P450 3A7target
DB09061CannabidiolSerotonin N-acetyltransferasetarget
DB09061CannabidiolN-acylethanolamine-hydrolyzing acid amidasetarget
DB09061CannabidiolCytochrome P450 1A2enzyme
DB09061CannabidiolCytochrome P450 1B1enzyme
DB09061CannabidiolCytochrome P450 2A6enzyme
DB09061CannabidiolCytochrome P450 2B6enzyme
DB09061CannabidiolCytochrome P450 2C8enzyme
DB09061CannabidiolCytochrome P450 2E1enzyme
DB09061CannabidiolCytochrome P450 3A7enzyme
DB09061CannabidiolUDP-glucuronosyltransferase 1-7enzyme
DB09061CannabidiolUDP-glucuronosyltransferase 1-9enzyme
DB09061CannabidiolUDP-glucuronosyltransferase 2B7enzyme
DB09061CannabidiolUDP-glucuronosyltransferase 2B17enzyme
DB09061CannabidiolP-glycoprotein 1transporter
DB09061CannabidiolCytochrome P450 2J2enzyme
DB09061CannabidiolLiver carboxylesterase 1enzyme
DB00349ClobazamCytochrome P450 2C19enzyme
DB00349ClobazamCytochrome P450 3A4enzyme
DB00349ClobazamCytochrome P450 2B6enzyme
DB00349ClobazamCytochrome P450 2C18enzyme
DB00349ClobazamP-glycoprotein 1transporter
DB00349ClobazamGABA(A) Receptortarget
DB00349ClobazamCytochrome P450 2D6enzyme
DB00349ClobazamGABA(A) Receptor Benzodiazepine Binding Sitetarget
DB00349ClobazamSerum albumincarrier
DB00349ClobazamAlpha-1-acid glycoprotein 1carrier
DB00349ClobazamCytochrome P450 2C9enzyme
DB00349ClobazamUDP-glucuronosyltransferase 1-4enzyme
DB00349ClobazamUDP-glucuronosyltransferase 1-6enzyme
DB00349ClobazamUDP-glucuronosyltransferase 2B4enzyme
DB00349ClobazamUDP-glucuronosyltransferase 1-1enzyme
DB00349ClobazamCytochrome P450 1A2enzyme
DB00349ClobazamCytochrome P450 2C8enzyme
DB00349ClobazamCytochrome P450 3A5enzyme
DB00349ClobazamCytochrome P450 3A7enzyme
DB00574Fenfluramine5-hydroxytryptamine receptor 2Ctarget
DB00574Fenfluramine5-hydroxytryptamine receptor 2Btarget
DB00574FenfluramineCytochrome P450 2D6enzyme
DB00574FenfluramineSodium-dependent serotonin transportertarget
DB00574Fenfluramine5-hydroxytryptamine receptor 2Atarget
DB00574Fenfluramine5-hydroxytryptamine receptor 1Dtarget
DB00574FenfluramineSigma non-opioid intracellular receptor 1target
DB00574Fenfluramine5-hydroxytryptamine receptor 1Atarget
DB00574FenfluramineCytochrome P450 1A2enzyme
DB00574FenfluramineCytochrome P450 2B6enzyme
DB00574FenfluramineCytochrome P450 2C9enzyme
DB00574FenfluramineCytochrome P450 2C19enzyme
DB00574FenfluramineCytochrome P450 3A4enzyme
DB00574FenfluramineCytochrome P450 3A5enzyme
DB01320FosphenytoinSodium channel protein type 5 subunit alphatarget
DB01320FosphenytoinCytochrome P450 2C19enzyme
DB01320FosphenytoinCytochrome P450 2B6enzyme
DB01320FosphenytoinCytochrome P450 2C9enzyme
DB01320FosphenytoinCytochrome P450 3A4enzyme
DB01320FosphenytoinSerum albumincarrier
DB01320FosphenytoinCytochrome P450 1A2enzyme
DB01320FosphenytoinUDP-glucuronosyltransferase 1-6enzyme
DB01320FosphenytoinUDP-glucuronosyltransferase 1-9enzyme
DB01320FosphenytoinThyroxine-binding globulincarrier
DB05087GanaxoloneGABA(A) Receptortarget
DB05087GanaxoloneCytochrome P450 3A4enzyme
DB05087GanaxoloneCytochrome P450 3A5enzyme
DB05087GanaxoloneCytochrome P450 2B6enzyme
DB05087GanaxoloneCytochrome P450 2C19enzyme
DB05087GanaxoloneCytochrome P450 2D6enzyme
DB00252PhenytoinSodium channel protein type 5 subunit alphatarget
DB00252PhenytoinSodium channel protein type 1 subunit alphatarget
DB00252PhenytoinCytochrome P450 2C8enzyme
DB00252PhenytoinCytochrome P450 2C19enzyme
DB00252PhenytoinCytochrome P450 2C9enzyme
DB00252PhenytoinCytochrome P450 2B6enzyme
DB00252PhenytoinCytochrome P450 3A5enzyme
DB00252PhenytoinSerum albumincarrier
DB00252PhenytoinCytochrome P450 3A4enzyme
DB00252PhenytoinSolute carrier organic anion transporter family member 1C1transporter
DB00252PhenytoinP-glycoprotein 1transporter
DB00252PhenytoinCanalicular multispecific organic anion transporter 1transporter
DB00252PhenytoinCytochrome P450 11B1, mitochondrialenzyme
DB00252PhenytoinCytochrome P450 3A7enzyme
DB00252PhenytoinNuclear receptor subfamily 1 group I member 2target
DB00252PhenytoinSodium channel subunit beta-1target
DB00252PhenytoinSodium channel protein type 3 subunit alphatarget
DB00252PhenytoinUDP-glucuronosyltransferase 1-1enzyme
DB00252PhenytoinUDP-glucuronosyltransferase 1-6enzyme
DB00252PhenytoinUDP-glucuronosyltransferase 1-9enzyme
DB00252PhenytoinThyroxine-binding globulincarrier
DB00252PhenytoinPotassium voltage-gated channel subfamily H member 2target
DB00252PhenytoinVoltage-dependent L-type calcium channeltarget
DB00252PhenytoinSodium channel protein type 2 subunit alphatarget
DB00252PhenytoinSodium channel protein type 8 subunit alphatarget
DB00252PhenytoinGABA(A) Receptortarget
DB00252PhenytoinCytochrome P450 1A2enzyme
DB00252PhenytoinCytochrome P450 2A6enzyme
DB00252PhenytoinCytochrome P450 2D6enzyme
DB00252PhenytoinCytochrome P450 2E1enzyme
DB00252PhenytoinEpoxide hydrolase 1enzyme
DB00252PhenytoinUDP-glucuronosyltransferase 1-4enzyme
DB00252PhenytoinCatechol O-methyltransferaseenzyme
DB00252PhenytoinNAD(P)H dehydrogenase [quinone] 1enzyme
DB00252PhenytoinCytochrome P450 2C18enzyme
DB09118StiripentolCytochrome P450 2C19enzyme
DB09118StiripentolCytochrome P450 2D6enzyme
DB09118StiripentolCytochrome P450 3A4enzyme
DB09118StiripentolCytochrome P450 1A2enzyme
DB09118StiripentolCytochrome P450 2C9enzyme
DB09118StiripentolGABA(A) Receptortarget
DB09118StiripentolL-lactate dehydrogenase A chaintarget
DB09118StiripentolL-lactate dehydrogenase B chaintarget
DB09118StiripentolCytochrome P450 2B6enzyme
DB09118StiripentolCytochrome P450 2C8enzyme
DB09118StiripentolP-glycoprotein 1transporter
DB09118StiripentolATP-binding cassette sub-family G member 2transporter
DB00599ThiopentalGamma-aminobutyric acid receptor subunit alpha-1target
DB00599ThiopentalFatty-acid amide hydrolase 1target
DB00599ThiopentalGamma-aminobutyric acid receptor subunit alpha-2target
DB00599ThiopentalGamma-aminobutyric acid receptor subunit alpha-3target
DB00599ThiopentalGamma-aminobutyric acid receptor subunit alpha-4target
DB00599ThiopentalGamma-aminobutyric acid receptor subunit alpha-5target
DB00599ThiopentalGamma-aminobutyric acid receptor subunit alpha-6target
DB00599ThiopentalNeuronal acetylcholine receptor subunit alpha-4target
DB00599ThiopentalNeuronal acetylcholine receptor subunit alpha-7target
DB00599ThiopentalGlutamate receptor 2target
DB00599ThiopentalGlutamate receptor ionotropic, kainate 2target
DB00599ThiopentalCytochrome P450 3A Subfamilyenzyme
DB00599ThiopentalMuscarinic acetylcholine receptor M3target
DB00599ThiopentalCytochrome P450 2C19enzyme
DB00697TizanidineAlpha-2 adrenergic receptorstarget
DB00697TizanidineCytochrome P450 1A2enzyme
DB00697TizanidineNischarintarget
DB00697TizanidineAlpha-1 adrenergic receptorstarget
DB00273TopiramateGamma-aminobutyric acid receptor subunit alpha-1target
DB00273TopiramateVoltage-gated sodium channel alpha subunittarget
DB00273TopiramateCarbonic anhydrase 2target
DB00273TopiramateCarbonic anhydrase 4target
DB00273TopiramateKainate receptorstarget
DB00273TopiramateCytochrome P450 2C19enzyme
DB00273TopiramateCytochrome P450 3A4enzyme
DB00273TopiramateCarbonic anhydrase 1target
DB00273TopiramateCarbonic anhydrase 3target
DB00273TopiramateVoltage gated L-type calcium channeltarget
DB00273TopiramateVoltage-dependent R-type calcium channeltarget
DB00273TopiramateSerum albumincarrier
DB00273TopiramateP-glycoprotein 1transporter
DB00273Topiramate5'-AMP-activated protein kinasetransporter
DrugDrug NamePhaseStatusCount
DB00829Diazepam0Completed1
DB00683Midazolam0Completed1
DB00747Scopolamine0Recruiting1
DB00887Bumetanide1Completed1
DB09061Cannabidiol1Completed2
DB01202Levetiracetam1Completed1
DB00683Midazolam1Completed1
DB00776Oxcarbazepine1Completed2
DB06201Rufinamide1Completed1
DB00273Topiramate1Completed1
DB00313Valproic acid1Completed1
DB09061Cannabidiol1 / 2Completed1
DB00555Lamotrigine1 / 2Completed1
DB01202Levetiracetam1 / 2Completed5
DB08883Perampanel1 / 2Completed1
DB00316Acetaminophen2Completed1
DB00490Buspirone2Terminated1
DB00349Clobazam2Completed1
DB00829Diazepam2Completed1
DB00254Doxycycline2Unknown Status1
DB01050Ibuprofen2Completed1
DB01202Levetiracetam2Completed2
DB14009Medical Cannabis2Recruiting1
DB00683Midazolam2Completed1
DB08883Perampanel2Completed1
DB00230Pregabalin2Completed1
DB12646SGS-7422Completed1
DB12367Selurampanel2Completed1
DB00273Topiramate2Completed5
DB00169Cholecalciferol2 / 3Completed1
DB01202Levetiracetam2 / 3Withdrawn1
DB00186Lorazepam2 / 3Withdrawn1
DB09061Cannabidiol3Completed3
DB00564Carbamazepine3Completed2
DB12338Carisbamate3Recruiting1
DB12338Carisbamate3Terminated1
DB00349Clobazam3Completed1
DB00829Diazepam3Completed1
DB00593Ethosuximide3Completed1
DB04953Ezogabine3Completed2
DB00996Gabapentin3Completed1
DB00555Lamotrigine3Completed2
DB01202Levetiracetam3Not Yet Recruiting1
DB01202Levetiracetam3Terminated1
DB00186Lorazepam3Completed1
DB00683Midazolam3Recruiting1
DB00230Pregabalin3Completed1
DB00273Topiramate3Completed10
DB00273Topiramate3Terminated1
DB00302Tranexamic acid3Terminated1
DB00313Valproic acid3Completed2
DB00829Diazepam4Not Yet Recruiting1
DB04953Ezogabine4Terminated1
DB06218Lacosamide4Terminated1
DB01202Levetiracetam4Completed2
DB01202Levetiracetam4Terminated1
DB01202Levetiracetam4Unknown Status1
DB01202Levetiracetam4Withdrawn1
DB00683Midazolam4Completed1
DB00683Midazolam4Not Yet Recruiting1
DB08883Perampanel4Recruiting1
DB00252Phenytoin4Terminated3
DB00230Pregabalin4Completed1
DB00273Topiramate4Completed1
DB00802AlfentanilNot AvailableCompleted1
DB00479AmikacinNot AvailableCompleted1
DB00513Aminocaproic acidNot AvailableCompleted1
DB00559BosentanNot AvailableCompleted1
DB00201CaffeineNot AvailableRecruiting1
DB09061CannabidiolNot AvailableRecruiting1
DB00564CarbamazepineNot AvailableCompleted1
DB09157Carbon dioxideNot AvailableRecruiting1
DB01413CefepimeNot AvailableCompleted1
DB00369CidofovirNot AvailableCompleted1
DB00537CiprofloxacinNot AvailableCompleted1
DB00363ClozapineNot AvailableCompleted1
DB00151CysteineNot AvailableWithdrawn1
DB00633DexmedetomidineNot AvailableCompleted1
DB00828FosfomycinNot AvailableCompleted1
DB00502HaloperidolNot AvailableCompleted1
DB01221KetamineNot AvailableCompleted1
DB00598LabetalolNot AvailableCompleted1
DB06218LacosamideNot AvailableCompleted1
DB06218LacosamideNot AvailableEnrolling by Invitation1
DB01202LevetiracetamNot AvailableCompleted7
DB01202LevetiracetamNot AvailableWithdrawn1
DB08815LurasidoneNot AvailableCompleted1
DB00422MethylphenidateNot AvailableRecruiting1
DB00959MethylprednisoloneNot AvailableCompleted1
DB01618MolindoneNot AvailableCompleted1
DB00607NafcillinNot AvailableCompleted1
DB01115NifedipineNot AvailableCompleted1
DB00776OxcarbazepineNot AvailableCompleted3
DB00497OxycodoneNot AvailableCompleted1
DB00312PentobarbitalNot AvailableCompleted1
DB08883PerampanelNot AvailableCompleted1
DB00319PiperacillinNot AvailableCompleted1
DB13831Potassium permanganateNot AvailableCompleted1
DB00818PropofolNot AvailableCompleted1
DB00899RemifentanilNot AvailableCompleted1
DB00728RocuroniumNot AvailableCompleted1
DB00658SevelamerNot AvailableCompleted1
DB00421SpironolactoneNot AvailableCompleted1
DB01606TazobactamNot AvailableCompleted1
DB00684TobramycinNot AvailableCompleted1
DB00273TopiramateNot AvailableCompleted2
DB00302Tranexamic acidNot AvailableActive Not Recruiting1
DB00302Tranexamic acidNot AvailableCompleted1
DB00313Valproic acidNot AvailableCompleted2
DB00512VancomycinNot AvailableCompleted1
DB01339VecuroniumNot AvailableCompleted1
DB00661VerapamilNot AvailableUnknown Status1
DB00682WarfarinNot AvailableCompleted1
DB00246ZiprasidoneNot AvailableCompleted1
DB00425ZolpidemNot AvailableCompleted1