Treatment-resistant Schizophrenia

Also known as: Schizophrenia, Treatment-Resistant / Treatment Resistant Schizophrenia / Schizophrenia, unspecified / Schizophrenia NOS / Dementia praecox / Schizophrenic disorders (disorder) / Unspecified schizophrenia / Unspecified schizophrenia, unspecified state / Schizophrenia / Schizophrenia (disorder)

DrugDrug NameDrug Description
DB00363ClozapineAn atypical or second-generation antipsychotic drug used in treatment-resistant schizophrenia and to decrease suicide risk in schizophrenic patients.
DrugDrug NameTargetType
DB00363ClozapineDopamine D4 receptortarget
DB00363ClozapineHistamine H1 receptortarget
DB00363ClozapineDopamine D2 receptortarget
DB00363ClozapineNeuron-specific vesicular protein calcyontarget
DB00363ClozapineHistamine H4 receptortarget
DB00363Clozapine5-hydroxytryptamine receptor 2Atarget
DB00363Clozapine5-hydroxytryptamine receptor 1Atarget
DB00363Clozapine5-hydroxytryptamine receptor 2Ctarget
DB00363ClozapineDopamine D1 receptortarget
DB00363ClozapineCytochrome P450 1A2enzyme
DB00363ClozapineCytochrome P450 2D6enzyme
DB00363ClozapineDopamine D3 receptortarget
DB00363ClozapineMuscarinic acetylcholine receptor M1target
DB00363ClozapineMuscarinic acetylcholine receptor M2target
DB00363ClozapineMuscarinic acetylcholine receptor M3target
DB00363ClozapineMuscarinic acetylcholine receptor M4target
DB00363ClozapineMuscarinic acetylcholine receptor M5target
DB00363Clozapine5-hydroxytryptamine receptor 1Btarget
DB00363Clozapine5-hydroxytryptamine receptor 1Dtarget
DB00363Clozapine5-hydroxytryptamine receptor 1Etarget
DB00363Clozapine5-hydroxytryptamine receptor 3Atarget
DB00363Clozapine5-hydroxytryptamine receptor 6target
DB00363Clozapine5-hydroxytryptamine receptor 7target
DB00363ClozapineAlpha-1A adrenergic receptortarget
DB00363ClozapineAlpha-1B adrenergic receptortarget
DB00363ClozapineAlpha-2A adrenergic receptortarget
DB00363ClozapineAlpha-2B adrenergic receptortarget
DB00363ClozapineAlpha-2C adrenergic receptortarget
DB00363ClozapineCytochrome P450 2C9enzyme
DB00363ClozapineP-glycoprotein 1transporter
DB00363ClozapineCytochrome P450 3A4enzyme
DB00363ClozapineCytochrome P450 2C19enzyme
DB00363ClozapineDimethylaniline monooxygenase [N-oxide-forming] 3enzyme
DB00363ClozapineUDP-glucuronosyltransferase 1-4enzyme
DB00363ClozapineCytochrome P450 1A1enzyme
DB00363ClozapineCytochrome P450 2A6enzyme
DB00363ClozapineCytochrome P450 2C8enzyme
DB00363ClozapineGlutathione S-transferase Ptarget
DB00363ClozapineAlpha-1-acid glycoprotein 1carrier
DB00363ClozapineSerum albumincarrier
DB00363ClozapineDopamine D5 receptortarget
DB00363ClozapineGamma-aminobutyric acid type B receptor subunit 1target
DB00363ClozapineGamma-aminobutyric acid type B receptor subunit 2target
DB00363ClozapineSolute carrier family 22 member 1transporter
DB00363ClozapineSolute carrier family 22 member 2transporter
DB00363ClozapineSolute carrier family 22 member 3transporter
DB00363ClozapineGamma-aminobutyric acid receptor subunit alpha-1target
DB00363ClozapineGamma-aminobutyric acid receptor subunit beta-1target
DB00363ClozapineGamma-aminobutyric acid receptor subunit gamma-1target
DrugDrug NamePhaseStatusCount
DB00740Riluzole0Recruiting1
DB00073Rituximab1Completed1
DB00966Telmisartan2Terminated1
DB06288Amisulpride3Unknown Status1
DB00363Clozapine3Unknown Status1
DB00334Olanzapine3Terminated1
DB00734Risperidone3Terminated1
DB06288Amisulpride4Completed1
DB01238Aripiprazole4Not Yet Recruiting1
DB01238Aripiprazole4Recruiting1
DB06016Cariprazine4Recruiting1
DB00363Clozapine4Completed1
DB00363Clozapine4Recruiting1
DB00514Dextromethorphan4Recruiting1
DB08815Lurasidone4Recruiting1
DB00334Olanzapine4Recruiting1
DB01267Paliperidone4Not Yet Recruiting1
DB01267Paliperidone4Recruiting1
DB01224Quetiapine4Recruiting1
DB00734Risperidone4Recruiting1
DB00246Ziprasidone4Recruiting1
DB00802AlfentanilNot AvailableCompleted1
DB00479AmikacinNot AvailableCompleted1
DB00513Aminocaproic acidNot AvailableCompleted1
DB06288AmisulprideNot AvailableNot Yet Recruiting1
DB01238AripiprazoleNot AvailableNot Yet Recruiting1
DB00559BosentanNot AvailableCompleted1
DB01413CefepimeNot AvailableCompleted1
DB00369CidofovirNot AvailableCompleted1
DB00537CiprofloxacinNot AvailableCompleted1
DB00363ClozapineNot AvailableCompleted1
DB00828FosfomycinNot AvailableCompleted1
DB00502HaloperidolNot AvailableCompleted1
DB00598LabetalolNot AvailableCompleted1
DB08815LurasidoneNot AvailableCompleted1
DB00959MethylprednisoloneNot AvailableCompleted1
DB01618MolindoneNot AvailableCompleted1
DB00607NafcillinNot AvailableCompleted1
DB01115NifedipineNot AvailableCompleted1
DB00334OlanzapineNot AvailableNot Yet Recruiting1
DB00497OxycodoneNot AvailableCompleted1
DB00312PentobarbitalNot AvailableCompleted1
DB00319PiperacillinNot AvailableCompleted1
DB00734RisperidoneNot AvailableNot Yet Recruiting1
DB00728RocuroniumNot AvailableCompleted1
DB00658SevelamerNot AvailableCompleted1
DB00421SpironolactoneNot AvailableCompleted1
DB01606TazobactamNot AvailableCompleted1
DB00684TobramycinNot AvailableCompleted1
DB00302Tranexamic acidNot AvailableCompleted1
DB00512VancomycinNot AvailableCompleted1
DB01339VecuroniumNot AvailableCompleted1
DB00682WarfarinNot AvailableCompleted1
DB00246ZiprasidoneNot AvailableCompleted1
DB00425ZolpidemNot AvailableCompleted1