Design of enzyme inhibitors using iterative protein crystallographic analysis.
Article Details
- CitationCopy to clipboard
Appelt K, Bacquet RJ, Bartlett CA, Booth CL, Freer ST, Fuhry MA, Gehring MR, Herrmann SM, Howland EF, Janson CA, et al.
Design of enzyme inhibitors using iterative protein crystallographic analysis.
J Med Chem. 1991 Jul;34(7):1925-34.
- PubMed ID
- 2066965 [ View in PubMed]
- Abstract
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DrugBank Data that Cites this Article
- Binding Properties
Drug Target Property Measurement pH Temperature (°C) 10-Propargyl-5,8-Dideazafolic Acid Thymidylate synthase Ki (nM) 12 N/A N/A Details