Showing BioInteractions for Doxefazepam (DB13837)

BioInteractor utilizes data on drug-target, -enzyme and -transporter associations to provide insight on drug-drug interactions. It allows you to identify, for instance, which drugs act similarly on the same target. Such drugs may have additive pharmacodynamic effects if given concomitantly. Conversely, two drugs may antagonize the beneficial effects of each other by having opposite actions on a specific drug target. BioInteractor uses ranked drug-enzyme association information to predict enzyme-mediated drug interactions that may be clinically relevant.
Interacting GroupInteracting Drugs
Doxefazepam is a GABA(A) Receptor positive allosteric modulator
1GABA(A) Receptor positive allosteric modulators1,2-Benzodiazepine, Adinazolam, Alprazolam, Bentazepam, Brexanolone, Bromazepam, Brotizolam, Butabarbital, Butalbital, Camazepam, Chlordiazepoxide, Cinazepam, Cinolazepam, Clobazam, Clonazepam, Clorazepic acid, Clotiazepam, Cloxazolam, Delorazepam, Desflurane, Diazepam, Estazolam, Eszopiclone, Ethchlorvynol, Ethyl loflazepate, Etizolam, Etomidate, Flumazenil, Flunitrazepam, Flurazepam, Glutethimide, Halazepam, Halothane, Isoflurane, Ketazolam, Loprazolam, Lorazepam, Lormetazepam, Medazepam, Meprobamate, Metharbital, Methoxyflurane, Methyprylon, Mexazolam, Midazolam, Nitrazepam, Nordazepam, Oxazepam, Oxazepam acetate, Pentobarbital, Pinazepam, Prazepam, Primidone, Propofol, Quazepam, Remimazolam, Sevoflurane, Stiripentol, Talbutal, Temazepam, Triazolam
2GABA(A) Receptor positive modulatorsAcamprosate
3GABA(A) Receptor potentiatorsEnflurane
4GABA(A) Receptor bindersAmoxapine, Memantine
5GABA(A) Receptor antagonistsApalutamide, Lamotrigine, Prasterone, Thiocolchicoside
6GABA(A) Receptor agonistsStiripentol, Taurine
7GABA(A) Receptor inducersLamotrigine
8GABA(A) Receptor inhibitorsMedroxyprogesterone acetate
Interacting GroupInteracting Drugs
Doxefazepam is a GABA(A) Receptor Benzodiazepine Binding Site ligand
1GABA(A) Receptor Benzodiazepine Binding Site partial agonistsAdipiplon
2GABA(A) Receptor Benzodiazepine Binding Site ligands1,2-Benzodiazepine, 5,7,2′-trihydroxy-6,8-dimethoxyflavone, Adinazolam, Alprazolam, Bentazepam, Bromazepam, Brotizolam, Camazepam, Chlordiazepoxide, Cinazepam, Cinolazepam, Clobazam, Clonazepam, Clorazepic acid, Clotiazepam, Cloxazolam, Delorazepam, Diazepam, Estazolam, Ethyl loflazepate, Etizolam, Flunitrazepam, Flurazepam, Halazepam, Ketazolam, Loprazolam, Lorazepam, Lormetazepam, Medazepam, Mexazolam, Midazolam, Nitrazepam, Nordazepam, Oxazepam, Oxazepam acetate, Pinazepam, Prazepam, Quazepam, Remimazolam, Temazepam, Triazolam
3GABA(A) Receptor Benzodiazepine Binding Site inhibitorsLamotrigine, Olanzapine