Histamine H3 Antagonists

Name
Histamine H3 Antagonists
Accession Number
DBCAT002803
Description

Not Available

Drugs
DrugDrug Description
PF-03654746PF-03654746 has been investigated for the treatment of Narcolepsy, Schizophrenia, Tourette's Syndrome, and Excessive Daytime Sleepiness.
BavisantBavisant has been used in trials studying the basic science and treatment of Alcoholism, Pharmacokinetics, Drug Interactions, Attention Deficit Hyperactivity Disorder, and Attention Deficit Disorders With Hyperactivity.
PF-03654764PF-03654764 has been used in trials studying the basic science and treatment of Allergic Rhinitis.
JNJ-39220675JNJ-39220675 has been used in trials studying the treatment of Allergic Rhinitis.
ViloxazineA selective norepinephrine reuptake inhibitor indicated for the treatment of Attention Deficit Hyperactivity Disorder (ADHD) in adults in children.
PitolisantAn antagonist and inverse agonist at the histamine H3 receptor that is used to treat narcolepsy in adults.
Drugs & Drug Targets
DrugTargetType
ViloxazineSodium-dependent noradrenaline transportertarget
ViloxazineCytochrome P450 1A2enzyme
ViloxazineCytochrome P450 2D6enzyme
ViloxazineUDP-glucuronosyltransferase 1-9enzyme
ViloxazineUDP-glucuronosyltransferase 2B15enzyme
ViloxazineCytochrome P450 2B6enzyme
ViloxazineCytochrome P450 3A4enzyme
ViloxazineCytochrome P450 3A5enzyme
ViloxazineMultidrug and toxin extrusion protein 1transporter
Viloxazine5-hydroxytryptamine receptor 2Btarget
Viloxazine5-hydroxytryptamine receptor 2Ctarget
ViloxazineAlpha-1B adrenergic receptortarget
ViloxazineBeta-2 adrenergic receptortarget
ViloxazineAmine oxidase [flavin-containing] Atarget
ViloxazineAmine oxidase [flavin-containing] Btarget
ViloxazineHistamine H1 receptortarget
ViloxazineHistamine H2 receptortarget
ViloxazineMuscarinic acetylcholine receptor M1target
ViloxazineMuscarinic acetylcholine receptor M2target
ViloxazineMuscarinic acetylcholine receptor M3target
ViloxazineMuscarinic acetylcholine receptor M4target
PitolisantHistamine H3 receptortarget
PitolisantCytochrome P450 3A4enzyme
PitolisantCytochrome P450 2D6enzyme
PitolisantCytochrome P450 1A2enzyme
PitolisantCytochrome P450 2B6enzyme
PitolisantSolute carrier family 22 member 1transporter
PitolisantPotassium voltage-gated channel subfamily H member 2target
PitolisantSerum albumincarrier
PitolisantAlpha-1-acid glycoprotein 1carrier