| DB01544 | Flunitrazepam | approved, illicit | yes | potentiator | Details |
| DB00829 | Diazepam | approved, illicit, investigational, vet_approved | yes | potentiator | Details |
| DB01567 | Fludiazepam | experimental, illicit | yes | potentiator | Details |
| DB01558 | Bromazepam | approved, illicit, investigational | yes | potentiator | Details |
| DB00371 | Meprobamate | approved, illicit | yes | agonist | Details |
| DB00683 | Midazolam | approved, illicit | yes | potentiator | Details |
| DB00690 | Flurazepam | approved, illicit, investigational | yes | potentiator | Details |
| DB04903 | Pagoclone | investigational | unknown | | Details |
| DB05087 | Ganaxolone | investigational | unknown | | Details |
| DB00404 | Alprazolam | approved, illicit, investigational | unknown | ligand | Details |
| DB00842 | Oxazepam | approved | yes | potentiator | Details |
| DB00425 | Zolpidem | approved | unknown | agonist | Details |
| DB00402 | Eszopiclone | approved, investigational | unknown | agonist | Details |
| DB00231 | Temazepam | approved, investigational | yes | potentiator | Details |
| DB01595 | Nitrazepam | approved | yes | potentiator | Details |
| DB00897 | Triazolam | approved, investigational | yes | potentiator | Details |
| DB01198 | Zopiclone | approved | yes | potentiator | Details |
| DB01559 | Clotiazepam | approved, illicit | yes | potentiator | Details |
| DB01588 | Prazepam | approved, illicit | yes | potentiator | Details |
| DB01594 | Cinolazepam | experimental | yes | potentiator | Details |
| DB01589 | Quazepam | approved, illicit | yes | potentiator | Details |
| DB01215 | Estazolam | approved, illicit | yes | potentiator | Details |
| DB00801 | Halazepam | approved, illicit, withdrawn | yes | potentiator | Details |
| DB00546 | Adinazolam | experimental | yes | potentiator | Details |
| DB01351 | Amobarbital | approved, illicit | yes | potentiator | Details |
| DB00312 | Pentobarbital | approved, investigational, vet_approved | yes | potentiator | Details |
| DB00241 | Butalbital | approved, illicit | yes | potentiator | Details |
| DB00306 | Talbutal | approved, illicit | yes | potentiator | Details |
| DB00418 | Secobarbital | approved, vet_approved | yes | potentiator | Details |
| DB00463 | Metharbital | withdrawn | yes | potentiator | Details |
| DB00599 | Thiopental | approved, vet_approved | yes | potentiator | Details |
| DB00794 | Primidone | approved, vet_approved | yes | potentiator | Details |
| DB00849 | Methylphenobarbital | approved | yes | potentiator | Details |
| DB01352 | Aprobarbital | experimental, illicit | yes | potentiator | Details |
| DB01353 | Butobarbital | approved, illicit | yes | potentiator | Details |
| DB01354 | Heptabarbital | experimental | yes | potentiator | Details |
| DB01355 | Hexobarbital | experimental | yes | potentiator | Details |
| DB01483 | Barbital | illicit | yes | potentiator | Details |
| DB01496 | Barbituric acid derivative | experimental, illicit | yes | potentiator | Details |
| DB01346 | Quinidine barbiturate | approved | yes | potentiator | Details |
| DB00898 | Ethanol | approved | unknown | | Details |
| DB09166 | Etizolam | experimental | yes | agonist | Details |
| DB13872 | Lormetazepam | approved | yes | positive allosteric modulator | Details |
| DB13994 | AZD-7325 | investigational | yes | positive allosteric modulator | Details |