Reaction: Baclofen to 1 product

Reaction
Reaction type
deamination
Direction
Major circulating metabolite?
Yes
Spontaneous?
No
Activity
inactive
References
  1. Sanchez-Ponce R, Wang LQ, Lu W, von Hehn J, Cherubini M, Rush R: Metabolic and Pharmacokinetic Differentiation of STX209 and Racemic Baclofen in Humans. Metabolites. 2012 Sep 11;2(3):596-613. doi: 10.3390/metabo2030596. [Article]
  2. EMC Summary of Product Characteristics: Baclofen Oral Tablets [Link]
Comments
Not Available
Enzymes
Not Available