Neuroactive Steroid Gamma-Aminobutyric Acid (GABA) A Receptor Positive Modulators

Name
Neuroactive Steroid Gamma-Aminobutyric Acid (GABA) A Receptor Positive Modulators
Accession Number
DBCAT005699
Description

Neuroactive steroid agents which positively modulate GABA-A receptors.

Drugs
DrugDrug Description
BrexanoloneBrexanolone is a synthetic neuroactive steroid gamma-aminobutyric acid A (GABA(a)) receptor positive modulator indicated for the treatment of postpartum depression (PPD) in adult women [FDA Label][A176080, A176083, F4063, F4066, F4072].
Drugs & Drug Targets
DrugTargetType
BrexanoloneGABA(A) Receptortarget
BrexanoloneAldose reductaseenzyme