A New Era in Oncology: Tennessee's $20 Million Leap into Radiopharmaceutical Research
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Drug Name
Type
Name
target
enzyme
carrier
transporter
Clear
2-[1-(4-chlorobenzoyl)-5-methoxy-2-methyl-1H-indol-3-yl]-n-[(1S)-1-(hydroxymethyl)propyl]acetamide
target
Prostaglandin G/H synthase 1
Details
+/-METHYL 4-(AMINOIMINOMETHYL)-BETA-[3- INH (AMINOIMINO)PHENYL]BENZENE PENTANOATE
target
Trypsin-1
Details
[4-(4-PHENYL-PIPERIDIN-1-YL)-BENZENESULFONYLAMINO]-ACETIC ACID
target
Stromelysin-1
Details
[2-(5-Mercapto-[1,3,4]thiadiazol-2-ylcarbamoyl)-1-phenyl-ethyl]-carbamic acid benzyl ester
target
Stromelysin-1
Details
2-[3-(5-Mercapto-[1,3,4]thiadiazol-2yl)-ureido]-N-methyl-3-pentafluorophenyl-propionamide
target
Stromelysin-1
Details
2-(ACETYL-HYDROXY-AMINO)-4-METHYL-PENTANOIC ACID METHYL ESTER
target
Thermolysin
Details
(RP,SP)-O-(2R)-(1-PHENOXYBUT-2-YL)-METHYLPHOSPHONIC ACID CHLORIDE
target
Lipase
Details
N-[(1R)-3-(4-HYDROXYPHENYL)-1-METHYLPROPYL]-2-(2-PHENYL-1H-INDOL-3-YL)ACETAMIDE
target
Estrogen receptor alpha
Details
Indoxyl sulfate
carrier
Serum albumin
Details
N~3~-[3-(1H-INDOL-6-YL)BENZYL]PYRIDINE-2,3-DIAMINE
target
Beta-secretase 1
Details
N~3~-[5-(1H-INDOL-6-YL)-2-(PYRIDIN-2-YLMETHOXY)BENZYL]PYRIDINE-2,3-DIAMINE
target
Beta-secretase 1
Details
H-89
target
cAMP-dependent protein kinase inhibitor alpha
Details
H-89
target
Interferon-induced, double-stranded RNA-activated protein kinase
Details
H-89
target
cAMP-dependent protein kinase catalytic subunit alpha
Details
H-89
target
Serine/threonine-protein kinase haspin
Details
5-(2-methylpiperazine-1-sulfonyl)isoquinoline
target
cAMP-dependent protein kinase catalytic subunit alpha
Details
5-(2-methylpiperazine-1-sulfonyl)isoquinoline
target
cAMP-dependent protein kinase inhibitor alpha
Details
N-[2-(METHYLAMINO)ETHYL]-5-ISOQUINOLINESULFONAMIDE
target
cAMP-dependent protein kinase inhibitor alpha
Details
N-[2-(METHYLAMINO)ETHYL]-5-ISOQUINOLINESULFONAMIDE
target
cAMP-dependent protein kinase catalytic subunit alpha
Details
{4-[(CARBOXYMETHOXY)CARBONYL]-3,3-DIOXIDO-1-OXONAPHTHO[1,2-D]ISOTHIAZOL-2(1H)-YL}ACETIC ACID
target
Aldose reductase
Details
2-(CARBOXYMETHYL)-1-OXO-1,2-DIHYDRONAPHTHO[1,2-D]ISOTHIAZOLE-4-CARBOXYLIC ACID 3,3-DIOXIDE
target
Aldose reductase
Details
5-(3-{3-[3-HYDROXY-2-(METHOXYCARBONYL)PHENOXY]PROPENYL}PHENYL)-4-(HYDROXYMETHYL)ISOXAZOLE-3-CARBOXYLIC ACID
target
Tyrosine-protein phosphatase non-receptor type 1
Details
ISOTHIAZOLIDINONE ANALOG
target
Tyrosine-protein phosphatase non-receptor type 1
Details
(2S)-2-{[3-(3-aminophenyl)imidazo[1,2-b]pyridazin-6-yl]amino}-3-methylbutan-1-ol
target
Serine/threonine-protein kinase haspin
Details
4-{[5-chloro-4-(1H-indol-3-yl)pyrimidin-2-yl]amino}-N-ethylpiperidine-1-carboxamide
target
Mitogen-activated protein kinase 10
Details
N-anthracen-2-yl-5-methyl[1,2,4]triazolo[1,5-a]pyrimidin-7-amine
target
Dihydroorotate dehydrogenase (quinone), mitochondrial
Details
(2R)-3-{[(BENZYLAMINO)CARBONYL]AMINO}-2-HYDROXYPROPANOIC ACID
target
Chymotrypsin-like elastase family member 1
Details
5-methyl-N-[4-(trifluoromethyl)phenyl][1,2,4]triazolo[1,5-a]pyrimidin-7-amine
target
Dihydroorotate dehydrogenase (quinone), mitochondrial
Details
SU-11652
target
Calcium/calmodulin-dependent protein kinase type 1G
Details
(3Z)-1-[(6-fluoro-4H-1,3-benzodioxin-8-yl)methyl]-4-[(E)-2-phenylethenyl]-1H-indole-2,3-dione 3-oxime
target
Mitogen-activated protein kinase 10
Details
Displaying targets
21211 - 21240
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