Agitation

Also known as: Agitational state / Agitated states / Agitated state / Excitement abnormal / Feeling agitated (finding) / Agitated

DrugDrug NameDrug Description
DB00543AmoxapineA tricyclic antidepressant used in the treatment of neurotic or reactive depressive disorders and endogenous or psychotic depression.
DB01238AripiprazoleAn atypical antipsychotic used in the treatment of a wide variety of mood and psychotic disorders, such as schizophrenia, bipolar I, major depressive disorder, irritability associated with autism, and Tourette's syndrome.
DB09128BrexpiprazoleA serotonin–dopamine activity modulator used in the treatment of major depressive disorder as an adjunct, schizophrenia, and agitation associated with dementia due to Alzheimer’s disease.
DB00633DexmedetomidineAn alpha-2 agonist used for sedation during various procedures.
DB00450DroperidolA butyrophenone derivative and dopamine antagonist used to prevent and treat postoperative nausea and vomiting.
DB00186LorazepamA short-acting benzodiazepine commonly used to treat panic disorders, severe anxiety, and seizures.
DB13437MedazepamA long-acting benzodiazepine used for its sedative and anxiolytic properties.
DB00457PrazosinAn alpha-blocker that causes a decrease in total peripheral resistance and is used to treat hypertension.
DB00831TrifluoperazineA phenothiazine used to treat depression, anxiety, and agitation.
DB00246ZiprasidoneAn atypical antipsychotic used to manage schizophrenia, bipolar mania, and agitation in patients with schizophrenia.
DB01624ZuclopenthixolAn antipsychotic indicated for the management of schizophrenia. The acuphase formulation is indicated for initial treatment of acute psychosis or exacerbation of psychosis, while the depot formulation is best for maintenance.
DrugDrug NameTargetType
DB00543AmoxapineSodium-dependent serotonin transportertarget
DB00543AmoxapineSodium-dependent noradrenaline transportertarget
DB00543AmoxapineAlpha-2A adrenergic receptortarget
DB00543AmoxapineDopamine D2 receptortarget
DB00543AmoxapineAlpha-1A adrenergic receptortarget
DB00543AmoxapineDopamine D1 receptortarget
DB00543AmoxapineMuscarinic acetylcholine receptor M1target
DB00543AmoxapineGamma-aminobutyric acid receptor subunit alpha-1target
DB00543AmoxapineAlpha-1-acid glycoprotein 1carrier
DB00543AmoxapineCytochrome P450 2D6enzyme
DB00543Amoxapine5-hydroxytryptamine receptor 2Atarget
DB00543Amoxapine5-hydroxytryptamine receptor 2Ctarget
DB00543Amoxapine5-hydroxytryptamine receptor 6target
DB00543Amoxapine5-hydroxytryptamine receptor 7target
DB00543AmoxapineDopamine D3 receptortarget
DB00543AmoxapineDopamine D4 receptortarget
DB00543AmoxapineHistamine H1 receptortarget
DB00543AmoxapineAlpha-1 adrenergic receptorstarget
DB00543AmoxapineMuscarinic acetylcholine receptortarget
DB00543Amoxapine5-hydroxytryptamine receptor 2Btarget
DB00543Amoxapine5-hydroxytryptamine receptor 3Atarget
DB00543Amoxapine5-hydroxytryptamine receptor 1Atarget
DB00543Amoxapine5-hydroxytryptamine receptor 1Btarget
DB00543AmoxapineAlpha-2 adrenergic receptorstarget
DB00543AmoxapineHistamine H4 receptortarget
DB00543AmoxapineGABA(A) Receptortarget
DB00543AmoxapineSodium-dependent dopamine transportertarget
DB01238AripiprazoleDopamine D2 receptortarget
DB01238Aripiprazole5-hydroxytryptamine receptor 1Atarget
DB01238Aripiprazole5-hydroxytryptamine receptor 2Atarget
DB01238AripiprazoleCytochrome P450 3A4enzyme
DB01238AripiprazoleCytochrome P450 2D6enzyme
DB01238Aripiprazole5-hydroxytryptamine receptor 1Btarget
DB01238Aripiprazole5-hydroxytryptamine receptor 1Dtarget
DB01238Aripiprazole5-hydroxytryptamine receptor 1Etarget
DB01238AripiprazoleDopamine D1 receptortarget
DB01238AripiprazoleDopamine D5 receptortarget
DB01238AripiprazoleDopamine D3 receptortarget
DB01238AripiprazoleDopamine D4 receptortarget
DB01238Aripiprazole5-hydroxytryptamine receptor 2Ctarget
DB01238Aripiprazole5-hydroxytryptamine receptor 3Atarget
DB01238Aripiprazole5-hydroxytryptamine receptor 6target
DB01238Aripiprazole5-hydroxytryptamine receptor 7target
DB01238AripiprazoleHistamine H1 receptortarget
DB01238AripiprazoleAlpha-1A adrenergic receptortarget
DB01238AripiprazoleAlpha-1B adrenergic receptortarget
DB01238AripiprazoleAlpha-2A adrenergic receptortarget
DB01238AripiprazoleAlpha-2B adrenergic receptortarget
DB01238AripiprazoleAlpha-2C adrenergic receptortarget
DB01238AripiprazoleCytochrome P450 3A5enzyme
DB01238AripiprazoleCytochrome P450 3A7enzyme
DB01238AripiprazoleSerum albumincarrier
DB01238Aripiprazole5-hydroxytryptamine receptor 2Btarget
DB01238Aripiprazole5-hydroxytryptamine receptor 5Atarget
DB01238AripiprazoleBeta-1 adrenergic receptortarget
DB01238AripiprazoleBeta-2 adrenergic receptortarget
DB01238AripiprazoleHistamine H2 receptortarget
DB01238AripiprazoleHistamine H3 receptortarget
DB01238AripiprazoleHistamine H4 receptortarget
DB01238AripiprazoleMuscarinic acetylcholine receptor M1target
DB01238AripiprazoleMuscarinic acetylcholine receptor M2target
DB01238AripiprazoleMuscarinic acetylcholine receptor M3target
DB01238AripiprazoleMuscarinic acetylcholine receptor M4target
DB01238AripiprazoleMuscarinic acetylcholine receptor M5target
DB01238AripiprazoleKappa-type opioid receptortarget
DB01238AripiprazoleMu-type opioid receptortarget
DB01238AripiprazoleDelta-type opioid receptortarget
DB01238AripiprazoleGlutamate (NMDA) receptortarget
DB01238AripiprazoleSodium-dependent dopamine transportertarget
DB01238AripiprazoleSodium-dependent serotonin transportertarget
DB01238AripiprazoleP-glycoprotein 1transporter
DB01238AripiprazoleATP-binding cassette sub-family G member 2transporter
DB09128BrexpiprazoleCytochrome P450 2D6enzyme
DB09128BrexpiprazoleCytochrome P450 3A4enzyme
DB09128Brexpiprazole5-hydroxytryptamine receptor 1Atarget
DB09128BrexpiprazoleDopamine D2 receptortarget
DB09128Brexpiprazole5-hydroxytryptamine receptor 2Atarget
DB09128BrexpiprazoleAlpha-2C adrenergic receptortarget
DB09128BrexpiprazoleAlpha-1B adrenergic receptortarget
DB09128BrexpiprazoleMultidrug and toxin extrusion protein 2transporter
DB09128BrexpiprazoleSerum albumincarrier
DB09128BrexpiprazoleAlpha-1-acid glycoprotein 1carrier
DB09128BrexpiprazoleDopamine D3 receptortarget
DB09128Brexpiprazole5-hydroxytryptamine receptor 2Btarget
DB09128Brexpiprazole5-hydroxytryptamine receptor 7target
DB09128BrexpiprazoleAlpha-1A adrenergic receptortarget
DB09128BrexpiprazoleAlpha-1D adrenergic receptortarget
DB09128BrexpiprazoleHistamine H1 receptortarget
DB09128BrexpiprazoleMuscarinic acetylcholine receptor M1target
DB00633DexmedetomidineAlpha-2A adrenergic receptortarget
DB00633DexmedetomidineCytochrome P450 2E1enzyme
DB00633DexmedetomidineCytochrome P450 1A2enzyme
DB00633DexmedetomidineCytochrome P450 1A1enzyme
DB00633DexmedetomidineCytochrome P450 2D6enzyme
DB00450DroperidolDopamine D2 receptortarget
DB00450DroperidolAlpha-1A adrenergic receptortarget
DB00186LorazepamUDP-glucuronosyltransferase 2B15enzyme
DB00186LorazepamGABA(A) Receptortarget
DB00186LorazepamCytochrome P450 3A4enzyme
DB00186LorazepamGABA(A) Receptor Benzodiazepine Binding Sitetarget
DB13437MedazepamGABA(A) Receptortarget
DB13437MedazepamGABA(A) Receptor Benzodiazepine Binding Sitetarget
DB00457PrazosinAlpha-1A adrenergic receptortarget
DB00457PrazosinAlpha-1B adrenergic receptortarget
DB00457PrazosinAlpha-1D adrenergic receptortarget
DB00457PrazosinPotassium voltage-gated channel subfamily H member 2target
DB00457PrazosinAlpha-1-acid glycoprotein 1carrier
DB00457PrazosinSolute carrier family 22 member 1transporter
DB00457PrazosinSolute carrier family 22 member 3transporter
DB00457PrazosinP-glycoprotein 1transporter
DB00457PrazosinATP-binding cassette sub-family G member 2transporter
DB00457PrazosinAlpha-2A adrenergic receptortarget
DB00457PrazosinAlpha-2B adrenergic receptortarget
DB00457PrazosinAlpha-1 adrenergic receptorstarget
DB00831TrifluoperazineDopamine D2 receptortarget
DB00831TrifluoperazineAlpha-1A adrenergic receptortarget
DB00831TrifluoperazineNeuron-specific vesicular protein calcyontarget
DB00831TrifluoperazineXanthine dehydrogenase/oxidaseenzyme
DB00831TrifluoperazineUDP-glucuronosyltransferase 1-4enzyme
DB00831TrifluoperazineCytochrome P450 1A2enzyme
DB00831TrifluoperazineP-glycoprotein 1transporter
DB00831TrifluoperazineCalmodulintarget
DB00831TrifluoperazineTroponin C, slow skeletal and cardiac musclestarget
DB00831TrifluoperazineProtein S100-A4target
DB00246ZiprasidoneAlpha-1A adrenergic receptortarget
DB00246ZiprasidoneDopamine D2 receptortarget
DB00246Ziprasidone5-hydroxytryptamine receptor 2Ctarget
DB00246ZiprasidoneDopamine D3 receptortarget
DB00246Ziprasidone5-hydroxytryptamine receptor 1Atarget
DB00246Ziprasidone5-hydroxytryptamine receptor 1Dtarget
DB00246ZiprasidoneHistamine H1 receptortarget
DB00246Ziprasidone5-hydroxytryptamine receptor 2Atarget
DB00246ZiprasidoneDopamine D4 receptortarget
DB00246Ziprasidone5-hydroxytryptamine receptor 7target
DB00246ZiprasidoneCytochrome P450 3A4enzyme
DB00246ZiprasidoneAlpha-2A adrenergic receptortarget
DB00246ZiprasidoneAlpha-1B adrenergic receptortarget
DB00246ZiprasidoneAlpha-2B adrenergic receptortarget
DB00246ZiprasidoneAlpha-2C adrenergic receptortarget
DB00246ZiprasidoneDopamine D1 receptortarget
DB00246ZiprasidoneDopamine D5 receptortarget
DB00246ZiprasidoneMuscarinic acetylcholine receptor M1target
DB00246ZiprasidoneMuscarinic acetylcholine receptor M2target
DB00246ZiprasidoneMuscarinic acetylcholine receptor M3target
DB00246ZiprasidoneMuscarinic acetylcholine receptor M4target
DB00246ZiprasidoneMuscarinic acetylcholine receptor M5target
DB00246Ziprasidone5-hydroxytryptamine receptor 1Btarget
DB00246Ziprasidone5-hydroxytryptamine receptor 1Etarget
DB00246Ziprasidone5-hydroxytryptamine receptor 6target
DB00246ZiprasidoneAldehyde oxidaseenzyme
DB00246ZiprasidoneSerum albumincarrier
DB00246ZiprasidoneP-glycoprotein 1transporter
DB00246ZiprasidoneAlpha-1-acid glycoprotein 1carrier
DB00246Ziprasidone5-hydroxytryptamine 3 receptortarget
DB00246Ziprasidone5-hydroxytryptamine receptor 5Atarget
DB01624ZuclopenthixolDopamine D1 receptortarget
DB01624ZuclopenthixolDopamine D5 receptortarget
DB01624ZuclopenthixolDopamine D2 receptortarget
DB01624ZuclopenthixolCytochrome P450 2D6enzyme
DB01624ZuclopenthixolAlpha-1A adrenergic receptortarget
DB01624ZuclopenthixolAlpha-2A adrenergic receptortarget
DB01624Zuclopenthixol5-hydroxytryptamine receptor 2Atarget
DB01624ZuclopenthixolHistamine H1 receptortarget
DB01624ZuclopenthixolCytochrome P450 3A4enzyme
DrugDrug NamePhaseStatusCount
DB00633Dexmedetomidine1Completed1
DB09061Cannabidiol2Recruiting1
DB00633Dexmedetomidine2Completed2
DB00633Dexmedetomidine2Terminated1
DB00633Dexmedetomidine2Withdrawn1
DB00514Dextromethorphan2Completed1
DB00502Haloperidol2Completed1
DB14509Lithium carbonate2Completed1
DB04870Oleoyl-estrone2Terminated1
DB00908Quinidine2Completed1
DB11344(+)-menthol2 / 3Completed1
DB00316Acetaminophen2 / 3Completed1
DB14283Angelica archangelica root2 / 3Completed1
DB00921Buprenorphine2 / 3Completed1
DB15649Carbomer2 / 3Completed1
DB00633Dexmedetomidine2 / 3Completed1
DB10344Ginger2 / 3Completed1
DB00502Haloperidol2 / 3Completed1
DB16021Levosulpiride2 / 3Completed1
DB00295Morphine2 / 3Completed1
DB00486Nabilone2 / 3Completed1
DB02701Nicotinamide2 / 3Completed1
DB00230Pregabalin2 / 3Completed1
DB09446Safflower oil2 / 3Completed1
DB00215Citalopram3Completed1
DB00633Dexmedetomidine3Completed4
DB00633Dexmedetomidine3Terminated1
DB00502Haloperidol3Completed1
DB00186Lorazepam3Completed1
DB00486Nabilone3Recruiting1
DB00334Olanzapine3Completed1
DB01224Quetiapine3Terminated1
DB06140SUVN-5023Recruiting1
DB00313Valproic acid3Terminated1
DB06216Asenapine4Completed1
DB00245Benzatropine4Completed1
DB00477Chlorpromazine4Completed1
DB00633Dexmedetomidine4Completed3
DB00633Dexmedetomidine4Not Yet Recruiting1
DB00633Dexmedetomidine4Recruiting1
DB00633Dexmedetomidine4Unknown Status2
DB01175Escitalopram4Completed1
DB00813Fentanyl4Completed1
DB00502Haloperidol4Completed3
DB00502Haloperidol4Withdrawn1
DB01221Ketamine4Completed1
DB01221Ketamine4Withdrawn1
DB00186Lorazepam4Completed1
DB00653Magnesium sulfate4Unknown Status1
DB01065Melatonin4Completed1
DB00370Mirtazapine4Completed1
DB00844Nalbuphine4Recruiting1
DB01069Promethazine4Completed1
DB00818Propofol4Completed2
DB01224Quetiapine4Completed1
DB00899Remifentanil4Completed1
DB00899Remifentanil4Unknown Status1
DB00734Risperidone4Completed3
DB00734Risperidone4Withdrawn1
DB00296Ropivacaine4Completed1
DB01236Sevoflurane4Completed1
DB00656Trazodone4Withdrawn1
DB00246Ziprasidone4Withdrawn1
DB00611ButorphanolNot AvailableUnknown Status1
DB00633DexmedetomidineNot AvailableCompleted2
DB00813FentanylNot AvailableCompleted1
DB00502HaloperidolNot AvailableCompleted1
DB00502HaloperidolNot AvailableTerminated1
DB00683MidazolamNot AvailableCompleted3
DB00334OlanzapineNot AvailableTerminated1