Showing BioInteractions for Gavestinel (DB06741)
BioInteractor utilizes data on drug-target, -enzyme and -transporter associations to provide insight on drug-drug interactions. It allows you to identify, for instance, which drugs act similarly on the same target. Such drugs may have additive pharmacodynamic effects if given concomitantly. Conversely, two drugs may antagonize the beneficial effects of each other by having opposite actions on a specific drug target. BioInteractor uses ranked drug-enzyme association information to predict enzyme-mediated drug interactions that may be clinically relevant.
Interacting Group | Interacting Drugs | |
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Gavestinel is a Glutamate (NMDA) receptor antagonist | ||
1 | Glutamate (NMDA) receptor antagonists | Acamprosate, Enflurane, Memantine |
2 | Glutamate (NMDA) receptor blockers | Magnesium carbonate |
3 | Glutamate (NMDA) receptor ligands | Aripiprazole, Magnesium acetate tetrahydrate |
4 | Glutamate (NMDA) receptor inhibitors | Fluciclovine (18F) |
Interacting Group | Interacting Drugs | |
---|---|---|
Gavestinel is a UDP-glucuronosyltransferase 1-3 substrate | ||
1 | UDP-glucuronosyltransferase 1-3 substrates | Ambrisentan, Anastrozole, Atorvastatin, Baloxavir marboxil, Candesartan, Candesartan cilexetil, Cyproheptadine, Delafloxacin, Dexibuprofen, Diclofenac, Dolutegravir, Eltrombopag, Empagliflozin, Enasidenib, Etodolac, Ezetimibe, Ezogabine, Flurbiprofen, Fluvastatin, Gemfibrozil, Hydromorphone, Ibuprofen, Irbesartan, Letermovir, Licofelone, Lorlatinib, Losartan, Lovastatin, Mitiglinide, Morphine, Muraglitazar, Naldemedine, Nalmefene, Naproxen, Pitavastatin, Simvastatin, Telmisartan, Troglitazone, Valproic acid |
2 | UDP-glucuronosyltransferase 1-3 inhibitors | Deferasirox, Dovitinib, Flunitrazepam, Gemfibrozil |
Interacting Group | Interacting Drugs | |
---|---|---|
Gavestinel is a UDP-glucuronosyltransferase 2B4 substrate | ||
1 | UDP-glucuronosyltransferase 2B4 substrates | Canagliflozin, Carvedilol, Cenobamate, Codeine, Dapagliflozin, Dexibuprofen, Dextromethorphan, Diclofenac, Flurbiprofen, Gemfibrozil, Ibuprofen, Morphine |