HIV Integrase Inhibitors

Name
HIV Integrase Inhibitors
Accession Number
DBCAT001873
Description

Inhibitors of HIV INTEGRASE, an enzyme required for integration of viral DNA into cellular DNA.

Drugs
DrugDrug Description
RaltegravirAn antiretroviral agent used for the treatment of HIV infections in conjunction with other antiretrovirals.
DolutegravirAn antiviral agent used for the treatment of HIV-1 infections in combination with other antiretroviral agents.
ElvitegravirAn antiretroviral agent used in combination with other antiretrovirals for the treatment of HIV-1 infection in antiretroviral treatment-experienced adults.
HIV Integrase InhibitorHIV Integrase Inhibitor is under investigation in clinical trial NCT00397566 (A Multiple Ascending Dose Study of BMS-707035 in HIV-1 Infected Subjects).
CabotegravirAn HIV-1 integrase inhibitor used for treatment and pre-exposure prophylaxis of HIV-1 infection.
Drugs & Drug Targets
DrugTargetType
RaltegravirUDP-glucuronosyltransferase 1-1enzyme
RaltegravirIntegrasetarget
DolutegravirUDP-glucuronosyltransferase 1-1enzyme
DolutegravirCytochrome P450 3A Subfamilyenzyme
DolutegravirIntegrasetarget
DolutegravirSolute carrier family 22 member 2transporter
DolutegravirUDP-glucuronosyltransferase 1-3enzyme
DolutegravirUDP-glucuronosyltransferase 1-9enzyme
DolutegravirATP-binding cassette sub-family G member 2transporter
DolutegravirSolute carrier family 22 member 6transporter
DolutegravirSolute carrier family 22 member 8transporter
DolutegravirP-glycoprotein 1transporter
DolutegravirMultidrug and toxin extrusion protein 1transporter
DolutegravirSerum albumincarrier
Dolutegraviralpha1-acid glycoproteincarrier
ElvitegravirIntegrasetarget
ElvitegravirCytochrome P450 3A4enzyme
ElvitegravirUDP-glucuronosyltransferase 1-1enzyme
CabotegravirSolute carrier family 22 member 6transporter
CabotegravirSolute carrier family 22 member 8transporter
CabotegravirUDP-glucuronosyltransferase 1-1enzyme
CabotegravirUDP-glucuronosyltransferase 1-9enzyme
CabotegravirP-glycoprotein 1transporter
CabotegravirATP-binding cassette sub-family G member 2transporter
CabotegravirSerum albumincarrier
CabotegravirIntegrasetarget