cAMP-dependent protein kinase regulatory subunit

Details

Name
cAMP-dependent protein kinase regulatory subunit
Synonyms
  • cAMP-dependent protein kinase regulatory subunit, putative
Gene Name
PKAr
Organism
Plasmodium falciparum (isolate 3D7)
Amino acid sequence
>lcl|BSEQ0051530|cAMP-dependent protein kinase regulatory subunit
MGNVCTWRQGKEKAGDDNSQVIKDKELQNEFKTFEQKMRSNKKNAHEGDMNNDGEDDRYK
FSRGFSLSKKPSKTKIPITKTDSEILDGLDYSEMSKQVLMTLNKKNILNDDGSSDGNDTD
VHSMFDRKEIERKVLDLESIHFIQKKRLSVSAEAYGDWNKKIDNFIPKVYKKDEKEKAKI
REALNESFLFNHLNKKEFEIIVNAFFDKNVEKGVNIINEGDYGDLLYVIDQGEVEIYKTK
ENNKKEVLTVLKSKDVFGELALLYNSKRAATATALTKCHLWALDRESFTYIIKDMVAKKR
KMYEDILSHVNILKDMDPYERCKVADCLKSKSYNDGEIIIKEGEEGDTFFILIDGNAVAS
KDNKVIKTYTKGDYFGELALLKNKPRAATIKAQNFCQVVYLDRKSFKRLLGPIEDILHRN
VENYKKVLNELGLDTTCIDEN
Number of residues
441
Molecular Weight
50832.44
Theoretical pI
Not Available
GO Classification
Functions
cAMP binding / cAMP-dependent protein kinase activity / cAMP-dependent protein kinase regulator activity
Components
cAMP-dependent protein kinase complex
General Function
Not Available
Specific Function
Camp binding
Pfam Domain Function
Transmembrane Regions
Not Available
Cellular Location
Not Available
Gene sequence
>lcl|BSEQ0051531|cAMP-dependent protein kinase regulatory subunit (PKAr)
ATGGGCAATGTGTGCACATGGAGACAAGGGAAAGAAAAAGCAGGTGACGATAATTCACAA
GTAATAAAAGATAAAGAATTACAAAACGAGTTTAAAACATTCGAACAAAAAATGAGAAGT
AATAAAAAAAATGCTCATGAAGGAGATATGAATAATGATGGTGAAGATGATAGATATAAA
TTTTCCAGAGGTTTTTCATTAAGTAAAAAACCAAGTAAAACTAAAATACCGATTACCAAA
ACGGATAGTGAAATATTAGATGGATTGGATTATTCTGAAATGAGTAAACAAGTTCTTATG
ACTTTAAATAAAAAAAATATACTTAATGACGACGGTTCAAGCGACGGTAACGACACAGAT
GTTCACAGCATGTTCGATAGGAAAGAAATAGAGAGAAAGGTATTGGATTTAGAAAGTATA
CATTTCATACAGAAGAAAAGATTATCTGTGAGTGCCGAAGCATATGGTGACTGGAATAAA
AAGATTGATAATTTTATTCCTAAAGTTTATAAGAAAGATGAAAAAGAAAAGGCCAAGATA
AGAGAAGCATTGAATGAATCCTTTTTGTTTAATCATTTAAATAAGAAAGAATTTGAAATT
ATTGTAAATGCATTTTTTGATAAAAATGTAGAAAAAGGGGTTAATATTATAAATGAAGGA
GATTATGGAGATTTATTATATGTTATAGATCAAGGTGAAGTTGAAATATATAAAACAAAA
GAAAATAATAAAAAAGAAGTATTAACAGTATTAAAATCTAAAGATGTTTTTGGAGAATTA
GCCTTATTATATAATTCTAAAAGAGCTGCAACAGCTACAGCCTTAACCAAATGCCATTTA
TGGGCCTTAGATAGAGAATCTTTTACATATATAATAAAAGATATGGTTGCTAAGAAAAGA
AAAATGTATGAAGATATTCTTAGTCATGTAAATATTTTAAAAGACATGGATCCATATGAA
AGATGTAAAGTTGCTGATTGCTTAAAATCTAAAAGTTATAATGATGGAGAAATTATTATT
AAAGAAGGAGAAGAAGGAGATACATTTTTTATCCTTATAGATGGAAATGCTGTAGCTTCT
AAAGATAATAAAGTCATCAAAACTTATACAAAGGGAGATTACTTTGGAGAATTAGCTCTT
CTCAAAAATAAACCAAGAGCTGCTACCATAAAAGCACAAAATTTTTGTCAAGTCGTCTAT
TTAGATAGAAAAAGTTTCAAAAGATTATTAGGACCTATTGAGGATATATTACATAGAAAT
GTTGAAAATTACAAAAAAGTTCTGAACGAATTAGGTTTGGATACAACTTGTATTGATGAA
AATTAA
Chromosome Location
Not Available
Locus
Not Available
External Identifiers
ResourceLink
UniProtKB IDQ7KQK0
UniProtKB Entry NameQ7KQK0_PLAF7
General References
  1. Gardner MJ, Hall N, Fung E, White O, Berriman M, Hyman RW, Carlton JM, Pain A, Nelson KE, Bowman S, Paulsen IT, James K, Eisen JA, Rutherford K, Salzberg SL, Craig A, Kyes S, Chan MS, Nene V, Shallom SJ, Suh B, Peterson J, Angiuoli S, Pertea M, Allen J, Selengut J, Haft D, Mather MW, Vaidya AB, Martin DM, Fairlamb AH, Fraunholz MJ, Roos DS, Ralph SA, McFadden GI, Cummings LM, Subramanian GM, Mungall C, Venter JC, Carucci DJ, Hoffman SL, Newbold C, Davis RW, Fraser CM, Barrell B: Genome sequence of the human malaria parasite Plasmodium falciparum. Nature. 2002 Oct 3;419(6906):498-511. [Article]
  2. Littler DR, Bullen HE, Harvey KL, Beddoe T, Crabb BS, Rossjohn J, Gilson PR: Disrupting the Allosteric Interaction between the Plasmodium falciparum cAMP-dependent Kinase and Its Regulatory Subunit. J Biol Chem. 2016 Dec 2;291(49):25375-25386. doi: 10.1074/jbc.M116.750174. Epub 2016 Oct 13. [Article]

Drug Relations

Drug Relations
DrugBank IDNameDrug groupPharmacological action?ActionsDetails
DB11638Artenimolapproved, experimental, investigationalunknownligandDetails