| DB01567 | Fludiazepam | experimental, illicit | yes | potentiator | Details |
| DB00371 | Meprobamate | approved, illicit | yes | agonist | Details |
| DB04903 | Pagoclone | investigational | unknown | | Details |
| DB05087 | Ganaxolone | investigational | unknown | | Details |
| DB00425 | Zolpidem | approved | unknown | agonist | Details |
| DB00402 | Eszopiclone | approved, investigational | unknown | agonist | Details |
| DB01198 | Zopiclone | approved | yes | potentiator | Details |
| DB01351 | Amobarbital | approved, illicit | yes | potentiator | Details |
| DB00312 | Pentobarbital | approved, investigational, vet_approved | yes | potentiator | Details |
| DB00241 | Butalbital | approved, illicit | yes | potentiator | Details |
| DB00306 | Talbutal | approved, illicit | yes | potentiator | Details |
| DB00418 | Secobarbital | approved, vet_approved | yes | potentiator | Details |
| DB00463 | Metharbital | withdrawn | yes | potentiator | Details |
| DB00599 | Thiopental | approved, vet_approved | yes | potentiator | Details |
| DB00794 | Primidone | approved, vet_approved | yes | potentiator | Details |
| DB00849 | Methylphenobarbital | approved | yes | potentiator | Details |
| DB01352 | Aprobarbital | experimental, illicit | yes | potentiator | Details |
| DB01353 | Butobarbital | approved, illicit | yes | potentiator | Details |
| DB01354 | Heptabarbital | experimental | yes | potentiator | Details |
| DB01355 | Hexobarbital | experimental | yes | potentiator | Details |
| DB01483 | Barbital | illicit | yes | potentiator | Details |
| DB01496 | Dihydro-2-thioxo-5-((5-(2-(trifluoromethyl)phenyl)-2-furanyl)methyl)-4,6(1H,5H)-pyrimidinedione | experimental, illicit | yes | potentiator | Details |
| DB01346 | Quinidine barbiturate | approved | yes | potentiator | Details |
| DB00898 | Ethanol | approved | unknown | | Details |
| DB13994 | AZD-7325 | investigational | yes | positive allosteric modulator | Details |