Genitourinary Smooth Muscle Relaxants

Name
Genitourinary Smooth Muscle Relaxants
Accession Number
DBCAT003744
Description

Not Available

Drugs
DrugDrug Description
TolterodineA muscarinic receptor antagonist used to treat overactive bladder with urinary incontinence, urgency, and frequency.
VibegronA beta-3 adrenergic agonist the treatment of overactive bladder (OAB) with symptoms of urge urinary incontinence, urgency, and urinary frequency in adults.
Drugs & Drug Targets
DrugTargetType
TolterodineMuscarinic acetylcholine receptor M1target
TolterodineMuscarinic acetylcholine receptor M2target
TolterodineMuscarinic acetylcholine receptor M3target
TolterodineCytochrome P450 2D6enzyme
TolterodineCytochrome P450 3A4enzyme
TolterodineCytochrome P450 2C9enzyme
TolterodineCytochrome P450 2C19enzyme
TolterodineMuscarinic acetylcholine receptor M4target
TolterodineMuscarinic acetylcholine receptor M5target
VibegronBeta-3 adrenergic receptortarget
VibegronCytochrome P450 3A4enzyme
VibegronP-glycoprotein 1transporter