Purinergic P1 Receptor Agonists

Name
Purinergic P1 Receptor Agonists
Accession Number
DBCAT001025
Description

Compounds that bind to and stimulate PURINERGIC P1 RECEPTORS.

Drugs
DrugDrug Description
AdenosineA medication used in myocardial perfusion scintigraphy and to treat supraventricular tachycardia.
RegadenosonA coronary vasodilator used in radionuclide myocardial perfusion imaging (MPI).
BinodenosonFor cardiac pharmacologic stress SPECT imaging, which is used to diagnose coronary artery disease.
TecadenosonInvestigated for use/treatment in arrhythmia and atrial fibrillation.
NamodenosonNamodenoson has been used in trials studying the treatment of Chronic Hepatitis C and Hepatocellular Carcinoma.
Drugs & Drug Targets
DrugTargetType
AdenosineAdenosine receptor A3target
AdenosineAdenosine deaminaseenzyme
AdenosineAdenosine kinaseenzyme
AdenosineAdenosine receptor A1target
AdenosineAdenosine receptor A2atarget
AdenosineAdenosine receptor A2btarget
AdenosineSolute carrier family 28 member 3transporter
AdenosineEquilibrative nucleoside transporter 1transporter
AdenosineEquilibrative nucleoside transporter 2transporter
AdenosineEquilibrative nucleoside transporter 3transporter
AdenosineEquilibrative nucleoside transporter 4transporter
AdenosineSodium/nucleoside cotransporter 1transporter
AdenosineSodium/nucleoside cotransporter 2transporter
AdenosineGap junction alpha-1 proteintransporter
AdenosineAdenylate kinase isoenzyme 1enzyme
AdenosineNucleoside diphosphate kinase Aenzyme
AdenosineNucleoside diphosphate kinase Benzyme
AdenosinePurine nucleoside phosphorylaseenzyme
AdenosineXanthine dehydrogenase/oxidaseenzyme
AdenosineSerum albumincarrier
RegadenosonAdenosine receptor A2atarget
BinodenosonAdenosine receptor A2atarget
TecadenosonAdenosine receptor A1target