Displaying drugs 1 - 25 of 398 in total
Leuprolide
Leuprolide is a synthetic 9-residue peptide analogue of gonadotropin-releasing hormone (GnRH). Unlike the endogenous decapeptide GnRH, leuprolide contains a single D-amino acid (D-leucyl) residue, which helps to increase its circulating half-life from three to four minutes to approximately three hours. As a GnRH mimic, leuprolide is capable of binding to...
Approved
Investigational
Matched Name: … Leuprolide …
Matched Description: … Leuprolide is a synthetic 9-residue peptide analogue of gonadotropin-releasing hormone (GnRH). ... Unlike the endogenous decapeptide GnRH, leuprolide contains a single D-amino acid (D-leucyl) residue, ... [A203222] As a GnRH mimic, leuprolide is capable of binding to the GnRH receptor (GnRHR) and inducing …
Matched Mixtures name: … Leuprolide Acetate ... Leuprolide Acetate ... Leuprolide Acetate …
Matched Salts name: … Leuprolide acetate ... Leuprolide mesylate …
Matched Products: … Leuprolide Acetate ... Leuprolide Acetate Depot ... Leuprolide Acetate Injection …
Matched Description: … Leuprolide is a synthetic 9-residue peptide analogue of gonadotropin-releasing hormone (GnRH). ... Unlike the endogenous decapeptide GnRH, leuprolide contains a single D-amino acid (D-leucyl) residue, ... [A203222] As a GnRH mimic, leuprolide is capable of binding to the GnRH receptor (GnRHR) and inducing …
Matched Mixtures name: … Leuprolide Acetate ... Leuprolide Acetate ... Leuprolide Acetate …
Matched Salts name: … Leuprolide acetate ... Leuprolide mesylate …
Matched Products: … Leuprolide Acetate ... Leuprolide Acetate Depot ... Leuprolide Acetate Injection …
Aluminum acetate
Approved
Investigational
Matched Synonyms: … Aluminum acetate …
Matched Name: … Aluminum acetate …
Matched Products: … Humco Aluminum Acetate Burrow …
Matched Name: … Aluminum acetate …
Matched Products: … Humco Aluminum Acetate Burrow …
Oxyphenisatin acetate
Oxyphenisatin acetate is the pro-drug of oxyphenisatin (3,3-bis(4-hydroxyphenyl)-1H-indol-2-one). The FDA withdrew its approval for the use of oxyphenisatin acetate due to safety reasons.
Approved
Investigational
Withdrawn
Matched Synonyms: … Oxyphenisatin acetate ... Oxyphenisatine acetate …
Matched Name: … Oxyphenisatin acetate …
Matched Iupac: … 4-{3-[4-(acetyloxy)phenyl]-2-oxo-2,3-dihydro-1H-indol-3-yl}phenyl acetate …
Matched Description: … Oxyphenisatin acetate is the pro-drug of [oxyphenisatin] (3,3-bis(4-hydroxyphenyl)-1H-indol-2-one). ... The FDA withdrew its approval for the use of oxyphenisatin acetate due to safety reasons.[L43942] …
Matched Name: … Oxyphenisatin acetate …
Matched Iupac: … 4-{3-[4-(acetyloxy)phenyl]-2-oxo-2,3-dihydro-1H-indol-3-yl}phenyl acetate …
Matched Description: … Oxyphenisatin acetate is the pro-drug of [oxyphenisatin] (3,3-bis(4-hydroxyphenyl)-1H-indol-2-one). ... The FDA withdrew its approval for the use of oxyphenisatin acetate due to safety reasons.[L43942] …
Cyproterone acetate
An anti-androgen that, in the form of its acetate (cyproterone acetate), also has progestational properties. It is used in the treatment of hypersexuality in males, as a palliative in prostatic carcinoma, and, in combination with estrogen, for the therapy of severe acne and hirsutism in females.
Approved
Investigational
Matched Synonyms: … Cyproterone acetate ... Cyproterone 17-O-acetate …
Matched Name: … Cyproterone acetate …
Matched Iupac: … acetyl-9-chloro-2,16-dimethyl-6-oxopentacyclo[9.7.0.0^{2,8}.0^{3,5}.0^{12,16}]octadeca-7,9-dien-15-yl acetate …
Matched Description: … An anti-androgen that, in the form of its acetate (cyproterone acetate), also has progestational properties …
Matched Name: … Cyproterone acetate …
Matched Iupac: … acetyl-9-chloro-2,16-dimethyl-6-oxopentacyclo[9.7.0.0^{2,8}.0^{3,5}.0^{12,16}]octadeca-7,9-dien-15-yl acetate …
Matched Description: … An anti-androgen that, in the form of its acetate (cyproterone acetate), also has progestational properties …
Zinc acetate
Approved
Investigational
Matched Synonyms: … Zinc(II) acetate ... Zinc acetate anhydrous …
Matched Name: … Zinc acetate …
Matched Mixtures name: … Diphenhydramine HCl, Zinc Acetate ... Diphenhydramine HCI and Zinc Acetate ... Diphenhydramine HCl and Zinc Acetate …
Matched Salts name: … Zinc acetate dihydrate …
Matched Categories: … zinc acetate …
Matched Name: … Zinc acetate …
Matched Mixtures name: … Diphenhydramine HCl, Zinc Acetate ... Diphenhydramine HCI and Zinc Acetate ... Diphenhydramine HCl and Zinc Acetate …
Matched Salts name: … Zinc acetate dihydrate …
Matched Categories: … zinc acetate …
Megestrol acetate
17-Hydroxy-6-methylpregna-3,6-diene-3,20-dione. A progestational hormone used most commonly as the acetate ester. As the acetate, it is more potent than progesterone both as a progestagen and as an ovulation inhibitor. It has also been used in the palliative treatment of breast cancer.
Approved
Investigational
Vet approved
Matched Synonyms: … Megestrol acetate ... 17-Hydroxy-6-methylpregna-4,6-diene-3,20-dione 17-acetate ... 17α-Hydroxy-6-methylpregna-4,6-diene-3,20-dione acetate …
Matched Name: … Megestrol acetate …
Matched Iupac: … ,11S,14R,15S)-14-acetyl-2,8,15-trimethyl-5-oxotetracyclo[8.7.0.0²,⁷.0¹¹,¹⁵]heptadeca-6,8-dien-14-yl acetate …
Matched Description: … A progestational hormone used most commonly as the acetate ester. ... As the acetate, it is more potent than progesterone both as a progestagen and as an ovulation inhibitor …
Matched Products: … Megestrol Acetate ... Megestrol acetate ... MEGESTROL ACETATE …
Matched Name: … Megestrol acetate …
Matched Iupac: … ,11S,14R,15S)-14-acetyl-2,8,15-trimethyl-5-oxotetracyclo[8.7.0.0²,⁷.0¹¹,¹⁵]heptadeca-6,8-dien-14-yl acetate …
Matched Description: … A progestational hormone used most commonly as the acetate ester. ... As the acetate, it is more potent than progesterone both as a progestagen and as an ovulation inhibitor …
Matched Products: … Megestrol Acetate ... Megestrol acetate ... MEGESTROL ACETATE …
Magnesium acetate
Approved
Matched Synonyms: … Mg(II) acetate ... Magnesium di(acetate) …
Matched Name: … Magnesium acetate …
Matched Name: … Magnesium acetate …
alpha-Tocopherol acetate
Alpha-tocopherol is the primary form of vitamin E that is preferentially used by the human body to meet appropriate dietary requirements. In particular, the RRR-alpha-tocopherol (or sometimes called the d-alpha-tocopherol stereoisomer) stereoisomer is considered the natural formation of alpha-tocopherol and generally exhibits the greatest bioavailability out of all of the...
Approved
Matched Synonyms: … Tocopherol acetate ... Tocopheryl acetate ... Vitamin E acetate …
Matched Name: … alpha-Tocopherol acetate …
Matched Description: … Moreover, RRR-alpha-tocopherol acetate is a relatively stabilized form of vitamin E that is most commonly ... Alpha-tocopherol acetate is subsequently most commonly indicated for dietary supplementation in individuals …
Matched Name: … alpha-Tocopherol acetate …
Matched Description: … Moreover, RRR-alpha-tocopherol acetate is a relatively stabilized form of vitamin E that is most commonly ... Alpha-tocopherol acetate is subsequently most commonly indicated for dietary supplementation in individuals …
Segesterone acetate
Segesterone acetate is a steroidal progestin or synthetic progesterone and a 19-norprogesterone derivative with no CH3 group radical in position 6 . In animal studies, segesterone acetate was shown to be one of the most potent progestins . It mediates progestational activity 100 times higher than that of progesterone ....
Approved
Experimental
Investigational
Matched Synonyms: … Segesterone acetate ... 17-Hydroxy-16-methylene-19-norpregn-4-ene-3,20-dione acetate …
Matched Name: … Segesterone acetate …
Matched Iupac: … methylidene-7-oxo-1H,2H,3H,3aH,3bH,4H,5H,7H,8H,9H,9aH,9bH,10H,11H,11aH-cyclopenta[a]phenanthren-1-yl acetate …
Matched Description: … Segesterone acetate is a steroidal progestin or synthetic progesterone and a 19-norprogesterone derivative ... In animal studies, segesterone acetate was shown to be one of the most potent progestins [A37090]. ... Segesterone acetate binds selectively to progesterone receptors and not androgen receptors [A37083]. …
Matched Name: … Segesterone acetate …
Matched Iupac: … methylidene-7-oxo-1H,2H,3H,3aH,3bH,4H,5H,7H,8H,9H,9aH,9bH,10H,11H,11aH-cyclopenta[a]phenanthren-1-yl acetate …
Matched Description: … Segesterone acetate is a steroidal progestin or synthetic progesterone and a 19-norprogesterone derivative ... In animal studies, segesterone acetate was shown to be one of the most potent progestins [A37090]. ... Segesterone acetate binds selectively to progesterone receptors and not androgen receptors [A37083]. …
Nomegestrol acetate
Nomegestrol acetate, also known as NOMAC, is a progestin used in oral contraceptives, menopausal hormone therapy, and for the treatment of gynecological disorders.
Approved
Investigational
Matched Synonyms: … Nomegestrol acetate ... 17-alpha-Hydroxy-6-methyl-19-norpregna-4,6-diene-3,20-dione acetate …
Matched Name: … Nomegestrol acetate …
Matched Iupac: … acetyl-5,11a-dimethyl-7-oxo-1H,2H,3H,3aH,3bH,7H,8H,9H,9aH,9bH,10H,11H,11aH-cyclopenta[a]phenanthren-1-yl acetate …
Matched Description: … Nomegestrol acetate, also known as NOMAC, is a progestin used in oral contraceptives, menopausal hormone …
Matched Name: … Nomegestrol acetate …
Matched Iupac: … acetyl-5,11a-dimethyl-7-oxo-1H,2H,3H,3aH,3bH,7H,8H,9H,9aH,9bH,10H,11H,11aH-cyclopenta[a]phenanthren-1-yl acetate …
Matched Description: … Nomegestrol acetate, also known as NOMAC, is a progestin used in oral contraceptives, menopausal hormone …
Resorcinol monoacetate
Approved
Experimental
Matched Synonyms: … Resorcinol acetate …
Matched Iupac: … 3-hydroxyphenyl acetate …
Matched Iupac: … 3-hydroxyphenyl acetate …
Levacetylmethadol
Levacetylmethadol is a narcotic analgesic with a long onset and duration of action. It is used mainly in the treatment of narcotic dependence.
Levacetylmethadol was withdrawn from use in the European Union due to its high risk of QT interval prolongation. The production of levacetylmethadol in the US has ceased...
Approved
Investigational
Withdrawn
Matched Synonyms: … Levomethadyl acetate ... Levo-methadyl acetate ... (1S,4S)-4-(dimethylamino)-1-ethyl-2,2-diphenylpentyl acetate …
Matched Iupac: … (3S,6S)-6-(dimethylamino)-4,4-diphenylheptan-3-yl acetate …
Matched Iupac: … (3S,6S)-6-(dimethylamino)-4,4-diphenylheptan-3-yl acetate …
Dexmethylphenidate
Dexmethylphenidate is the dextrorotary form of methylphenidate introduced in 2002 . It is a norepinephrine-dopamine reuptake inhibitor (NDRI) and thus a psychostimulant . It is used for treatment of Attention Deficit Hyperactivity Disorder (ADHD)[Label,A177181]. The d-isomer is thought to have greater effect with fewer side effects than the l-isomer or...
Approved
Investigational
Matched Synonyms: … methyl (R)-phenyl[(R)-piperidin-2-yl]acetate …
Matched Iupac: … methyl (2R)-2-phenyl-2-[(2R)-piperidin-2-yl]acetate …
Matched Iupac: … methyl (2R)-2-phenyl-2-[(2R)-piperidin-2-yl]acetate …
Cabazitaxel
Cabazitaxel is a taxoid synthesized from 10-deacetylbaccatin III, a compound isolated from the yew tree. As a second-generation semisynthetic microtubule inhibitor, cabazitaxel stabilizes microtubules and induces tumour cell death. Due to its low affinity for the P-glycoprotein (P-gp) efflux pump, cabazitaxel can more readily penetrate the blood–brain barrier compared to...
Approved
Matched Synonyms: … -TRIYL 4-ACETATE 2-BENZOATE 13-((2R,3S)-3-(((TERT-BUTOXY)CARBONYL)AMINO)-2-HYDROXY-3-PHENYLPROPANOATE …
Diltiazem
Diltiazem is a benzothiazepine derivative with antihypertensive and vasodilating properties. Approved in 1982 by the FDA, it is a member of the non-dihydropyridine calcium channel blockers drug class. It works through various mechanisms of action, but it primarily works by inhibiting the calcium influx into cardiac and vascular smooth muscle...
Approved
Investigational
Matched Synonyms: … cis-5-[2-(dimethylamino)ethyl]-2,3-dihydro-3-hydroxy-2-(p-methoxyphenyl)-1,5-benzothiazepin-4(5H)-one acetate ... -5-(2-(dimethylamino)ethyl)-2-(4-methoxyphenyl)-4-oxo-2,3,4,5-tetrahydrobenzo[b][1,4]thiazepin-3-yl acetate …
Matched Iupac: … 3S)-5-[2-(dimethylamino)ethyl]-2-(4-methoxyphenyl)-4-oxo-2,3,4,5-tetrahydro-1,5-benzothiazepin-3-yl acetate …
Matched Iupac: … 3S)-5-[2-(dimethylamino)ethyl]-2-(4-methoxyphenyl)-4-oxo-2,3,4,5-tetrahydro-1,5-benzothiazepin-3-yl acetate …
Abiraterone
Abiraterone is a potent, irreversible, and selective inhibitor of 17 αhydroxylase/C17,20-lyase (CYP17), an enzyme expressed in testicular, adrenal, and prostatic tumour tissues, to regulate androgen biosynthesis.[A3811, A260880, L40968] Abiraterone was first approved by the FDA and EMA on April, July, and September 2011, respectively. It is used to treat metastatic...
Approved
Matched Description: … abiraterone has poor oral bioavailability and is susceptible to hydrolysis by esterases, abiraterone acetate …
Matched Salts name: … Abiraterone acetate …
Matched Products: … Abiraterone Acetate ... Abiraterone acetate ... Abiratred Abiraterone Acetate Tablets 250mg …
Matched Salts name: … Abiraterone acetate …
Matched Products: … Abiraterone Acetate ... Abiraterone acetate ... Abiratred Abiraterone Acetate Tablets 250mg …
Norethisterone
Norethisterone, also known as norethindrone, is a synthetic progestational hormone belonging to the 19-nortestosterone-derived class of progestins. It is further classified as a second-generation progestin, along with levonorgestrel and its derivatives, and is the active form of several other progestins including norethynodrel and lynestrenol. Norethisterone mimics the actions of endogenous...
Approved
Matched Mixtures name: … Estradiol / Norethindrone Acetate ... Estradiol / Norethindrone Acetate ... Estradiol / Norethindrone Acetate …
Matched Salts name: … Norethisterone acetate …
Matched Products: … Norethindrone Acetate ... Norethindrone acetate …
Matched Salts name: … Norethisterone acetate …
Matched Products: … Norethindrone Acetate ... Norethindrone acetate …
Ulipristal
Ulipristal is a selective progesterone receptor modulator used for the purposes of emergency contraception (Ella) and for the treatment of uterine fibroids (Fibristal). It is a derivative of 19-norprogesterone and has both antagonistic and partial agonist activity at the progesterone receptor. It also binds to glucocorticoid receptor, however compared to...
Approved
Matched Salts name: … Ulipristal acetate …
Matched Products: … Ulipristal Acetate Gedeon Richter ... Ulipristal acetate Hexal 30 mg - Filmtabletten …
Matched Products: … Ulipristal Acetate Gedeon Richter ... Ulipristal acetate Hexal 30 mg - Filmtabletten …
Methylprednisolone
Methylprednisolone is a prednisolone derivative glucocorticoid with higher potency than prednisone. It was first described in the literature in the late 1950s.[A188811,A188814]
Methylprednisolone was granted FDA approval on 24 October 1957. In the outbreak of COVID-19, low dose methylprednisolone-based therapy was successful in treating COVID-19-associated pneumonia in one patient with...
Approved
Vet approved
Matched Salts name: … Methylprednisolone acetate …
Matched Products: … Methylprednisolone Acetate ... Methylprednisolone acetate ... Methylprednisolone Acetate Injectable Suspension USP …
Matched Products: … Methylprednisolone Acetate ... Methylprednisolone acetate ... Methylprednisolone Acetate Injectable Suspension USP …
Desmopressin
Desmopressin (dDAVP), a synthetic analogue of 8-arginine vasopressin (ADH), is an antidiuretic peptide drug modified by deamination of 1-cysteine and substitution of 8-L-arginine by 8-D-arginine. ADH is an endogenous pituitary hormone that has a crucial role in the control of the water content in the body. Upon release from the...
Approved
Matched Description: … The active ingredient in most formulations is desmopressin acetate. ... Nocdurna, or desmopressin acetate, was approved by the FDA on June 21st, 2018 for the treatment of nocturia …
Matched Salts name: … Desmopressin acetate ... Desmopressin acetate anhydrous …
Matched Products: … Desmopressin Acetate ... Desmopressin acetate …
Matched Salts name: … Desmopressin acetate ... Desmopressin acetate anhydrous …
Matched Products: … Desmopressin Acetate ... Desmopressin acetate …
Betamethasone
Betamethasone is a long-acting corticosteroid with immunosuppressive and antiinflammatory properties. It can be used topically to manage inflammatory skin conditions such as eczema, and parenterally to manage several disease states including autoimmune disorders. Betamethasone has potent glucocorticoid activity and negligible mineralocorticoid activity.
Approved
Vet approved
Matched Mixtures name: … Betamethasone Sodium Phosphate and Betamethasone Acetate ... Betamethasone Sodium Phosphate and Betamethasone Acetate ... Betamethasone Sodium Phosphate and Betamethasone Acetate …
Matched Salts name: … Betamethasone acetate …
Matched Salts name: … Betamethasone acetate …
Zuclopenthixol
Zuclopenthixol, also known as Zuclopentixol or Zuclopenthixolum, is an antipsychotic agent. Zuclopenthixol is a thioxanthene-based neuroleptic with therapeutic actions similar to the phenothiazine antipsychotics. It is an antagonist at D1 and D2 dopamine receptors. Major brands of zuclopenthixol are Cisordinol, Acuphase, and Clopixol. This drug is a liquid. This compound...
Approved
Investigational
Matched Salts name: … Zuclopenthixol acetate …
alpha-Tocopherol succinate
Alpha-tocopherol is the primary form of vitamin E that is preferentially used by the human body to meet appropriate dietary requirements. In particular, the RRR-alpha-tocopherol (or sometimes called the d-alpha-tocopherol stereoisomer) stereoisomer is considered the natural formation of alpha-tocopherol and generally exhibits the greatest bioavailability out of all of the...
Approved
Nutraceutical
Vet approved
Tesamorelin
Tesamorelin is a stabilized synthetic peptide analogue of the hypothalamic peptide, Growth Hormone Releasing Hormone (GHRH) indicated for the reduction of excess abdominal fat in HIV-infected patients with lipodystrophy. Lipodystrophy is a metabolic condition characterized by insulin resistance, fat redistribution, and hyperlipidemia associated with antiretroviral therapy for HIV infection.
Approved
Investigational
Matched Salts name: … Tesamorelin acetate …
Prednisolone
Prednisolone is a glucocorticoid similar to cortisol used for its anti-inflammatory, immunosuppressive, anti-neoplastic, and vasoconstrictive effects. Prednisolone was granted FDA approval on 21 June 1955.
Approved
Vet approved
Matched Products: … STERILE PREDNISOLONE ACETATE SUSPENSION …
Displaying drugs 1 - 25 of 398 in total