Histamine-3 (H3) Receptor Antagonists/Inverse Agonists

Name
Histamine-3 (H3) Receptor Antagonists/Inverse Agonists
Accession Number
DBCAT005677
Description

Not Available

Drugs
DrugDrug Description
PitolisantAn antagonist and inverse agonist at the histamine H3 receptor that is used to treat narcolepsy in adults.
Drugs & Drug Targets
DrugTargetType
PitolisantHistamine H3 receptortarget
PitolisantCytochrome P450 3A4enzyme
PitolisantCytochrome P450 2D6enzyme
PitolisantCytochrome P450 1A2enzyme
PitolisantCytochrome P450 2B6enzyme
PitolisantSolute carrier family 22 member 1transporter
PitolisantPotassium voltage-gated channel subfamily H member 2target
PitolisantSerum albumincarrier
PitolisantAlpha-1-acid glycoprotein 1carrier