Kidney Transplant Rejection

Also known as: Rejection; Transplant, Kidney / Renal Transplant Rejection / Acute allograft nephropathy / Renal transplant rejection (disorder)

DrugDrug NameDrug Description
DB00087AlemtuzumabA monoclonal anti-CD52 antibody used in the treatment of B-cell chronic lymphocytic leukemia and relapsing forms of multiple sclerosis.
DB09312Antilymphocyte immunoglobulin (horse)A primarily IgG immune globulin used to manage allograft rejection in renal transplant patients.
DB00993AzathioprineAn immunosuppressant used to prevent renal transplant rejection, treat rheumatoid arthritis, Crohn's disease, and ulcerative colitis.
DB06681BelataceptA selective T-cell costimulation blocker used in the prophylaxis of organ rejection in adult patients receiving a kidney transplant.
DB00091CyclosporineA steroid-sparing immunosuppressant used in organ and bone marrow transplants as well as inflammatory conditions such as ulcerative colitis, rheumatoid arthritis, and atopic dermatitis.
DB01590EverolimusA mammalian target of rapamycin (mTOR) kinase inhibitor used to treat various types of malignancies.
DB01024Mycophenolic acidAn immunosuppressant used to prevent organ transplant rejections.
DB00864TacrolimusA calcineurin inhibitor used to prevent organ transplant rejection and to treat moderate to severe atopic dermatitis.
DrugDrug NameTargetType
DB00087AlemtuzumabCAMPATH-1 antigentarget
DB00087AlemtuzumabLow affinity immunoglobulin gamma Fc region receptor III-Btarget
DB00087AlemtuzumabLow affinity immunoglobulin gamma Fc region receptor III-Atarget
DB00087AlemtuzumabHigh affinity immunoglobulin gamma Fc receptor Itarget
DB00087AlemtuzumabLow affinity immunoglobulin gamma Fc region receptor II-atarget
DB00087AlemtuzumabLow affinity immunoglobulin gamma Fc region receptor II-btarget
DB00087AlemtuzumabLow affinity immunoglobulin gamma Fc region receptor II-ctarget
DB00993AzathioprineThiopurine S-methyltransferaseenzyme
DB00993AzathioprineXanthine dehydrogenase/oxidaseenzyme
DB00993AzathioprineGlutathione S-transferase A1enzyme
DB00993AzathioprineGlutathione S-transferase A2enzyme
DB00993AzathioprineGlutathione S-transferase Mu 1enzyme
DB00993AzathioprineRas-related C3 botulinum toxin substrate 1target
DB00993AzathioprineCytochrome P450 1A2enzyme
DB00993AzathioprineHypoxanthine-guanine phosphoribosyltransferaseenzyme
DB00993AzathioprineNucleotide triphosphate diphosphatase NUDT15enzyme
DB00993AzathioprineEquilibrative nucleoside transporter 2transporter
DB00993AzathioprineSolute carrier family 28 member 3transporter
DB00993AzathioprineP-glycoprotein 1transporter
DB00993AzathioprineSolute carrier family 43 member 3transporter
DB00993AzathioprineSerum albumincarrier
DB00993AzathioprineInosine-5'-monophosphate dehydrogenase 1enzyme
DB00993AzathioprineInosine-5'-monophosphate dehydrogenase 2enzyme
DB00993AzathioprineGMP synthase [glutamine-hydrolyzing]enzyme
DB00993AzathioprineInosine triphosphate pyrophosphataseenzyme
DB06681BelataceptT-lymphocyte activation antigen CD86target
DB06681BelataceptT-lymphocyte activation antigen CD80target
DB00091CyclosporineCalcium signal-modulating cyclophilin ligandtarget
DB00091CyclosporinePeptidyl-prolyl cis-trans isomerase Atarget
DB00091CyclosporineCalcineurin subunit B type 2target
DB00091CyclosporineCytochrome P450 3A5enzyme
DB00091CyclosporineCytochrome P450 3A4enzyme
DB00091CyclosporineP-glycoprotein 1transporter
DB00091CyclosporineBile salt export pumptransporter
DB00091CyclosporineIleal sodium/bile acid cotransportertransporter
DB00091CyclosporineSodium/bile acid cotransportertransporter
DB00091CyclosporineSolute carrier family 22 member 6transporter
DB00091CyclosporineMultidrug resistance-associated protein 7transporter
DB00091CyclosporineCanalicular multispecific organic anion transporter 1transporter
DB00091CyclosporineATP-binding cassette sub-family G member 2transporter
DB00091CyclosporineSolute carrier organic anion transporter family member 1B1transporter
DB00091CyclosporineCytochrome P450 2C19enzyme
DB00091CyclosporineCytochrome P450 2D6enzyme
DB00091CyclosporinePeptidyl-prolyl cis-trans isomerase F, mitochondrialtarget
DB00091CyclosporineSolute carrier organic anion transporter family member 1B3transporter
DB01590EverolimusSerine/threonine-protein kinase mTORtarget
DB01590EverolimusCytochrome P450 3A4enzyme
DB01590EverolimusSolute carrier organic anion transporter family member 1B1transporter
DB01590EverolimusSolute carrier organic anion transporter family member 1B3transporter
DB01590EverolimusSolute carrier organic anion transporter family member 1A2transporter
DB01590EverolimusCytochrome P450 2D6enzyme
DB01590EverolimusP-glycoprotein 1transporter
DB01024Mycophenolic acidInosine-5'-monophosphate dehydrogenase 2target
DB01024Mycophenolic acidInosine-5'-monophosphate dehydrogenase 1target
DB01024Mycophenolic acidUDP-glucuronosyltransferase 1-1enzyme
DB01024Mycophenolic acidUDP-glucuronosyltransferase 1-9enzyme
DB01024Mycophenolic acidUDP-glucuronosyltransferase 2B7enzyme
DB01024Mycophenolic acidUDP-glucuronosyltransferase 1-7enzyme
DB01024Mycophenolic acidUDP-glucuronosyltransferase 1-6enzyme
DB01024Mycophenolic acidSerum albumincarrier
DB01024Mycophenolic acidUDP-glucuronosyltransferase 1-8enzyme
DB01024Mycophenolic acidUDP-glucuronosyltransferase 1-10enzyme
DB01024Mycophenolic acidCytochrome P450 3A4enzyme
DB01024Mycophenolic acidCytochrome P450 3A5enzyme
DB01024Mycophenolic acidCytochrome P450 2C8enzyme
DB00864TacrolimusPeptidyl-prolyl cis-trans isomerase FKBP1Atarget
DB00864TacrolimusCytochrome P450 3A4enzyme
DB00864TacrolimusCytochrome P450 3A5enzyme
DB00864TacrolimusP-glycoprotein 1transporter
DB00864TacrolimusATP-binding cassette sub-family A member 5transporter
DB00864TacrolimusSerum albumincarrier
DB00864TacrolimusAlpha-1-acid glycoprotein 1carrier
DB00864TacrolimusSolute carrier organic anion transporter family member 1B1transporter
DrugDrug NamePhaseStatusCount
DB00864Tacrolimus0Terminated2
DB15726Human Umbilical Cord Mesenchymal Stem Cells1Terminated1
DB15726Human Umbilical Cord Mesenchymal Stem Cells1Unknown Status1
DB08879Belimumab1 / 2Completed1
DB00188Bortezomib1 / 2Completed1
DB16741Bortezomib D-mannitol1 / 2Completed1
DB12849Clazakizumab1 / 2Active Not Recruiting1
DB09331Daratumumab1 / 2Completed1
DB12010Fostamatinib1 / 2Recruiting1
DB00688Mycophenolate mofetil1 / 2Withdrawn1
DB00073Rituximab1 / 2Completed1
DB00864Tacrolimus1 / 2Withdrawn1
DB00098Antithymocyte immunoglobulin (rabbit)2Completed2
DB06681Belatacept2Completed1
DB01590Everolimus2Unknown Status1
DB08868Fingolimod2Enrolling by Invitation1
DB15726Human Umbilical Cord Mesenchymal Stem Cells2Unknown Status1
DB15258Imlifidase2Completed1
DB00065Infliximab2Completed1
DB11228Methylcellulose2Enrolling by Invitation1
DB00959Methylprednisolone2Completed1
DB12821Perflubutane2Completed1
DB00860Prednisolone2Completed1
DB00864Tacrolimus2Completed2
DB00864Tacrolimus2Enrolling by Invitation1
DB00864Tacrolimus2Recruiting1
DB16974Tegoprubart2Enrolling by Invitation1
DB16974Tegoprubart2Recruiting1
DB00688Mycophenolate mofetil2 / 3Not Yet Recruiting1
DB00864Tacrolimus2 / 3Not Yet Recruiting2
DB00098Antithymocyte immunoglobulin (rabbit)3Not Yet Recruiting1
DB00098Antithymocyte immunoglobulin (rabbit)3Terminated1
DB00074Basiliximab3Not Yet Recruiting1
DB17310Heme arginate3Terminated1
DB00028Human immunoglobulin G3Active Not Recruiting1
DB18513MDR-1013Active Not Recruiting1
DB00959Methylprednisolone3Active Not Recruiting1
DB00688Mycophenolate mofetil3Not Yet Recruiting1
DB01024Mycophenolic acid3Not Yet Recruiting1
DB00073Rituximab3Active Not Recruiting1
DB09153Sodium chloride3Terminated1
DB00864Tacrolimus3Not Yet Recruiting1
DB00098Antithymocyte immunoglobulin (rabbit)4Completed2
DB00098Antithymocyte immunoglobulin (rabbit)4Recruiting3
DB00993Azathioprine4Recruiting1
DB00074Basiliximab4Completed2
DB00074Basiliximab4Recruiting2
DB06681Belatacept4Completed2
DB06681Belatacept4Recruiting1
DB11799Bictegravir4Active Not Recruiting1
DB00091Cyclosporine4Terminated1
DB00879Emtricitabine4Active Not Recruiting1
DB01590Everolimus4Completed2
DB01590Everolimus4Recruiting1
DB01590Everolimus4Terminated1
DB01590Everolimus4Unknown Status1
DB00959Methylprednisolone4Recruiting1
DB00688Mycophenolate mofetil4Recruiting2
DB00688Mycophenolate mofetil4Terminated1
DB01024Mycophenolic acid4Completed3
DB01024Mycophenolic acid4Not Yet Recruiting1
DB01024Mycophenolic acid4Recruiting1
DB01024Mycophenolic acid4Terminated1
DB01024Mycophenolic acid4Unknown Status1
DB00635Prednisone4Completed2
DB00635Prednisone4Recruiting2
DB00635Prednisone4Unknown Status1
DB00877Sirolimus4Completed1
DB00864Tacrolimus4Active Not Recruiting2
DB00864Tacrolimus4Completed3
DB00864Tacrolimus4Recruiting1
DB00864Tacrolimus4Terminated1
DB09299Tenofovir alafenamide4Active Not Recruiting1
DB00098Antithymocyte immunoglobulin (rabbit)Not AvailableCompleted1
DB00074BasiliximabNot AvailableCompleted1
DB00074BasiliximabNot AvailableNot Yet Recruiting1
DB06681BelataceptNot AvailableNot Yet Recruiting1
DB06215FerumoxytolNot AvailableCompleted1
DB15258ImlifidaseNot AvailableTerminated1
DB00688Mycophenolate mofetilNot AvailableNot Yet Recruiting1
DB00073RituximabNot AvailableCompleted1
DB00864TacrolimusNot AvailableRecruiting2