Reaction: Entrectinib to 1 product

Reaction
Reaction type
reduction
Direction
Major circulating metabolite?
No
Spontaneous?
No
Activity
unknown
References
  1. Attwa MW, Kadi AA, Alrabiah H, Darwish HW: LC-MS/MS reveals the formation of iminium and quinone methide reactive intermediates in entrectinib metabolism: In vivo and in vitro metabolic investigation. J Pharm Biomed Anal. 2018 Oct 25;160:19-30. doi: 10.1016/j.jpba.2018.07.032. Epub 2018 Jul 22. [Article]
Comments
Not Available
Enzymes
Not Available