Reaction: Cyclosporine to 3 products

Reaction
Reaction type
oxidation
Direction
Major circulating metabolite?
No
Spontaneous?
No
Activity
active
References
  1. Barbarino JM, Staatz CE, Venkataramanan R, Klein TE, Altman RB: PharmGKB summary: cyclosporine and tacrolimus pathways. Pharmacogenet Genomics. 2013 Oct;23(10):563-85. doi: 10.1097/FPC.0b013e328364db84. [Article]
  2. Neoral (Cyclosporine) FDA Label [Link]
Comments
Not Available
Enzymes
EnzymeKmVmaxRole
Cytochrome P450 3A4Not AvailableNot Availableconfirmed
Cytochrome P450 3A5Not AvailableNot Availableconfirmed