Showing BioInteractions for Apomorphine (DB00714)
BioInteractor utilizes data on drug-target, -enzyme and -transporter associations to provide insight on drug-drug interactions. It allows you to identify, for instance, which drugs act similarly on the same target. Such drugs may have additive pharmacodynamic effects if given concomitantly. Conversely, two drugs may antagonize the beneficial effects of each other by having opposite actions on a specific drug target. BioInteractor uses ranked drug-enzyme association information to predict enzyme-mediated drug interactions that may be clinically relevant.
Interacting Group | Interacting Drugs | |
---|---|---|
Apomorphine is a Dopamine D1 receptor agonist | ||
1 | Dopamine D1 receptor antagonists | Acepromazine, Amoxapine, Aripiprazole, Asenapine, Carphenazine, Chlorpromazine, Chlorprothixene, Clozapine, Flupentixol, Fluphenazine, Haloperidol, Iloperidone, Lisuride, Loxapine, Methotrimeprazine, Methylergometrine, Olanzapine, Paliperidone, Periciazine, Perphenazine, Pipamperone, Pipotiazine, Quetiapine, Risperidone, Tetrahydropalmatine, Thioproperazine, Thioridazine, Thiothixene, Triflupromazine, Ziprasidone, Zuclopenthixol |
2 | Dopamine D1 receptor agonists | Bromocriptine, Cabergoline, Dopamine, Fenoldopam, Levodopa, Minaprine, Pergolide, Rotigotine |
3 | Dopamine D1 receptor partial agonists | Aripiprazole, Phenylpropanolamine |
4 | Dopamine D1 receptor ligands | Aripiprazole |
Interacting Group | Interacting Drugs | |
---|---|---|
Apomorphine is a Dopamine D4 receptor agonist | ||
1 | Dopamine D4 receptor antagonists | Amoxapine, Aripiprazole, Asenapine, Bromocriptine, Buspirone, Clozapine, Flibanserin, Flupentixol, Iloperidone, Methotrimeprazine, Olanzapine, Paliperidone, Perospirone, Pipamperone, Remoxipride, Sulpiride, Ziprasidone |
2 | Dopamine D4 receptor agonists | Cabergoline, Dopamine, Flibanserin, Levodopa, Lisuride, Pergolide, Pramipexole, Ropinirole, Rotigotine |
3 | Dopamine D4 receptor partial agonists | Aripiprazole |
4 | Dopamine D4 receptor ligands | Quetiapine |
5 | Dopamine D4 receptor binders | Chlorpromazine, Loxapine |
Interacting Group | Interacting Drugs | |
---|---|---|
Apomorphine is a Dopamine D3 receptor agonist | ||
1 | Dopamine D3 receptor antagonists | Amisulpride, Amoxapine, Aripiprazole, AS-8112, Asenapine, Blonanserin, Buspirone, Chlorprothixene, Clozapine, Domperidone, Flupentixol, Iloperidone, Methotrimeprazine, Olanzapine, Paliperidone, Pimozide, Remoxipride, Sulpiride, Yohimbine, Ziprasidone |
2 | Dopamine D3 receptor agonists | Bromocriptine, Cabergoline, Captodiame, Cariprazine, Dopamine, Levodopa, Lisuride, Pergolide, Pramipexole, Ropinirole, Rotigotine, Tianeptine |
3 | Dopamine D3 receptor partial agonists | Aripiprazole, Cariprazine, Dihydro-alpha-ergocryptine |
4 | Dopamine D3 receptor inverse agonists | Haloperidol |
5 | Dopamine D3 receptor ligands | Quetiapine, Sarizotan |
6 | Dopamine D3 receptor inhibitors | Chlorpromazine |
7 | Dopamine D3 receptor binders | Loxapine, Mianserin |
8 | Dopamine D3 receptor blockers | Tiapride |
Interacting Group | Interacting Drugs | |
---|---|---|
Apomorphine is a Dopamine D5 receptor agonist | ||
1 | Dopamine D5 receptor agonists | Bromocriptine, Cabergoline, Dopamine, Fenoldopam, Levodopa, Pergolide, Rotigotine |
2 | Dopamine D5 receptor antagonists | Aripiprazole, Carphenazine, Lisuride, Methotrimeprazine, Olanzapine, Ziprasidone, Zuclopenthixol |
3 | Dopamine D5 receptor partial agonists | Aripiprazole |
4 | Dopamine D5 receptor ligands | Aripiprazole, Quetiapine |
5 | Dopamine D5 receptor inhibitors | Chlorpromazine |
6 | Dopamine D5 receptor binders | Loxapine |
Interacting Group | Interacting Drugs | |
---|---|---|
Apomorphine is a Alpha-2C adrenergic receptor agonist | ||
1 | Alpha-2C adrenergic receptor antagonists | Aripiprazole, Asenapine, Brexpiprazole, Cabergoline, Carvedilol, Celiprolol, Clozapine, Dronedarone, Fenoldopam, Iloperidone, Lurasidone, Methotrimeprazine, Mianserin, Phenoxybenzamine, Pizotifen, Quetiapine, Risperidone, Yohimbine, Ziprasidone |
2 | Alpha-2C adrenergic receptor agonists | Agmatine, Brimonidine, Bromocriptine, Clonidine, Droxidopa, Ephedra sinica root, Metamfetamine, Norepinephrine, Oxymetazoline, Paliperidone, Racepinephrine, Xylometazoline |
3 | Alpha-2C adrenergic receptor binders | Loxapine, Tolazoline |
Interacting Group | Interacting Drugs | |
---|---|---|
Apomorphine is a Alpha-2B adrenergic receptor agonist | ||
1 | Alpha-2B adrenergic receptor antagonists | Aripiprazole, Asenapine, Cabergoline, Carvedilol, Celiprolol, Clozapine, Dronedarone, Fenoldopam, Methotrimeprazine, Mianserin, Paliperidone, Phenoxybenzamine, Pizotifen, Quetiapine, Risperidone, Rotigotine, Yohimbine, Ziprasidone |
2 | Alpha-2B adrenergic receptor agonists | Apraclonidine, Brimonidine, Bromocriptine, Clonidine, Droxidopa, Ephedra sinica root, Epinephrine, Etomidate, Metamfetamine, Norepinephrine, Oxymetazoline, Racepinephrine, Xylometazoline |
3 | Alpha-2B adrenergic receptor ligands | Aripiprazole |
4 | Alpha-2B adrenergic receptor binders | Guanabenz, Guanfacine, Loxapine, Prazosin, Tolazoline |
Interacting Group | Interacting Drugs | |
---|---|---|
Apomorphine is a 5-hydroxytryptamine receptor 2B agonist | ||
1 | 5-hydroxytryptamine receptor 2B antagonists | Amoxapine, Asenapine, Cariprazine, Clomipramine, Cyclobenzaprine, Doxepin, Lisuride, Methysergide, Minaprine, Pizotifen, PRX-08066, Tegaserod, Triflupromazine, Yohimbine |
2 | 5-hydroxytryptamine receptor 2B agonists | Bromocriptine, Cabergoline, Dihydroergotamine, Fenfluramine, Lysergic acid diethylamide, Midomafetamine, Paroxetine, Pergolide, Zolmitriptan |
3 | 5-hydroxytryptamine receptor 2B binders | Mianserin |
4 | 5-hydroxytryptamine receptor 2B inverse agonists | Aripiprazole |
Interacting Group | Interacting Drugs | |
---|---|---|
Apomorphine is a 5-hydroxytryptamine receptor 1D agonist | ||
1 | 5-hydroxytryptamine receptor 1D agonists | Almotriptan, Bromocriptine, Cabergoline, Dihydroergotamine, Eletriptan, Ergotamine, Fenfluramine, Frovatriptan, Lisuride, Lofexidine, Naratriptan, Oxymetazoline, Pergolide, Rizatriptan, Sumatriptan, Zolmitriptan |
2 | 5-hydroxytryptamine receptor 1D antagonists | Aripiprazole, Clozapine, Paliperidone, Pizotifen, Risperidone, Ziprasidone |
3 | 5-hydroxytryptamine receptor 1D ligands | Aripiprazole, Quetiapine |
4 | 5-hydroxytryptamine receptor 1D partial agonists | Yohimbine |
5 | 5-hydroxytryptamine receptor 1D binders | Amitriptyline, Loxapine, Trimipramine |
Interacting Group | Interacting Drugs | |
---|---|---|
Apomorphine is a 5-hydroxytryptamine receptor 1B agonist | ||
1 | 5-hydroxytryptamine receptor 1B agonists | Almotriptan, Bromocriptine, Cabergoline, Dihydroergotamine, Eletriptan, Ergotamine, Frovatriptan, Lisuride, Naratriptan, Oxymetazoline, Pergolide, Rizatriptan, Sumatriptan, Zolmitriptan |
2 | 5-hydroxytryptamine receptor 1B antagonists | Amoxapine, Aripiprazole, Asenapine, Clozapine, Penbutolol, Pizotifen, Ziprasidone |
3 | 5-hydroxytryptamine receptor 1B ligands | Aripiprazole, Quetiapine |
4 | 5-hydroxytryptamine receptor 1B partial agonists | Vortioxetine, Yohimbine |
5 | 5-hydroxytryptamine receptor 1B binders | Amitriptyline, Loxapine, Methysergide |
Interacting Group | Interacting Drugs | |
---|---|---|
Apomorphine is a Catechol O-methyltransferase substrate | ||
1 | Catechol O-methyltransferase inhibitors | Entacapone, Opicapone, Testosterone propionate, Tolcapone |
2 | Catechol O-methyltransferase substrates | Conjugated estrogens, Diethylstilbestrol, Dobutamine, Dopamine, Echinacoside, Epinephrine, Estradiol, Ethinylestradiol, Methyldopa, Micafungin, Phenytoin |
3 | Catechol O-methyltransferase cofactors | Ademetionine |
4 | Catechol O-methyltransferase inducers | Nylidrin |
Interacting Group | Interacting Drugs | |
---|---|---|
Apomorphine is a Sulfotransferase 1A1 substrate | ||
1 | Sulfotransferase 1A1 substrates | Acetaminophen, Polyethylene glycol 400, Propacetamol, Tamoxifen, Thyroid, porcine, Tibolone |
Interacting Group | Interacting Drugs | |
---|---|---|
Apomorphine is a Sulfotransferase 1A2 substrate | ||
1 | Sulfotransferase 1A2 substrates | Thyroid, porcine |
Interacting Group | Interacting Drugs | |
---|---|---|
Apomorphine is a Sulfotransferase 1A3/1A4 substrate | ||
1 | Sulfotransferase 1A3/1A4 substrates | Acetaminophen, Curcumin sulfate, Ethinylestradiol, Phenylephrine, Propacetamol, Thyroid, porcine |
Interacting Group | Interacting Drugs | |
---|---|---|
Apomorphine is a Estrogen sulfotransferase substrate | ||
1 | Estrogen sulfotransferase inhibitors | Cyclizine |
2 | Estrogen sulfotransferase substrates | Curcumin sulfate, Ethinylestradiol, Propacetamol, Tamoxifen, Thyroid, porcine |
Interacting Group | Interacting Drugs | |
---|---|---|
Apomorphine is a Sulfotransferase family cytosolic 1B member 1 substrate | ||
1 | Sulfotransferase family cytosolic 1B member 1 substrates | Curcumin sulfate, Thyroid, porcine |
Interacting Group | Interacting Drugs | |
---|---|---|
Apomorphine is a UDP-glucuronosyltransferases (UGTs) substrate | ||
1 | UDP-glucuronosyltransferases (UGTs) substrates | Estradiol, Fostemsavir, Lamotrigine, Terbutaline |
2 | UDP-glucuronosyltransferases (UGTs) inducers | Estradiol, Primidone, Ritonavir |
3 | UDP-glucuronosyltransferases (UGTs) inhibitors | Curcumin sulfate |
Interacting Group | Interacting Drugs | |
---|---|---|
Apomorphine is a Synaptic vesicular amine transporter inducer | ||
1 | Synaptic vesicular amine transporter inhibitors | 4-Methoxyamphetamine, Amphetamine, Deserpidine, Deutetrabenazine, Ephedra sinica root, Ephedrine, Isometheptene, Metamfetamine, Midomafetamine, MMDA, Rauwolfia serpentina root, Reserpine, Tetrabenazine |
2 | Synaptic vesicular amine transporter inducers | Benzphetamine, Dextroamphetamine |
3 | Synaptic vesicular amine transporter binders | Norepinephrine |