Moderate, severe, Vasomotor Symptoms caused by Menopause

Also known as: Moderate, severe Vasomotor Symptoms caused by Menopause

DrugDrug NameDrug Description
DB00977EthinylestradiolAn estradiol used as a contraceptive.
DB00717NorethisteroneA synthetic second-generation progestin used for contraception, prevention of endometrial hyperplasia in hormone replacement therapy, and in the treatment of other hormone-mediated illnesses such as endometriosis.
DrugDrug NameTargetType
DB00977EthinylestradiolEstrogen receptor alphatarget
DB00977EthinylestradiolNuclear receptor subfamily 1 group I member 2target
DB00977EthinylestradiolCytochrome P450 3A4enzyme
DB00977EthinylestradiolCytochrome P450 2C8enzyme
DB00977EthinylestradiolBile salt export pumptransporter
DB00977EthinylestradiolSodium/bile acid cotransportertransporter
DB00977EthinylestradiolCanalicular multispecific organic anion transporter 1transporter
DB00977EthinylestradiolP-glycoprotein 1transporter
DB00977EthinylestradiolUDP-glucuronosyltransferase 1-1enzyme
DB00977EthinylestradiolCytochrome P450 2C19enzyme
DB00977EthinylestradiolUDP-glucuronosyltransferase 1-4enzyme
DB00977EthinylestradiolUDP-glucuronosyltransferase 1-9enzyme
DB00977EthinylestradiolCytochrome P450 2C9enzyme
DB00977EthinylestradiolCytochrome P450 1A2enzyme
DB00977EthinylestradiolEstrogen sulfotransferaseenzyme
DB00977EthinylestradiolSulfotransferase 1A3/1A4enzyme
DB00977EthinylestradiolCytochrome P450 3A5enzyme
DB00977EthinylestradiolUDP-glucuronosyltransferase 2B7enzyme
DB00977EthinylestradiolUDP-glucuronosyltransferase 1-3enzyme
DB00977EthinylestradiolCatechol O-methyltransferaseenzyme
DB00977EthinylestradiolSolute carrier organic anion transporter family member 1A2transporter
DB00977EthinylestradiolSerum albumincarrier
DB00977EthinylestradiolSex hormone-binding globulincarrier
DB00717NorethisteroneProgesterone receptortarget
DB00717NorethisteroneP-glycoprotein 1transporter
DB00717NorethisteroneCytochrome P450 2C19enzyme
DB00717NorethisteroneSerum albumincarrier
DB00717NorethisteroneSex hormone-binding globulincarrier
DB00717NorethisteroneAldo-keto reductase family 1 member C4enzyme
DB00717Norethisterone3 beta-hydroxysteroid dehydrogenase/Delta 5-->4-isomerase type 2enzyme
DB00717Norethisterone3-oxo-5-alpha-steroid 4-dehydrogenaseenzyme
DB00717Norethisterone3-oxo-5-beta-steroid 4-dehydrogenaseenzyme
DB00717NorethisteroneCytochrome P450 3A4enzyme
DB00717NorethisteroneCytochrome P450 1A2enzyme
DB00717NorethisteroneCytochrome P450 2A6enzyme
DB00717NorethisteroneGlucocorticoid receptortarget
DB00717NorethisteroneAndrogen receptortarget
DrugDrug NamePhaseStatusCount