Showing BioInteractions for Histamine (DB05381)

BioInteractor utilizes data on drug-target, -enzyme and -transporter associations to provide insight on drug-drug interactions. It allows you to identify, for instance, which drugs act similarly on the same target. Such drugs may have additive pharmacodynamic effects if given concomitantly. Conversely, two drugs may antagonize the beneficial effects of each other by having opposite actions on a specific drug target. BioInteractor uses ranked drug-enzyme association information to predict enzyme-mediated drug interactions that may be clinically relevant.
Interacting GroupInteracting Drugs
Histamine is a Histamine H1 receptor agonist
1Histamine H1 receptor antagonistsAceprometazine, Acrivastine, Alcaftadine, Alimemazine, Amitriptyline, Amoxapine, Antazoline, Aripiprazole, Aripiprazole lauroxil, Asenapine, Astemizole, Azatadine, Azelastine, Benzatropine, Benzquinamide, Bepotastine, Bilastine, Bromodiphenhydramine, Brompheniramine, Buclizine, Butriptyline, Carbinoxamine, Cariprazine, Cetirizine, Chlorcyclizine, Chloropyramine, Chlorpheniramine, Chlorpromazine, Chlorprothixene, Cinnarizine, Clemastine, Clofedanol, Clozapine, Cyclizine, Cyproheptadine, Desipramine, Desloratadine, Dexbrompheniramine, Dexchlorpheniramine maleate, Dimenhydrinate, Dimetindene, Diphenhydramine, Diphenylpyraline, Dosulepin, Doxepin, Doxylamine, Emedastine, Epinastine, Fexofenadine, Flunarizine, Iloperidone, Imipramine, Isothipendyl, Ketotifen, Lamotrigine, Levocabastine, Levocetirizine, Loratadine, Lorpiprazole, Maprotiline, Meclizine, Mepyramine, Mequitazine, Methdilazine, Methotrimeprazine, Mianserin, Mirtazapine, Nortriptyline, Olanzapine, Olopatadine, Orphenadrine, Paliperidone, Phenindamine, Pizotifen, Prochlorperazine, Promazine, Promethazine, Propiomazine, Quetiapine, Risperidone, Rupatadine, Terfenadine, Tesmilifene, Thonzylamine, Trazodone, Trimipramine, Tripelennamine, Triprolidine, Ziprasidone, Zuclopenthixol
2Histamine H1 receptor inverse agonistsEsmirtazapine, Hydroxyzine, Perospirone, Pheniramine
3Histamine H1 receptor agonistsBetahistine, Tolazoline
4Histamine H1 receptor inhibitorsEscitalopram, Levocetirizine, Paroxetine
5Histamine H1 receptor bindersCitalopram, Loxapine
Interacting GroupInteracting Drugs
Histamine is a Histamine H2 receptor agonist
1Histamine H2 receptor agonistsBetazole, Tolazoline
2Histamine H2 receptor antagonistsAsenapine, Cimetidine, Doxepin, Epinastine, Famotidine, Methantheline, Metiamide, Nizatidine, Olopatadine, Promethazine, Ranitidine, Roxatidine acetate
3Histamine H2 receptor bindersLoxapine
4Histamine H2 receptor blockersAmitriptyline
5Histamine H2 receptor inhibitorsAzelastine
6Histamine H2 receptor ligandsAripiprazole
Interacting GroupInteracting Drugs
Histamine is a Histamine H3 receptor agonist
1Histamine H3 receptor antagonistsBetahistine, Olopatadine, Pitolisant
2Histamine H3 receptor inverse agonistsPitolisant
3Histamine H3 receptor ligandsAripiprazole
Interacting GroupInteracting Drugs
Histamine is a Histamine H4 receptor agonist
1Histamine H4 receptor antagonistsClozapine
2Histamine H4 receptor bindersAmitriptyline, Amoxapine, Chlorpromazine, Doxepin, Loxapine, Mianserin
3Histamine H4 receptor inverse agonistsPheniramine
4Histamine H4 receptor ligandsAripiprazole
Interacting GroupInteracting Drugs
Histamine is a Histamine N-methyltransferase substrate
1Histamine N-methyltransferase inhibitorsAmodiaquine, Harmaline, Quinacrine, S-adenosyl-L-homocysteine
2Histamine N-methyltransferase bindersS-adenosyl-L-homocysteine
Interacting GroupInteracting Drugs
Histamine is a Solute carrier family 22 member 2 substrate
1Solute carrier family 22 member 2 inhibitorsAbemaciclib, Amantadine, Amiloride, Aminohippuric acid, Amiodarone, Apalutamide, Baricitinib, Bupropion, Chlorpheniramine, Choline, Choline salicylate, Cimetidine, Cisplatin, Clopidogrel, Cocaine, Desipramine, Dexchlorpheniramine maleate, Dinoprostone, Diphenhydramine, Disopyramide, Dolutegravir, Dopamine, Dronedarone, Enasidenib, Erdafitinib, Estradiol, Estradiol acetate, Estradiol benzoate, Estradiol cypionate, Estradiol dienanthate, Estradiol valerate, Famotidine, Flurazepam, Grepafloxacin, Guanidine, Imatinib, Imipramine, Isavuconazole, Lamotrigine, Lenvatinib, Levofloxacin, Linagliptin, Metformin, Methylene blue, Metoprolol, Nicotine, Norepinephrine, Osilodrostat, Oxprenolol, Pemigatinib, Phenformin, Phenoxybenzamine, Pimagedine, Probenecid, Procainamide, Progesterone, Propranolol, Quinacrine, Quinidine, Quinine, Rimegepant, Salmeterol, Tafenoquine, Thiamine, Tirbanibulin, Trilaciclib, Tucatinib, Ubrogepant, Vandetanib, Varenicline
2Solute carrier family 22 member 2 substratesAgmatine, Amantadine, Choline, Choline salicylate, Cimetidine, Cisplatin, Dalfampridine, Dofetilide, Dopamine, Epinephrine, Guanfacine, Lamivudine, Linagliptin, Memantine, Metformin, Nafamostat, Norepinephrine, Oxaliplatin, Pramipexole, Ranitidine, Reserpine, Sulpiride, Terbutaline, Tetraethylammonium, Tipiracil, Varenicline
Interacting GroupInteracting Drugs
Histamine is a Solute carrier family 22 member 2 inhibitor
1Solute carrier family 22 member 2 inhibitorsAbemaciclib, Amantadine, Amiloride, Aminohippuric acid, Amiodarone, Apalutamide, Baricitinib, Bupropion, Chlorpheniramine, Choline, Choline salicylate, Cimetidine, Cisplatin, Clopidogrel, Cocaine, Desipramine, Dexchlorpheniramine maleate, Dinoprostone, Diphenhydramine, Disopyramide, Dolutegravir, Dopamine, Dronedarone, Enasidenib, Erdafitinib, Estradiol, Estradiol acetate, Estradiol benzoate, Estradiol cypionate, Estradiol dienanthate, Estradiol valerate, Famotidine, Flurazepam, Grepafloxacin, Guanidine, Imatinib, Imipramine, Isavuconazole, Lamotrigine, Lenvatinib, Levofloxacin, Linagliptin, Metformin, Methylene blue, Metoprolol, Nicotine, Norepinephrine, Osilodrostat, Oxprenolol, Pemigatinib, Phenformin, Phenoxybenzamine, Pimagedine, Probenecid, Procainamide, Progesterone, Propranolol, Quinacrine, Quinidine, Quinine, Rimegepant, Salmeterol, Tafenoquine, Thiamine, Tirbanibulin, Trilaciclib, Tucatinib, Ubrogepant, Vandetanib, Varenicline
2Solute carrier family 22 member 2 substratesAgmatine, Amantadine, Choline, Choline salicylate, Cimetidine, Cisplatin, Dalfampridine, Dofetilide, Dopamine, Epinephrine, Guanfacine, Lamivudine, Linagliptin, Memantine, Metformin, Nafamostat, Norepinephrine, Oxaliplatin, Pramipexole, Ranitidine, Reserpine, Sulpiride, Terbutaline, Tetraethylammonium, Tipiracil, Varenicline
Interacting GroupInteracting Drugs
Histamine is a Solute carrier family 22 member 3 inhibitor
1Solute carrier family 22 member 3 inhibitorsCholine, Choline salicylate, Cimetidine, Clonidine, Desipramine, Dopamine, Estradiol, Estradiol acetate, Estradiol benzoate, Estradiol cypionate, Estradiol dienanthate, Estradiol valerate, Formoterol, Guanidine, Imipramine, Irinotecan, Linagliptin, Melphalan, Metamfetamine, Nicotine, Norepinephrine, Phenoxybenzamine, Prazosin, Procainamide, Progesterone, Salmeterol, Vincristine
2Solute carrier family 22 member 3 substratesAdefovir dipivoxil, Agmatine, Amphetamine, Cimetidine, Guanidine, Lamivudine, Metformin, Norepinephrine, Oxaliplatin, Sulpiride, Testosterone cypionate, Testosterone enanthate
Interacting GroupInteracting Drugs
Histamine is a Solute carrier family 22 member 5 inhibitor
1Solute carrier family 22 member 5 inhibitorsAcetylcholine, Aldosterone, Aminohippuric acid, Ampicillin, Arginine, Azidocillin, Benzylpenicillin, Cefadroxil, Cefalotin, Cefdinir, Cefepime, Cefixime, Cefradine, Ceftazidime, Cephalexin, Cephaloglycin, Choline, Choline salicylate, Cimetidine, Clonidine, Creatine, Cyclacillin, Dactinomycin, Desipramine, Diphenhydramine, Dopamine, Furosemide, Grepafloxacin, Guanidine, Levamlodipine, Lidocaine, Lomefloxacin, Metamfetamine, Methacholine, Niacin, Nicotine, Norepinephrine, Norfloxacin, Ofloxacin, Probenecid, Procainamide, Quinidine, Quinine, Sparfloxacin, Thiamine, Valproic acid, Verapamil
2Solute carrier family 22 member 5 substratesAmphetamine, Formoterol, Ipratropium, Levocarnitine, Terbutaline, Tiotropium