Androstan Derivatives

DrugDrug NameDrug Description
DB00621OxandroloneAn androgenic hormone used to treat muscle loss from prolonged corticosteroid treatment and to treat bone pain associated with osteoporosis.
DB06412OxymetholoneAn anabolic steroid used for the treatment of types of anemia, such as acquired aplastic anemia, congenital aplastic anemia, myelofibrosis, and the hypoplastic anemias.
DB06718StanozololStanozolol is a synthetic anabolic steroid with therapeutic uses in treating C1-inhibitor deficient hereditary angioedema. C1-inhibitor is a protease that inhibits the complement system (part of the innate immune system),...
DB12787NorethandroloneNorethandrolone is under investigation in clinical trial NCT00700544 (Treatment Outcome in Elderly Patients).
DB13484QuinboloneNot Annotated
DB13586MetandienoneNot Annotated
DB13710MetenoloneNot Annotated
DB01708PrasteroneA steroid formulated as a vaginal insert indicated for the treatment of moderate to severe dyspareunia associated with menopausal vulvar and vaginal atrophy.
DB02901StanoloneA potent androgenic metabolite of testosterone. Dihydrotestosterone (DHT) is generated by a 5-alpha reduction of testosterone. Unlike testosterone, DHT cannot be aromatized to estradiol therefore DHT is considered a pure...
DrugDrug NameTargetType
DB00621OxandroloneAndrogen receptortarget
DB00621OxandroloneCytochrome P450 2C9enzyme
DB06412OxymetholoneAndrogen receptortarget
DB06412OxymetholoneSerum albumincarrier
DB06412OxymetholoneSex hormone-binding globulincarrier
DB06412OxymetholoneNatriuretic peptides Btarget
DB06412OxymetholoneAmine oxidase [flavin-containing] Aenzyme
DB06412OxymetholoneCytochrome P450 2D6enzyme
DB06412Oxymetholone3-oxo-5-alpha-steroid 4-dehydrogenase 1enzyme
DB06412OxymetholoneCytochrome P450 3A4enzyme
DB06412OxymetholoneCytochrome P450 3A5enzyme
DB06412OxymetholoneCytochrome P450 3A7enzyme
DB06412OxymetholoneCytochrome P450 3A43enzyme
DB06718StanozololGlucocorticoid binding proteinstarget
DB06718StanozololAndrogen receptortarget
DB01708PrasteroneSteroid Delta-isomerasetarget
DB01708PrasteroneBile salt sulfotransferasetarget
DB01708PrasteroneCholesterol oxidasetarget
DB01708PrasteroneEstradiol 17-beta-dehydrogenase 1target
DB01708PrasteroneSulfotransferase family cytosolic 2B member 1target
DB01708PrasteroneCytochrome P450 3A7enzyme
DB01708PrasteronePeroxisome proliferator-activated receptor alphatarget
DB01708PrasteroneEstrogen receptor alphatarget
DB01708PrasteroneSigma non-opioid intracellular receptor 1target
DB01708PrasteroneEstrogen receptor betatarget
DB01708PrasteroneNuclear receptor subfamily 1 group I member 2target
DB01708PrasteroneNuclear receptor subfamily 1 group I member 3target
DB01708PrasteroneGABA-A receptor (anion channel)target
DB01708PrasteroneNMDA receptortarget
DB01708PrasteroneAndrogen receptortarget
DB02901StanoloneSex hormone-binding globulincarrier
DB02901StanoloneAndrogen receptortarget
DB02901StanoloneEstradiol 17-beta-dehydrogenase 1target
DB02901StanoloneP-glycoprotein 1transporter
DB02901StanoloneCholesterol side-chain cleavage enzyme, mitochondrialenzyme
DB02901StanoloneSteroid 17-alpha-hydroxylase/17,20 lyaseenzyme
DB02901StanoloneCytochrome P450 19A1enzyme
DB02901StanoloneEstrogen receptor alphatarget
DB02901StanoloneMineralocorticoid receptortarget