Receptors, LHRH, antagonists & inhibitors

Name
Receptors, LHRH, antagonists & inhibitors
Accession Number
DBCAT002787  (DBCAT003827)
Description

Not Available

Drugs
DrugDrug Description
RelugolixAn oral GnRH receptor antagonist for androgen deprivation therapy in the treatment of advanced prostate cancer.
Drugs & Drug Targets
DrugTargetType
RelugolixSerum albumincarrier
RelugolixAlpha-1-acid glycoprotein 1carrier
RelugolixP-glycoprotein 1transporter
RelugolixATP-binding cassette sub-family G member 2transporter
RelugolixCytochrome P450 3A Subfamilyenzyme
RelugolixCytochrome P450 2C8enzyme
RelugolixCytochrome P450 2B6enzyme
RelugolixGonadotropin-releasing hormone receptortarget