Opioid Dependence

Also known as: Opioid type dependence / Opioid dependent / Opioid Dependency / Dependence, Opioid / Opioid-Related Disorders / Opioid type dependence, unspecified use / Opiate Dependence / Opioid dependence (disorder) / Dependence on opiates / Opioid related disorders / Drug Dependence / Unspecified drug dependence / Drug dependence, unspecified / Addiction to drugs / Dependent drug abuse (disorder) / Drug addiction / Dependence drug (NOS) / Drug dependence NOS / Psychoactive substance dependence (disorder)

DrugDrug NameDrug Description
DB00921BuprenorphineA partial opioid agonist used for management of severe pain that is not responsive to alternative treatments. Also used for maintenance treatment of opioid addiction.
DB04465LactoseAn additive and filler found in various products to maintain structure and consistency.
DB01183NaloxoneAn opioid receptor antagonist used to rapidly reverse an opioid overdose. Also included in some drug formulations as an abuse deterrent to prevent injection.
DB00704NaltrexoneA narcotic antagonist used in opioid overdose.
DrugDrug NameTargetType
DB00921BuprenorphineKappa-type opioid receptortarget
DB00921BuprenorphineMu-type opioid receptortarget
DB00921BuprenorphineCytochrome P450 3A4enzyme
DB00921BuprenorphineCytochrome P450 2D6enzyme
DB00921BuprenorphineP-glycoprotein 1transporter
DB00921BuprenorphineATP-binding cassette sub-family G member 2transporter
DB00921BuprenorphineCytochrome P450 2C9enzyme
DB00921BuprenorphineCytochrome P450 3A5enzyme
DB00921BuprenorphineCytochrome P450 2C8enzyme
DB00921BuprenorphineCytochrome P450 3A7enzyme
DB00921BuprenorphineDelta-type opioid receptortarget
DB00921BuprenorphineCytochrome P450 2C18enzyme
DB00921BuprenorphineCytochrome P450 2C19enzyme
DB00921BuprenorphineNociceptin receptortarget
DB04465LactoseBeta-galactosidasetarget
DB04465LactoseGlycosyltransferase 6 domain-containing protein 1target
DB04465LactoseGlycolipid transfer proteintarget
DB04465LactoseHydrolasetarget
DB04465LactoseEndo-1,4-beta-xylanase Atarget
DB04465LactoseGalectin-3target
DB04465LactoseSialidasetarget
DB04465LactoseBeta-galactosidasetarget
DB01183NaloxoneMu-type opioid receptortarget
DB01183NaloxoneEstrogen receptor alphatarget
DB01183NaloxoneCyclic AMP-responsive element-binding protein 1target
DB01183NaloxoneDelta-type opioid receptortarget
DB01183NaloxoneSolute carrier organic anion transporter family member 1A2transporter
DB01183NaloxoneP-glycoprotein 1transporter
DB01183NaloxoneKappa-type opioid receptortarget
DB01183NaloxoneCytochrome P450 3A4enzyme
DB01183NaloxoneSerum albumincarrier
DB01183NaloxoneToll-like receptor 4target
DB01183NaloxoneLiver carboxylesterase 1target
DB01183NaloxoneUDP-glucuronosyltransferase 1-1enzyme
DB01183NaloxoneCytochrome P450 2C18enzyme
DB01183NaloxoneCytochrome P450 2C19enzyme
DB00704NaltrexoneMu-type opioid receptortarget
DB00704NaltrexoneKappa-type opioid receptortarget
DB00704NaltrexoneDelta-type opioid receptortarget
DB00704NaltrexoneUDP-glucuronosyltransferase 1-1enzyme
DB00704NaltrexoneSigma non-opioid intracellular receptor 1target
DrugDrug NamePhaseStatusCount
DB00704Naltrexone0Completed1
DB00497Oxycodone0Terminated1
DB00107Oxytocin0Completed1
DB00734Risperidone0Terminated1
DB09034Suvorexant0Recruiting1
DB00246Ziprasidone0Terminated1
DB00673Aprepitant1Completed1
DB00921Buprenorphine1Completed4
DB00260Cycloserine1Completed1
DB01264Darunavir1Completed1
DB00343Diltiazem1Completed1
DB01319Fosamprenavir1Completed1
DB00996Gabapentin1Completed1
DB00327Hydromorphone1Completed1
DB00270Isradipine1Completed1
DB16956L-Acetylleucine1Completed1
DB06218Lacosamide1Recruiting1
DB04948Lofexidine1Completed3
DB04871Lorcaserin1Completed1
DB00333Methadone1Completed3
DB01183Naloxone1Completed3
DB00704Naltrexone1Completed2
DB00704Naltrexone1Not Yet Recruiting1
DB01115Nifedipine1Completed1
DB00615Rifabutin1Completed1
DB01045Rifampicin1Completed1
DB00503Ritonavir1Completed1
DB01273Varenicline1Completed1
DB00661Verapamil1Completed1
DB00921Buprenorphine1 / 2Completed2
DB00575Clonidine1 / 2Completed1
DB00270Isradipine1 / 2Completed1
DB14158Microcrystalline cellulose1 / 2Completed1
DB00295Morphine1 / 2Completed1
DB01183Naloxone1 / 2Completed1
DB00704Naltrexone1 / 2Completed1
DB00107Oxytocin1 / 2Completed1
DB00193Tramadol1 / 2Completed1
DB00316Acetaminophen2Recruiting1
DB00921Buprenorphine2Active Not Recruiting1
DB00921Buprenorphine2Completed5
DB00921Buprenorphine2Not Yet Recruiting1
DB00190Carbidopa2Recruiting1
DB00907Cocaine2Completed1
DB00318Codeine2Recruiting1
DB00822Disulfiram2Completed2
DB00996Gabapentin2Completed2
DB00956Hydrocodone2Recruiting1
DB00741Hydrocortisone2Completed1
DB05266Ibudilast2Completed1
DB01221Ketamine2Terminated1
DB01202Levetiracetam2Completed2
DB01235Levodopa2Recruiting1
DB00742Mannitol2Completed1
DB01043Memantine2Completed1
DB04817Metamizole2Recruiting1
DB00333Methadone2Completed2
DB00295Morphine2Recruiting1
DB01183Naloxone2Completed2
DB00704Naltrexone2Completed3
DB00704Naltrexone2Not Yet Recruiting1
DB00788Naproxen2Recruiting1
DB00497Oxycodone2Recruiting1
DB01192Oxymorphone2Recruiting1
DB00860Prednisolone2Terminated1
DB11664Psilocybin2Not Yet Recruiting1
DB09034Suvorexant2Completed1
DB00193Tramadol2Recruiting1
DB00297Bupivacaine2 / 3Unknown Status1
DB00921Buprenorphine2 / 3Completed3
DB00470Dronabinol2 / 3Completed1
DB00668Epinephrine2 / 3Unknown Status1
DB04948Lofexidine2 / 3Recruiting1
DB01043Memantine2 / 3Completed2
DB00333Methadone2 / 3Completed1
DB01183Naloxone2 / 3Completed2
DB00704Naltrexone2 / 3Completed2
DB00704Naltrexone2 / 3Terminated1
DB00921Buprenorphine3Completed10
DB00921Buprenorphine3Terminated2
DB00921Buprenorphine3Unknown Status1
DB00921Buprenorphine3Withdrawn2
DB01156Bupropion3Completed1
DB01452Diamorphine3Completed2
DB00327Hydromorphone3Completed1
DB04948Lofexidine3Completed1
DB00333Methadone3Completed4
DB00295Morphine3Completed1
DB01183Naloxone3Completed5
DB01183Naloxone3Withdrawn2
DB00704Naltrexone3Completed1
DB11130Opium3Completed1
DB00936Salicylic acid3Completed1
DB00936Salicylic acid3Unknown Status1
DB11799Bictegravir4Unknown Status1
DB00297Bupivacaine4Completed1
DB00921Buprenorphine4Completed5
DB00921Buprenorphine4Enrolling by Invitation1
DB00921Buprenorphine4Not Yet Recruiting1
DB00921Buprenorphine4Recruiting1
DB09065Cobicistat4Unknown Status1
DB06700Desvenlafaxine4Completed1
DB09101Elvitegravir4Unknown Status1
DB00879Emtricitabine4Unknown Status1
DB00996Gabapentin4Completed1
DB00281Lidocaine4Terminated1
DB01183Naloxone4Completed4
DB01183Naloxone4Enrolling by Invitation1
DB01183Naloxone4Recruiting1
DB00704Naltrexone4Completed2
DB08934Sofosbuvir4Unknown Status1
DB09299Tenofovir alafenamide4Unknown Status1
DB11613Velpatasvir4Unknown Status1
DB00921BuprenorphineNot AvailableActive Not Recruiting1
DB00921BuprenorphineNot AvailableNot Yet Recruiting1
DB00813FentanylNot AvailableUnknown Status1
DB00951IsoniazidNot AvailableActive Not Recruiting1
DB00333MethadoneNot AvailableActive Not Recruiting1
DB01017MinocyclineNot AvailableCompleted1
DB01183NaloxoneNot AvailableActive Not Recruiting1
DB00704NaltrexoneNot AvailableCompleted1
DB00497OxycodoneNot AvailableActive Not Recruiting1
DB00935OxymetazolineNot AvailableActive Not Recruiting1
DB01201RifapentineNot AvailableActive Not Recruiting1
DB00759TetracyclineNot AvailableCompleted1