Atherosclerotic Cardiovascular Disease

Also known as: Atherosclerotic Cardiovascular Diseases / Atheromatosis / Atherosclerotic heart disease of native coronary artery / Atherosclerosis / Atherosclerosis (morphologic abnormality) / Arteriosclerotic vascular disease (disorder) / Arteriosclerosis / Arteriosclerosis (morphologic abnormality) / Vascular sclerosis (morphologic abnormality)

DrugDrug NameDrug Description
DB00945Acetylsalicylic acidA salicylate used to treat pain, fever, inflammation, migraines, and reducing the risk of major adverse cardiovascular events.
DB11936Bempedoic acidA drug used in conjunction with lifestyle modification and/or other agents for the treatment of refractory hypercholesterolemia.
DB14901InclisiranA PCSK9-targeting short interfering RNA (siRNA) that lowers plasma LDL-cholesterol levels.
DB01098RosuvastatinAn HMG-CoA reductase inhibitor used to lower lipid levels and reduce the risk of cardiovascular disease including myocardial infarction and stroke.
DrugDrug NameTargetType
DB00945Acetylsalicylic acidProstaglandin G/H synthase 1target
DB00945Acetylsalicylic acidProstaglandin G/H synthase 2target
DB00945Acetylsalicylic acidAldo-keto reductase family 1 member C1target
DB00945Acetylsalicylic acidSolute carrier family 22 member 6transporter
DB00945Acetylsalicylic acidP-glycoprotein 1transporter
DB00945Acetylsalicylic acidCytochrome P450 2C19enzyme
DB00945Acetylsalicylic acidCytochrome P450 2C9enzyme
DB00945Acetylsalicylic acid5'-AMP-activated protein kinasetarget
DB00945Acetylsalicylic acidEndothelin-1 receptortarget
DB00945Acetylsalicylic acidCellular tumor antigen p53target
DB00945Acetylsalicylic acid78 kDa glucose-regulated proteintarget
DB00945Acetylsalicylic acidRibosomal protein S6 kinase alpha-3target
DB00945Acetylsalicylic acidNF-kappa-B inhibitor alphatarget
DB00945Acetylsalicylic acidTumor necrosis factor-inducible gene 6 proteintarget
DB00945Acetylsalicylic acidCaspase-1target
DB00945Acetylsalicylic acidCaspase-3target
DB00945Acetylsalicylic acidInhibitor of nuclear factor kappa-B kinase subunit betatarget
DB00945Acetylsalicylic acidExtracellular signal-regulated kinase (ERK)target
DB00945Acetylsalicylic acidG1/S-specific cyclin-D1target
DB00945Acetylsalicylic acidMyc proto-oncogene proteintarget
DB00945Acetylsalicylic acidProliferating cell nuclear antigentarget
DB00945Acetylsalicylic acidCyclin Atarget
DB00945Acetylsalicylic acidUDP-glucuronosyltransferase 1-6enzyme
DB00945Acetylsalicylic acidArylamine N-acetyltransferase 2enzyme
DB00945Acetylsalicylic acidSolute carrier family 22 member 8transporter
DB00945Acetylsalicylic acidSialidase-1target
DB11936Bempedoic acidATP-citrate synthasetarget
DB11936Bempedoic acidVery long-chain acyl-CoA synthetaseenzyme
DB11936Bempedoic acidSolute carrier organic anion transporter family member 1B1transporter
DB11936Bempedoic acidCanalicular multispecific organic anion transporter 2transporter
DB11936Bempedoic acidSolute carrier organic anion transporter family member 1B3transporter
DB11936Bempedoic acidUDP-glucuronosyltransferase 2B7enzyme
DB11936Bempedoic acidNUAK family SNF1-like kinase 2enzyme
DB14901InclisiranProprotein convertase subtilisin/kexin type 9target
DB01098Rosuvastatin3-hydroxy-3-methylglutaryl-coenzyme A reductasetarget
DB01098RosuvastatinCytochrome P450 2C9enzyme
DB01098RosuvastatinMultidrug resistance-associated protein 4transporter
DB01098RosuvastatinSolute carrier organic anion transporter family member 1A2transporter
DB01098RosuvastatinSolute carrier organic anion transporter family member 1B3transporter
DB01098RosuvastatinSolute carrier organic anion transporter family member 2B1transporter
DB01098RosuvastatinCystine/glutamate transportertransporter
DB01098RosuvastatinSolute carrier organic anion transporter family member 1B1transporter
DB01098RosuvastatinBile salt export pumptransporter
DB01098RosuvastatinATP-binding cassette sub-family G member 2transporter
DB01098RosuvastatinSerum albumincarrier
DB01098RosuvastatinCanalicular multispecific organic anion transporter 1transporter
DB01098RosuvastatinSolute carrier family 22 member 8transporter
DB01098RosuvastatinSodium/bile acid cotransportertransporter
DB01098RosuvastatinIntegrin alpha-Ltarget
DrugDrug NamePhaseStatusCount
DB01373Calcium1Recruiting1
DB01098Rosuvastatin1Recruiting1
DB09303Evolocumab2Completed2
DB09303Evolocumab2Recruiting1
DB14901Inclisiran2Completed2
DB18728Olezarsen2Completed1
DB12520Plozalizumab2Withdrawn1
DB12849Clazakizumab2 / 3Active Not Recruiting1
DB09302Alirocumab3Completed1
DB06630Anacetrapib3Active Not Recruiting1
DB00335Atenolol3Completed1
DB11936Bempedoic acid3Completed4
DB00999Hydrochlorothiazide3Completed1
DB14901Inclisiran3Active Not Recruiting2
DB14901Inclisiran3Completed2
DB00563Methotrexate3Completed1
DB14890Obicetrapib3Active Not Recruiting1
DB14890Obicetrapib3Recruiting1
DB00275Olmesartan3Completed1
DB00052Somatotropin3Unknown Status1
DB00945Acetylsalicylic acid4Completed1
DB00125Arginine4Terminated1
DB01076Atorvastatin4Completed1
DB01076Atorvastatin4Recruiting1
DB09303Evolocumab4Completed2
DB09303Evolocumab4Not Yet Recruiting1
DB17310Heme arginate4Terminated1
DB14901Inclisiran4Not Yet Recruiting1
DB00945Acetylsalicylic acidNot AvailableCompleted1
DB06630AnacetrapibNot AvailableCompleted1
DB01076AtorvastatinNot AvailableRecruiting1
DB01076AtorvastatinNot AvailableUnknown Status1
DB09303EvolocumabNot AvailableActive Not Recruiting1
DB00973EzetimibeNot AvailableActive Not Recruiting1
DB00973EzetimibeNot AvailableRecruiting1
DB14901InclisiranNot AvailableActive Not Recruiting2
DB08860PitavastatinNot AvailableRecruiting1