Showing BioInteractions for Betahistine (DB06698)

BioInteractor utilizes data on drug-target, -enzyme and -transporter associations to provide insight on drug-drug interactions. It allows you to identify, for instance, which drugs act similarly on the same target. Such drugs may have additive pharmacodynamic effects if given concomitantly. Conversely, two drugs may antagonize the beneficial effects of each other by having opposite actions on a specific drug target. BioInteractor uses ranked drug-enzyme association information to predict enzyme-mediated drug interactions that may be clinically relevant.
Interacting GroupInteracting Drugs
Betahistine is a Histamine H1 receptor agonist
1Histamine H1 receptor antagonistsAceprometazine, Acrivastine, Alcaftadine, Alimemazine, Amitriptyline, Amoxapine, Antazoline, Aripiprazole, Aripiprazole lauroxil, Asenapine, Astemizole, Azatadine, Azelastine, Benzatropine, Benzquinamide, Bepotastine, Bilastine, Bromodiphenhydramine, Brompheniramine, Buclizine, Butriptyline, Carbinoxamine, Cariprazine, Cetirizine, Chlorcyclizine, Chloropyramine, Chlorpheniramine, Chlorpromazine, Chlorprothixene, Cinnarizine, Clemastine, Clofedanol, Clozapine, Cyclizine, Cyproheptadine, Desipramine, Desloratadine, Dexbrompheniramine, Dexchlorpheniramine maleate, Dimenhydrinate, Dimetindene, Diphenhydramine, Diphenylpyraline, Dosulepin, Doxepin, Doxylamine, Emedastine, Epinastine, Fexofenadine, Flunarizine, Iloperidone, Imipramine, Isothipendyl, Ketotifen, Lamotrigine, Levocabastine, Levocetirizine, Loratadine, Lorpiprazole, Maprotiline, Meclizine, Mepyramine, Mequitazine, Methdilazine, Methotrimeprazine, Mianserin, Mirtazapine, Nortriptyline, Olanzapine, Olopatadine, Orphenadrine, Paliperidone, Phenindamine, Pizotifen, Prochlorperazine, Promazine, Promethazine, Propiomazine, Quetiapine, Risperidone, Rupatadine, Terfenadine, Tesmilifene, Thonzylamine, Trazodone, Trimipramine, Tripelennamine, Triprolidine, Ziprasidone, Zuclopenthixol
2Histamine H1 receptor inverse agonistsEsmirtazapine, Hydroxyzine, Perospirone, Pheniramine
3Histamine H1 receptor agonistsHistamine, Tolazoline
4Histamine H1 receptor inhibitorsEscitalopram, Levocetirizine, Paroxetine
5Histamine H1 receptor bindersCitalopram, Loxapine
Interacting GroupInteracting Drugs
Betahistine is a Histamine H3 receptor antagonist
1Histamine H3 receptor agonistsHistamine
2Histamine H3 receptor antagonistsOlopatadine, Pitolisant
3Histamine H3 receptor inverse agonistsPitolisant
4Histamine H3 receptor ligandsAripiprazole
Interacting GroupInteracting Drugs
Betahistine is a Monoamine oxidase substrate
1Monoamine oxidase inhibitorsAmphetamine, Procaine, Procarbazine
2Monoamine oxidase cofactorsCopper
3Monoamine oxidase antagonistsMoclobemide
4Monoamine oxidase substratesEpinephrine, Escitalopram, Rauwolfia serpentina root