Also known as: Headache / Cephalgia / Cephalalgia / Headaches / Head Pain / [D]Headache / Headache NOS / Pain head / Facial pain NOS
DrugDrug NameDrug Description
DB00945Acetylsalicylic acidThe prototypical analgesic used in the treatment of mild to moderate pain. It has anti-inflammatory and antipyretic properties and acts as an inhibitor of cyclooxygenase which results in the inhibition of the biosynthesis of prostaglandins. Acetylsalicylic acid also inhibits platelet aggregation and is used in the prevention of arterial and venous thrombosis. (From Martindale, The Extra Pharmacopoeia, 30th ed, p5)
DB06681BelataceptBelatacept is a soluble fusion protein, which links the extracellular domain of human cytotoxic T-lymphocyte-associated antigen 4 (CTLA-4) to the modified Fc (hinge, CH2, and CH3 domains) portion of human immunoglobulin G1 (IgG1). Structurally, abatacept is a glycosylated fusion protein with a MALDI-MS molecular weight of 92,300 Da and it is a homodimer of two homologous polypeptide chains of 357 amino acids each. It is produced through recombinant DNA technology in mammalian CHO cells. The drug has activity as a selective co-stimulation modulator with inhibitory activity on T lymphocytes. It is approved for the treatment of rheumatoid arthritis. Belatacept selectively blocks the process of T-cell activation. It was developed by Bristol-Myers-Squibb. It differs from abatacept (Orencia) by only 2 amino acids. FDA approved on June 15, 2011.
DB00083Botulinum Toxin Type APurified botulinum toxin from Clostridium botulinum, purified from culture via dialysis and acid precipitation.
DB01050IbuprofenIbuprofen, a propionic acid derivative, is a prototypical nonsteroidal anti-inflammatory agent (NSAIA) with analgesic and antipyretic properties.
DB09054IdelalisibIdelalisib is a phosphoinositide 3-kinase inhibitor indicated in the treatment of chronic lymphocytic leukemia (CLL), relapsed follicular B-cell non-Hodgkin lymphoma (FL), and relapsed small lymphocytic lymphoma (SLL). For the treatment of relapsed CLL, it is currently indicated as a second-line agent in combination with rituximab in patients for whom rituximab alone would be considered appropriate therapy due to other co-morbidities, while in the treatment of FL and SLL it is intended to be used in patients who have received at least two prior systemic therapies. More specifically, idelalisib targets P110δ, the delta isoform of the enzyme phosphatidylinositol-4,5-bisphosphate 3-kinase, also known as PI-3K. The PI-3Ks are a family of enzymes involved in cellular functions such as cell growth, proliferation, differentiation, motility, survival and intracellular trafficking, which in turn are involved in cancer. In contrast to the other class IA PI3Ks p110α and p110β, p110δ is principally expressed in leukocytes (white blood cells) and is important for the function of T cells, B cell, mast cells and neutrophils. By inhibiting this enzyme, idelalisib induces apoptosis of malignant cells and inhibits several cell signaling pathways, including B-cell receptor (BCR) signaling and C-X-C chemokine receptors type 5 and type 4 signalling, which are involved in trafficking and homing of B-cells to the lymph nodes and bone marrow. Treatment of lymphoma cells with idelalisib has been shown to result in inhibition of chemotaxis and adhesion, and reduced cell viability.
DB00788NaproxenAn anti-inflammatory agent with analgesic and antipyretic properties. Both the acid and its sodium salt are used in the treatment of rheumatoid arthritis and other rheumatic or musculoskeletal disorders, dysmenorrhea, and acute gout.
DrugDrug NameTargetType
DB00945Acetylsalicylic acidProstaglandin G/H synthase 1target
DB00945Acetylsalicylic acidProstaglandin G/H synthase 2target
DB00945Acetylsalicylic acidSerum albumincarrier
DB00945Acetylsalicylic acidAldo-keto reductase family 1 member C1target
DB00945Acetylsalicylic acidSolute carrier family 22 member 6transporter
DB00945Acetylsalicylic acidMultidrug resistance protein 1transporter
DB00945Acetylsalicylic acidSolute carrier family 22 member 7transporter
DB00945Acetylsalicylic acidCytochrome P450 2C19enzyme
DB00945Acetylsalicylic acidCytochrome P450 2C8enzyme
DB00945Acetylsalicylic acidCytochrome P450 2C9enzyme
DB00945Acetylsalicylic acid5'-AMP-activated protein kinasetarget
DB00945Acetylsalicylic acidEndothelin-1 receptortarget
DB00945Acetylsalicylic acidInhibitor of nuclear factor kappa-B kinase subunit betatarget
DB00945Acetylsalicylic acidCellular tumor antigen p53target
DB00945Acetylsalicylic acid78 kDa glucose-regulated proteintarget
DB00945Acetylsalicylic acidRibosomal protein S6 kinase alpha-3target
DB00945Acetylsalicylic acidNF-kappa-B inhibitor alphatarget
DB00945Acetylsalicylic acidNuclear factor NF-kappa-Btarget
DB06681BelataceptT-lymphocyte activation antigen CD86target
DB06681BelataceptT-lymphocyte activation antigen CD80target
DB00083Botulinum Toxin Type ASynaptosomal-associated protein 25target
DB00083Botulinum Toxin Type ARho-related GTP-binding protein RhoBtarget
DB01050IbuprofenProstaglandin G/H synthase 1target
DB01050IbuprofenProstaglandin G/H synthase 2target
DB01050IbuprofenCytochrome P450 2C9enzyme
DB01050IbuprofenSerum albumincarrier
DB01050IbuprofenMultidrug resistance-associated protein 4transporter
DB01050IbuprofenMultidrug resistance-associated protein 1transporter
DB01050IbuprofenSolute carrier organic anion transporter family member 1A2transporter
DB01050IbuprofenSolute carrier family 22 member 6transporter
DB01050IbuprofenSolute carrier family 22 member 8transporter
DB01050IbuprofenSolute carrier family 22 member 11transporter
DB01050IbuprofenSolute carrier organic anion transporter family member 2B1transporter
DB01050IbuprofenMultidrug resistance protein 1transporter
DB01050IbuprofenUDP-glucuronosyltransferase 1-1enzyme
DB01050IbuprofenUDP-glucuronosyltransferase 1-3enzyme
DB01050IbuprofenUDP-glucuronosyltransferase 1-9enzyme
DB01050IbuprofenUDP-glucuronosyltransferase 2B4enzyme
DB01050IbuprofenUDP-glucuronosyltransferase 2B7enzyme
DB01050IbuprofenCytochrome P450 2C8enzyme
DB01050IbuprofenCytochrome P450 2C19enzyme
DB01050IbuprofenProstaglandin G/H synthase 1enzyme
DB01050IbuprofenProstaglandin G/H synthase 2enzyme
DB01050IbuprofenApoptosis regulator Bcl-2target
DB01050IbuprofenThrombomodulintarget
DB01050IbuprofenTissue-type plasminogen activatortarget
DB01050IbuprofenFatty acid-binding protein, intestinaltarget
DB01050IbuprofenPeroxisome proliferator-activated receptor gammatarget
DB01050IbuprofenCystic fibrosis transmembrane conductance regulatortarget
DB01050IbuprofenSolute carrier family 15 member 1target
DB01050IbuprofenPeroxisome proliferator-activated receptor alphatarget
DB09054IdelalisibAldehyde oxidaseenzyme
DB09054IdelalisibCytochrome p450 3A subfamilyenzyme
DB09054IdelalisibUDP-glucuronosyltransferase 1A4enzyme
DB09054IdelalisibUDP-glucuronosyltransferase 1A1enzyme
DB09054IdelalisibCytochrome P450 2C8enzyme
DB09054IdelalisibCytochrome P450 2C19enzyme
DB09054IdelalisibCytochrome P450 2B6enzyme
DB09054IdelalisibCytochrome P450 3A4enzyme
DB09054IdelalisibPhosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit delta isoform (P110δ)target
DB09054IdelalisibATP-binding cassette sub-family G member 2transporter
DB09054IdelalisibMultidrug resistance protein 1transporter
DB09054IdelalisibSolute carrier organic anion transporter family member 1B1transporter
DB09054IdelalisibSolute carrier organic anion transporter family member 1B3transporter
DB00788NaproxenProstaglandin G/H synthase 1target
DB00788NaproxenProstaglandin G/H synthase 2target
DB00788NaproxenSerum albumincarrier
DB00788NaproxenCytochrome P450 2C9enzyme
DB00788NaproxenCytochrome P450 1A2enzyme
DB00788NaproxenSolute carrier organic anion transporter family member 1A2transporter
DB00788NaproxenSolute carrier family 22 member 6transporter
DB00788NaproxenCytochrome P450 2C8enzyme
DB00788NaproxenUDP-glucuronosyltransferase 1-1enzyme
DB00788NaproxenUDP-glucuronosyltransferase 2B7enzyme
DB00788NaproxenPeptostreptococcal albumin-binding proteintarget
DrugDrug NamePhaseStatusCount
DB01240Epoprostenol1Terminated1
DB00457Prazosin1 / 2Recruiting1
DB09153Sodium Chloride1 / 2Completed1
DB09145Water1 / 2Completed1
DB00297Bupivacaine2Completed1
DB09157Carbon dioxide2Completed1
DB00633Dexmedetomidine2Completed1
DB12158Filorexant2Completed1
DB00273Topiramate2Completed1
DB00653Magnesium Sulfate2 / 3Withdrawn1
DB01233Metoclopramide2 / 3Withdrawn1
DB00316Acetaminophen3Terminated1
DB00945Acetylsalicylic acid3Terminated1
DB00321Amitriptyline3Terminated1
DB00321Amitriptyline3Unknown Status1
DB00083Botulinum Toxin Type A3Completed1
DB00297Bupivacaine3Completed1
DB00201Caffeine3Unknown Status1
DB01234Dexamethasone3Recruiting1
DB01234Dexamethasone3Terminated1
DB01075Diphenhydramine3Recruiting1
DB01050Ibuprofen3Unknown Status1
DB01221Ketamine3Recruiting1
DB01221Ketamine3Terminated1
DB00465Ketorolac3Recruiting1
DB01233Metoclopramide3Recruiting1
DB00788Naproxen3Withdrawn2
DB00952Naratriptan3Withdrawn2
DB06614Peramivir3Completed1
DB06614Peramivir3Terminated1
DB00860Prednisolone3Completed1
DB00433Prochlorperazine3Terminated1
DB00571Propranolol3Completed1
DB00669Sumatriptan3Completed1
DB00273Topiramate3Completed4
DB00273Topiramate3Terminated1
DB00316Acetaminophen4Completed1
DB00945Acetylsalicylic acid4Completed1
DB00321Amitriptyline4Terminated1
DB00297Bupivacaine4Recruiting1
DB01234Dexamethasone4Recruiting1
DB01075Diphenhydramine4Completed1
DB01628Etoricoxib4Completed1
DB01628Etoricoxib4Unknown Status1
DB00813Fentanyl4Not Yet Recruiting1
DB00502Haloperidol4Active Not Recruiting1
DB01050Ibuprofen4Completed1
DB01221Ketamine4Completed1
DB00465Ketorolac4Completed1
DB01233Metoclopramide4Completed1
DB00904Ondansetron4Completed1
DB00230Pregabalin4Withdrawn1
DB00433Prochlorperazine4Completed1
DB00433Prochlorperazine4Recruiting1
DB00571Propranolol4Terminated1
DB00852Pseudoephedrine4Completed1
DB09153Sodium Chloride4Active Not Recruiting1
DB09153Sodium Chloride4Recruiting1
DB08816Ticagrelor4Recruiting1
DB00273Topiramate4Completed1
DB00273Topiramate4Terminated1
DB00620Triamcinolone4Recruiting1
DB00316AcetaminophenNot AvailableCompleted1
DB00819AcetazolamideNot AvailableCompleted1
DB00802AlfentanilNot AvailableRecruiting1
DB01238AripiprazoleNot AvailableRecruiting1
DB00181BaclofenNot AvailableEnrolling by Invitation1
DB00083Botulinum Toxin Type ANot AvailableActive Not Recruiting1
DB00083Botulinum Toxin Type ANot AvailableCompleted1
DB00297BupivacaineNot AvailableEnrolling by Invitation1
DB06774CapsaicinNot AvailableEnrolling by Invitation1
DB00411CarbacholNot AvailableCompleted2
DB00438CeftazidimeNot AvailableRecruiting1
DB00369CidofovirNot AvailableRecruiting1
DB00537CiprofloxacinNot AvailableRecruiting1
DB00363ClozapineNot AvailableRecruiting1
DB00318CodeineNot AvailableCompleted1
DB00924CyclobenzaprineNot AvailableEnrolling by Invitation1
DB01234DexamethasoneNot AvailableRecruiting1
DB00829DiazepamNot AvailableRecruiting1
DB00586DiclofenacNot AvailableEnrolling by Invitation1
DB12789DinoprostNot AvailableCompleted1
DB00917DinoprostoneNot AvailableCompleted1
DB01075DiphenhydramineNot AvailableCompleted1
DB00668EpinephrineNot AvailableEnrolling by Invitation1
DB01240EpoprostenolNot AvailableUnknown Status1
DB00712FlurbiprofenNot AvailableEnrolling by Invitation1
DB01320FosphenytoinNot AvailableRecruiting1
DB00996GabapentinNot AvailableEnrolling by Invitation1
DB00502HaloperidolNot AvailableRecruiting1
DB01109HeparinNot AvailableRecruiting1
DB00327HydromorphoneNot AvailableRecruiting1
DB01050IbuprofenNot AvailableCompleted1
DB01221KetamineNot AvailableCompleted1
DB01221KetamineNot AvailableEnrolling by Invitation1
DB01202LevetiracetamNot AvailableRecruiting1
DB00281LidocaineNot AvailableEnrolling by Invitation1
DB08815LurasidoneNot AvailableRecruiting1
DB09337Medical airNot AvailableCompleted1
DB00814MeloxicamNot AvailableEnrolling by Invitation1
DB00825MentholNot AvailableCompleted1
DB00825MentholNot AvailableEnrolling by Invitation1
DB00760MeropenemNot AvailableRecruiting1
DB00959MethylprednisoloneNot AvailableRecruiting1
DB01233MetoclopramideNot AvailableCompleted1
DB00683MidazolamNot AvailableRecruiting1
DB01618MolindoneNot AvailableRecruiting1
DB00295MorphineNot AvailableRecruiting1
DB00622NicardipineNot AvailableRecruiting1
DB00334OlanzapineNot AvailableRecruiting2
DB00198OseltamivirNot AvailableRecruiting1
DB09140OxygenNot AvailableCompleted1
DB00652PentazocineNot AvailableCompleted1
DB00312PentobarbitalNot AvailableRecruiting1
DB00750PrilocaineNot AvailableEnrolling by Invitation1
DB00818PropofolNot AvailableRecruiting1
DB01224QuetiapineNot AvailableRecruiting1
DB00734RisperidoneNot AvailableRecruiting1
DB00533RofecoxibNot AvailableCompleted1
DB00296RopivacaineNot AvailableCompleted1
DB00669SumatriptanNot AvailableEnrolling by Invitation1
DB00373TimololNot AvailableRecruiting1
DB00697TizanidineNot AvailableEnrolling by Invitation1
DB00684TobramycinNot AvailableRecruiting1
DB00273TopiramateNot AvailableEnrolling by Invitation1
DB00273TopiramateNot AvailableRecruiting1
DB00273TopiramateNot AvailableWithdrawn1
DB00313Valproic AcidNot AvailableRecruiting1
DB00682WarfarinNot AvailableRecruiting1
DB01593ZincNot AvailableCompleted1
DB00246ZiprasidoneNot AvailableRecruiting1