Cystic Fibrosis Transmembrane Conductance Regulator Potentiators

Name
Cystic Fibrosis Transmembrane Conductance Regulator Potentiators
Accession Number
DBCAT003776  (DBCAT003486)
Description

Not Available

Drugs
DrugDrug Description
IvacaftorA cystic fibrosis transmembrane conductance regulator (CFTR) potentiator used alone or in combination products to treat cystic fibrosis in patients who have specific genetic mutations that are responsive to the medication.
Drugs & Drug Targets
DrugTargetType
IvacaftorCystic fibrosis transmembrane conductance regulatortarget
IvacaftorCytochrome P450 3A4enzyme
IvacaftorSerum albumincarrier
IvacaftorAlpha-1-acid glycoprotein 1carrier
IvacaftorP-glycoprotein 1transporter
IvacaftorCytochrome P450 3A5enzyme
IvacaftorCytochrome P450 2C9enzyme