Identification of the first retinoid X, receptor homodimer antagonist.
Article Details
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Canan Koch SS, Dardashti LJ, Hebert JJ, White SK, Croston GE, Flatten KS, Heyman RA, Nadzan AM
Identification of the first retinoid X, receptor homodimer antagonist.
J Med Chem. 1996 Aug 16;39(17):3229-34.
- PubMed ID
- 8765503 [ View in PubMed]
- Abstract
Not Available
DrugBank Data that Cites this Article
- Binding Properties
Drug Target Property Measurement pH Temperature (°C) Tretinoin Retinoic acid receptor RXR-alpha Ki (nM) 8 N/A N/A Details Tretinoin Retinoic acid receptor RXR-beta Ki (nM) 9 N/A N/A Details Tretinoin Retinoic acid receptor RXR-gamma Ki (nM) 14 N/A N/A Details