| DB04851 | Biricodar dicitrate | investigational | unknown | | Details |
| DB00317 | Gefitinib | approved, investigational | unknown | substrateinhibitor | Details |
| DB04216 | Quercetin | experimental, investigational | unknown | inhibitor | Details |
| DB00661 | Verapamil | approved | unknown | inhibitor | Details |
| DB03467 | Naringenin | experimental | unknown | inhibitor | Details |
| DB01030 | Topotecan | approved, investigational | unknown | substrateinhibitor | Details |
| DB01051 | Novobiocin | approved, investigational, vet_approved | unknown | inhibitor | Details |
| DB00655 | Estrone | approved | unknown | inhibitor | Details |
| DB01232 | Saquinavir | approved, investigational | unknown | inhibitor | Details |
| DB00338 | Omeprazole | approved, investigational, vet_approved | unknown | inhibitor | Details |
| DB01094 | Hesperetin | approved | unknown | inhibitor | Details |
| DB01645 | Genistein | investigational | unknown | inhibitor | Details |
| DB00220 | Nelfinavir | approved | unknown | inhibitor | Details |
| DB01016 | Glyburide | approved | unknown | substrateinhibitor | Details |
| DB00255 | Diethylstilbestrol | approved, investigational | unknown | inhibitor | Details |
| DB00503 | Ritonavir | approved, investigational | unknown | inhibitor | Details |
| DB00175 | Pravastatin | approved | unknown | substrateinhibitor | Details |
| DB00997 | Doxorubicin | approved, investigational | unknown | substrateinhibitor | Details |
| DB00213 | Pantoprazole | approved | unknown | inhibitor | Details |
| DB00091 | Cyclosporine | approved, investigational, vet_approved | unknown | inhibitor | Details |
| DB04348 | Taurocholic Acid | experimental | unknown | inhibitor | Details |
| DB00619 | Imatinib | approved | unknown | substrateinhibitor | Details |
| DB00741 | Hydrocortisone | approved, vet_approved | unknown | inhibitor | Details |
| DB00783 | Estradiol | approved, investigational, vet_approved | unknown | inhibitor | Details |
| DB01204 | Mitoxantrone | approved, investigational | unknown | substrateinhibitor | Details |
| DB02115 | Daidzin | experimental | unknown | inhibitor | Details |
| DB00398 | Sorafenib | approved, investigational | unknown | substrateinhibitor | Details |
| DB01268 | Sunitinib | approved, investigational | unknown | inhibitor | Details |
| DB00470 | Dronabinol | approved, illicit | unknown | inhibitor | Details |
| DB00921 | Buprenorphine | approved, illicit, investigational, vet_approved | unknown | inhibitor | Details |
| DB00795 | Sulfasalazine | approved | unknown | substrateinhibitor | Details |
| DB00966 | Telmisartan | approved, investigational | unknown | inhibitor | Details |
| DB01234 | Dexamethasone | approved, investigational, vet_approved | unknown | inhibitor | Details |
| DB01254 | Dasatinib | approved, investigational | unknown | substrateinhibitor | Details |
| DB00457 | Prazosin | approved | unknown | substrateinhibitor | Details |
| DB00448 | Lansoprazole | approved, investigational | unknown | inhibitor | Details |
| DB01129 | Rabeprazole | approved, investigational | unknown | inhibitor | Details |
| DB04881 | Elacridar | investigational | unknown | inhibitor | Details |
| DB04868 | Nilotinib | approved, investigational | unknown | substrateinhibitor | Details |
| DB00530 | Erlotinib | approved, investigational | unknown | inhibitor | Details |
| DB05294 | Vandetanib | approved | unknown | inhibitor | Details |
| DB00709 | Lamivudine | approved, investigational | unknown | substrate | Details |
| DB00762 | Irinotecan | approved, investigational | unknown | substrate | Details |
| DB00773 | Etoposide | approved | unknown | substrate | Details |
| DB00970 | Dactinomycin | approved, investigational | unknown | substrate | Details |
| DB00286 | Conjugated estrogens | approved | unknown | substrate | Details |
| DB00439 | Cerivastatin | approved, withdrawn | unknown | substrate | Details |
| DB00624 | Testosterone | approved, investigational | unknown | substrate | Details |
| DB00675 | Tamoxifen | approved | unknown | substrate | Details |
| DB00669 | Sumatriptan | approved, investigational | unknown | substrate | Details |
| DB00694 | Daunorubicin | approved | unknown | substrate | Details |
| DB04540 | Cholesterol | approved, experimental, investigational | unknown | substrate | Details |
| DB00563 | Methotrexate | approved | unknown | substrate | Details |
| DB00158 | Folic Acid | approved, nutraceutical, vet_approved | unknown | substrate | Details |
| DB03496 | Alvocidib | experimental, investigational | unknown | substrate | Details |
| DB00541 | Vincristine | approved, investigational | unknown | substrate | Details |
| DB00444 | Teniposide | approved | unknown | substrate | Details |
| DB00698 | Nitrofurantoin | approved, vet_approved | unknown | substrate | Details |
| DB00602 | Ivermectin | approved, investigational, vet_approved | unknown | substrate | Details |
| DB04690 | Camptothecin | experimental | unknown | substrate | Details |
| DB00740 | Riluzole | approved, investigational | unknown | substrate | Details |
| DB00242 | Cladribine | approved, investigational | unknown | substrate | Details |
| DB00631 | Clofarabine | approved, investigational | unknown | substrate | Details |
| DB00526 | Oxaliplatin | approved, investigational | unknown | substrate | Details |
| DB06772 | Cabazitaxel | approved | unknown | inhibitor | Details |
| DB08860 | Pitavastatin | approved | unknown | substrate | Details |
| DB06589 | Pazopanib | approved | unknown | substrate | Details |
| DB08864 | Rilpivirine | approved | unknown | inhibitor | Details |
| DB08880 | Teriflunomide | approved | unknown | substrate | Details |
| DB01097 | Leflunomide | approved, investigational | unknown | substrate | Details |
| DB08881 | Vemurafenib | approved | unknown | substrate | Details |
| DB06605 | Apixaban | approved | unknown | substrate | Details |
| DB08828 | Vismodegib | approved, investigational | unknown | inhibitor | Details |
| DB08896 | Regorafenib | approved | unknown | inhibitor | Details |
| DB08901 | Ponatinib | approved, investigational | unknown | substrateinhibitor | Details |
| DB00973 | Ezetimibe | approved | unknown | substrate | Details |
| DB08912 | Dabrafenib | approved, investigational | unknown | substrateinhibitor | Details |
| DB00549 | Zafirlukast | approved, investigational | unknown | Antagonist | Details |
| DB00285 | Venlafaxine | approved | unknown | inducer | Details |
| DB00495 | Zidovudine | approved | unknown | substrate | Details |
| DB08916 | Afatinib | approved | unknown | substrateinhibitor | Details |
| DB00544 | Fluorouracil | approved | unknown | substrate | Details |
| DB00688 | Mycophenolate mofetil | approved, investigational | unknown | substrate | Details |
| DB00515 | Cisplatin | approved | unknown | substrate | Details |
| DB00958 | Carboplatin | approved | unknown | substrate | Details |
| DB01098 | Rosuvastatin | approved | unknown | substrate | Details |
| DB01229 | Paclitaxel | approved, vet_approved | unknown | substrate | Details |
| DB01248 | Docetaxel | approved, investigational | unknown | substrate | Details |
| DB08934 | Sofosbuvir | approved | no | substrate | Details |
| DB09078 | Lenvatinib | approved, investigational | no | substrate | Details |
| DB09054 | Idelalisib | approved | no | substrate | Details |
| DB09065 | Cobicistat | approved | yes | inhibitor | Details |
| DB09291 | Rolapitant | approved, investigational | no | inhibitor | Details |
| DB09102 | Daclatasvir | approved, investigational | unknown | inhibitor | Details |
| DB05239 | Cobimetinib | approved, investigational | unknown | weak inhibitor | Details |
| DB09330 | Osimertinib | approved | no | substrate | Details |
| DB11363 | Alectinib | approved, investigational | no | inhibitor | Details |
| DB08931 | Riociguat | approved | yes | substrate | Details |
| DB09183 | Dasabuvir | approved | unknown | inhibitor | Details |
| DB11581 | Venetoclax | approved, investigational | no | substrate | Details |
| DB06654 | Safinamide | approved, investigational | unknown | substrate | Details |
| DB11613 | Velpatasvir | approved, investigational | no | substrateinhibitor | Details |
| DB06290 | Simeprevir | approved | unknown | substrateinhibitor | Details |
| DB09027 | Ledipasvir | approved | no | transporter | Details |
| DB09296 | Ombitasvir | approved, investigational | no | substrate | Details |
| DB11943 | Delafloxacin | approved, investigational | no | substrate | Details |
| DB01685 | Topiroxostat | approved, investigational | unknown | inhibitor | Details |
| DB12026 | Voxilaprevir | approved, investigational | no | substrateinhibitor | Details |
| DB13874 | Enasidenib | approved, investigational | unknown | substrateinhibitor | Details |
| DB13878 | Pibrentasvir | approved, investigational | unknown | substrateinhibitor | Details |
| DB13879 | Glecaprevir | approved, investigational | unknown | substrateinhibitor | Details |
| DB12483 | Copanlisib | approved, investigational | unknown | substrate | Details |
| DB12001 | Abemaciclib | approved, investigational | unknown | substrateinhibitor | Details |
| DB12070 | Letermovir | approved, investigational | no | inhibitor | Details |
| DB12267 | Brigatinib | approved, investigational | no | substrateinhibitor | Details |
| DB08930 | Dolutegravir | approved | no | substrate | Details |
| DB12332 | Rucaparib | approved, investigational | unknown | substrateinhibitor | Details |
| DB11817 | Baricitinib | approved, investigational | unknown | substrateinhibitor | Details |
| DB09061 | Cannabidiol | approved, investigational | unknown | inhibitor | Details |
| DB11827 | Ertugliflozin | approved, investigational | unknown | substrate | Details |
| DB13943 | Testosterone cypionate | approved | unknown | substrate | Details |
| DB13944 | Testosterone enanthate | approved | unknown | substrate | Details |
| DB13946 | Testosterone undecanoate | approved, investigational | unknown | substrate | Details |
| DB13952 | Estradiol acetate | approved, investigational, vet_approved | unknown | inhibitor | Details |
| DB13953 | Estradiol benzoate | approved, investigational, vet_approved | unknown | inhibitor | Details |
| DB13954 | Estradiol cypionate | approved, investigational, vet_approved | unknown | inhibitor | Details |
| DB13955 | Estradiol dienanthate | approved, investigational, vet_approved | unknown | inhibitor | Details |
| DB13956 | Estradiol valerate | approved, investigational, vet_approved | unknown | inhibitor | Details |
| DB11901 | Apalutamide | approved, investigational | unknown | inducer | Details |
| DB11633 | Isavuconazole | approved, investigational | unknown | inhibitor | Details |
| DB14011 | Nabiximols | approved | unknown | inhibitor | Details |
| DB14009 | Medical Cannabis | experimental | unknown | inhibitor | Details |