Diagnostic Radiopharmaceuticals

Name
Diagnostic Radiopharmaceuticals
Accession Number
DBCAT002128
Description

Not Available

ATC Classification
Drugs
DrugDrug Description
Indium In-111 imciromab pentetateIndium In-111 imciromab pentetate is a mouse monoclonal antibody labelled with the radioisotope Indium-111 which was used for cardiac imaging under the trade name Myoscint, but was withdrawn in 1993.
Indium In-111 satumomab pendetideFor diagnosis of extrahepatic malignant cancers
Capromab pendetideA monoclonal anti-prostate specific membrane antigen antibody used in imaging kits to target radioactive agents to malignant prostate tissue.
Technetium Tc-99m arcitumomabFor imaging colorectal tumors
Ioflupane I-123A radiopharmaceutical used in single photon emission computed tomography (SPECT) brain imaging to help diagnose patients with suspected Parkinsonian syndromes.
Technetium Tc-99m mebrofeninA diagnostic radiopharmaceutical agent used during hepatobiliary imaging tests.
Technetium Tc-99m medronateA diagnostic radiopharmaceutical agent used as a bone imaging agent to delineate areas of altered osteogenesis.
Technetium Tc-99m oxidronateTechnetium Tc-99m oxidronate is indicated in adult and pediatric patients to be used in skeletal imaging for diagnosis of areas that can present altered osteogenesis. When administered intravenously, it is...
Florbetaben F-18A radiopharmaceutical diagnostic agent used during Positron Emission Tomography (PET) imaging of the brain to estimate β-amyloid neuritic plaque density in adult patients to diagnose the causes of cognitive impairment.
Florbetapir (18F)A radiopharmaceutical diagnostic agent used during Positron Emission Tomography (PET) imaging of the brain to estimate β-amyloid neuritic plaque density in adult patients to diagnose the causes of cognitive impairment.
Flutemetamol (18F)A radiopharmaceutical diagnostic agent used during Positron Emission Tomography (PET) imaging of the brain to estimate β-amyloid neuritic plaque density in adult patients to diagnose the causes of cognitive impairment.
Technetium Tc-99m tetrofosminTechnetium-99m tetrofosmin is indicated for the diagnosis of heart abnormalities by exercise myocardial scintigraphy. The exercise myocardial scintigraphy is an established method for the diagnosis of the severity of coronary...
Technetium Tc-99m sestamibiA radiopharmaceutical diagnostic agent used in nuclear medicine imaging tests to detect coronary artery disease and evaluate myocardial function.
Technetium Tc-99m exametazimeA radiopharmaceutical diagnostic agent used as an adjunct for scintigraphy in the detection of altered regional cerebral perfusion in stroke.
Technetium Tc-99m disofeninA radiopharmaceutical diagnostic agent used for hepatobiliary scans.
Technetium Tc-99m pyrophosphateA radiopharmaceutical diagnostic agent used for diagnostic imaging scans for the bones, heart, and gastrointestinal tract.
Technetium Tc-99m tilmanoceptA radiopharmaceutical diagnostic imaging agent indicated with or without scintigraphic imaging for lymphatic mapping and guiding sentinel lymph node biopsy.
Iodide I-131A radioisotopic agent used for the treatment of hyperthyroidism and thyroid carcinomas that take up iodine.
Technetium Tc-99m pertechnetateA radiocontrast agent used for the identification of various organs, including but not limited to the brain, thyroid, placenta, and bladder.
Xenon-133An inhaled radionuclide used to measure lung function and organ blood flow.
Technetium Tc-99m sulfur colloidA radiopharmaceutical diagnostic agent used for the localization of lymph nodes, evaluation of peritoneovenous (LeVeen) shunt patency, imaging areas of functioning reticuloendothelial cells, and gastrointestinal imaging.
Fluoride ion F-18A diagnostic radiopharmaceutical agent used as a bone imaging agent to delineate areas of altered osteogenesis.
Iodide I-123A radiopharmaceutical diagnostic agent used for the evaluation of the thyroid function and/or morphology.
Indium In-111 pentetateA radiopharmaceutical diagnostic agent used for radionuclide cisternography.
Technetium Tc-99m succimerA radioactive diagnostic agent used as an aid in the scintigraphic evaluation of renal parenchymal disorders.
Krypton Kr 81mNot Annotated
Iodohippurate sodium I-123Not Annotated
Iofetamine I-123Not Annotated
Fludeoxyglucose (18F)A radiopharmaceutical agent used for positron emission tomography (PET) imaging in oncology, cardiology, and neurology.
Technetium Tc-99m etifeninA radiopharmaceutical indicated in imaging studies of the liver and biliary tract.
Iodine (131I) norcholesterolA radioiodine-labeled cholesterol analogue that accumulates in areas where steroid hormones are produced and is used in certain diagnostic procedures.
Ferric (59Fe) citrateNot Annotated
Selenium (75Se) norcholesterolA radiopharmaceutical indicated in nuclear imaging studies of the digestive system.
Iodocholesterol (131I)Not Annotated
Fluorodopa (18F)Fluorodopa F 18 is indicated for use with positron emission tomography (PET) to visualize dopaminergic nerve terminals in the striatum for the evaluation of adult patients with suspected Parkinsonian syndromes...
SulesomabMarket product is Tc99m-labeled murine antibody fragment for nuclear imaging of activated granulocytes.
IobenguaneA radiopharmaceutical agent used for the diagnosis of primary and metastatic pheochromocytoma or neuroblastoma.
Technetium Tc-99m etidronateNot Annotated
Indium In-111 pentetreotideIndium In 111 pentetreotide (Octreoscan) has been used in trials studying the diagnostic of SARCOIDOSIS, Solid Tumors, and cushing syndrome.
Fluciclovine (18F)A radiolabelled L-leucine derivative used to image tumors, especially in the prostate.
Edotreotide gallium Ga-68A radioactive diagnostic agent used in PET scans for somatostatin receptor positive neuroendocrine tumors in adult and pediatric patients.
Iodohippurate sodium I-131Not Annotated
Fluorocholine F-18A radiopharmaceutical indicated in PET scans of the prostate.
Gallium Ga-68 gozetotideA radiopharmaceutical agent used in the diagnosis of prostate-specific membrane antigen (PSMA) positive lesions in male patients during positron emission tomography.
Thallous chloride Tl-201A radioisotope indicated for cardiac perfusion scintigraphy
Piflufolastat F 18A radiopharmaceutical diagnostic agent used with PET to image PSMA-positive lesions for the diagnosis of metastatic or recurrent prostate cancer.
Methionine C-11Not Annotated
Flortaucipir F-18A small lipophilic tracer containing [18F]fluoride capable of crossing the blood-brain barrier and binding to aggregated tau protein; used in PET imaging for the diagnosis of Alzheimer's disease.
Flotufolastat F-18A radiopharmaceutical diagnostic agent used in PET imaging to visualize PSMA-positive lesions in men with prostate cancer with suspected metastasis or recurrence.
FET F-18FET F-18 is under investigation in clinical trial NCT01756352 (FET-PET for Evaluation of Response of Recurrent GBM to Avastin).
Drugs & Drug Targets
DrugTargetType
Indium In-111 satumomab pendetideTumor-associated glycoprotein 72 (TAG-72)target
Capromab pendetideGlutamate carboxypeptidase 2target
Technetium Tc-99m arcitumomabCarcinoembryonic antigen-related cell adhesion molecule 1target
Ioflupane I-123Sodium-dependent dopamine transportertransporter
Technetium Tc-99m mebrofeninSolute carrier organic anion transporter family member 1B1transporter
Technetium Tc-99m mebrofeninSolute carrier organic anion transporter family member 1B3transporter
Technetium Tc-99m oxidronateSerum albumincarrier
Florbetaben F-18Cytochrome P450 2J2enzyme
Florbetaben F-18Leukotriene-B(4) omega-hydroxylase 1enzyme
Florbetaben F-18Amyloid beta A4 proteintarget
Florbetapir (18F)Amyloid beta A4 proteintarget
Flutemetamol (18F)Amyloid beta A4 proteintarget
Technetium Tc-99m tetrofosminP-glycoprotein 1carrier
Technetium Tc-99m sestamibiP-glycoprotein 1transporter
Technetium Tc-99m sestamibiMultidrug resistance-associated protein 1transporter
Technetium Tc-99m pyrophosphateHydroxyapatitetarget
Technetium Tc-99m pyrophosphateAmorphous calcium phosphatetarget
Technetium Tc-99m tilmanoceptMacrophage mannose receptor 1target
Technetium Tc-99m succimerSodium-dependent phosphate transporter 1transporter
Technetium Tc-99m succimerSodium-dependent phosphate transporter 2transporter
Fludeoxyglucose (18F)Hexokinase-1enzyme
Fludeoxyglucose (18F)Solute carrier family 2, facilitated glucose transporter member 4transporter
Fludeoxyglucose (18F)Solute carrier family 2, facilitated glucose transporter member 2transporter
Fludeoxyglucose (18F)Solute carrier family 2, facilitated glucose transporter member 1transporter
Fludeoxyglucose (18F)Solute carrier family 2, facilitated glucose transporter member 3transporter
Fludeoxyglucose (18F)Solute carrier family 2, facilitated glucose transporter member 9transporter
Fludeoxyglucose (18F)Solute carrier family 2, facilitated glucose transporter member 5transporter
Fludeoxyglucose (18F)Solute carrier family 2, facilitated glucose transporter member 6transporter
Fludeoxyglucose (18F)Solute carrier family 2, facilitated glucose transporter member 7transporter
Fludeoxyglucose (18F)Solute carrier family 2, facilitated glucose transporter member 8transporter
Fludeoxyglucose (18F)Solute carrier family 2, facilitated glucose transporter member 10transporter
Fludeoxyglucose (18F)Solute carrier family 2, facilitated glucose transporter member 11transporter
Fludeoxyglucose (18F)Solute carrier family 2, facilitated glucose transporter member 12transporter
Fluorodopa (18F)Aromatic-L-amino-acid decarboxylaseenzyme
IobenguaneSodium-dependent noradrenaline transportertransporter
Fluciclovine (18F)Neutral amino acid transporter B(0)target
Fluciclovine (18F)Y+L amino acid transporter 1target
Fluciclovine (18F)Cationic amino acid transporter 3target
Fluciclovine (18F)Glutamate (NMDA) receptortarget
Fluciclovine (18F)Glutamate receptor 1target
Fluciclovine (18F)Glutamate receptor 2target
Fluciclovine (18F)Glutamate receptor 3target
Fluciclovine (18F)Glutamate receptor 4target
Fluciclovine (18F)Multidrug resistance-associated protein 4transporter
Edotreotide gallium Ga-68Somatostatin receptor type 2target
Edotreotide gallium Ga-68Somatostatin receptor type 1target
Edotreotide gallium Ga-68Somatostatin receptor type 5target
Edotreotide gallium Ga-68Somatostatin receptor type 3target
Gallium Ga-68 gozetotideProstate-specific antigentarget
Piflufolastat F 18Glutamate carboxypeptidase 2target
Flortaucipir F-18Microtubule-associated protein tautarget
Flortaucipir F-18Amine oxidase [flavin-containing] Atarget
Flortaucipir F-18Amine oxidase [flavin-containing] Btarget
Flotufolastat F-18Glutamate carboxypeptidase 2target