Angina Pectoris

Also known as: Angina pectoris, unspecified / Anginal syndrome / Stenocardia / Anginal pain / Anginal discomfort / Angina syndrome / Ischaemic chest pain / Ischemic chest pain (finding) / Ischemic chest pain / Angina (disorder)

DrugDrug NameDrug Description
DB00335AtenololA synthetic beta-1 selective blocker used in the management of hypertension and chronic angina, and to reduce mortality in known or suspected myocardial infarction in hemodynamically stable patients.
DB09231BenidipineA synthetic dihydropyridine calcium channel blocker used to treat hypertension and angina pectoris.
DB04846CeliprololA beta-blocker for the management of hypertension and angina pectoris.
DB09401IsosorbideA vasodilator used for the prevention and treatment of angina pectoris due to coronary artery disease. It was previously used to reduce intraocular pressure.
DB00883Isosorbide dinitrateA vasodilator used to treat angina in coronary artery disease.
DB01020Isosorbide mononitrateA nitrate used to prevent and treat angina and to treat angina caused by coronary artery disease.
DB00264MetoprololA beta-blocker used in the treatment of hypertension and angina, and used to reduce mortality due to myocardial infarction.
DB09282MolsidomineA long-acting vasodilator used to treat angina pectoris, including in association with left heart failure and acute myocardial infarction.
DB01203NadololA non-selective beta-adrenergic antagonist used for the management of arrhythmias, angina pectoris, and hypertension.
DB09220NicorandilA vasodilatory drug that functions through potassium channels and intracellular cGMP concentrations commonly used to treat angina.
DB00727NitroglycerinA nitrate vasodilator used to treat or prevent angina, heart failure, hypertension, and anal fissures.
DB00960PindololA beta adrenoceptor antagonist used to treat hypertension, edema, ventricular tachycardias, and atrial fibrillation.
DB00571PropranololA non-selective beta adrenergic antagonist used to treat hypertension, angina, atrial fibrillation, myocardial infarction, migraine, essential tremor, hypertrophic subaortic stenosis, and pheochromocytoma.
DB09069TrimetazidineA piperazine derivative indicated as an adjunct therapy in symptomatic treatment of stable angina pectoris.
DrugDrug NameTargetType
DB00335AtenololBeta-1 adrenergic receptortarget
DB00335AtenololBeta-2 adrenergic receptortarget
DB00335AtenololCytochrome P450 2D6enzyme
DB00335AtenololBile salt export pumptransporter
DB00335AtenololSerum albumincarrier
DB09231BenidipineVoltage-dependent L-type calcium channeltarget
DB09231BenidipineVoltage-dependent N-type calcium channel subunit alpha-1Btarget
DB09231BenidipineVoltage-dependent T-type calcium channeltarget
DB09231BenidipineCytochrome P450 3A4enzyme
DB09231BenidipineCytochrome P450 3A5enzyme
DB04846CeliprololBeta-1 adrenergic receptortarget
DB04846CeliprololBeta-2 adrenergic receptortarget
DB04846CeliprololBeta-3 adrenergic receptortarget
DB04846CeliprololAlpha-2A adrenergic receptortarget
DB04846CeliprololAlpha-2B adrenergic receptortarget
DB04846CeliprololAlpha-2C adrenergic receptortarget
DB04846CeliprololCytochrome P450 2D6enzyme
DB09401IsosorbideGuanylate cyclasetarget
DB00883Isosorbide dinitrateAtrial natriuretic peptide receptor 1target
DB00883Isosorbide dinitrateCytochrome P450 2E1enzyme
DB01020Isosorbide mononitrateGuanylate cyclase soluble subunit alpha-2target
DB01020Isosorbide mononitrateGlutathione S-transferase Mu 1enzyme
DB01020Isosorbide mononitrateXanthine dehydrogenase/oxidaseenzyme
DB01020Isosorbide mononitrateAlcohol dehydrogenase class-3enzyme
DB00264MetoprololBeta-1 adrenergic receptortarget
DB00264MetoprololCytochrome P450 2D6enzyme
DB00264MetoprololBeta-2 adrenergic receptortarget
DB00264MetoprololSolute carrier family 22 member 2transporter
DB00264MetoprololSerum albumincarrier
DB00264MetoprololCytochrome P450 3A4enzyme
DB00264MetoprololBeta adrenergic receptortarget
DB09282MolsidomineGuanylate cyclase soluble subunit alpha-2target
DB09282MolsidomineGuanylate cyclase soluble subunit alpha-2enzyme
DB09282MolsidominecGMP-specific 3',5'-cyclic phosphodiesteraseenzyme
DB01203NadololBeta-1 adrenergic receptortarget
DB01203NadololBeta-2 adrenergic receptortarget
DB01203NadololP-glycoprotein 1transporter
DB01203NadololPOU domain, class 2, transcription factor 1transporter
DB01203NadololPOU domain, class 2, transcription factor 2transporter
DB01203NadololMultidrug and toxin extrusion protein 1transporter
DB01203NadololMultidrug and toxin extrusion protein 2transporter
DB01203Nadololalpha1-acid glycoproteincarrier
DB09220NicorandilATP-binding cassette sub-family C member 9target
DB00727NitroglycerinAtrial natriuretic peptide receptor 1target
DB00727NitroglycerinAldehyde dehydrogenase, mitochondrialenzyme
DB00960PindololBeta-1 adrenergic receptortarget
DB00960PindololBeta-2 adrenergic receptortarget
DB00960Pindolol5-hydroxytryptamine receptor 1Atarget
DB00960Pindolol5-hydroxytryptamine receptor 1Btarget
DB00960PindololCytochrome P450 2D6enzyme
DB00960PindololBeta-3 adrenergic receptortarget
DB00960PindololUDP-glucuronosyltransferases (UGTs)enzyme
DB00960PindololSulfotransferaseenzyme
DB00960PindololSolute carrier family 22 member 2transporter
DB00960Pindololalpha1-acid glycoproteincarrier
DB00571PropranololBeta-1 adrenergic receptortarget
DB00571PropranololBeta-2 adrenergic receptortarget
DB00571PropranololBeta-3 adrenergic receptortarget
DB00571Propranolol5-hydroxytryptamine receptor 1Atarget
DB00571Propranolol5-hydroxytryptamine receptor 1Btarget
DB00571PropranololCytochrome P450 1A2enzyme
DB00571PropranololCytochrome P450 2D6enzyme
DB00571PropranololAlpha-1-acid glycoprotein 1carrier
DB00571PropranololCytochrome P450 2C19enzyme
DB00571PropranololCytochrome P450 3A4enzyme
DB00571PropranololCytochrome P450 3A5enzyme
DB00571PropranololCytochrome P450 3A7enzyme
DB00571PropranololSolute carrier family 22 member 2transporter
DB00571PropranololP-glycoprotein 1transporter
DB00571PropranololCytochrome P450 1A1enzyme
DB00571PropranololAmine oxidase [flavin-containing] Aenzyme
DB00571PropranololSerum albumincarrier
DB09069TrimetazidineSerum albumincarrier
DB09069Trimetazidine3-ketoacyl-CoA thiolase, mitochondrialtarget
DrugDrug NamePhaseStatusCount
DB01016Glyburide1Completed1
DB05760Telcagepant1Completed1
DB12228Telcagepant1Completed1
DB00640Adenosine1 / 2Completed1
DB00062Albumin human2Completed1
DB00335Atenolol2Unknown Status1
DB04945Hemoglobin2Completed1
DB09106Hydroxyethyl Starch2Completed1
DB09083Ivabradine2Unknown Status1
DB09236Lacidipine2Completed1
DB00583Levocarnitine2Completed1
DB11816Omecamtiv Mecarbil2Completed1
DB01229Paclitaxel2Completed1
DB00945Acetylsalicylic acid3Completed1
DB00009Alteplase3Completed1
DB00758Clopidogrel3Terminated1
DB00975Dipyridamole3Completed1
DB01109Heparin3Completed1
DB09083Ivabradine3Completed1
DB14304Panax notoginseng root3Completed1
DB00243Ranolazine3Completed1
DB00054Abciximab4Completed1
DB00945Acetylsalicylic acid4Completed1
DB09302Alirocumab4Unknown Status1
DB00381Amlodipine4Completed1
DB00126Ascorbic acid4Unknown Status1
DB00335Atenolol4Completed1
DB01076Atorvastatin4Completed1
DB00006Bivalirudin4Completed1
DB00758Clopidogrel4Completed2
DB00758Clopidogrel4Terminated1
DB00758Clopidogrel4Unknown Status1
DB01120Gliclazide4Withdrawn1
DB01109Heparin4Completed1
DB00999Hydrochlorothiazide4Completed1
DB00159Icosapent4Unknown Status1
DB00264Metoprolol4Completed1
DB09220Nicorandil4Withdrawn1
DB00727Nitroglycerin4Completed1
DB00727Nitroglycerin4Unknown Status1
DB01132Pioglitazone4Completed1
DB06209Prasugrel4Terminated1
DB06209Prasugrel4Unknown Status1
DB00243Ranolazine4Completed1
DB00243Ranolazine4Withdrawn1
DB00412Rosiglitazone4Terminated1
DB00412Rosiglitazone4Withdrawn1
DB01098Rosuvastatin4Completed1
DB01098Rosuvastatin4Unknown Status2
DB00203Sildenafil4Completed1
DB00624Testosterone4Completed1
DB08816Ticagrelor4Completed1
DB08816Ticagrelor4Unknown Status1
DB00381AmlodipineNot AvailableCompleted1
DB06692AprotininNot AvailableCompleted1
DB01076AtorvastatinNot AvailableCompleted1
DB00796Candesartan cilexetilNot AvailableTerminated1
DB00758ClopidogrelNot AvailableTerminated1
DB00966TelmisartanNot AvailableTerminated1