Showing BioInteractions for Carisoprodol (DB00395)

BioInteractor utilizes data on drug-target, -enzyme and -transporter associations to provide insight on drug-drug interactions. It allows you to identify, for instance, which drugs act similarly on the same target. Such drugs may have additive pharmacodynamic effects if given concomitantly. Conversely, two drugs may antagonize the beneficial effects of each other by having opposite actions on a specific drug target. BioInteractor uses ranked drug-enzyme association information to predict enzyme-mediated drug interactions that may be clinically relevant.
Interacting GroupInteracting Drugs
Carisoprodol is a Gamma-aminobutyric acid receptor subunit alpha-1 activator
1Gamma-aminobutyric acid receptor subunit alpha-1 potentiatorsAmobarbital, Aprobarbital, Barbital, Butalbital, Butobarbital, Dihydro-2-thioxo-5-((5-(2-(trifluoromethyl)phenyl)-2-furanyl)methyl)-4,6(1H,5H)-pyrimidinedione, Dihydroquinidine barbiturate, Eszopiclone, Fludiazepam, Heptabarbital, Hexobarbital, Metharbital, Methylphenobarbital, Pentobarbital, Phenobarbital, Primidone, Quinidine barbiturate, Secobarbital, Talbutal, Thiopental, Zaleplon, Zopiclone
2Gamma-aminobutyric acid receptor subunit alpha-1 agonistsEthanol, Etomidate, Glutethimide, Isoflurane, Meprobamate, Methoxyflurane, Methyprylon, Progabide, Sevoflurane, Thiamylal, Topiramate, Zolpidem
3Gamma-aminobutyric acid receptor subunit alpha-1 antagonistsAmoxapine, Flumazenil, Methohexital, Picrotoxin
4Gamma-aminobutyric acid receptor subunit alpha-1 negative modulatorsGinkgo biloba
Interacting GroupInteracting Drugs
Carisoprodol is a Gamma-aminobutyric acid receptor subunit alpha-1 modulator
1Gamma-aminobutyric acid receptor subunit alpha-1 potentiatorsAmobarbital, Aprobarbital, Barbital, Butalbital, Butobarbital, Dihydro-2-thioxo-5-((5-(2-(trifluoromethyl)phenyl)-2-furanyl)methyl)-4,6(1H,5H)-pyrimidinedione, Dihydroquinidine barbiturate, Eszopiclone, Fludiazepam, Heptabarbital, Hexobarbital, Metharbital, Methylphenobarbital, Pentobarbital, Phenobarbital, Primidone, Quinidine barbiturate, Secobarbital, Talbutal, Thiopental, Zaleplon, Zopiclone
2Gamma-aminobutyric acid receptor subunit alpha-1 agonistsEthanol, Etomidate, Glutethimide, Isoflurane, Meprobamate, Methoxyflurane, Methyprylon, Progabide, Sevoflurane, Thiamylal, Topiramate, Zolpidem
3Gamma-aminobutyric acid receptor subunit alpha-1 antagonistsAmoxapine, Flumazenil, Methohexital, Picrotoxin
4Gamma-aminobutyric acid receptor subunit alpha-1 negative modulatorsGinkgo biloba
Interacting GroupInteracting Drugs
Carisoprodol is a Gamma-aminobutyric acid receptor subunit beta-2 modulator
1Gamma-aminobutyric acid receptor subunit beta-2 potentiatorsFludiazepam, Fospropofol, Propofol
2Gamma-aminobutyric acid receptor subunit beta-2 negative modulatorsGinkgo biloba
Interacting GroupInteracting Drugs
Carisoprodol is a Gamma-aminobutyric acid receptor subunit alpha-5 modulator
1Gamma-aminobutyric acid receptor subunit alpha-5 agonistsEszopiclone, Meprobamate
2Gamma-aminobutyric acid receptor subunit alpha-5 potentiatorsAmobarbital, Aprobarbital, Barbital, Butalbital, Butobarbital, Dihydro-2-thioxo-5-((5-(2-(trifluoromethyl)phenyl)-2-furanyl)methyl)-4,6(1H,5H)-pyrimidinedione, Fludiazepam, Heptabarbital, Hexobarbital, Metharbital, Methylphenobarbital, Pentobarbital, Primidone, Secobarbital, Talbutal, Thiopental, Zopiclone
3Gamma-aminobutyric acid receptor subunit alpha-5 antagonistsFlumazenil
Interacting GroupInteracting Drugs
Carisoprodol is a Gamma-aminobutyric acid receptor subunit alpha-3 modulator
1Gamma-aminobutyric acid receptor subunit alpha-3 agonistsEszopiclone, Meprobamate, Zolpidem
2Gamma-aminobutyric acid receptor subunit alpha-3 potentiatorsAmobarbital, Aprobarbital, Barbital, Butalbital, Butobarbital, Dihydro-2-thioxo-5-((5-(2-(trifluoromethyl)phenyl)-2-furanyl)methyl)-4,6(1H,5H)-pyrimidinedione, Fludiazepam, Heptabarbital, Hexobarbital, Metharbital, Methylphenobarbital, Pentobarbital, Primidone, Secobarbital, Talbutal, Thiopental, Zopiclone
3Gamma-aminobutyric acid receptor subunit alpha-3 positive allosteric modulatorsAZD-7325
Interacting GroupInteracting Drugs
Carisoprodol is a Cytochrome P450 2C19 substrate
1Cytochrome P450 2C19 substrates(R)-warfarin, (S)-Warfarin, Acenocoumarol, Adinazolam, Albendazole, Almotriptan, Ambrisentan, Aminophenazone, Amiodarone, Amitriptyline, Antipyrine, Apixaban, Aprepitant, Arformoterol, Artemether, Asunaprevir, Atomoxetine, Axitinib, Azelastine, Barbital, Binimetinib, Bioallethrin, Bortezomib, Brivaracetam, Bromazepam, Bupivacaine, Cannabidiol, Capravirine, Cenobamate, Chlorpropamide, Cilostazol, Cisapride, Citalopram, Clobazam, Clomethiazole, Clomipramine, Clopidogrel, Clotiazepam, Clozapine, Cyclophosphamide, Dapsone, Dexibuprofen, Dexlansoprazole, Dexrabeprazole, Dextromethorphan, Diazepam, Diclofenac, Diltiazem, Diphenhydramine, Doxazosin, Doxepin, Eletriptan, Enasidenib, Encorafenib, Enfuvirtide, Escitalopram, Esketamine, Esomeprazole, Estradiol, Estradiol acetate, Estradiol benzoate, Estradiol cypionate, Estradiol dienanthate, Estradiol valerate, Etizolam, Etravirine, Fedratinib, Fenfluramine, Flunitrazepam, Fluoxetine, Formoterol, Fosphenytoin, Gliclazide, Glyburide, Guanfacine, Haloperidol, Hexobarbital, Hydrocodone, Ibuprofen, Ifosfamide, Imatinib, Imipramine, Indomethacin, Ixazomib, Ketobemidone, Labetalol, Lacosamide, Lansoprazole, Lapatinib, Levomilnacipran, Lofexidine, Lonafarnib, Loratadine, Lorcaserin, Lorlatinib, Lovastatin, Lumiracoxib, Lynestrenol, Macitentan, Medical Cannabis, Melatonin, Meperidine, Mephenytoin, Methadone, Methsuximide, Methylene blue, Methylphenobarbital, Moclobemide, Nabiximols, Nebivolol, Nelfinavir, Nicotine, Nilutamide, Norethisterone, Nortriptyline, Oliceridine, Omeprazole, Ospemifene, Oxiconazole, Oxymetazoline, Pantoprazole, Paroxetine, Pentamidine, Pentobarbital, Perphenazine, Phenacetin, Phenobarbital, Phenytoin, Piperaquine, Pipotiazine, Pirfenidone, Prasugrel, Praziquantel, Primidone, Progesterone, Proguanil, Promazine, Propofol, Propranolol, Quazepam, Quetiapine, Quinine, Rabeprazole, Ramelteon, Rilpivirine, Romidepsin, Rupatadine, Selegiline, Selumetinib, Seratrodast, Sertraline, Sildenafil, Simvastatin, St. John's Wort, Stiripentol, Tamoxifen, Tapentadol, Teniposide, Terbinafine, Testosterone, Testosterone cypionate, Testosterone enanthate, Testosterone undecanoate, Thalidomide, Thiopental, Thioridazine, Ticlopidine, Timolol, Tipranavir, Tofacitinib, Tolbutamide, Tolterodine, Trabectedin, Triclabendazole, Trimethadione, Trimipramine, Valproic acid, Verapamil, Vilazodone, Voriconazole, Vortioxetine, Voxelotor, Warfarin, Zolpidem, Zonisamide
2Cytochrome P450 2C19 inhibitorsAbiraterone, Alpelisib, Amiodarone, Amitriptyline, Amprenavir, Aprepitant, Armodafinil, Artenimol, Atorvastatin, Avasimibe, Azelastine, Benzbromarone, Bicalutamide, Bortezomib, Buprenorphine, Carbamazepine, Casimersen, Cenobamate, Chloramphenicol, Cimetidine, Cisapride, Citalopram, Clascoterone, Clevidipine, Clinafloxacin, Clozapine, Curcumin sulfate, Cyclosporine, Dabrafenib, Delavirdine, Dexlansoprazole, Diazepam, Dimethyl sulfoxide, Dosulepin, Dovitinib, Duloxetine, Elexacaftor, Enasidenib, Eslicarbazepine, Eslicarbazepine acetate, Esomeprazole, Ethambutol, Ethanol, Ethinylestradiol, Etoricoxib, Etravirine, Felbamate, Fenofibrate, Fluconazole, Fluoxetine, Fluvastatin, Fluvoxamine, Gefitinib, Gemfibrozil, Gestodene, Idelalisib, Imipramine, Indomethacin, Isavuconazole, Isoniazid, Ketoconazole, Lansoprazole, Lenvatinib, Letrozole, Lobeglitazone, Lonafarnib, Lopinavir, Loratadine, Losartan, Luliconazole, Lynestrenol, Manidipine, Memantine, Menadione, Mephenytoin, Methimazole, Methsuximide, Methylene blue, Miconazole, Midostaurin, Moclobemide, Modafinil, Naloxegol, Nicardipine, Nilutamide, Nilvadipine, Olanzapine, Omeprazole, Oritavancin, Osilodrostat, Oxcarbazepine, Pantoprazole, Phenelzine, Piperaquine, Progesterone, Quinine, Rabeprazole, Rifamycin, Rilpivirine, Rucaparib, Safinamide, Seproxetine, Sertraline, Sildenafil, Sitaxentan, Somapacitan, Somatotropin, Sorafenib, Stiripentol, Sulfanilamide, Telmisartan, Thalidomide, Ticlopidine, Tioconazole, Tipranavir, Tirbanibulin, Topiramate, Topiroxostat, Tranylcypromine, Triclabendazole, Troglitazone, Ubrogepant, Valproic acid, Vismodegib, Voriconazole, Warfarin, Zafirlukast, Zonisamide, Zucapsaicin
3Cytochrome P450 2C19 inducersAcetylsalicylic acid, Aminoglutethimide, Apalutamide, Artemether, Barbital, Betamethasone, Budesonide, Carbamazepine, Dabrafenib, Dexamethasone, Dexamethasone acetate, Efavirenz, Enzalutamide, Hydrocortisone, Hydroxyprogesterone caproate, Letermovir, Lumacaftor, Methylprednisolone, Midostaurin, Nelfinavir, Norethisterone, Opicapone, Phenobarbital, Phenytoin, Prednisolone phosphate, Prednisone, Primidone, Rifabutin, Rifampicin, Rifamycin, Rifapentine, Rifaximin, Ritonavir, Secobarbital, St. John's Wort